GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,008 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(193 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
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Found 5977 products of "GPCR/G-Protein"
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Gastrin I, rat
CAS:Gastrin I, rat is a peptide hormone that effectively stimulates gastric acid secretion.Formula:C94H128N22O31S2Color and Shape:SolidMolecular weight:2126.3Neuropeptide Y (3-36) (porcine)
CAS:Neuropeptide Y (3-36) (porcine) is a potent, selective agonist at NPY Y2 receptors, increasing feeding in rats.Formula:C176H271N53O54Color and Shape:SolidMolecular weight:3993.36Kisspeptin-54(human) TFA
Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.Formula:C258H401N79O78·C2HF3O2Color and Shape:SolidMolecular weight:5971.45Cyclic SSTR agonist octreotide
Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .Formula:C53H71N11O14S2Color and Shape:SolidMolecular weight:1150.33[Asu1,6-Arg8]Vasopressin
CAS:[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.Formula:C48H68N14O12Color and Shape:SolidMolecular weight:1033.14(2R,2R)-PF-07258669
CAS:(2R,2R)-PF-07258669' is an antagonist for the MC4R (melanocortin 4 receptor), primarily studied for its role in regulating appetite and energy expenditure.
Formula:C25H27FN6O2Color and Shape:SolidMolecular weight:462.52Melanostatin, frog
CAS:Melanostatin, frog, is an inhibitor of α-melanocyte-stimulating hormone (α-MSH) release, with an IC50 of 60 nM [1] [2].Formula:C189H285N53O57SColor and Shape:SolidMolecular weight:4243.67α-CGRP(human) TFA
α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as aFormula:C165H268F3N51O51S2Color and Shape:SolidMolecular weight:3903.33Neuropeptide Y (3-36) (human, rat)
CAS:Neuropeptide Y (3-36) is a Y2 receptor agonist that limits norepinephrine release, produced by DPP4 from NPY.Formula:C175H269N53O54SColor and Shape:SolidMolecular weight:4011.5Endothelin 1 (swine, human), Alexa Fluor 488-labeled
Synthetic human/swine Endothelin 1 peptide, tagged with Alexa Fluor 488, acts as a strong vasoconstrictor via ET A/B receptors.Color and Shape:SolidMolecular weight:2848.4Amylin (IAPP), feline TFA
Amylin (IAPP), feline TFA: 37-amino acid peptide; inhibits insulin/glucagon; secreted by pancreatic β-cells.Formula:C167H271F3N52O56S2Color and Shape:SolidMolecular weight:4024.47d[Cha4]-AVP TFA
d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.Formula:C52H72F3N13O13S2Color and Shape:SolidMolecular weight:1208.33(Pro34)-Peptide YY (human)
CAS:(Pro34)-Peptide YY (human) is a highly Y 1 -selective full agonist of Peptide YY /neuropeptide Y receptors [1] .Formula:C194H294N54O56Color and Shape:SolidMolecular weight:4278.73Lys-[Hyp3]-Bradykinin
CAS:Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.Formula:C56H85N17O13Color and Shape:SolidMolecular weight:1204.38des-Gln14-Ghrelin TFA
Des-Gln14-Ghrelin TFA, a ligand for GHSR, boosts [Ca2+]i with an EC50 of 2.4 nM in CHO-GHSR62 cells.Formula:C144H238F3N43O42Color and Shape:SolidMolecular weight:3300.69Neurokinin A(4-10) TFA
Neurokinin A (4-10) TFA is a tachykinin NK 2 receptor agonist [1] .Formula:C36H55F3N8O12SColor and Shape:SolidMolecular weight:880.93Tirzepatide TFA
Tirzepatide TFA, a GIP and GLP-1 agonist, targets type 2 diabetes treatment.Formula:C227H349F3N48O70Color and Shape:SolidMolecular weight:4927.47OXA(17-33) TFA
OXA(17-33) TFA: Potent OX1 agonist, ~23x more selective for OX1 (EC50=8.29nM) than OX2 (187nM).Formula:C81H126F3N23O24Color and Shape:SolidMolecular weight:1863Spantide I TFA
Spantide I TFA is a selective NK1 antagonist (230 nM); much less for NK2 (8150 nM); it modulates cytokines to prevent corneal perforation.Formula:C77H109F3N20O15Color and Shape:SolidMolecular weight:1611.81a-Helical Corticotropin Releasing Factor (12-41)
CAS:α-Helical CRF (12-41), a 30-aa analog, curbs CRF's ACTH-stimulating effect.Formula:C152H251N43O47S2Color and Shape:SolidMolecular weight:3497.01
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