Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,715 products)
- Apoptosis(6,164 products)
- Cell Cycle/Checkpoint(4,727 products)
- Chromatin/Epigenetics(2,400 products)
- Cytoskeletal Signaling(1,492 products)
- DNA Damage/DNA Repair(2,928 products)
- Endocrinology/Hormones(3,653 products)
- Enzyme(3,661 products)
- GPCR/G-Protein(8,861 products)
- Immunology and Inflammation(3,801 products)
- Influenza Virus(299 products)
- JAK/STAT signaling(412 products)
- MAPK Signaling(1,239 products)
- Membrane Transporter/Ion Channel(2,979 products)
- Metabolism(10,029 products)
- Microbiology/Virology(7,445 products)
- Neuroscience(10,281 products)
- Other Inhibitors(36,478 products)
- Oxidation-Reduction(44 products)
- PI3K/Akt/mTOR Signaling(1,443 products)
- Proteases/Proteasome(1,695 products)
- Stem Cell and Derivatives(829 products)
- Tyrosine Kinase/Adaptors(2,035 products)
- Ubiquitination(1,693 products)
Show 16 more subcategories
Found 66676 products of "Inhibitors"
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Demethyleneberberine chloride
CAS:Demethyleneberberine chloride, a natural mitochondria-targeted antioxidant, mitigates colitis in mice and suppresses inflammatory responses by blocking the NF-Formula:C19H18ClNO4Purity:98%Color and Shape:SolidMolecular weight:359.8PDE5-IN-42
CAS:PDE5-IN-42 is a selective inhibitor of second-generation phosphodiesterase type 5 (PDE5).Formula:C23H31N7O3Purity:98%Color and Shape:SolidMolecular weight:453.54GLUT4 activator 1
CAS:GLUT4 activator 1 is a potent glucose transporter type 4 (GLUT4) translocation activator (EC50: 0.14 μM).Formula:C23H21FN4O3SPurity:98%Color and Shape:SolidMolecular weight:452.5PCSK9-IN-20
CAS:<p>PCSK9-IN-20 (Compound 3i) is a PCSK9 inhibitor exhibiting an IC50 value of 3.96 µM, shown to reduce PCSK9 and enhance LDLR protein levels in vitro [1].</p>Formula:C27H32N6O5S2Color and Shape:SolidMolecular weight:584.71ICMT-IN-38
CAS:<p>ICMT-IN-38 (Compound 42) is an ICMT inhibitor, demonstrating an IC50 value of 0.049 μM [1].</p>Formula:C22H28ClNOColor and Shape:SolidMolecular weight:357.92INX-SM-56
CAS:<p>INX-SM-56 is a cytotoxin designed for the synthesis of an anti-VISTA (V-region Immunoglobulin-containing Suppressor of T cell Activation [1]) antibody-agent</p>Formula:C32H36N2O6SColor and Shape:SolidMolecular weight:576.7cis-Indatraline hydrochloride
CAS:Cis-indatraline hydrochloride (cis-Lu 19-005) is an active compound utilized in the research of neurodegenerative diseases [1].Formula:C16H16Cl3NColor and Shape:SolidMolecular weight:328.66(R)-FT709
CAS:<p>(R)-FT709 is an active compound utilized in cancer research [1].</p>Formula:C23H22N4O7SColor and Shape:SolidMolecular weight:498.51PZ-1190
CAS:<p>PZ-1190, a multitarget ligand for serotonin and dopamine receptors, exhibits potential antipsychotic activity in rodents [1].</p>Formula:C27H30N4O2S2Purity:98%Color and Shape:SolidMolecular weight:506.68DC_AC50
CAS:"DC_AC50 inhibits Atox1/CCS to reduce cancer cell growth and prevent chemotherapy resistance."Formula:C17H12BrF2N3OSPurity:99.84% - 99.9%Color and Shape:SolidMolecular weight:424.26BD-AcAc 2
CAS:BD-AcAc 2 (Ketone Ester) is a ketone monoester and can be used as a source of oral nutritional ketones.Formula:C8H16O4Purity:99.62%Color and Shape:SolidMolecular weight:176.21IM156
CAS:IM156, a Metformin derivative, activates AMPK, enhances cognition in aging animals, and inhibits OXPHOS in solid tumor research.Formula:C13H16F3N5OPurity:99.67%Color and Shape:SolidMolecular weight:315.29CXCR2 antagonist 2
CAS:<p>CXCR2 antagonist 2 is a potent CXCR2 antagonist for cancer immunotherapy with an IC 50 value of 95 nM.</p>Formula:C17H17FN2O4SColor and Shape:SolidMolecular weight:364.39Fosthiazate
CAS:<p>Fosthiazate is a broad-spectrum nematicide that combats a range of plant parasitic nematodes such as Meloidogyne spp., Globodera spp., and Pratylenchus spp., by</p>Formula:C9H18NO3PS2Purity:97.78%Color and Shape:SolidMolecular weight:283.35Dothiepin
CAS:Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancingFormula:C19H21NSPurity:98%Color and Shape:SolidMolecular weight:295.44BMS-262084
CAS:BMS-262084 is a potent selective β-lactam trypsin inhibitor with therapeutic potential in the treatment of asthma.Formula:C18H31N7O5Color and Shape:SolidMolecular weight:425.48KUNG38
CAS:KUNG38 is a purine-based inhibitor of Grp94.Formula:C18H16Cl2N2O5Purity:98%Color and Shape:SolidMolecular weight:411.24AZD4747
CAS:<p>AZD4747 is an inhibitor of the mutant GTPase KRASG12C that hasial antitumor activity for the study of pancreatic and colorectal adenocarcinoma.</p>Formula:C24H22ClFN2O3Purity:99.36%Color and Shape:SolidMolecular weight:440.89O-allyl-AP
O-allyl-AP is a neuroprotective and proliferative agent with significantly higher stimulatory effect than that of allopregnanolone.Formula:C24H38O2Color and Shape:SolidMolecular weight:358.57Mps1-IN-10
CAS:<p>Mps1-IN-6 (Compound 9) is a highly effective Mps1 inhibitor with an IC50 value of 6.4 nM and exhibits significant anti-proliferation and anti-tumor effects on</p>Formula:C24H27N7O2Color and Shape:SolidMolecular weight:445.52THR-β modulator-1
CAS:<p>THR-β Modulator-1 (Compound 1a) is a potent modulator of the thyroid hormone receptor β, utilized in the study of thyroid hormone receptor-associated disorders</p>Formula:C17H14Cl2N6O4Color and Shape:SolidMolecular weight:437.24D1N52
CAS:D1N52 is a potent inhibitor of the SARS-CoV-2 3CL protease, demonstrating an inhibitory concentration half-maximal (IC50) value of 0.53 μM [1].Formula:C20H13F4N5O3Purity:98%Color and Shape:SolidMolecular weight:447.34G-5555
CAS:<p>G-5555 is a potent inhibitor of p21-activated kinase 1 (PAK1) (Kis: 3.7 nM and 11 nM for PAK1 and PAK2, respectively).</p>Formula:C25H25ClN6O3Purity:99.76% - 99.84%Color and Shape:SolidMolecular weight:492.96E6130
CAS:E6130 may be effective in the treatment of inflammatory bowel disease and is a highly selective CX3CR1 regulator for oral administration.Formula:C28H37ClF3N3O3Color and Shape:SolidMolecular weight:556.06Tecarfarin sodium
CAS:Tecarfarin sodium is a novel orally active non-competitive vitamin K epoxide reductase antagonist. Tecarfarin sodium has the antithrombotic activity.Formula:C21H13F6NaO5Purity:98%Color and Shape:SolidMolecular weight:482.316CEPN
CAS:<p>6CEPN is a Cyclooxygenase-1 inhibitor that acts by suppressing colorectal cancer growth.</p>Formula:C23H18O5Color and Shape:SolidMolecular weight:374.39L-ANAP
CAS:<p>L-ANAP is a polarity-sensitive and genetically encodable fluorescent unnatural amino acid.</p>Formula:C15H16N2O3Purity:98%Color and Shape:SolidMolecular weight:272.3T-00127_HEV1
CAS:T-00127_HEV1 is an inhibitor of phosphatidylinositol 4-kinase III beta(PI4KIIIβ, IC50 = 60 nM).Formula:C22H29N5O3Purity:99.89%Color and Shape:SolidMolecular weight:411.5TAK-659
CAS:TAK-659 is a spleen tyrosine kinase (SYK) inhibitor.Formula:C17H21FN6OPurity:98%Color and Shape:SolidMolecular weight:344.39Mal-Pc
CAS:Mal-Pc, a maleimide phthalocyanine, depletes GSH to reduce aggregation and boost ROS, improving PDT against cancer.Formula:C46H28N10O8SiPurity:98%Color and Shape:SolidMolecular weight:876.86AGN 194310
CAS:AGN 194310 (VTP-194310) is retinioic acid receptors (RARs) pan-antagonist. The Kd values of 3 nM, 2 nM, 5 nM for RARα, RARβ, RARγ, respectively[1][2].Formula:C28H24O2SColor and Shape:SolidMolecular weight:424.55Pim-1 kinase inhibitor 5
CAS:<p>Pim-1 kinase inhibitor 5 (Compound 4c), with an IC50 of 0.61 μM, exhibits cytotoxicity against various cancer cell lines, including HepG2, MCF-7, PC3, and HCT-</p>Formula:C22H13Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:406.26LEQ-506 HCl (1204975-42-7 free base)
LEQ506 is an orally bioavailable small-molecule Smoothened antagonist. It also has a potential antineoplastic activity.Formula:C27H31Cl2N5OPurity:98%Color and Shape:SolidMolecular weight:512.481-Deazaadenosine
CAS:1-Deazaadenosine, an adenosine deaminase inhibitor (Ki: 0.66 μM), may treat cancer, particularly lymphoproliferative disorders.Formula:C11H14N4O4Purity:98%Color and Shape:SolidMolecular weight:266.25JNK3 inhibitor-3
CAS:JNK3 Inhibitor-3 selectively blocks JNK3 (>4.1 nM), crosses the blood-brain barrier, is orally active, and improves memory in dementia mice.Formula:C26H25N7O2Purity:98%Color and Shape:SolidMolecular weight:467.52GGTI-2133
CAS:GGTI-2133: potent GGTase I inhibitor, IC50=38 nM; blocks inflammatory cell invasion in mice asthma.Formula:C27H28N4O3Purity:99.75%Color and Shape:SolidMolecular weight:456.54AAK1-IN-3
CAS:<p>AAK1-IN-3: Brain-penetrant AAK1 inhibitor for neuropathic pain research; IC50=11 nM.</p>Formula:C20H20N4Color and Shape:SolidMolecular weight:316.44A3-SC8
CAS:<p>4A3-SC8 is a modular, degradable dendrimer facilitating the extension of survival in aggressive liver cancer models through the delivery of small RNAs [1].</p>Formula:C75H139N3O16S4Purity:99.87%Color and Shape:SolidMolecular weight:1467.18MCT1-IN-3
CAS:<p>MCT1-IN-3 is a monocarboxylate transporter 1 (MCT1) inhibitor.</p>Formula:C22H19N3O4Purity:99.35%Color and Shape:SoildMolecular weight:389.4MK-0674
CAS:MK-0674 is a cathepsin K inhibitor (IC50: 0.4 nM) that inhibits Cat B, Cat F, Cat L, and Cat S for metabolism-related diseases.Formula:C26H27F6N3O2Purity:97.3% - 99.91%Color and Shape:SolidMolecular weight:527.5αvβ1 integrin-IN-1
CAS:<p>αvβ1 integrin-IN-1 is a potent and selective inhibitor of αvβ1 integrin (IC50 of 0.63 nM) with antifibrotic effects.</p>Formula:C26H34N6O6SPurity:99.74% - >99.99%Color and Shape:SolidMolecular weight:558.65Moracin C
CAS:<p>Moracin C, a natural compound found in Morus mesozygia, Morus alba var.</p>Formula:C19H18O4Purity:99.77% - >99.99%Color and Shape:SolidMolecular weight:310.34Melengestrol acetate
CAS:<p>Melengestrol acetate is a derivative of progesterone and acts as a corticosteroid hormone.</p>Formula:C25H32O4Purity:98.68% - 98.79%Color and Shape:SolidMolecular weight:396.52STAT6-IN-2
CAS:STAT6-IN-2(R)-84 is a STAT6 inhibitor that inhibits the secretion of eotaxin-3 and the tyrosine phosphorylation of STAT6.Formula:C28H31N5O2Purity:99.67%Color and Shape:SolidMolecular weight:469.58Tefinostat
CAS:<p>Tefinostat (CHR-2845) is a potent monocyte/macrophage-targeted histone deacetylase (HDAC) inhibitor.</p>Formula:C28H37N3O5Purity:99.83%Color and Shape:SolidMolecular weight:495.61Rovatirelin
CAS:Rovatirelin (S-0373) is a TRH analog that improves motor dysfunction in a rat model of cytosine arabinoside-induced spinal cerebellar degeneration.Formula:C16H22N4O4SPurity:99.59%Color and Shape:SolidMolecular weight:366.43L-DABA hydrobromide
CAS:<p>L-DABA hydrobromide (L-2,4-Diaminobutyric acid hydrobromide) , GABA transaminase inhibitor with antitumor and anticonvulsant activity.</p>Formula:C4H11BrN2O2Purity:99.11%Color and Shape:SolidMolecular weight:199.05MB-07811
CAS:<p>MB-07811 (VK-2809) is an orally active HepDirect prodrug of MB07344 with cholesterol and triglycerides lowering activity.</p>Formula:C28H32ClO5PPurity:99.74% - 99.94%Color and Shape:SolidMolecular weight:514.98PARP-1-IN-4
CAS:<p>PARP-1-IN-4 is a potent PARP-1 inhibitor with potential see anti-tumor activity, and inhibition of PARP-1 may be used in cancer development.</p>Formula:C22H15Cl2N3O2Purity:99.82%Color and Shape:SolidMolecular weight:424.28Tematropium
CAS:Tematropium (CDDD3602) possesses anticholinergic effects and can be used in neurological studies.Formula:C21H31NO8SPurity:99.89%Color and Shape:SolidMolecular weight:457.54TPN171
CAS:<p>TPN171 is potent PDE5 inhibitor with subnanomolar potency for PDE5 and good selectivity over PDE6, which has the potential for the treatment of pulmonary</p>Formula:C24H35N5O3Purity:>99.99%Color and Shape:SolidMolecular weight:441.572,4′-Dichloroacetanilide
CAS:<p>2,4′-Dichloroacetanilide (2-chloro-N-(4-chlorophenyl)acetamide) has antifungal activity and inhibits T. asteroides with a MIC value of 6.25 μg/mL.</p>Formula:C8H7Cl2NOPurity:99.36%Color and Shape:SolidMolecular weight:204.05LY3295668
CAS:<p>LY3295668 (AK-01) is a selective inhibitor of Aurora A with Kis of 0.8 nM and 1038 nM for Aurora A and B, respectively.</p>Formula:C24H26ClF2N5O2Purity:99.68%Color and Shape:SolidMolecular weight:489.95PSB-603
CAS:<p>PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.</p>Formula:C24H25ClN6O4SPurity:97.13%Color and Shape:SolidMolecular weight:529.01LTβR-IN-1
CAS:LTβR-IN-1 is a potent and selective lymphin β receptor (LTβR) inhibitor.Formula:C18H16N4O2Purity:98.93%Color and Shape:SolidMolecular weight:320.35PI3K-IN-54
CAS:<p>Compound 10w, a substituted pyrazolo[1,5-a]pyrimidinamide compound, is a ZSTK474 analog that shows anticancer activity against HeLa cells.</p>Formula:C20H24F2N8O3Purity:98.15%Color and Shape:SolidMolecular weight:462.45Baxdrostat
CAS:<p>Baxdrostat is an aldosterone synthase inhibitor.</p>Formula:C22H25N3O2Purity:99.8%Color and Shape:SolidMolecular weight:363.45Calcium channel-modulator-1
CAS:<p>Calcium channel-modulator-1 is a calcium channel-modulator (IC50:0.8 μM) with specialisation to block aortic constriction.</p>Formula:C26H24Cl2N2O7SPurity:99.95%Color and Shape:SolidMolecular weight:579.45ABR-238901
CAS:ABR-238901 is an oral, active S100A8/A9 blocker that inhibits the interaction of S100A8/A9 with its receptors RAGE(receptor for advanced glycation end productsFormula:C11H9BrClN3O4SPurity:98.63% - 98.71%Color and Shape:SolidMolecular weight:394.63Sembragiline
CAS:<p>Sembragiline (EVT-302) is a selective MAO-B inhibitor for the study of Alzheimer's disease (AD).</p>Formula:C19H19FN2O3Purity:99.49% - 99.49%Color and Shape:SolidMolecular weight:342.36TAK-020
CAS:TAK-020 is a potent covalent inhibitor of Btk with potential antitumor activity for the study of rheumatoid arthritis and immune-related diseases.Formula:C18H17N5O3Purity:98.66%Color and Shape:SolidMolecular weight:351.36Osemozotan HCl
CAS:Osemozotan is a 5-HT1A receptor agonist potentially for the treatment of generalized anxiety disorder.Formula:C19H22ClNO5Purity:98.87% - 99.63%Color and Shape:SolidMolecular weight:379.84UCL-TRO-1938
CAS:<p>UCL-TRO-1938 is a subtype-selective PI3Kα allosteric activator with cardioprotective and neuroregenerative effects.</p>Formula:C27H32N6OPurity:99.95%Color and Shape:SolidMolecular weight:456.58BGB-8035
CAS:<p>BGB-8035 is a BTK inhibitor with antitumor activity that inhibits BTK, TEC, and EGFR.BGB-8035 is used in the study of tumors and autoimmune diseases.</p>Formula:C24H31N5O4Purity:96.74%Color and Shape:SolidMolecular weight:453.53VU0661013
CAS:<p>VU0661013 is an effective and selective inhibitor of MCL-1.</p>Formula:C39H39Cl2N5O4Purity:99.04%Color and Shape:SolidMolecular weight:712.66Bupivacaine hydrochloride monohydrate
CAS:Bupivacaine hydrochloride monohydrate is an NMDA receptor inhibitor that inhibits SCN5A channels and is commonly used in the study of chronic pain.Formula:C18H31ClN2O2Purity:99.91%Color and Shape:SolidMolecular weight:342.9ALDH2 modulator 1
CAS:<p>ALDH2 modulator 1 is a potent and orally active modulator of acetaldehyde dehydrogenase-2 (ALDH2), which reduces blood alcohol levels in mice.</p>Formula:C18H18ClFN2O3Purity:99.68%Color and Shape:SoildMolecular weight:364.8Xanthine oxidase-IN-10
CAS:Xanthine oxidase-IN-10 (XO8 analog) is a xanthine oxidase (XO) inhibitor for the study of gout.Formula:C10H8N2OSPurity:99.16%Color and Shape:SolidMolecular weight:204.25Ac-YVAD-AOM
CAS:<p>Ac-YVAD-AOM is a selective and potent caspase-1 inhibitor showing antitumor activity and potential analgesic activity.</p>Formula:C33H42N4O10Purity:98%Color and Shape:SolidMolecular weight:654.71Aderamastat
CAS:<p>Aderamastat (FP-025) is an orally active matrix metalloproteinase 12 (MMP-12) inhibitor indicated for the study of allergic asthma, COPD and pulmonary fibrosis.</p>Formula:C21H18N2O4SPurity:99.35%Color and Shape:SolidMolecular weight:394.44GI 181771
CAS:<p>GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used in studies about obesity.</p>Formula:C34H31N5O6Purity:95.02%Color and Shape:SolidMolecular weight:605.64CCR3 antagonist 1
CAS:CCR3 antagonist 1 is a potent CCR3 antagonist, used for the research of inflammatory and immunologic diseases.Formula:C19H21Cl2N3O4S2Purity:98.28%Color and Shape:SolidMolecular weight:490.42CMP-Sialic acid sodium salt
CAS:CMP-Sialic acid, a sodium salt, inhibits UDP-GlcNAc 2-epimerase allosterically and serves as a sialyltransferase substrate.Formula:C20H30N4NaO16PPurity:98.32%Color and Shape:SolidMolecular weight:636.43AY 77
CAS:<p>AY 77: Potent, selective PAR2 agonist, favors Ca2+ (ec50=40nM) & ERK1/2 (ec50=2μM), boosts breast cancer cell migration.</p>Formula:C21H32N4O4Purity:99.7%Color and Shape:SolidMolecular weight:404.5PDDC inhibitor
CAS:PDDC inhibitor (Phenyl (R)-(1-(3-(3,4-dimethoxyphenyl)-2,6-dimethylimidazo[1,2-b]pyridazin-8-yl)pyrrolidin-3-yl)carbamate) is an nSMase2 inhibitor.Formula:C27H29N5O4Purity:96.09% - 99.39%Color and Shape:SolidMolecular weight:487.55IN-1130
CAS:IN-1130: ALK5 inhibitor, IC50 - 5.3 nM (Smad3), 36 nM (casein), 4.3 μM (p38α MAPK).Formula:C25H20N6OPurity:99.79%Color and Shape:SolidMolecular weight:420.47Jarin-1
CAS:Jarin-1: JAR1 inhibitor, blocks bioactive JA production in plants, IC50 3.8 μM.Formula:C28H29N3O4Purity:99.82%Color and Shape:SolidMolecular weight:471.55Camonsertib
CAS:<p>Camonsertib (RP-3500) is a novel, potent and selective ATR kinase inhibitor (ATRi) that exhibits potent antitumor effects with an IC50: 1.00 nM in biochemical assays.Cost-effective and quality-assured.</p>Formula:C21H26N6O3Purity:99.6% - 99.93%Color and Shape:SolidMolecular weight:410.47Rislenemdaz
CAS:Rislenemdaz (CERC-301) (CERC-301) is an antagonist of the N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B).Formula:C19H23FN4O2Purity:98.18%Color and Shape:SolidMolecular weight:358.41WAY-620147
CAS:<p>WAY-620147 inhibits Monoamine Oxidase and can be used for the study of neurological disorders.</p>Formula:C12H16BrN3O2Purity:99.55%Color and Shape:SolidMolecular weight:314.18INT-777
CAS:INT-777 (S-EMCA) is a potent TGR5 agonist with an EC50 of 0.82 μM.Formula:C27H46O5Purity:99.89%Color and Shape:SolidMolecular weight:450.65EMD57033
CAS:EMD57033 activates cardiac troponin C, enhances Ca2+ sensitivity to boost heart contraction.Formula:C22H23N3O4SPurity:97.24% - 99.11%Color and Shape:SolidMolecular weight:425.5ADS032
CAS:ADS032 (BT-032) is an NLRP1 and NLRP3 inhibitor with anti-inflammatory activity for the study of respiratory inflammation or infection.Formula:C22H29NO4SPurity:98.37%Color and Shape:SolidMolecular weight:403.54JWG-071
CAS:JWG-071: First ERK5 kinase probe, BET inhibitor, 1 μM BRD4 IC, boosts ERK5 function and BRD4 selectivity.Formula:C34H44N8O3Purity:99.83%Color and Shape:SolidMolecular weight:612.777-BIA
CAS:7-BIA is a receptor-type protein tyrosine phosphatase D (PTPRD) inhibitor with anti-addictive properties and can be used in the study of neuropathic pain.Formula:C15H18O6Purity:≥98% - ≥98%Color and Shape:SolidMolecular weight:294.3AZA197
CAS:AZA197 (AZA-197) is a selective Cdc42 inhibitor.Formula:C24H36N6Purity:99.08%Color and Shape:SolidMolecular weight:408.58Enerisant
CAS:Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.Formula:C22H30N4O3Purity:99.7%Color and Shape:SoildMolecular weight:398.50Dalzanemdor
CAS:<p>Dalzanemdor (SAGE-718) is an NMDA receptor-positive modulator of metabolism that can be used to study Huntington's chorea, Alzheimer's disease, and cognitive</p>Formula:C27H43F3O2Purity:98.2% - >99.99%Color and Shape:SolidMolecular weight:456.62p-Ethynylphenylalanine
CAS:p-Ethynylphenylalanine (4-Ethynyl-L-phenylalanine), a tryptophan hydroxylase (TPH) inhibitor, is competitive, effective, selective, and reversible, with a Ki ofFormula:C11H11NO2Purity:99.44%Color and Shape:SolidMolecular weight:189.21Enpp-1-IN-16
CAS:Enpp-1-IN-16 is an ENPP1 inhibitor, yo anti-cancer activity.Enpp-1-IN-16 can be used to study insulin resistance and chondrocalcinosis.Formula:C23H32N4O4Purity:99.87%Color and Shape:SolidMolecular weight:428.52Kras4B G12D-IN-1
CAS:Kras4B G12D-IN-1 is an inhibitor of Kras4B G12D with anticancer activity.Kras4B G12D-IN-1 inhibits Kras protein expression.Formula:C16H21ClN2O4SPurity:99.75%Color and Shape:SolidMolecular weight:372.87GW 833972A
CAS:<p>GW 833972A: selective CB2 agonist; reduces neural depolarization and citric acid cough in animals.</p>Formula:C18H14Cl2F3N5OPurity:99.93%Color and Shape:SoildMolecular weight:444.24CDC801
CAS:<p>CDC801 is an inhibitor of PDE4 and TNF-α with IC50s of 1.1 μM and 2.5 μM, respectively.</p>Formula:C23H24N2O5Purity:99.61%Color and Shape:SolidMolecular weight:408.45Funapide
CAS:Funapide (TV 45070) is a potent Nav1.7 inhibitor, potentially treating inflammation and various pains.Formula:C22H14F3NO5Purity:99.91%Color and Shape:SolidMolecular weight:429.35α-(difluoromethyl)-DL-Arginine
CAS:<p>α-(difluoromethyl)-DL-Arginine (RMI 71897) is an enzyma-activated, irreversible inhibitor of arginine decarboxylase for E.</p>Formula:C7H14F2N4O2Purity:99.77% - 99.78%Color and Shape:SolidMolecular weight:224.21WAY-600
CAS:<p>WAY-600 is a potent, ATP-competitive and selective inhibitor of mTOR with IC50 of 9 nM; blocks mTORC1/P-S6K(T389) and mTORC2/P-AKT(S473) but not P-AKT(T308).</p>Formula:C28H30N8OPurity:99.88%Color and Shape:SolidMolecular weight:494.59RS 8359
CAS:RS 8359 is a selective MAO-A reversible inhibitor with a 2200:1 A:B ratio, exhibiting antidepressant effects.Formula:C14H12N4OPurity:99.3%Color and Shape:SolidMolecular weight:252.27MC4033
CAS:MC4033 exhibits inhibitory concentration 50 (IC50) values of 39.4 µM in HCT116, 52.1 µM in H1299, 41 µM in A549, and 30.1 µM in U937 [1].Formula:C16H13N3O3Purity:98.16%Color and Shape:SolidMolecular weight:295.29Vidupiprant
CAS:Vidupiprant (AMG 853) is an effective dual antagonist of CRTH2 and prostanoid D receptor with IC50s of 8 nM and 35 nM in human plasma.Formula:C28H27Cl2FN2O6SPurity:98.88%Color and Shape:SolidMolecular weight:609.49Debio-0123
CAS:Debio-0123: potent, specific oral WEE1 inhibitor; IC50 in low nanomolar; boosts DNA damage & Carboplatin's anti-cancer effects.Formula:C26H28Cl2N6OPurity:99.93%Color and Shape:SolidMolecular weight:511.45A7132
CAS:A7132 is an antibacterial agent and possesses broad and potent antibacterial activity.Formula:C19H16F2N4O3Purity:96.64%Color and Shape:SolidMolecular weight:386.35HBED-CC-tris(tert-butyl ester)
CAS:<p>HBED-CC-tris(tert-butyl ester) is a monovalent variant of HBED-CC that can be used for tumor imaging.</p>Formula:C38H56N2O10Purity:99.9%Color and Shape:SolidMolecular weight:700.859AMG 579
CAS:AMG 579 is an efficacious and selective inhibitor of PDE10A (IC50 = 0.1 nM).Formula:C25H23N5O3Purity:99.87%Color and Shape:SolidMolecular weight:441.48CF53
CAS:CF53: potent, selective oral BET inhibitor; Ki <1 nM, Kd 2.2 nM, IC50 2 nM for BRD4 BD1; high affinity for BRD2/3/4/BRDT; effective anti-tumor agent.Formula:C24H25N7O2Purity:99.72%Color and Shape:SolidMolecular weight:443.5PD-L1-IN-3
CAS:PD-L1-IN-3 is a PD-1/PD-L1 inhibitor for the study of tumors and immune diseases.Formula:C19H15ClFN2OSPurity:99.47%Color and Shape:SoildMolecular weight:373.85CINPA1
CAS:CINPA1 selectively inhibits CAR with IC50 of 70 nM, useful in CAR function studies.Formula:C23H29N3O3Purity:99.98%Color and Shape:SolidMolecular weight:395.49CPI-360
CAS:<p>CPI-360 is a small molecule EZH2 inhibitor (IC50: 0.002 μM, EC50: 0.080 μM) that shows antitumor activity in an EZH200-dependent tumor xenograft model.</p>Formula:C25H31N3O4Purity:99.52%Color and Shape:SolidMolecular weight:437.53VH032
CAS:VH032 is a VHL/HIF-1α inhibitor and PROTAC precursor targeting VHL for ubiquitination.Formula:C24H32N4O4SPurity:99.72%Color and Shape:SolidMolecular weight:472.6Zongertinib
CAS:Zongertinib is a human HER2-selective tyrosine kinase inhibitor, a novel TK that is highly selective for covalent binding to the HER2 tyrosine kinase domain (Formula:C29H29N9O2Purity:98.24%Color and Shape:SolidMolecular weight:535.6Ifebemtinib
CAS:Ifebemtinib (BI-853520) is an adhesion plaque kinase inhibitor with anti-tumour activity for the study of breast cancer.Formula:C28H28F4N6O4Purity:98.84% - 99.85%Color and Shape:SolidMolecular weight:588.55Antiviral agent 34
CAS:Antiviral Agent 34 is an antiviral compound that inhibits influenza virus and inhibits the proliferation of influenza virus by modulating RNA polymerase.Formula:C29H33N3O2SPurity:99.51%Color and Shape:SoildMolecular weight:487.66Fluspirilene
CAS:Fluspirilene is a long-acting antipsychotic for schizophrenia, inhibiting L-type calcium channels (IC50: 0.03 μM).Formula:C29H31F2N3OPurity:99.59%Color and Shape:SolidMolecular weight:475.57Soraprazan
CAS:BS3 Crosslinker (Bis(sulfosuccinimidyl)suberate) is an ADC linker that can be used to synthesize antibody-coupled active molecules.Formula:C21H25N3O3Purity:97.69% - 99.84%Color and Shape:SolidMolecular weight:367.44Lartesertib
CAS:<p>Lartesertib (ATM Inhibitor-5) is an inhibitor of the serine/threonine protein kinase ATM with potential anticancer activity and can be used to study lung cancer</p>Formula:C23H21FN6O3Purity:99.9%Color and Shape:SolidMolecular weight:448.45VGSCs-IN-1
CAS:<p>VGSCs-IN-1, a VGSC inhibitor and Riluzole analog, exhibits good blocking activity on Nav1.4 and can be used to study cellular excitability disorders.</p>Formula:C12H12F3N3OSPurity:99.88%Color and Shape:SolidMolecular weight:303.3Roxifiban acetate
CAS:Roxifiban acetate（DMP 754 acetate） is a potent GP IIb / IIIa antagonist that exhibits antiplatelet aggregation activity via immune mediation and can be used inFormula:C23H33N5O8Purity:97.91% - 98.36%Color and Shape:SolidMolecular weight:507.54FHT-1015
CAS:<p>FHT-1205 is a potent inhibitor (IC50 ≤ 10 nM) of SMARCA4/SMARCA2 ATPase (BRG1 and BRM).</p>Formula:C25H25N5O4S3Purity:98.57%Color and Shape:SolidMolecular weight:555.69XY028-140
CAS:<p>XY028-140 is a selective CDK4/6 inhibitor and degrader, acting via PROTAC with ligands for Cereblon and CDK in cancer cells.</p>Formula:C39H40N10O7Purity:98.59%Color and Shape:SolidMolecular weight:760.8KER047
CAS:ALK2-IN-4, a highly effective ALK2 inhibitor.Formula:C26H30FN7OPurity:98.49% - >99.99%Color and Shape:SolidMolecular weight:475.560990CL
CAS:0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMPFormula:C21H21N5Purity:98.99%Color and Shape:SolidMolecular weight:343.42h-NTPDase-IN-2
CAS:h-NTPDase-IN-2 is a broad-spectrum NTPDase inhibitor that inhibits multiple h-NTPDas isoforms.Formula:C19H16N4SPurity:99.58%Color and Shape:SolidMolecular weight:332.42UC-764864
CAS:UC-764864, a UBE2N inhibitor, impedes the enzymatic activity of UBE2N and exhibits cytotoxic effects through the disruption of UBE2N-dependent signaling inFormula:C19H18N2OSPurity:99.3%Color and Shape:SolidMolecular weight:322.42SMN-C3
CAS:SMN-C3 (MV8T2MCK57) is an orally active modulator of SMN2 splicing, and has the potential to treat spinal muscular atrophy (SMA).Formula:C24H28N6OPurity:99.01% - 99.05%Color and Shape:SolidMolecular weight:416.52CGP-20712
CAS:CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.Formula:C23H25F3N4O5Purity:99.40% - 99.58%Color and Shape:SolidMolecular weight:494.46AZD4573
CAS:AZD4573 is an effective and selective CDK9 inhibitor (IC50: <4 nM). It enables transient target engagement for the treatment of hematologic malignancies.Formula:C22H28ClN5O2Purity:99% - 99.51%Color and Shape:SolidMolecular weight:429.94Zidesamtinib
CAS:<p>Zidesamtinib (NVL-520) is a ROS1 fusion and resistance mutation inhibitor that inhibits ROS1 and can be used to study non-small cell lung cancer.</p>Formula:C22H22FN7OPurity:99.74%Color and Shape:SolidMolecular weight:419.455Cudetaxestat
CAS:<p>Cudetaxestat (BLD-0409) is a potent inhibitor of orally active autotaxin.</p>Formula:C21H15Cl2F2N3O2SPurity:99.9%Color and Shape:SolidMolecular weight:482.33α1 adrenoceptor-MO-1
CAS:<p>α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.</p>Formula:C20H24ClN5OPurity:99.20% - 99.29%Color and Shape:SolidMolecular weight:385.89PDE9-IN-(S)-C33
CAS:<p>PDE9-IN-(S)-C33: potent PDE9 inhibitor with 11 nM IC50, for CNS diseases and diabetes study.</p>Formula:C18H20ClN5OPurity:98.75%Color and Shape:SolidMolecular weight:357.84SB 216641 hydrochloride
CAS:SB 216641 hydrochloride (SB-216641A) is a 5-HT1B/D receptor antagonist with anxiolytic properties.Formula:C28H31ClN4O4Purity:98.06% - 99.23%Color and Shape:SolidMolecular weight:523.02Nothofagin
CAS:Nothofagin: Antioxidant, anti-inflammatory, prevents clotting, inhibits leukocyte activity, may treat vascular inflammation.Formula:C21H24O10Purity:98.51%Color and Shape:SolidMolecular weight:436.41GW274150
CAS:<p>GW274150: selective oral iNOS inhibitor (Kd=40 nM), low activity on eNOS/nNOS, protective in acute lung injury.</p>Formula:C8H17N3O2SPurity:96.43%Color and Shape:SolidMolecular weight:219.3ALK-IN-27
CAS:Neladalkib (NVL-655) is an ALK inhibitor with antitumor activity for the study of non-small cell cancers.Formula:C23H22ClFN6OPurity:99.71%Color and Shape:SolidMolecular weight:452.91CGP 78608 hydrochloride
CAS:<p>CGP 78608 hydrochloride: NMDA receptor antagonist (IC50=6 nM), anticonvulsant, enhances GluN1/GluN3A currents (EC50=26.3 nM).</p>Formula:C11H14BrClN3O5PPurity:99.85%Color and Shape:SolidMolecular weight:414.58NSC697923
CAS:NSC-697923 inhibits UBE2N, triggers p53-dependent and JNK-mediated apoptosis, blocks DNA damage and NF-κB signaling in neuroblastoma cells.Formula:C11H9NO5SPurity:97% - 99.84%Color and Shape:SolidMolecular weight:267.26CXCR2-IN-1
CAS:<p>CXCR2-IN-1 has a pIC50 of 9.3 and is a CXCR2 antagonist of the central nervous system penetration agent.</p>Formula:C19H20Cl2FN3O4SPurity:99.89%Color and Shape:SolidMolecular weight:476.35BMS-212122
CAS:BMS-212122 inhibits MTP, reduces lipids and plaque in animal tests.Formula:C43H36F6N4O2Purity:99.85%Color and Shape:SolidMolecular weight:754.76FIIN-1
CAS:FIIN-1 (FGFR irreversible inhibitor-1) is an irreversible and selective FGFR inhibitor with Kd of 2.8, 6.9, 5.4, 120, 32 and 120 nM for FGFR1, FGFR2, FGFR3,Formula:C32H39Cl2N7O4Purity:98.75%Color and Shape:SolidMolecular weight:656.6SynuClean-D
CAS:<p>SynuClean-D prevents α-synuclein clumps, breaks fibrils & protects neurons in Parkinson’s models.</p>Formula:C13H5F3N4O5Purity:99.64% - 99.96%Color and Shape:SolidMolecular weight:354.2AZ PFKFB3 26
CAS:<p>AZ PFKFB3 26 is an effective and selective PFKFB3 inhibitor with an IC50 of 23 nM. The IC50s for PFKFB1 and PFKFB2 are 2.06 and 0.384 μM, respectively.</p>Formula:C24H26N4O2Purity:99.85%Color and Shape:SolidMolecular weight:402.49Philanthotoxin 74 dihydrochloride
CAS:<p>Philanthotoxin 74 dihydrochloride is an antagonist of AMPAR with IC50s of 263 and 296 nM for GluR3 and GluR1.</p>Formula:C24H44Cl2N4O3Purity:99.75%Color and Shape:SolidMolecular weight:507.54(±)-CPSI-1306
CAS:(±)-CPSI-1306 (2-(3-(2,4-Difluorophenyl)-4,5-dihydroisoxazol-5-yl)-1-morpholinoethan-1-one) is a macrophage migration inhibitory factor (MIF) antagonist and canFormula:C15H16F2N2O3Purity:97.46%Color and Shape:SolidMolecular weight:310.3EGFR/ErbB-2 inhibitor-1
CAS:<p>EGFR/ErbB-2 inhibitor-1 is a selective ErbB2/HER2 inhibitor that effectively blocks ErbB2 and HER2 signaling.</p>Formula:C23H15ClFN3OS2Purity:98.93%Color and Shape:SolidMolecular weight:467.97Varespladib methyl
CAS:Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.Formula:C22H22N2O5Purity:99.42% - 99.97%Color and Shape:SolidMolecular weight:394.42DGAT-1 inhibitor 2
CAS:DGAT-1 inhibitor 2: effective against obesity, targets enzyme in triglyceride synthesis for diabetes treatment.Formula:C24H28N4O3Purity:98.36%Color and Shape:SolidMolecular weight:420.5BTK inhibitor 1
CAS:<p>BTK inhibitor 1 (Compound 27) is a BTK inhibitor (IC50: 0.11 nM) with an inhibitory effect on B-cell activation in hWB with an IC50 of 2 nM.</p>Formula:C24H23FN8O2Purity:98.24% - 98.91%Color and Shape:SolidMolecular weight:474.49LE135
CAS:LE135: RARα/RARβ antagonist (Ki: 1.4 μM/220 nM), favors RARβ, selective vs RARγ/RXRs; also activates TRPV1/TRPA1 (EC50s: 2.5/20 μM).Formula:C29H30N2O2Purity:97.94%Color and Shape:SolidMolecular weight:438.56CE-224535
CAS:CE-224535 (PF-04905428) is a selective antagonist of P2X7 receptor. CE-224535 can be used in disease-modifying antirheumatic studies.Formula:C22H29ClN4O6Purity:99.68%Color and Shape:SolidMolecular weight:480.94Iptacopan
CAS:Iptacopan (LNP023) is an inhibitor with high affinity to factor B, with a KD value of 7.9 nM and an IC50 value of 10 nM. Cost-effective and quality-assured.Formula:C25H30N2O4Purity:99.07% - >99.99%Color and Shape:SolidMolecular weight:422.52Terbufibrol
CAS:<p>Terbufibrol reduces the levels of serum total cholesterol in normal and hypercholesterolemic male rats.</p>Formula:C20H24O5Purity:98.345%Color and Shape:SolidMolecular weight:344.4Didesmethyl cariprazine
CAS:<p>Didesmethyl cariprazine, Cariprazine's active metabolite, treats schizophrenia/bipolar with D3/D2 affinity; half-life 1-3 weeks.</p>Formula:C19H28Cl2N4OPurity:99.52%Color and Shape:SolidMolecular weight:399.36RH01386
CAS:<p>RH01386, a small molecule, prevents ER stress in β cells, inhibits proapoptotic genes, and may treat type 2 diabetes by restoring insulin secretion.</p>Formula:C18H15F3N4O3SPurity:99.16% - 99.67%Color and Shape:SolidMolecular weight:424.4Rheb inhibitor NR1
CAS:Rheb inhibitor NR1 is a Rheb inhibitor and selective mTORC1 inhibitor that promotes phosphorylation of S473pAKT.Formula:C25H19BrCl2N2O3SPurity:99.72%Color and Shape:SolidMolecular weight:578.3CGS 15435
CAS:CGS 15435: potent TxA2 synthase inhibitor, IC50=1 nM; less selective for PGI2 synthase, COX, and liposynthase.Formula:C20H21ClN2O2Purity:99.86%Color and Shape:SolidMolecular weight:356.85Ac-DEVD-CHO
CAS:Ac-DEVD-CHO is a specific Caspase-3 inhibitor (Ki: 230 pM).Ac-DEVD-CHO has an inhibitory effect in SLNT-induced apoptosis.Formula:C20H30N4O11Purity:98.69%Color and Shape:SolidMolecular weight:502.47GP 1a
CAS:<p>GP 1a: potent CB2 receptor agonist (EC50=7.1), 30x CB2 over CB1 preference, boosts P-ERK1/2, aids skin healing, anti-inflammatory.</p>Formula:C23H22Cl2N4OPurity:99.79%Color and Shape:SolidMolecular weight:441.35K777
CAS:K777: Oral cysteine protease inhibitor, CYP3A4 blocker (IC50=60 nM), CCR4 antagonist, anti-Trypanosoma cruzi, antiviral, halts EBOV/SARS-CoV entry (IC50<1 nM).Formula:C32H38N4O4SPurity:98.43% - 99.14%Color and Shape:SolidMolecular weight:574.73HIV-1 inhibitor-54
CAS:HIV-1 inhibitor-54: potent anti-HIV (EC50: 32 nM), targets WT HIV-1 IIIB in MT-4 cells for infection research.Formula:C27H30N6O4SPurity:98.05% - 99.39%Color and Shape:SoildMolecular weight:534.63CU-CPD107
CAS:<p>CU-CPD107 selectively activates TLR8 and ssRNA, inhibits TLR8 with R848 (IC50=13.7 μM), and coactivates with ssRNA.</p>Formula:C16H21IN2O2Purity:98%Color and Shape:SolidMolecular weight:400.25CFTR corrector 4
CAS:Potent, oral CFTR corrector 4 targets cystic fibrosis, increasing cell surface CFTR levels.Formula:C29H27F2NO7Purity:99.32%Color and Shape:SolidMolecular weight:539.52Lotiglipron
CAS:<p>Lotiglipron (PF-07081532) is a GLP-1R agonist that lowers blood glucose and may be used in the study of type 2 diabetes mellitus (T2DM) and excess obesity.</p>Formula:C31H31ClN4O5Purity:98.3%Color and Shape:SolidMolecular weight:575.05Toxoflavin
CAS:Toxoflavin (Xanthothricin) is an antagonist of transcription factor 4 (TCF4)/β-catenin complex. Toxoflavin also acts as an inhibitor of KDM4A.Formula:C7H7N5O2Purity:98.24% - 99.7%Color and Shape:SolidMolecular weight:193.16HIF-2α agonist 2
CAS:HIF-2α agonist 2 is an HIF-2α agonist with an EC50 value of 1.68 μM for HIF-2α.Formula:C13H8Br2N2O2SPurity:98.87%Color and Shape:SoildMolecular weight:416.09Cis-22a
CAS:Cis-22a: selective TRPV6 inhibitor (IC50=0.32μM), halts T47D breast cancer cell growth.Formula:C24H30F3N3O2Purity:99.99%Color and Shape:SolidMolecular weight:449.51DHX9-IN-2
CAS:<p>DHX9-IN-2 is an inhibitor targeting ATP-dependent RNA de-helicase A (DHX9) with anticancer and antitumor activity for cancer research.</p>Formula:C18H16ClN3O3S2Purity:98%Color and Shape:SolidMolecular weight:421.92Reldesemtiv
CAS:<p>Reldesemtiv (CK-2127107) boosts exercise capacity, targeting fast muscle troponin, EC50 3.4 μM.</p>Formula:C19H18F2N6OPurity:97.27%Color and Shape:SolidMolecular weight:384.38AS2717638
CAS:AS2717638: oral LPA5 antagonist, IC50 38 nM, reduces PGF2α/PGE2/AMPA allodynia.Formula:C25H25N3O5Purity:99.23%Color and Shape:SolidMolecular weight:447.48ZY-19489
CAS:<p>ZY-19489: Antimalarial, potential single-dose cure, FDA orphan drug status.</p>Formula:C24H32FN9Purity:>99.99%Color and Shape:SoildMolecular weight:465.57Exarafenib
CAS:Exarafenib (RAF/KIN_2787) is an oral pan-RAF inhibitor with antitumor properties, targeting MAPK signaling in cancer research.Formula:C26H34F3N5O3Purity:98.36% - 99.84%Color and Shape:SolidMolecular weight:521.58JAK-IN-3
CAS:JAK-IN-3 is a potent JAK inhibitor that inhibits JAK3, JAK1, TYK2, and JAK2, and can be used for the study of immune system disorders.Formula:C18H20N4O3Purity:98.04% - 98.19%Color and Shape:SolidMolecular weight:340.38AVP-13358
CAS:AVP-13358: a CD23/IgE inhibitor for treating immune, infection, and ENT disorders.Formula:C30H29N5O2Purity:98.45%Color and Shape:SolidMolecular weight:491.58DuP-697
CAS:DuP-697 is an irreversible, specific COX-2 inhibitor with IC50 values of 10 nM and 800 nM for human COX-2 and COX-1.Cost-effective and quality-assured.Formula:C17H12BrFO2S2Purity:99.92%Color and Shape:SolidMolecular weight:411.31Msr-Ratio
CAS:<p>Msr-Ratio is a probe for tracking MSR activity, with 375 nm excitation and 550 nm emission, used in vitro and in cells.</p>Formula:C18H14O3SPurity:98.93%Color and Shape:SolidMolecular weight:310.37PA452
CAS:<p>PA452 is a selective antagonist of retinoic X receptor (RXR) and suppresses the effect of Retinoic acid on Th1/Th2 development.</p>Formula:C26H37N3O3Purity:97.14%Color and Shape:SolidMolecular weight:439.59MK-2461
CAS:MK-2461 is a novel inhibitor that targets multiple proteins and competitively binds to ATP sites, specifically inhibiting the activated c-Met protein with anFormula:C24H25N5O5SPurity:95.41% - 99.67%Color and Shape:SolidMolecular weight:495.55hRIO2 kinase ligand-1
CAS:hRIO2 kinase ligand-1 is a potent ligand for hRIO2 kinase (Kd: 520 nM).Formula:C17H14N2OPurity:99.89%Color and Shape:SolidMolecular weight:262.31Clazosentan
CAS:Clazosentan (Ro 61-1790) is a selective ET_A receptor antagonist that inhibits ET-1 vasoconstriction and prevents cerebral vasospasm.Formula:C25H23N9O6SPurity:95.39% - >99.99%Color and Shape:SolidMolecular weight:577.57Elobixibat
CAS:Elobixibat (A 3309) blocks IBAT in mice/humans/dogs (IC50: 0.13/0.53/5.8 nM); used for constipation research.Formula:C36H45N3O7S2Purity:97.43% - 98.03%Color and Shape:SolidMolecular weight:695.89NMI 8739
CAS:<p>NMI 8739 (n-docosahexaenoyl dopamine) is an agonist of D2 autoreceptor.</p>Formula:C30H41NO3Purity:98.51%Color and Shape:SolidMolecular weight:463.65LNA-Adenosine
CAS:LNA-Adenosine (LNA-A) is a nucleoside analogue that acts as a ligand for adenosine A3 receptors.Formula:C11H13N5O4Purity:99.15%Color and Shape:SolidMolecular weight:279.25IMP-1710
CAS:IMP-1710 is a selective UCH-L1 inhibitor with an IC50 value of 38 nM in a fluorescence polarization assay.[1]Cost-effective and quality-assured.Formula:C23H19N5OPurity:99.3%Color and Shape:SolidMolecular weight:381.43IL-17 modulator 4
CAS:IL-17 modulator 4 is a prodrug of IL-17 modulator 1, which acts as a potent modulator of IL-17.Cost-effective and quality-assured.Formula:C27H34N6O2Purity:99.59%Color and Shape:SolidMolecular weight:474.6TCMDC-135051
CAS:TCMDC-135051: Selective PfCLK3 inhibitor, low toxicity, halts parasite growth & transmission; EC50=320 nM.Formula:C29H33N3O3Purity:99.05%Color and Shape:SolidMolecular weight:471.59A2B receptor antagonist 1
CAS:A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.Formula:C21H24N6O2Purity:99.53%Color and Shape:SolidMolecular weight:392.45CH6953755
CAS:CH6953755: oral YES1 kinase inhibitor, IC50 1.8 nM, potent, selective, anticancer, halts cell proliferation.Formula:C26H22F2N6O4SPurity:98.87%Color and Shape:SolidMolecular weight:552.55CCT365623
CAS:<p>CCT365623: oral Lysyl Oxidase inhibitor, potent, selective, good pharmacokinetics, anti-metastatic.</p>Formula:C18H17NO4S3Purity:97.299% - 99.49%Color and Shape:SolidMolecular weight:407.53Dechloro Rivaroxaban
CAS:<p>Dechloro Rivaroxaban is a Factor Xa inhibitor that inhibits free FXa and plasminogen and fibrin-associated FXa activity in humans.</p>Formula:C19H19N3O5SPurity:98.63%Color and Shape:SolidMolecular weight:401.44WAY-639228
CAS:<p>WAY-639228-A has potential antithrombotic and anticoagulant activity for the study of cerebral thrombosis.</p>Formula:C22H24N2O2SPurity:99.75%Color and Shape:SolidMolecular weight:380.5Salicyl-AMS
CAS:<p>Salicyl-AMS is an inhibitor of mycobacterium auxin biosynthesis that inhibits the growth of mycobacterium in the presence of iron deficiency in vitro.</p>Formula:C17H18N6O8SPurity:98.19%Color and Shape:SolidMolecular weight:466.43BuChE-IN-TM-10
CAS:TM-10: Potent BuChE inhibitor, IC50 8.9 nM, disaggregates Aβ, antioxidant, BBB penetrant, may treat Alzheimer's.Formula:C32H38N2O3Purity:99.54%Color and Shape:SolidMolecular weight:498.66E7016
CAS:<p>E7016 (GPI 21016) is an orally available PARP inhibitor. E7016 inhibits of DNA repair. E7016 can enhance tumor cell radiosensitivity in vitro and in vivo.</p>Formula:C20H19N3O3Purity:99.02%Color and Shape:SolidMolecular weight:349.38OPC-28326
CAS:OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Formula:C26H35N3O2Purity:99.79%Color and Shape:SolidMolecular weight:421.58BDP9066
CAS:BDP9066 is a potent and selective MRCK inhibitor, inhibits MRCKβ and MRCKα/β, and can be used for the prevention and treatment of skin cancer.Formula:C20H24N6Purity:98.18%Color and Shape:SolidMolecular weight:348.44R-(+)-EU-1180-453
CAS:R-(+)-EU-1180-453 is a novel GluN2C/D selective NMDAR-positive modulator for the study of neurological disorders.Formula:C22H21FN2O3Purity:99.63%Color and Shape:SolidMolecular weight:380.41Aneratrigine hydrochloride
CAS:Aneratrigine hydrochloride is a Nav 1.9 blocker that may be used to prevent or treat sodium channel blocker-related disorders.Formula:C19H21Cl2F2N5O2S2Purity:98.37% - 99.16%Color and Shape:SolidMolecular weight:524.43SAFit2
CAS:<p>SAFit2 is a highly potent and selective inhibitor of fk506 binding protein 51 (FKBP51).Cost-effective and quality-assured</p>Formula:C46H62N2O10Purity:98.16% - >99.99%Color and Shape:SolidMolecular weight:802.99Cis-N-Feruloyltyramine
CAS:Cis-N-Feruloyltyramine is a naturally occurring compound found in various plants that shows cytotoxicity against the P-388 cancer cell line.Formula:C18H19NO4Purity:97.43%Color and Shape:SolidMolecular weight:313.35Adomeglivant
CAS:Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.Formula:C32H36F3NO4Purity:99.91%Color and Shape:SolidMolecular weight:555.63Antiproliferative agent-36
CAS:<p>Antiproliferative agent-36 is a broad-spectrum anticancer benzothiazolylhydrazone-derived compound that inhibits cell proliferation.</p>Formula:C13H11N5SPurity:97.57%Color and Shape:SolidMolecular weight:269.33ERDRP-0519
CAS:ERDRP-0519 is an oral measles polymerase inhibitor, preventing disease in monkeys, with potent nanomolar efficacy against morbilliviruses.Formula:C23H30F3N5O4SPurity:98.64% - 98.71%Color and Shape:SolidMolecular weight:529.58
