Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(52 products)
- Calcium Channel(496 products)
- Chloride channel(49 products)
- GABA Receptor(336 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(277 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2290 products of "Membrane Transporter/Ion Channel"
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ABT-639 hydrochloride
CAS:<p>ABT-639 hydrochloride is a selective, novel T-type Ca2+ channel blocker.</p>Formula:C20H21Cl2F2N3O3SColor and Shape:SolidMolecular weight:492.36Acecainide hydrochloride
CAS:<p>Acecainide hydrochloride (NAPA) is the major hepatic metabolite of procainamide.Cost-effective and quality-assured.</p>Formula:C15H24ClN3O2Purity:98.023% - 99.81%Color and Shape:SolidMolecular weight:313.83TGN-020
CAS:<p>TGN-020 is an inhibitor of Aquaporin 4 (AQP4, IC50: 3.1 μM), the most abundant water channel in the brain.</p>Formula:C8H6N4OSPurity:99.54% - 99.99%Color and Shape:SolidMolecular weight:206.22PF 429242
CAS:<p>PF-429242 inhibits SREBP site 1 protease selectively (IC50: 0.175 μM); reduces cholesterol synthesis in CHO cells (IC50: 0.53 μM).</p>Formula:C25H35N3O2Purity:99.27%Color and Shape:SolidMolecular weight:409.56Polyoxyethylene stearate
CAS:<p>Polyoxyethylene stearate (POES) is an agent of non-ionic emulsifying.</p>Formula:C20H40O3Purity:n~9-10Color and Shape:Light Amber SemisolidMolecular weight:328.29775KPT276
CAS:<p>KPT276 (KPT 276) is an orally bioavailable selective inhibitor of nuclear export (SINE) that irreversibly bind to CRM1 and block the function of CRM1.</p>Formula:C16H10F8N4OPurity:99.89% - >99.99%Color and Shape:SolidMolecular weight:426.26Cinacalcet metabolite M4
CAS:<p>Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.</p>Formula:C10H12F3NPurity:97.13%Color and Shape:SolidMolecular weight:203.2Loreclezole hydrochloride
CAS:<p>Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.</p>Formula:C10H7Cl4N3Color and Shape:SolidMolecular weight:310.99Ocinaplon
CAS:<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Formula:C17H11N5OPurity:99.81%Color and Shape:SolidMolecular weight:301.3Esomeprazole
CAS:<p>Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.</p>Formula:C17H19N3O3SPurity:97.3%Color and Shape:SolidMolecular weight:345.42Bepridil free base
CAS:<p>Bepridil: Class IV anti-arrhythmic, calcium blocker, dilates coronary arteries.</p>Formula:C24H34N2OColor and Shape:SolidMolecular weight:366.54Ibutilide
CAS:<p>Ibutilide (U70226E) is an antiarrhythmic that prolongs action potential by blocking I Kr in AT-1 cells.</p>Formula:C20H36N2O3SColor and Shape:SolidMolecular weight:384.58Rimeporide hydrochloride
CAS:<p>Rimeporide hydrochloride (EMD-87580 hydrochloride) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.</p>Formula:C11H16ClN3O5S2Purity:99.82%Color and Shape:SolidMolecular weight:369.84Transdermal Peptide Disulfide Acetate
<p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>Formula:C42H68N14O18S2Purity:99.97%Color and Shape:SolidMolecular weight:1121.2Evenamide
CAS:<p>Evenamide (NW-3509) is a sodium channel blocker. Which shows efficacy in a broad spectrum of rodent models of psychosis, mania, depression, and aggressiveness.</p>Formula:C16H26N2O2Purity:96.74% - 99.15%Color and Shape:SolidMolecular weight:278.39FGH10019
CAS:<p>FGH10019 is a novel inhibitor of sterol regulatory element-binding protein (SREBP) ( IC50 :1 μM).</p>Formula:C18H19N3O2S2Purity:98.93%Color and Shape:SolidMolecular weight:373.49BTS
CAS:<p>BTS (N-Tosylbenzylamine) is a potent inhibitor of Ca2+-stimulated myosin S1 ATPase (IC50 : 5 μM) .</p>Formula:C14H15NO2SPurity:99.45%Color and Shape:White Crystalline SolidMolecular weight:261.34AM92016
CAS:<p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>Formula:C26H30Cl2N2O6SColor and Shape:SolidMolecular weight:569.49Disopyramide phosphate
CAS:<p>Disopyramide: Class 1a anti-arrhythmic, treats Ventricular Tachycardia, reduces heart muscle contractility.</p>Formula:C21H32N3O5PColor and Shape:SolidMolecular weight:437.47Icenticaftor
CAS:Icenticaftor (QBW251) is an orally active potentiator of CFTR channel.Formula:C12H13F6N3O3Purity:99.76%Color and Shape:SolidMolecular weight:361.24Metaflumizone
CAS:<p>Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.</p>Formula:C24H16F6N4O2Purity:98.73%Color and Shape:SolidMolecular weight:506.40KCNQ2/3 activator-1
CAS:<p>KCNQ2/3 activator-1 is a Kv7.2/Kv7.3 (KCNQ2/3) potassium channel activator.</p>Formula:C23H29FN2OPurity:99.16% - 99.47%Color and Shape:SolidMolecular weight:368.49Tiagabine hydrochloride hydrate
CAS:<p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>Formula:C20H28ClNO3S2Color and Shape:SolidMolecular weight:430.02UBP551
CAS:<p>UBP551 is a potent and selective NMDA receptors modulator.</p>Formula:C11H8O4Purity:98.69%Color and Shape:SolidMolecular weight:204.18Omecamtiv mecarbil
CAS:<p>Omecamtiv mecarbil (CK-1827452) has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic</p>Formula:C20H24FN5O3Purity:98% - 99.23%Color and Shape:SolidMolecular weight:401.43PAP-1
CAS:<p>PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).</p>Formula:C21H18O5Purity:99.35% - 99.75%Color and Shape:White SolidMolecular weight:350.36VU0134992
CAS:<p>VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μM</p>Formula:C20H31BrN2O2Purity:99.86%Color and Shape:SolidMolecular weight:411.38Gabazine free base
CAS:<p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>Formula:C15H17N3O3Color and Shape:SolidMolecular weight:287.31N-Me-aminopyrimidinone9
CAS:<p>N-Me-aminopyrimidinone9 is a sodium channel antagonist</p>Formula:C16H21N3OSPurity:99.21%Color and Shape:SolidMolecular weight:303.42GMQ hydrochloride
CAS:<p>GMQ hydrochloride, a potent ASIC modulator, activates ASIC3 at neutral pH and inhibits acid-induced peak current.</p>Formula:C10H12ClN5Purity:99.64%Color and Shape:SolidMolecular weight:237.692'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Formula:C16H14O4Purity:98.75%Color and Shape:SolidMolecular weight:270.28Linerixibat
CAS:<p>Linerixibat (GSK2330672) is a highly effective, nonabsorbable ASBT inhibitor. Linerixibat can lower glucose in an animal model of type 2 diabetes.</p>Formula:C28H38N2O7SPurity:98.5% - 99.98%Color and Shape:SolidMolecular weight:546.68Songorine
CAS:<p>Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.</p>Formula:C22H31NO3Purity:98% - 99.92%Color and Shape:SolidMolecular weight:357.49Acetoxyvalerensre
CAS:<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Formula:C17H24O4Purity:98.22%Color and Shape:SolidMolecular weight:292.37DQP 1105
CAS:<p>DQP 1105 is a NMDA receptor antagonist.</p>Formula:C29H24BrN3O4Purity:98.6%Color and Shape:SolidMolecular weight:558.42Arecaidine hydrochloride
CAS:<p>Arecaidine hydrochloride may have carcinogenesis.</p>Formula:C7H12ClNO2Purity:99.69% - ≥95%Color and Shape:SolidMolecular weight:177.63ML329
CAS:<p>ML329 is a small molecule inhibitor of MITF, inhibiting TRPM-1 promoter activity.</p>Formula:C16H12N2O4SPurity:98.96%Color and Shape:SolidMolecular weight:328.34ML204
CAS:<p>ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels.</p>Formula:C15H18N2Purity:98.1% - 99.72%Color and Shape:SolidMolecular weight:226.32QX-222 chloride
CAS:<p>QX-222 chloride (Lidocaine N-Methyl Hydrochloride) is a sodium channel blocker.</p>Formula:C13H21ClN2OPurity:97.37%Color and Shape:SolidMolecular weight:256.77Nateglinide
CAS:<p>Nateglinide is an oral drug for type 2 diabetes, stimulating insulin release; may cause rare acute liver injury.</p>Formula:C19H27NO3Purity:99.93% - 99.94%Color and Shape:White Crystalline PowderMolecular weight:317.42rac-BHFF
CAS:<p>rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.</p>Formula:C17H21F3O3Purity:99.69% - >99.99%Color and Shape:SolidMolecular weight:330.34TRPM8 antagonist WS-3
CAS:TRPM8 antagonist WS-3 (Cyclohexanecarboxamide) is an agonist of TRPM8( EC50 : 3.7 μM).Formula:C13H25NOPurity:97.64%Color and Shape:DrypowderMolecular weight:211.34CCTA-1523
CAS:<p>CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.</p>Formula:C16H15Cl2NO3Purity:99.71%Color and Shape:SolidMolecular weight:340.2TC-I2000
CAS:<p>TC-I2000 is an TRPM8 channel blocker. Inhibits icilin-induced TRPM8 channel activation in rTRPM8-expressing CHO cells with IC50 of 53 nM.</p>Formula:C23H18F4N2OPurity:99.778%Color and Shape:SolidMolecular weight:414.4Acamprosate calcium
CAS:<p>Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.</p>Formula:C10H20CaN2O8S2Purity:98% - 99.93%Color and Shape:White Odorless Or Nearly Odorless PowderMolecular weight:400.48α-Cyano-4-hydroxycinnamic acid
CAS:<p>α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvate</p>Formula:C10H7NO3Purity:99.8% - 99.86%Color and Shape:PowderMolecular weight:189.17Evifacotrep
CAS:<p>Evifacotrep: TRPC5 antagonist for neurological disease research (WO2020061162, compound 100).</p>Formula:C18H12ClF4N5O2Purity:98.6%Color and Shape:SolidMolecular weight:441.77A-967079
CAS:<p>A 967079 is a potent, selective, and bioavailable inhibitor of the TRPA1 channel, with IC50 values of 67 and 289 nM for the human and rat isoforms, respectively</p>Formula:C12H14FNOPurity:98.34% - 99.75%Color and Shape:SolidMolecular weight:207.24Nisoxetine
CAS:<p>Nisoxetine is a selective NET (noradrenaline transporter) inhibitor (Kd=0.76 nM) capable of blocking voltage-gated sodium channels.</p>Formula:C17H21NO2Color and Shape:SolidMolecular weight:271.35Afloqualone
CAS:<p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>Formula:C16H14FN3OPurity:99.72%Color and Shape:SolidMolecular weight:283.3IDRA-21
CAS:IDRA-21 is a positive AMPA receptor modulator.Formula:C8H9ClN2O2SPurity:99.73%Color and Shape:SolidMolecular weight:232.69DL-Menthol
CAS:<p>DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.</p>Formula:C10H20OPurity:99.74%Color and Shape:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Molecular weight:156.27RN-1734
CAS:<p>RN-1734 is selective TRPV4 channel antagonist(IC50 of 2.3 μM,5.9 μM,3.2 μM for hTRPV4, mTRPV4 and rTRPV4,respectively)</p>Formula:C14H22Cl2N2O2SPurity:99.1% - 99.3%Color and Shape:SolidMolecular weight:353.31MDR-652
CAS:<p>MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM for</p>Formula:C22H23ClFN3O2SPurity:99.96%Color and Shape:SolidMolecular weight:447.95JNJ-26990990
CAS:<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Formula:C9H10N2O2S2Purity:97.37%Color and Shape:SolidMolecular weight:242.32YHO-13177
CAS:<p>YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.</p>Formula:C20H22N2O3SPurity:98.78%Color and Shape:SolidMolecular weight:370.475,7-Dichlorokynurenic acid
CAS:5,7-Dichlorokynurenic acid (5,7-dichlorokynurenic acid sodium) is an NMDA receptor antagonist.Formula:C10H5Cl2NO3Purity:99.71%Color and Shape:SolidMolecular weight:258.06Flupirtine
CAS:<p>Flupirtine(D 9998) is a selective neuronal potassium channel opener as well as shows properties of NMDA receptor antagonist.</p>Formula:C15H17FN4O2Color and Shape:SolidMolecular weight:304.32BPU-11
CAS:<p>BPU-11 (Biphenyl Urea 11) is an HCN4 CLP ligand that acts by modulating channel function and completely abolishing the cAMP-induced shift in V1/2.</p>Formula:C32H31N5OPurity:99.16%Color and Shape:SolidMolecular weight:501.62AMG 517
CAS:<p>AMG 517 is an effective and specific TRPV1 antagonist, antagonizes proton (IC50: 0.76 nM), capsaicin (IC50: 0.62 nM) and heat activation (IC50: 1.3 nM) of TRPV1</p>Formula:C20H13F3N4O2SPurity:99.77% - 99.85%Color and Shape:SolidMolecular weight:430.4Loreclezole
CAS:<p>Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.</p>Formula:C10H6Cl3N3Purity:99.78%Color and Shape:SolidMolecular weight:274.53Kavain
CAS:<p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>Formula:C14H14O3Purity:99.93% - ≥95%Color and Shape:SolidMolecular weight:230.26RQ-00203078
CAS:<p>RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist.</p>Formula:C21H13ClF6N2O5SPurity:98% - 99.6%Color and Shape:SolidMolecular weight:554.85Blebbistatin
CAS:<p>Blebbistatin ((±)-Blebbistatin) is a non-muscle myosin II (NMII)-selective and non-muscle myosin heavy chain 9 (MYH9)-specific inhibitor.Cost-effective and quality-assured.</p>Formula:C18H16N2O2Purity:99.88% - 99.97%Color and Shape:Bright Yellow SolidMolecular weight:292.33KM 91104
CAS:<p>KM 91104 is a cell permeable inhibitor of V-ATPase. KM91104 specifically targets the interaction between V-ATPase subunit A3 and subunit B2.</p>Formula:C14H12N2O4Purity:99.04%Color and Shape:SolidMolecular weight:272.26λ-Cyhalothrin
CAS:<p>λ-Cyhalothrin (Icon) is a type II synthetic pyrethroid insecticide featuring a high-efficiency, broad-spectrum formula with an α-cyano group.</p>Formula:C23H19ClF3NO3Purity:99.76%Color and Shape:SolidMolecular weight:449.85Tezacaftor
CAS:<p>Tezacaftor (VX661) is a small molecule that can be used as a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) gene function.</p>Formula:C26H27F3N2O6Purity:98.84% - >99.99%Color and Shape:SolidMolecular weight:520.5Esomeprazole magnesium salt
CAS:<p>Esomeprazole magnesium, an oral proton pump inhibitor, curbs gastric acid by blocking H+, K+-ATPase; used in treating GERD.</p>Formula:C17H21MgN3O3SColor and Shape:SolidMolecular weight:371.74Guanidinoethyl sulfonate
CAS:<p>Guanidinoethyl sulfonate (Taurocyamine) is a competitive glycine receptor antagonist.</p>Formula:C3H9N3O3SPurity:99.43% - 99.47%Color and Shape:SolidMolecular weight:167.19Prilocaine
CAS:<p>Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of</p>Formula:C13H20N2OPurity:98.49%Color and Shape:Needles SolidMolecular weight:220.31Imidazenil
CAS:<p>Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.</p>Formula:C18H12BrFN4OPurity:98.4%Color and Shape:SolidMolecular weight:399.22Rimtuzalcap
CAS:<p>Rimtuzalcap (CAD-1883), a selective modulator for SK channels, may treat movement disorders like SCA and ET.</p>Formula:C18H24F2N6OPurity:99.64%Color and Shape:SolidMolecular weight:378.42Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Formula:C20H29N3O5SPurity:99.39% - ≥95%Color and Shape:SolidMolecular weight:423.53CFTR(inh)-172
CAS:<p>CFTR(inh)-172 (CFTR Inhibitor-172) is a voltage-independent, selective CFTR inhibitor.</p>Formula:C18H10F3NO3S2Purity:98% - 99.72%Color and Shape:SolidMolecular weight:409.4Elobixibat hydrate
CAS:<p>Elobixibat hydrate, an IBAT inhibitor, IC50: 0.53 nM (human), 0.13 nM (mouse), 5.8 nM (canine); for CIC research.</p>Formula:C36H47N3O8S2Color and Shape:SolidMolecular weight:713.9Eperisone hydrochloride
CAS:<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Formula:C17H26ClNOPurity:99.80%Color and Shape:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TasteMolecular weight:295.85Ilaprazole sodium
CAS:<p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>Formula:C19H17N4NaO2SPurity:99.06%Color and Shape:SolidMolecular weight:388.42Tiagabine
CAS:<p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>Formula:C20H25NO2S2Purity:99.25%Color and Shape:White To Off-White Crystalline SolidMolecular weight:375.55Cis-ACBD
CAS:<p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>Formula:C6H9NO4Purity:99.77%Color and Shape:SolidMolecular weight:159.14Guan-fu base A hydrochloride(1394-48-5 free base)
CAS:<p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>Formula:C24H32NO6ClPurity:99.9%Color and Shape:SolidMolecular weight:465.97Piperazine
CAS:<p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>Formula:C4H10N2Color and Shape:SolidMolecular weight:86.14GlyH-101
CAS:<p>GlyH-101 is a cell-permeable glycinyl hydrazone compound that blocks CFTR with Ki of 1.4 uM.</p>Formula:C19H15Br2N3O3Purity:98.71% - 98.78%Color and Shape:SolidMolecular weight:493.15Quadrol
CAS:<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Formula:C14H32N2O4Purity:99.91% - 99.92%Color and Shape:Viscous Liquid Liquid ViscousMolecular weight:292.41S107
CAS:<p>S107 stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>Formula:C11H15NOSPurity:99.90%Color and Shape:SolidMolecular weight:209.31Sepimostat dimethanesulfonate
CAS:<p>Sepimostat dimethanesulfonate (FUT-187) is a neuroprotective NR2B receptor antagonist with an inhibition Ki of 27.7 μM.</p>Formula:C23H27N5O8S2Color and Shape:SolidMolecular weight:565.62Tetrabenazine methanesulfonate
CAS:<p>Tetrabenazine methanesulfonate: ex-antipsychotic/therapy for movement disorders, blocks neurotransmitter uptake, labels vesicle transport.</p>Formula:C20H31NO6SPurity:98%Color and Shape:SolidMolecular weight:413.53Vanillyl butyl ether
CAS:<p>Vanillyl butyl ether (Butyl vanillyl ether) (VBE)is a capsaicin analogue,induce sensory irritation in humans,Vanillyl butyl ether is an alkoxy-substituted</p>Formula:C12H18O3Purity:99.57%Color and Shape:Yellowish Liquid LiquidMolecular weight:210.27DL-AP5
CAS:<p>DL-AP5 is the racemic form of a selective N-methyl-D-aspartate (NMDA) receptor antagonist with anticonvulsant effects.</p>Formula:C5H12NO5PPurity:99.33%Color and Shape:White Fine Crystalline PowderMolecular weight:197.13RY785
CAS:<p>RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.</p>Formula:C21H20N4O2SPurity:99.78%Color and Shape:SolidMolecular weight:392.47Parimifasor
CAS:<p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>Formula:C18H11Cl2F4N5OPurity:96.77% - 98.97%Color and Shape:SolidMolecular weight:460.21Felbamate
CAS:<p>Felbamate (W-554) is an Anti-epileptic Agent.</p>Formula:C11H14N2O4Purity:99% - >99.99%Color and Shape:White Powder SolidMolecular weight:238.24DL-Willardiine
CAS:<p>DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate.</p>Formula:C7H9N3O4Purity:99.83%Color and Shape:SolidMolecular weight:199.16A2793
CAS:<p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>Formula:C13H12ClNO3Purity:98.54%Color and Shape:SolidMolecular weight:265.69HC067047 Hydrochloride(883031-03-6 free base)
CAS:HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.Formula:C26H29ClF3N3O2Purity:99.95%Color and Shape:SolidMolecular weight:507.98Dotinurad
CAS:Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).Formula:C14H9Cl2NO4SPurity:97.43% - 98.04%Color and Shape:SolidMolecular weight:358.2Azumolene sodium anhydrous
CAS:<p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>Formula:C13H8BrN4NaO3Color and Shape:SolidMolecular weight:371.13Lesinurad
CAS:<p>Lesinurad (RDEA594), a selective uric acid reabsorption inhibitor, is used to treat gout without causing liver damage.</p>Formula:C17H14BrN3O2SPurity:99.83% - 99.86%Color and Shape:SolidMolecular weight:404.28Thiocolchicoside
CAS:<p>Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.</p>Formula:C27H33NO10SPurity:99.11% - 99.39%Color and Shape:SolidMolecular weight:563.62Flupirtine maleate
CAS:<p>Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.</p>Formula:C15H17FN4O2·C4H4O4Purity:99.5% - 99.9%Color and Shape:Off-White Crystalline PowderMolecular weight:420.39Levcromakalim
CAS:<p>Levcromakalim (BRL 38227) is an activator of the ATP-sensitive K+ channel.</p>Formula:C16H18N2O3Purity:99.74%Color and Shape:SolidMolecular weight:286.33ML213
CAS:<p>ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,</p>Formula:C17H23NOPurity:>99.99%Color and Shape:SolidMolecular weight:257.37YHO-13351
CAS:YHO-13351 is an ABCG2 inhibitor that induces sensitization of cancer stem cells/initiating-like side population cells to irinotecan.Formula:C27H37N3O7S2Purity:97.88%Color and Shape:SolidMolecular weight:579.73Lomerizine
CAS:<p>Lomerizine, a blocker of diphenylmethylpiperazine Ca2+ channel, is used to prevent migraines.</p>Formula:C27H30F2N2O3Color and Shape:SolidMolecular weight:468.54Pico145
CAS:<p>Pico145 (HC-608) is a remarkable inhibitor of TRPC1/4/5 channels.</p>Formula:C23H20ClF3N4O5Purity:99.06%Color and Shape:SolidMolecular weight:524.88p-Hydroxybenzaldehyde
CAS:1.Formula:C7H6O2Purity:99.05% - 99.86%Color and Shape:SolidMolecular weight:122.12Selinexor (KPT-330)
CAS:<p>Selinexor (KPT-330) is an orally available, small molecule inhibitor of CRM1 (exportin 1 or XPO1), with potential antineoplastic activity.</p>Formula:C17H11F6N7OPurity:98% - 99.97%Color and Shape:SolidMolecular weight:443.31TRAM-34
CAS:<p>TRAM-34 (Triarylmethane-34), an effective and specific inhibitor of the intermediate-conductance Ca2+-activated K+ channel, does not block cytochrome P450.</p>Formula:C22H17ClN2Purity:99.01% - 99.91%Color and Shape:SolidMolecular weight:344.84BI 01383298
CAS:<p>BI 01383298 is a selective inhibitor of the sodium-citrate co-transporter (SLC13A5).</p>Formula:C19H19Cl2FN2O3SPurity:99.71%Color and Shape:SolidMolecular weight:445.34Unifiram
CAS:<p>Unifiram boosts cognition, enhances rat hippocampal signals (EC50=27 nM), and ups ACh in rat cortex.</p>Formula:C13H15FN2O3SPurity:99.9%Color and Shape:SolidMolecular weight:298.33TRPM4-IN-1
CAS:<p>TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.</p>Formula:C15H11Cl2NO4Purity:97.22%Color and Shape:SolidMolecular weight:340.16GLPG1837
CAS:<p>GLPG1837 (ABBV-974) is an effective CFTR potentiator, with EC50s of 3 nM and 339 nM for F508del and G551D CFTR, respectively.</p>Formula:C16H20N4O3SPurity:99.64% - 99.91%Color and Shape:SolidMolecular weight:348.42Caroverine hydrochloride
CAS:Caroverine HCL: Blocks NMDA/AMPA receptors, antioxidant, calcium-blocker, and vasorelaxant, used for tinnitus research.Formula:C22H28ClN3O2Purity:98.37% - 98.75%Color and Shape:SolidMolecular weight:401.9VU590 HCl
CAS:<p>VU590 is a small molecule inhibitor of KCNJ1 (IC50 = 294 nM).</p>Formula:C24H34Cl2N4O7Color and Shape:SolidMolecular weight:561.457Tricaine methanesulfonate
CAS:<p>Tricaine methanesulfonate (TMS/MS-222) is an anesthetic used in hatcheries and studies to immobilize fish for marking, transport, and invasive procedures.</p>Formula:C10H15NO5SPurity:99.259% - 99.86%Color and Shape:White PowderMolecular weight:261.30CTP disodium dihydrate
CAS:<p>CTP disodium dihydrate is an agonist of P2X4 purinergic receptor</p>Formula:C9H18N3Na2O16P3Purity:98.51%Color and Shape:White Crystalline PowderMolecular weight:563.15Methyl homoveratrate
CAS:<p>Methyl homoveratrate, a McN5691 (RWJ-26240) metabolite detected in vivo in plasma, urine, and fecal extracts, functions as a voltage-sensitive calcium channel</p>Formula:C11H14O4Purity:99.48%Color and Shape:SolidMolecular weight:210.23Quinine hydrobromide
CAS:<p>Quinidine: oral, selective P450db inhibitor, K+ channel blocker (IC50=19.9μM), antiarrhythmic, used in malaria research.</p>Formula:C20H25BrN2O2Color and Shape:SolidMolecular weight:405.336SSD114 HCl
CAS:<p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>Formula:C18H21ClF3N3OPurity:99.03% - 99.95%Color and Shape:SolidMolecular weight:387.83BzATP triethylammonium salt
CAS:<p>BzATP triethylammonium salt is a P2X7 receptor agonist.</p>Formula:C30H39N6O15P3Purity:95% - 99.57%Color and Shape:SolidMolecular weight:816.59MK6-83
CAS:<p>MK6-83 is the transient receptor potential channel ML3 agonist.</p>Formula:C16H20N2O2S2Purity:99.5%Color and Shape:SolidMolecular weight:336.47ICA-121431
CAS:<p>ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.</p>Formula:C23H19N3O3S2Purity:98.06%Color and Shape:SolidMolecular weight:449.55Sodium ionophore III
CAS:<p>Sodium ionophore III (ETH2120) is a Na+ ionophore suitable for the test of sodium activity in plasma, serum, and blood.</p>Formula:C34H52N2O4Purity:99.51% - 99.78%Color and Shape:SolidMolecular weight:552.79Vonoprazan
CAS:<p>Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer and</p>Formula:C17H16FN3O2SPurity:99.87% - 99.92%Color and Shape:SolidMolecular weight:345.39Eniporide hydrochloride
CAS:<p>Eniporide hydrochloride (EMD-96785 hydrochloride) serves as a robust inhibitor of the sodium/hydrogen (Na+/H+) exchange process.</p>Formula:C14H17ClN4O3SColor and Shape:SolidMolecular weight:356.83Esomeprazole hemistrontium
CAS:<p>Esomeprazole hemistrontium, potent oral proton pump inhibitor, reduces gastric acid by blocking H+, K+-ATPase.</p>Formula:C34H36N6O6S2SrColor and Shape:SolidMolecular weight:776.44O4I1
CAS:<p>O4I1 is an effective Oct3/4 inducer.</p>Formula:C16H15NO2Purity:96.25% - 99.47%Color and Shape:SolidMolecular weight:253.39-Phenanthrol
CAS:<p>9-Phenanthrol is inhibitor of the transient receptor potential melastatin 4 (TRPM) channel, a Ca2+ -activated non-selective cation channel.</p>Formula:C14H10OPurity:98.48%Color and Shape:SolidMolecular weight:194.23Ononetin
CAS:<p>Ononetin (2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone) is a TRPM3 channel blocker(IC50: 0.3 μM).</p>Formula:C15H14O4Purity:98.06%Color and Shape:SolidMolecular weight:258.27Neramexane HCl
CAS:PAC is a cyclic amine used as a chiral auxiliary in various asymmetric syntheses.Formula:C11H24ClNPurity:95.00%Color and Shape:SolidMolecular weight:205.768NPPB
CAS:<p>NPPB is a chloride channel blocker with IC50 of 80 nM .</p>Formula:C16H16N2O4Purity:99.95%Color and Shape:Light Yellow To Yellow SolidMolecular weight:300.31Ivacaftor
CAS:<p>Ivacaftor (VX-770) (VX-770) is a potentiator of CFTR targeting G551D-CFTR (EC50: 100 nM) and F508del-CFTR (EC50: 25 nM) in Fisher rat thyroid cells,</p>Formula:C24H28N2O3Purity:99% - 99.98%Color and Shape:SolidMolecular weight:392.49Tiludronate
CAS:<p>Tiludronate, an oral bisphosphonate, treats metabolic bone disorders and inhibits osteoclasts.</p>Formula:C7H9ClO6P2SColor and Shape:SolidMolecular weight:318.61ML133 hydrochloride
CAS:<p>ML133 hydrochloride (ML133 HCl) is a selective potassium channel inhibitor for Kir2.1, has no effect on Kir1.1 and weak activity for Kir4.1 and Kir7.1.</p>Formula:C19H19NO·HClPurity:99.48%Color and Shape:SolidMolecular weight:313.82Selamectin
CAS:<p>Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in</p>Formula:C43H63NO11Purity:99.84%Color and Shape:SolidMolecular weight:769.96PF-4840154
CAS:<p>PF-4840154: potent TrpA1 agonist; EC50 of 97 nM (rat) & 23 nM (human); triggers nociception in mice.</p>Formula:C26H38N6O2Purity:>99.99%Color and Shape:SolidMolecular weight:466.62Myomodulin acetate(110570-93-9 free base)
<p>Myomodulin acetate is present in two identified aplysia neurons that contain myomodulin A the ARC motor neuron B16 and the abdominal neuron L10.</p>Formula:C38H71N11O10S2Purity:99.24%Color and Shape:SolidMolecular weight:906.17Esomeprazole potassium salt
CAS:<p>Esomeprazole potassium, a potent oral proton pump inhibitor, curbs acid secretion in stomach cells, aiding GERD research.</p>Formula:C17H18KN3O3SColor and Shape:SolidMolecular weight:383.51Flecainide acetate
CAS:<p>Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).</p>Formula:C19H24F6N2O5Purity:99.42%Color and Shape:SolidMolecular weight:474.39NS6180
CAS:<p>NS6180 is a potent and selective KCa3.1 channel inhibitor(IC50= 9 nM). It prevents T-cell activation and inflammation.</p>Formula:C16H12F3NOSPurity:99.83% - ≥95%Color and Shape:SolidMolecular weight:323.33Flecainide hydrochloride
CAS:<p>Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.</p>Formula:C17H21ClF6N2O3Purity:97.79%Color and Shape:SolidMolecular weight:450.81Rbin-1
CAS:<p>Rbin-1 (Ribozinoindole-1) is a potent,specific inhibitor of eukaryotic ribosome biogenesis.</p>Formula:C13H12N4SPurity:99.83%Color and Shape:SolidMolecular weight:256.33Enflurane
CAS:<p>Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.</p>Formula:C3H2ClF5OPurity:99.64%Color and Shape:Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As AnMolecular weight:184.49Azimilide Dihydrochloride
CAS:Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.Formula:C23H30Cl3N5O3Purity:97.59% - ≥95%Color and Shape:SolidMolecular weight:530.88Fipronil
CAS:<p>Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.</p>Formula:C12H4Cl2F6N4OSPurity:97.21%Color and Shape:Solid PowderMolecular weight:437.15KB-R7943 mesylate
CAS:<p>KB-R7943 mesylate is a widely used inhibitor of the reverse Na+/Ca2+ exchanger (NCXrev) with IC50 of 5.7±2.1 μM.</p>Formula:C17H21N3O6S2Purity:99.88% - ≥95%Color and Shape:SolidMolecular weight:427.5Nicainoprol
CAS:<p>Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent.</p>Formula:C21H27N3O3Purity:99.54%Color and Shape:SolidMolecular weight:369.46Amlodipine mesylate
CAS:<p>Amlodipine mesylate, an oral dihydropyridine Ca2+ blocker, treats angina, hypertension, and may be used in cancer research.</p>Formula:C21H29ClN2O8SColor and Shape:SolidMolecular weight:504.98DS-1971a
CAS:<p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>Formula:C20H21ClFN5O3SPurity:99.66%Color and Shape:SolidMolecular weight:465.93Jujuboside A
CAS:<p>Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.</p>Formula:C58H94O26Purity:98% - >99.99%Color and Shape:SolidMolecular weight:1207.35Rufinamide
CAS:<p>Rufinamide (E 2080), a triazole derivative, is used as voltage-gated sodium channel blocker for the treatment of seizure disorders.</p>Formula:C10H8F2N4OPurity:99.77% - >99.99%Color and Shape:White PowderMolecular weight:238.19Ibutilide Fumarate
CAS:<p>Ibutilide Fumarate is a class III antiarrhythmic, prolonging action potentials by enhancing sodium influx, and can extend QT interval.</p>Formula:(C20H36N2O3S)2·C4H4O4Purity:99.68% - 99.74%Color and Shape:SolidMolecular weight:885.23Ko 143
CAS:<p>Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).</p>Formula:C26H35N3O5Purity:99.01% - 99.89%Color and Shape:SolidMolecular weight:469.57BAY-8002
CAS:<p>BAY-8002 is a potent dual MCT1/2 inhibitor (IC50 values are 3, 8, and 12 nM at rat (C6), human (DLD-1) and mouse (4T1) MCT1 respectively).</p>Formula:C20H14ClNO5SPurity:98.7% - 99.13%Color and Shape:SolidMolecular weight:415.85Phe-Met-Arg-Phe, amide acetate
<p>Phe-Met-Arg-Phe amide acetate (ED50=23 nM) triggers K+ current in caudodorsal neurons, co-localizes with neuropeptide Y in brain areas.</p>Formula:C31H46N8O6SPurity:99.4%Color and Shape:SolidMolecular weight:658.82Benzamil
CAS:<p>Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.</p>Formula:C13H14ClN7OPurity:99.79%Color and Shape:SolidMolecular weight:319.75Tetraethylammonium chloride
CAS:<p>Tetraethylammonium chloride is a quaternary ammonium compound.</p>Formula:C8H20ClNPurity:≥95%Color and Shape:White Solid Solid Particulate/PowderMolecular weight:165.7SAR7334 hydrochloride
CAS:<p>SAR7334 hydrochloride is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Formula:C21H24Cl3N3OPurity:98%Color and Shape:SolidMolecular weight:440.79Pikamilone
CAS:<p>Pikamilone (Picamilon) is an intelligent medicine.</p>Formula:C10H12N2O3Purity:99.38%Color and Shape:White Crystalline PowderMolecular weight:208.21BRITE-338733
CAS:<p>BRITE-338733 is a novel inhibitor of ATPase. BRITE 338733 inhibits the expression of RecA in bacteria (IC50=4.7 μM) for the bacterial infections treatment.</p>Formula:C27H35N3O2Purity:99.85%Color and Shape:SolidMolecular weight:433.59Raxatrigine
CAS:Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.Formula:C18H19FN2O2Purity:98% - 99.43%Color and Shape:SolidMolecular weight:314.35VU590
CAS:<p>VU590 is an inhibitor of extrarenal medullary potassium ROMK.VU590 inhibits Kir7.1 and modulates uterine myometrial contractility and melanocortin signalling.</p>Formula:C24H32N4O7Purity:98.06%Color and Shape:SolidMolecular weight:488.53Darigabat
CAS:<p>Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.</p>Formula:C22H21FN4O3SPurity:98.42% - 99.29%Color and Shape:SolidMolecular weight:440.49Methionine
CAS:<p>Methionine (D-Methionine) (MRX-1024; D-Methionine) is an effective chemoprotective agent which can also inhibit the neuronal activity through GABAA receptor</p>Formula:C5H11NO2SPurity:99.13% - 99.62%Color and Shape:SolidMolecular weight:149.21Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Formula:C8H5F3N2OSPurity:99.71% - 99.88%Color and Shape:PowderMolecular weight:234.2VB124
CAS:<p>VB124 is an orally active, potent and selective MCT4 inhibitor. VB124 blocked lactate importand expor in MDA-MB-231 cells.Cost-effective and quality-assured.</p>Formula:C23H23ClN2O4Purity:99.21% - 99.57%Color and Shape:SoildMolecular weight:426.89Dimiracetam
CAS:<p>Dimiracetam, a NMDA-receptor antagonist, is used potentially for the treatment of neuropathic pain.</p>Formula:C6H8N2O2Purity:>99.99% - >99.99%Color and Shape:SolidMolecular weight:140.14ZT-1a
CAS:<p>ZT-1a is a SPAK inhibitor.ZT-1a inhibits SPAK.ZT-1a can be used for the prevention and treatment of neurodegenerative and neurocognitive disorders.</p>Formula:C22H15Cl3N2O2Purity:99.77%Color and Shape:SolidMolecular weight:445.73Mtb ATP synthase-IN-1
CAS:Mtb ATP synthase-IN-1 is a potent, low-toxicity M. tuberculosis inhibitor with good oral bioavailability and metabolic stability.Formula:C17H13N3O4Purity:98.28%Color and Shape:SolidMolecular weight:323.30CX717
CAS:<p>CX 717 is a positive allosteric modulator of AMPA receptor which has an antidepressant-like effect.</p>Formula:C11H11N3O3Purity:99.81%Color and Shape:SoildMolecular weight:233.23Lanicemine dihydrochloride
CAS:<p>Lanicemine dihydrochloride (AZD-6765 dihydrochloride) is an NMDA channel blocker with antidepressant activity and can be used to study neurological diseases.</p>Formula:C13H16Cl2N2Purity:98.37%Color and Shape:SolidMolecular weight:271.19SRI-41315
CAS:<p>SRI-41315 is an eRF1 degrader that acts as a molecular glue at the ribosomal decoding center.SRI-41315 induces extended pauses at the termination codon.</p>Formula:C22H19N3O2Purity:99.87%Color and Shape:SolidMolecular weight:357.41Ro 25-6981 Maleate
CAS:<p>Ro 25-6981 Maleate is an NMDA receptor antagonist used in the study of neurological disorders such as Parkinson's and epilepsy.</p>Formula:C26H33NO6Purity:99.42%Color and Shape:SolidMolecular weight:455.54Propoxycaine hydrochloride
CAS:Propoxycaine hydrochloride is an ester local anesthetic that inhibits voltage-gated sodium channels, modulates nerve impulses, and induces loss of sensation.Formula:C16H27ClN2O3Purity:97.25%Color and Shape:SolidMolecular weight:330.85JNJ-28583113
CAS:<p>JNJ-28583113 is a TRPM2 antagonist, inducing phosphorylation of GSK3α and β subunits, protecting cells from oxidative stress-induced cell death.</p>Formula:C19H21F3N2O2Purity:98.57%Color and Shape:SolidMolecular weight:366.38PF 03716556
CAS:<p>PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal reflux</p>Formula:C22H26N4O3Purity:99.79% - 99.85%Color and Shape:SolidMolecular weight:394.47HUP30
CAS:<p>HUP30 is a potent vasodilating agent. HUP30 can stimulate soluble guanylyl cyclase, activate K+ channels, and block extracellular Ca2+ influx.</p>Formula:C14H15N3O3SPurity:99.96%Color and Shape:SolidMolecular weight:305.35Bupivacaine
CAS:<p>Bupivacaine (AH-250) is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels</p>Formula:C18H28N2OPurity:99.83%Color and Shape:SolidMolecular weight:288.43N-Methyl-L-leucin
CAS:<p>N-Methyl-L-leucine ((S)-4-Methyl-2-(methylamino)pentanoic acid) is a novel calcium channel antagonist used in pain research.</p>Formula:C7H15NO2Purity:99.87%Color and Shape:SolidMolecular weight:145.2Safinamide
CAS:<p>Safinamide: reversible MAO-B inhibitor, enhances dopamine, blocks glutamate release, sodium, calcium channels; may treat Parkinson's, RLS, epilepsy.</p>Formula:C17H19FN2O2Purity:99.92%Color and Shape:SolidMolecular weight:302.34BL-1249
CAS:<p>BL-1249 is a selective and potent non-steroidal potassium channel activator with anti-inflammatory activity that activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2).</p>Formula:C17H17N5Purity:98% - 98.25%Color and Shape:SolidMolecular weight:291.35Doxapram
CAS:Doxapram (Dopram) is a respiratory stimulant that inhibits TASK-1, TASK-3, and TASK-1/TASK-3 heterodimer channels.Formula:C24H30N2O2Purity:99.42%Color and Shape:SolidMolecular weight:378.51Apinocaltamide
CAS:Apinocaltamide (ACT-709478) is an orally available and selective T-type calcium channel blocker that cross BBB for Cav3.1, Cav3.2, and Cav3.3,epilepsy.Formula:C22H18F3N5OPurity:99.80%Color and Shape:SolidMolecular weight:425.41Bupivacaine-d9
CAS:Bupivacaine-d9 is a deuterated compound of Bupivacaine. Bupivacaine has a CAS number of 38396-39-3. Bupivacaine is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels with the IC50 of 69.5 μM. Bupivacaine can be used for the research of chronic pain.Formula:C18H19D9N2OColor and Shape:SolidMolecular weight:297.48Eleclazine
CAS:<p>Eleclazine (GS-6615) is a novel and selective voltage-gated sodium channel inhibitor with antiarrhythmic properties that reduces peak sodium current (INaP).</p>Formula:C21H16F3N3O3Purity:98.67%Color and Shape:SolidMolecular weight:415.37SAR7334
CAS:<p>SAR7334 (TRCP6-IN-1) is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Formula:C21H22ClN3OPurity:99.62% - 99.71%Color and Shape:SolidMolecular weight:367.87FSC231
CAS:<p>FSC231 is a PICK1 inhibitor with analgesic activity, activating GSK-3β and ERK1/2.</p>Formula:C13H10Cl2N2O3Purity:99.66%Color and Shape:SolidMolecular weight:313.14Amlodipine hydrochloride
CAS:<p>Amlodipine hydrochloride is a salt of Amlodipine --- a medication used to lower blood pressure and prevent chest pain.</p>Formula:C20H26Cl2N2O5Color and Shape:SolidMolecular weight:445.34Amlodipine besilate impurity G
CAS:<p>Amlodipine besilate impurity G is a Calcium Channel antagonist with potential application in the study of neurological diseases and is an impurity in the</p>Formula:C17H18ClNO4Purity:98%Color and Shape:SolidMolecular weight:335.78Flavoxate
CAS:<p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>Formula:C24H25NO4Color and Shape:SolidMolecular weight:391.46Cinepazide
CAS:<p>Cinepazide: a vasodilator targeting adenosine A2 receptors, treats various vascular diseases.</p>Formula:C22H31N3O5Color and Shape:White PowderMolecular weight:417.5VGSC blocker-1
CAS:<p>VGSC blocker-1 inhibits 34.9% INa in nNav1.5 at 1 μM, reduces MDA-MB-231 invasion by 0.3%, non-toxic.</p>Formula:C24H32F2N2Color and Shape:SolidMolecular weight:386.52MCT-IN-1
CAS:<p>MCT-IN-1 (compound 2) acts as a potent inhibitor of the monocarboxylate transporter (MCT), demonstrating IC50 values of 9 nM for MCT1 and 14 nM for MCT4.</p>Formula:C19H26N2O3Color and Shape:SolidMolecular weight:330.42Eperisone
CAS:<p>Eperisone: a muscle relaxant for stiffness and pain, relaxes muscles, improves circulation, and mitigates pain by inhibiting reflexes and vasodilation.</p>Formula:C17H25NOColor and Shape:SolidMolecular weight:259.39Dofetilide D4
CAS:Dofetilide D4 (UK 68789 D4), a deuterium-labeled version of Dofetilide, is categorized as a Class III antiarrhythmic medication.Formula:C19H27N3O5S2Purity:98%Color and Shape:SolidMolecular weight:445.59Nifedipine-d6
CAS:<p>Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.</p>Formula:C17H18N2O6Purity:98%Color and Shape:SolidMolecular weight:352.37Propafenone D7 hydrochloride
CAS:<p>Propafenone D7 hydrochloride is the deuterium labeled Propafenone, and is a classic anti-arrhythmic medication.</p>Formula:C21H28ClNO3Purity:98%Color and Shape:SolidMolecular weight:384.95Topiramate D12
CAS:<p>Topiramate D12 is a deuterium labeled Topiramate. Topiramate is an agent of broad-spectrum antiepileptic. Topiramate is an antagonist of GluR5 receptor.</p>Formula:C12H21NO8SPurity:98%Color and Shape:SolidMolecular weight:351.44PBFI-AM
CAS:<p>PBFI-AM is a useful tool to determine intracellular K + content [1] .</p>Formula:C58H62N2O24Color and Shape:SolidMolecular weight:1171.11BAY-390
CAS:<p>BAY-390, a selective TRPA1 inhibitor, crosses species, penetrates brains, with IC50s: 16-82 nM. Used in inflammation research.</p>Formula:C13H15F4NOColor and Shape:SolidMolecular weight:277.26Bumetanide-d5
CAS:Bumetanide D5 is a deuterium-labeled Bumetanide. Bumetanide is a Na+-K+-Cl- (NKCC1) inhibitor (IC50s: 0.68 and 4.0 μM for hNKCC1A and hNKCC2A).Formula:C17H20N2O5SPurity:98%Color and Shape:SolidMolecular weight:369.45
