CymitQuimica logo
5-HT Receptor

5-HT Receptor

5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.

Found 940 products of "5-HT Receptor"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • TG6-10-1

    CAS:
    <p>TG6-10-1 is an EP2 antagonist.</p>
    Formula:C23H23F3N2O4
    Purity:99.66% - ≥95%
    Color and Shape:Solid
    Molecular weight:448.43
  • Puerarin

    CAS:
    <p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>
    Formula:C21H20O9
    Purity:98.90% - 99.21%
    Color and Shape:Yellow Brown Fine Powder
    Molecular weight:416.38
  • Rotigotine Hydrochloride

    CAS:
    <p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>
    Formula:C19H26ClNOS
    Purity:99.53% - 99.56%
    Color and Shape:Almost White To White Crystalline Powder
    Molecular weight:351.93
  • Rotigotine-

    CAS:
    <p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>
    Formula:C19H25NOS
    Purity:98.08% - 99.59%
    Color and Shape:Solid
    Molecular weight:315.47
  • MK 212 hydrochloride

    CAS:
    <p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>
    Formula:C8H11ClN4·HCl
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:235.12
  • Metadoxine

    CAS:
    <p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>
    Formula:C8H11NO3·C5H7NO3
    Purity:99.19%
    Color and Shape:Off-White Powder
    Molecular weight:298.29
  • Intepirdine

    CAS:
    <p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>
    Formula:C19H19N3O2S
    Purity:98% - 98.63%
    Color and Shape:Solid
    Molecular weight:353.44
  • Mosapride Citrate

    CAS:
    <p>Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.</p>
    Formula:C21H25ClFN3O3·C6H8O7
    Purity:99.70%
    Color and Shape:White Powder
    Molecular weight:614.02
  • GSK163090

    CAS:
    <p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>
    Formula:C25H29N5O
    Purity:99.2%
    Color and Shape:Solid
    Molecular weight:415.53
  • Tianeptine

    CAS:
    <p>Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>
    Formula:C21H25ClN2O4S
    Purity:99.04%
    Color and Shape:Solid
    Molecular weight:436.95
  • Niaprazine

    CAS:
    <p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>
    Formula:C20H25FN4O
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:356.44
  • BRL-15572 dihydrochloride

    CAS:
    <p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>
    Formula:C25H27ClN2O·2HCl
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:479.87
  • Dolasetron Mesylate hydrate

    CAS:
    <p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>
    Formula:C20H26N2O7S
    Purity:99.86% - 99.9%
    Color and Shape:Solid
    Molecular weight:438.49
  • PRX-08066

    CAS:
    <p>PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.</p>
    Formula:C19H17ClFN5S
    Purity:97.79% - 98.07%
    Color and Shape:Solid
    Molecular weight:401.89
  • Ipsapirone hydrochloride

    CAS:
    <p>Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.</p>
    Formula:C19H24ClN5O3S
    Color and Shape:Solid
    Molecular weight:437.94
  • Donitriptan Mesylate

    CAS:
    <p>Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.</p>
    Formula:C24H29N5O5S
    Color and Shape:Solid
    Molecular weight:499.58
  • Melitracen

    CAS:
    <p>Melitracen is a tricyclic antidepressant.</p>
    Formula:C21H25N
    Color and Shape:Solid
    Molecular weight:291.43
  • Abaperidone Hydrochloride

    CAS:
    <p>Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.</p>
    Formula:C25H26ClFN2O5
    Color and Shape:Solid
    Molecular weight:488.94
  • Melperone

    CAS:
    <p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>
    Formula:C16H22FNO
    Purity:98.84%
    Color and Shape:Solid
    Molecular weight:263.35
  • Cannabigerol

    CAS:
    <p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>
    Formula:C21H32O2
    Purity:99.59% - 99.92%
    Color and Shape:Solid
    Molecular weight:316.48
  • Temanogrel

    CAS:
    <p>Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).</p>
    Formula:C24H28N4O4
    Purity:99.24%
    Color and Shape:Solid
    Molecular weight:436.5
  • 2'-O-Methylisoliquiritigenin

    CAS:
    <p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>
    Formula:C16H14O4
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:270.28
  • Alprenolol hydrochloride

    CAS:
    <p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>
    Formula:C15H24ClNO2
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:285.81
  • idalopirdine

    CAS:
    <p>Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.</p>
    Formula:C20H19F5N2O
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:398.37
  • Nuciferine

    CAS:
    <p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>
    Formula:C19H21NO2
    Purity:98.76% - 99.79%
    Color and Shape:Solid
    Molecular weight:295.38
  • Naratriptan

    CAS:
    <p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>
    Formula:C17H25N3O2S
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:335.47
  • Methiothepin mesylate

    CAS:
    <p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>
    Formula:C21H28N2O3S3
    Purity:98% - 99.92%
    Color and Shape:Solid
    Molecular weight:452.65
  • Rotundine

    CAS:
    <p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>
    Formula:C21H25NO4
    Purity:99.8% - 99.91%
    Color and Shape:Off-White Solid
    Molecular weight:355.43
  • BMY 7378 dihydrochloride

    CAS:
    <p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>
    Formula:C22H33Cl2N3O3
    Purity:97.32% - 99.08%
    Color and Shape:Solid
    Molecular weight:458.42
  • F-15599

    CAS:
    <p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>
    Formula:C19H21ClF2N4O
    Purity:98.72%
    Color and Shape:Solid
    Molecular weight:394.85
  • Pirenperone

    CAS:
    <p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>
    Formula:C23H24FN3O2
    Purity:99.2%
    Color and Shape:Solid
    Molecular weight:393.45
  • 7-Amino-4-(trifluoromethyl)coumarin

    CAS:
    <p>7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.</p>
    Formula:C10H6F3NO2
    Purity:97.31% - 97.84%
    Color and Shape:Yellow Powder
    Molecular weight:229.16
  • Cariprazine

    CAS:
    <p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>
    Formula:C21H32Cl2N4O
    Purity:99.68% - 99.87%
    Color and Shape:Solid
    Molecular weight:427.41
  • Almotriptan Malate

    CAS:
    <p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>
    Formula:C17H25N3O2S·C4H6O5
    Purity:99.95%
    Color and Shape:Pale Yellow Solid
    Molecular weight:469.55
  • Escitalopram Oxalate

    CAS:
    <p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>
    Formula:C22H23FN2O5
    Purity:97.39% - 99.73%
    Color and Shape:White Solid
    Molecular weight:414.43
  • Serotonin hydrochloride

    CAS:
    <p>Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (</p>
    Formula:C10H13ClN2O
    Purity:98.05% - 99.93%
    Color and Shape:White To Cream Powder
    Molecular weight:212.676
  • Azaphen

    CAS:
    <p>Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.</p>
    Formula:C16H21Cl2N5O
    Purity:97.62%
    Color and Shape:Solid
    Molecular weight:370.28
  • Piboserod

    CAS:
    <p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>
    Formula:C22H31N3O2
    Purity:97.21% - 99.49%
    Color and Shape:Solid
    Molecular weight:369.5
  • Perospirone

    CAS:
    <p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>
    Formula:C23H30N4O2S
    Purity:99.23%
    Color and Shape:White Powder
    Molecular weight:426.57
  • SB399885

    CAS:
    <p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>
    Formula:C18H21Cl2N3O4S
    Purity:98.94%
    Color and Shape:Solid
    Molecular weight:446.35
  • LY334370

    CAS:
    <p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>
    Formula:C21H22FN3O
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:351.42
  • Sevoflurane

    CAS:
    <p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>
    Formula:C4H3F7O
    Purity:98%
    Color and Shape:Less Oil Colorless Oil
    Molecular weight:200.05
  • Geissoschizine methyl ether

    CAS:
    <p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>
    Formula:C22H26N2O3
    Purity:99.24% - 99.68%
    Color and Shape:Solid
    Molecular weight:366.45
  • Ansofaxine hydrochloride

    CAS:
    <p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>
    Formula:C24H32ClNO3
    Purity:99.57% - 99.77%
    Color and Shape:Solid
    Molecular weight:417.97
  • Tropisetron

    CAS:
    <p>Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.</p>
    Formula:C17H20N2O2
    Purity:99.68%
    Color and Shape:White Solid
    Molecular weight:284.35
  • Nelotanserin

    CAS:
    <p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>
    Formula:C18H15BrF2N4O2
    Purity:98.42% - 99.88%
    Color and Shape:Solid
    Molecular weight:437.24
  • Amitriptyline

    CAS:
    <p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>
    Formula:C20H23N
    Purity:98.24% - 99.64%
    Color and Shape:Crystals Solid
    Molecular weight:277.4
  • Brexpiprazole HCl

    CAS:
    <p>Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.</p>
    Formula:C25H27N3O2S·xHCl
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:433.6
  • Sarpogrelate hydrochloride

    CAS:
    <p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>
    Formula:C24H32ClNO6
    Purity:99.73%
    Color and Shape:Colorless Liquid
    Molecular weight:465.97
  • Lurasidone hydrochloride

    CAS:
    <p>Lurasidone HCl: Atypical antipsychotic, treats schizophrenia &amp; bipolar, affects dopamine, serotonin &amp; adrenergic receptors.</p>
    Formula:C28H36N4O2S·HCl
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:529.14
  • PRX-07034 hydrochloride

    CAS:
    <p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>
    Formula:C21H29Cl2N3O4S
    Purity:98.5%
    Color and Shape:Solid
    Molecular weight:490.44
  • Clozapine N-Oxide

    CAS:
    <p>View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.</p>
    Formula:C18H19ClN4O
    Purity:98.43% - 99.94%
    Color and Shape:Solid
    Molecular weight:342.82
  • Nemifitide acetate(173240-15-8 free base)


    <p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>
    Formula:C35H47FN10O8
    Purity:97.97%
    Color and Shape:Solid
    Molecular weight:754.85
  • Cinitapride

    CAS:
    <p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>
    Formula:C21H30N4O4
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:402.49
  • Pergolide mesylate

    CAS:
    <p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>
    Formula:C20H30N2O3S2
    Purity:99.70%
    Color and Shape:White To Off-White Solid
    Molecular weight:410.59
  • Dasotraline hydrochloride

    CAS:
    <p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>
    Formula:C16H16Cl3N
    Purity:98.92% - 99.6%
    Color and Shape:Solid
    Molecular weight:328.66
  • L-745870 trihydrochloride

    CAS:
    <p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>
    Formula:C18H22Cl4N4
    Purity:97.52%
    Color and Shape:Solid
    Molecular weight:436.21
  • 5-Benzyloxygramine

    CAS:
    <p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>
    Formula:C18H20N2O
    Purity:99.13%
    Color and Shape:Solid
    Molecular weight:280.36
  • N-Desmethylclozapine

    CAS:
    <p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>
    Formula:C17H17ClN4
    Purity:97.25% - 99.83%
    Color and Shape:Yellow Crystalline Solid
    Molecular weight:312.8
  • NGB 2904

    CAS:
    <p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>
    Formula:C28H29Cl2N3O
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:494.46
  • Chlorprothixene

    CAS:
    <p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>
    Formula:C18H18ClNS
    Purity:98.77% - 99.756%
    Color and Shape:Pale Yellow Crystals Solid
    Molecular weight:315.86
  • Piperacetazine

    CAS:
    <p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>
    Formula:C24H30N2O2S
    Purity:99.9% - 99.92%
    Color and Shape:Solid
    Molecular weight:410.57
  • Loxapine

    CAS:
    <p>Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.</p>
    Formula:C18H18ClN3O
    Purity:99.88%
    Color and Shape:Pale Yellowish Crystals From Petroleum Ether Solid
    Molecular weight:327.81
  • Brexpiprazole

    CAS:
    <p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>
    Formula:C25H27N3O2S
    Purity:99.06% - 99.96%
    Color and Shape:Solid
    Molecular weight:433.57
  • Jatrorrhizine

    CAS:
    <p>Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.</p>
    Formula:C20H20NO4
    Purity:97.18% - 99.06%
    Color and Shape:Solid
    Molecular weight:338.38
  • Urapidil

    CAS:
    <p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>
    Formula:C20H29N5O3
    Purity:99.85% - >99.99%
    Color and Shape:Solid
    Molecular weight:387.48
  • RS-127445 hydrochloride

    CAS:
    <p>RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).</p>
    Formula:C17H17ClFN3
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:317.79
  • Zacopride hydrochloride

    CAS:
    <p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>
    Formula:C15H20ClN3O2·HCl
    Purity:98.32%
    Color and Shape:Solid
    Molecular weight:346.26
  • 8-Hydroxy-DPAT hydrobromide

    CAS:
    <p>8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.</p>
    Formula:C16H26BrNO
    Purity:98.90% - 99.09%
    Color and Shape:Solid
    Molecular weight:328.29
  • SB-203186 hydrochloride

    CAS:
    <p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>
    Formula:C16H20N2O2·HCl
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:308.81
  • Myristicin

    CAS:
    <p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>
    Formula:C11H12O3
    Purity:99.828%
    Color and Shape:Liquid
    Molecular weight:192.21
  • Hypidone hydrochloride

    CAS:
    <p>Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor</p>
    Formula:C18H23ClN2O2
    Purity:99.82% - 99.93%
    Color and Shape:Solid
    Molecular weight:334.84
  • Vortioxetine

    CAS:
    <p>Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.</p>
    Formula:C18H22N2S
    Purity:99.34% - 99.34%
    Color and Shape:Solid
    Molecular weight:298.45
  • BRL 54443

    CAS:
    <p>BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).</p>
    Formula:C14H18N2O
    Purity:98.07%
    Color and Shape:Solid
    Molecular weight:230.31
  • 6-fluoro-DL-Tryptophan

    CAS:
    <p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>
    Formula:C11H11FN2O2
    Purity:99.25%
    Color and Shape:Off-White Powder
    Molecular weight:222.22
  • Serotonin

    CAS:
    <p>Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!</p>
    Formula:C10H12N2O
    Purity:97.47% - 99.92%
    Color and Shape:Solid
    Molecular weight:176.22
  • NAN-190 hydrobromide

    CAS:
    <p>NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.</p>
    Formula:C23H28BrN3O3
    Purity:95.20%
    Color and Shape:Solid
    Molecular weight:474.39
  • Perospirone hydrochloride

    CAS:
    <p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>
    Formula:C23H31ClN4O2S
    Purity:99.37%
    Color and Shape:White Solid
    Molecular weight:463
  • 3-AQC

    CAS:
    <p>3-AQC is a competitive antagonist of 5-HT3.</p>
    Formula:C20H21N5O4
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:395.41
  • AVN-101

    CAS:
    <p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>
    Formula:C21H25ClN2
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:340.89
  • SCH-23390 hydrochloride

    CAS:
    <p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>
    Formula:C17H19Cl2NO
    Purity:98% - 99.83%
    Color and Shape:Solid
    Molecular weight:324.24
  • Mosapride

    CAS:
    <p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>
    Formula:C21H25ClFN3O3
    Purity:99.56%
    Color and Shape:White To Off-White Crystalline Solid
    Molecular weight:421.89
  • Tianeptine sodium salt

    CAS:
    <p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>
    Formula:C21H24ClN2NaO4S
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:458.93
  • Vilazodone Hydrochloride

    CAS:
    <p>Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the</p>
    Formula:C26H27N5O2·HCl
    Purity:99.56% - >99.99%
    Color and Shape:Solid
    Molecular weight:477.99
  • Xaliproden hydrochloride

    CAS:
    <p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>
    Formula:C24H23ClF3N
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:417.89
  • lumateperone Tosylate

    CAS:
    <p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>
    Formula:C31H36FN3O4S
    Purity:95.83% - 99.95%
    Color and Shape:Solid
    Molecular weight:565.7
  • Cerlapirdine

    CAS:
    <p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>
    Formula:C22H23N3O3S
    Purity:98.77%
    Color and Shape:Solid
    Molecular weight:409.5
  • Cariprazine hydrochloride

    CAS:
    <p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>
    Formula:C21H33Cl3N4O
    Purity:99.78% - >99.99%
    Color and Shape:Solid
    Molecular weight:463.87
  • Lerisetron

    CAS:
    <p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>
    Formula:C18H20N4
    Purity:99.15% - 99.82%
    Color and Shape:Solid
    Molecular weight:292.38
  • Indophagolin

    CAS:
    <p>Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.</p>
    Formula:C19H15BrClF3N2O3S
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:523.75
  • Amperozide

    CAS:
    <p>Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.</p>
    Formula:C23H29F2N3O
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:401.49
  • Metoclopramide hydrochloride hydrate

    CAS:
    <p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>
    Formula:C14H25Cl2N3O3
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:354.27
  • Eltoprazine hydrochloride

    CAS:
    <p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>
    Formula:C12H17ClN2O2
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:256.73
  • Vortioxetine hydrobromide

    CAS:
    <p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>
    Formula:C18H22N2S·HBr
    Purity:98.85% - 99.98%
    Color and Shape:Solid
    Molecular weight:379.36
  • Azaphen dihydrochloride monohydrate

    CAS:
    <p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>
    Formula:C16H23Cl2N5O2
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:388.29
  • RS-67333

    CAS:
    <p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>
    Formula:C19H29ClN2O2
    Purity:99.24%
    Color and Shape:Solid
    Molecular weight:352.9
  • SB 243213

    CAS:
    <p>SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.</p>
    Formula:C22H19F3N4O2
    Purity:98.78% - 99.86%
    Color and Shape:Solid
    Molecular weight:428.41
  • (S)-Mirtazapine

    CAS:
    <p>(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.</p>
    Formula:C17H19N3
    Purity:99.37%
    Color and Shape:Solid
    Molecular weight:265.35
  • Renzapride

    CAS:
    <p>Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.</p>
    Formula:C16H22ClN3O2
    Purity:98.97% - 99.09%
    Color and Shape:Solid
    Molecular weight:323.82
  • Ketanserin tartrate

    CAS:
    <p>Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.</p>
    Formula:C26H28FN3O9
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:545.51
  • Tandospirone

    CAS:
    <p>Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.</p>
    Formula:C21H29N5O2
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:383.49
  • Setiptiline

    CAS:
    <p>Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.</p>
    Formula:C19H19N
    Purity:98.05% - 98.07%
    Color and Shape:Solid
    Molecular weight:261.36
  • Latrepirdine dihydrochloride

    CAS:
    <p>Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.</p>
    Formula:C21H25N3·2HCl
    Purity:98.45%
    Color and Shape:Solid
    Molecular weight:392.37
  • Rizatriptan

    CAS:
    <p>Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.</p>
    Formula:C15H19N5
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:269.35
  • (R)-Mirtazapine

    CAS:
    <p>(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.</p>
    Formula:C17H19N3
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:265.35
  • Rotigotine

    CAS:
    <p>Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.</p>
    Formula:C19H25NOS
    Purity:99.04% - 99.88%
    Color and Shape:Solid
    Molecular weight:315.47
  • LP-533401 hydrochloride

    CAS:
    <p>LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.</p>
    Formula:C27H23ClF4N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:562.94
  • Citalopram

    CAS:
    <p>Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.</p>
    Formula:C20H21FN2O
    Purity:99.78% - 99.89%
    Color and Shape:Solid
    Molecular weight:324.39
  • WAY-100635 maleate

    CAS:
    <p>WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).</p>
    Formula:C25H34N4O2·xC4H4O4
    Purity:>99.99%
    Color and Shape:White Solid
    Molecular weight:538.645
  • Jatrorrhizine chloride

    CAS:
    <p>Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.</p>
    Formula:C20H20ClNO4
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:373.8
  • S1RA

    CAS:
    <p>S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2</p>
    Formula:C20H23N3O2
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:337.42
  • Syk Inhibitor II

    CAS:
    <p>Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).</p>
    Formula:C14H15F3N6O
    Purity:97.63%
    Color and Shape:Solid
    Molecular weight:340.3
  • R 59-022

    CAS:
    <p>R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.</p>
    Formula:C27H26FN3OS
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:459.58
  • Cyproheptadine hydrochloride

    CAS:
    <p>Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.</p>
    Formula:C21H21N·HCl
    Purity:99.88% - 99.97%
    Color and Shape:Solid
    Molecular weight:323.86
  • Risperidone Mesylate

    CAS:
    <p>Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.</p>
    Formula:C24H31FN4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:506.59
  • Escitalopram

    CAS:
    <p>Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.</p>
    Formula:C20H21FN2O
    Purity:99.82%
    Color and Shape:White Or White Crystalline Powder
    Molecular weight:324.39
  • N-Methyl amisulpride

    CAS:
    <p>N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.</p>
    Formula:C18H29N3O4S
    Color and Shape:Solid
    Molecular weight:383.51
  • Keto Ziprasidone

    CAS:
    <p>Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.</p>
    Formula:C21H19ClN4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:426.92
  • Arazasetron HCl

    CAS:
    <p>Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.</p>
    Formula:C17H20ClN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:349.81
  • Brexpiprazole-d8

    CAS:
    <p>Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.</p>
    Formula:C25H27N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.62
  • Amitriptyline-d6 Hydrochloride

    CAS:
    <p>Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.</p>
    Formula:C20H18D6ClN
    Color and Shape:Solid
    Molecular weight:319.90
  • Mirtazapine D3

    CAS:
    <p>Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .</p>
    Formula:C17H19N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:268.37
  • 5-Methyltryptamine hydrochloride

    CAS:
    <p>5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.</p>
    Formula:C11H15ClN2
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:210.703
  • Penbutolol sulfate

    CAS:
    <p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>
    Formula:C18H29NO2H2O4S
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:340.47
  • Ketanserinol

    CAS:
    <p>Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.</p>
    Formula:C22H24FN3O3
    Color and Shape:Solid
    Molecular weight:397.44
  • 7-Desmethyl-3-hydroxyagomelatine

    CAS:
    <p>7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.</p>
    Formula:C14H15NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:245.27
  • Diclofensine

    CAS:
    <p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>
    Formula:C17H17Cl2NO
    Purity:97.01% - 98.13%
    Color and Shape:Solid
    Molecular weight:322.23
  • Hydroxy ziprasidone

    CAS:
    <p>Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.</p>
    Formula:C21H21ClN4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:428.94
  • Pardoprunox

    CAS:
    <p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>
    Formula:C12H15N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:233.27
  • SB 271046 hydrochloride

    CAS:
    <p>SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is &gt; 200-fold selective over 55 other receptors, enzymes and ion channels.</p>
    Formula:C20H22ClN3O3S2·HCl
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:488.45
  • Paroxetine hydrochloride hemihydrate

    CAS:
    <p>Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).</p>
    Formula:C38H44Cl2F2N2O7
    Purity:99.949%
    Color and Shape:Solid
    Molecular weight:749.67
  • Dolasetron Mesylate

    CAS:
    <p>Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following</p>
    Formula:C20H24N2O6S
    Purity:99.05%
    Color and Shape:White Powder
    Molecular weight:420.48
  • LY 344864

    CAS:
    <p>LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.</p>
    Formula:C21H22FN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.42
  • Ampreloxetine

    CAS:
    <p>Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.</p>
    Formula:C18H18F3NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.34
  • 2-Methyl-5-HT maleate

    CAS:
    <p>2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.</p>
    Formula:C15H18N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:306.31
  • Ro 04-6790

    CAS:
    <p>Ro 04-6790 is a 5-HT6 receptor antagonist.</p>
    Formula:C12H16N6O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:308.36
  • ST1936

    CAS:
    <p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>
    Formula:C13H17ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:236.74
  • Org37684

    CAS:
    <p>5-HT2 receptors agonist</p>
    Formula:C14H20ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:269.77
  • Donitriptan

    CAS:
    <p>Donitriptan 是一种 5-HT 受体激动剂,对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。</p>
    Formula:C23H25N5O2
    Purity:98.76%
    Color and Shape:Solid
    Molecular weight:403.48
  • AR-A 2

    CAS:
    <p>AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).</p>
    Formula:C27H36N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.6
  • AVN-322

    CAS:
    <p>AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.</p>
    Formula:C17H20ClN5O2S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:393.89
  • Alniditan dihydrochloride

    CAS:
    <p>Alniditan dihydrochloride is a potent 5-HT1D agonist and migraine-abortive agent.</p>
    Formula:C17H28Cl2N4O
    Color and Shape:Solid
    Molecular weight:375.34
  • Methiothepin maleate

    CAS:
    <p>Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.</p>
    Formula:C24H28N2O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.62
  • RS 56812 hydrochloride

    CAS:
    <p>5-HT3 partial agonist</p>
    Formula:C18H22ClN3O2
    Purity:98.62%
    Color and Shape:Solid
    Molecular weight:347.84
  • AL-37350A

    CAS:
    <p>AL-37350A is a 5-HT2 receptor-selective agonist with ocular hypotensive activity.</p>
    Formula:C14H18N2O
    Color and Shape:Solid
    Molecular weight:230.31
  • CUMI-101

    CAS:
    <p>CUMI-101 is an agonist of 5-HT1A receptor.</p>
    Formula:C19H27N5O3
    Color and Shape:Solid
    Molecular weight:373.45
  • Ifoxetine sulfate

    CAS:
    <p>Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.</p>
    Formula:C13H19NO2H2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:270.34
  • WAY 629 hydrochloride

    CAS:
    <p>5-HT2C agonist</p>
    Formula:C15H19ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:262.78
  • E55888

    CAS:
    <p>E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.</p>
    Formula:C16H23N3
    Color and Shape:Solid
    Molecular weight:257.37
  • Etoperidone hydrochloride

    CAS:
    <p>Etoperidone hydrochloride is an antidepressant agent.</p>
    Formula:C19H29Cl2N5O
    Color and Shape:Solid
    Molecular weight:414.37
  • LEK 8841

    CAS:
    <p>LEK 8841 is an ergoline derivative that is a potential antipsychotic.</p>
    Formula:C21H24BrN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:494.4
  • Clovoxamine

    CAS:
    <p>Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant and anticonvulsant activity.</p>
    Formula:C14H21ClN2O2
    Purity:99.44% - 99.75%
    Color and Shape:Solid
    Molecular weight:284.78
  • Lofepramine hydrochloride

    CAS:
    <p>Lofepramine is a serotonin and norepinephrine reuptake inhibitor. Lofepramine is also a psychotropic IMIPRAMINE derivative.</p>
    Formula:C26H28Cl2N2O
    Purity:98%
    Color and Shape:Off-White Solid
    Molecular weight:455.42
  • Alosetron ((Z)-2-butenedioate)

    CAS:
    <p>Alosetron (GR 68755) (Z)-2-butenedioate is a Serotonin 5HT3-receptor antagonist that is used in the treatment of irritable bowel syndrome.</p>
    Formula:C21H22N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.42
  • 5-Carboxamidotryptamine maleate

    CAS:
    <p>5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.</p>
    Formula:C15H17N3O5
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:319.31
  • SB-221284

    CAS:
    <p>5-HT2C/2B receptor antagonist</p>
    Formula:C16H14F3N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.36
  • PF-3246799

    CAS:
    <p>PF-3246799 is an effective and selective agonist of the 5-HT2C receptor.</p>
    Formula:C15H17N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:239.32
  • SB 272183

    CAS:
    <p>SB 272183 is a highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drug.</p>
    Formula:C29H28ClN5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.02
  • Amitriptylinoxide

    CAS:
    <p>Amitriptylinoxide is an antidepressant.</p>
    Formula:C20H23NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:293.4
  • GW-876167

    CAS:
    <p>GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.</p>
    Formula:C16H21N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.37
  • BGC 20-761

    CAS:
    <p>BGC20-761: selective 5-HT6/Dopamine antagonist; enhances memory, potential antipsychotic. K i - 5-HT6: 20 nM, 5-HT2A: 69 nM, D2: 140 nM.</p>
    Formula:C19H22N2O
    Color and Shape:Solid
    Molecular weight:294.39
  • EMDT

    CAS:
    <p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>
    Formula:C15H22N2O
    Purity:97.66% - 99.78%
    Color and Shape:Solid
    Molecular weight:246.35
  • Captodiame

    CAS:
    <p>Captodiame is an antihistamine agent.</p>
    Formula:C21H29NS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:359.59
  • S(-)-8-Hydroxy-DPAT hydrobromide

    CAS:
    <p>S(-)-8-Hydroxy-DPAT hydrobromide is an agonist of 5-HT1A serotonin receptor.</p>
    Formula:C16H26BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.29
  • SB-737050A

    CAS:
    <p>SB-737050A, a 5-HT antagonist, is used potentially for the treatment of schizophrenia.</p>
    Formula:C22H23ClN2O3S2
    Color and Shape:Solid
    Molecular weight:463.01
  • GSK-215083

    CAS:
    <p>GSK-215083: a PET quinoline-based 5-HT6 antagonist radioligand, binds 5HT6 in striatum and 5HT2A in frontal cortex.</p>
    Formula:C20H20FN3O2S
    Color and Shape:Solid
    Molecular weight:385.46
  • Adatanserin

    CAS:
    <p>Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.</p>
    Formula:C21H31N5O
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:369.5
  • EMD 386088 hydrochloride

    CAS:
    <p>EMD 386088 hydrochloride is a 5-HT6 receptor agonist.</p>
    Formula:C14H16Cl2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.2
  • SB-269970

    CAS:
    <p>SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).</p>
    Formula:C18H28N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.49
  • p-MPPF dihydrochloride

    CAS:
    <p>p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.</p>
    Formula:C25H29Cl2FN4O2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:507.43
  • QF0301B

    CAS:
    <p>QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.</p>
    Formula:C23H28N2O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:364.48
  • (4E)-SUN9221

    CAS:
    <p>(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity in</p>
    Formula:C25H31FN4O3
    Purity:97.79%
    Color and Shape:Solid
    Molecular weight:454.54
  • Mirisetron

    CAS:
    <p>Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.</p>
    Formula:C24H31N3O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:393.52
  • CP-809101

    CAS:
    <p>CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>
    Formula:C15H17ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:304.77
  • Eplivanserin

    CAS:
    <p>Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.</p>
    Formula:C19H21FN2O2
    Purity:97.04%
    Color and Shape:Solid
    Molecular weight:328.38
  • GR 113808

    CAS:
    <p>GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.</p>
    Formula:C19H27N3O4S
    Purity:98.16%
    Color and Shape:Solid
    Molecular weight:393.5
  • AS19

    CAS:
    <p>AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).</p>
    Formula:C18H25N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.41
  • PNU-282987 S enantiomer hydrochloride

    CAS:
    <p>(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.</p>
    Formula:C14H18Cl2N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:301.21
  • L-694,247

    CAS:
    <p>L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.</p>
    Formula:C20H21N5O3S
    Purity:98.36%
    Color and Shape:White Solid
    Molecular weight:411.48
  • 5-HT7 agonist 1

    CAS:
    <p>5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).</p>
    Formula:C19H20ClN3
    Purity:98.61%
    Color and Shape:Solid
    Molecular weight:325.84
  • Ziprasidone mesylate trihydrate

    CAS:
    <p>Ziprasidone mesylate hydrate is an oral 5-HT/D2 antagonist with Ki: D2=4.8nM, 5-HT2A=0.42nM, 5-HT1A=3.4nM in rats.</p>
    Formula:C22H31ClN4O7S2
    Color and Shape:Solid
    Molecular weight:563.08
  • Way 100289

    CAS:
    <p>Way 100289 is a selective 5-HT3 receptor antagonist.</p>
    Formula:C20H27N3O3
    Color and Shape:Solid
    Molecular weight:357.45
  • Cinitapride Hydrogen Tartrate

    CAS:
    <p>Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptors</p>
    Formula:C25H36N4O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:552.581
  • Zimelidine dihydrochloride

    CAS:
    <p>5-HT re-uptake inhibitor</p>
    Formula:C16H18BrClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.69
  • CP94253 hydrochloride

    CAS:
    <p>CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).</p>
    Formula:C15H20ClN3O
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:293.79
  • 5-HT6/5-HT2A receptor ligand-1

    CAS:
    <p>Compound 33 is a dual 5-HT6/5-HT2A antagonist with Ki values of 2 nM and 11 nM, respectively, useful in neuro/psychiatric research.</p>
    Formula:C21H19FN2O2
    Color and Shape:Solid
    Molecular weight:350.39
  • (Rac)-WAY-161503

    CAS:
    <p>(Rac)-WAY-161503 is a selective and high-affinity agonist of the 5-HT2C receptor (Ki: 4 nM; EC50: 12 nM), with anti-obesity and antidepressant effects.</p>
    Formula:C11H11Cl2N3O
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:272.13
  • Irindalone

    CAS:
    <p>IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.</p>
    Formula:C24H29FN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.51
  • Blonanserin HCl

    CAS:
    <p>Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.</p>
    Formula:C23H32Cl2FN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.42
  • Usmarapride free base

    CAS:
    <p>Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.</p>
    Formula:C21H29N5O2
    Purity:99.91% - 99.91%
    Color and Shape:Solid
    Molecular weight:383.49
  • Pruvanserin hydrochloride

    CAS:
    <p>Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.</p>
    Formula:C22H22ClFN4O
    Purity:99.6%
    Color and Shape:Solid
    Molecular weight:412.89
  • PNU-142633

    CAS:
    <p>PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; &gt;18,000 nM for 5-HT1B.</p>
    Formula:C24H30N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:422.52
  • RS 64459-193

    CAS:
    <p>RS 64459-193 has a high affinity for the 5-HT1A binding site.</p>
    Formula:C26H36Cl2N2O2
    Color and Shape:Solid
    Molecular weight:479.48
  • MHP 133

    CAS:
    <p>MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).</p>
    Formula:C17H20ClN5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.83
  • Repinotan HCl

    CAS:
    <p>Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.</p>
    Formula:C21H25ClN2O4S
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:436.95
  • Iloperidone hydrochloride

    CAS:
    <p>Iloperidone hydrochloride is a D(2)/5-HT(2) receptor antagonist. It is also an atypical antipsychotic for the treatment of schizophrenia symptoms.</p>
    Formula:C24H28ClFN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:462.95
  • TMPPAA

    CAS:
    <p>TMPPAA is an allosteric agonist of 5-HT3 receptor.</p>
    Formula:C15H21NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:247.33
  • Bifeprunox

    CAS:
    <p>Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.</p>
    Formula:C24H23N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.46
  • CJ 033466

    CAS:
    <p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>
    Formula:C19H28ClN5O
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:377.91
  • Isamoltane hemifumarate

    CAS:
    <p>5-HT1B antagonist</p>
    Formula:C16H22N202C4H404
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.4