GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(54 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
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Found 5981 products of "GPCR/G-Protein"
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GLP-1R agonist 15
CAS:GLP-1R agonist 15 (Compound 101) is a GLP-1 receptor agonist [1] .Formula:C46H47FN8O7SColor and Shape:SolidMolecular weight:874.98Glucagon-like peptide 1 (1-37), human TFA
Human Glucagon-like peptide 1 (1-37) TFA is a potent GLP-1 receptor agonist derived from proglucagon.Formula:C188H276N51F3O61Purity:98%Color and Shape:SolidMolecular weight:4283.5Neuromedin N
CAS:Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.Formula:C38H63N7O8Purity:98%Color and Shape:SolidMolecular weight:745.95(±)14(15)-EpETE
CAS:(±)14(15)-EpETE is an intestinal microbial lipid metabolite that attenuates cisplatin chemotherapy-induced nausea in rats by inhibiting Substance P release.Formula:C20H30O3Color and Shape:SolidMolecular weight:318.45CCR2 antagonist 1
CAS:CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM).Formula:C28H32BrF3N2OColor and Shape:SolidMolecular weight:549.47CCR8 antagonist 1
CAS:CCR8 antagonist 1 is an antagonist of C-C Motif Chemokine Receptor 8 (CCR8) with a Ki value of 1.6 nM.Formula:C26H29N3O5SPurity:99.51%Color and Shape:SolidMolecular weight:495.59Tamsolusin Hydrochloride
CAS:Tamsolusin Hydrochloride (YM 12617) is a highly selective alpha-1A adrenergic receptor antagonist used in the treatment of benign prostatic hypertrophy.Formula:C20H29ClN2O5SPurity:99.92%Color and Shape:SoildMolecular weight:444.97P2Y12R ligand-1
P2Y12R ligand-1 (Compound 41) is a high-affinity P2Y12 receptor ligand with a Ki of 17.1 nM. The [18F]-labeled version of P2Y12R ligand-1 is suitable for research involving brain PET imaging.Color and Shape:Odour SolidHemopressin(rat)
CAS:Peptide inhibitor for ep24.15, neurolysin & ACE with Ki 27.76, 3.43, 1.87 μM. Lowers blood pressure, modulates CB1 receptor, reduces pain & food intake.Formula:C53H77N13O12Purity:98%Color and Shape:SolidMolecular weight:1088.27Alkyne-βAG-TOCA
Alkyne-βAG-TOCA is an octreotide derivative that targets somatostatin receptor subtype 2 (SST2). It is utilized in the synthesis and research of radioconjugates (RDC).Formula:C48H65N11O15S2Color and Shape:SolidMolecular weight:1100.22Cetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Formula:C21H27Cl3N2O3Color and Shape:SolidMolecular weight:461.81[Lys8] Vasopressin Desglycinamide
CAS:[Lys8] Vasopressin Desglycinamide, a vasopressin analog, supports the maintenance of active and passive avoidance behavior and aids in the facilitation ofFormula:C44H63N11O12S2Color and Shape:SolidMolecular weight:1002.17Galanin (1-29)(rat, mouse)
CAS:Non-selective galanin agonist; Ki: GAL1-0.98, GAL2-1.48, GAL3-1.47 nM. Anticonvulsant, stops full seizures in rats.Formula:C141H211N43O41Purity:98%Color and Shape:White Lyophilized PowderMolecular weight:3164.499FR252384
CAS:FR252384 is an antagonist of the neuropeptide Y-Y5 receptor (IC50: 2.3 nM).Formula:C18H17N3Purity:98%Color and Shape:SolidMolecular weight:275.35GR231118 TFA
GR231118 TFA: potent Y1 antagonist (pKi 10.4), Y4 agonist (pEC50 8.6, pKi 9.6), weak Y2/Y5 agonist, high affinity for mouse Y6 (pKi 8.8).Formula:C112H171F3N34O26Molecular weight:2466.76α-helical CRF 9-41 acetate
<p>α-helical CRF 9-41 acetate is a competitive antagonist of CRF2 (KB = 100 nM) and a partial agonist of CRF1 (EC50 = 140 nM).</p>Purity:96.60%Color and Shape:SolidMolecular weight:#N/ARef: TM-TP2048L
1mg208.00€5mg500.00€10mg672.00€25mg1,017.00€50mg1,359.00€100mg1,853.00€200mg2,498.00€17-phenyl trinor Prostaglandin F2α methyl amide
CAS:17-phenyl trinor Prostaglandin F2α (17-phenyl trinor PGF2α) is a metabolically stable analog of PGF2α and is a potent agonist for the FP receptor, binding withFormula:C24H35NO4Color and Shape:SolidMolecular weight:401.547Xenin-8 TFA
Xenin-8 TFA, a C-terminal octapeptide derived from the 25-amino acid peptide Xenin belonging to the neurotensin/xenopsin family, is biologically active.T-kinin
CAS:T-kinin (Ile-Ser-bradykinin) is a bradykinin-containing peptide utilized in inflammation research [1] [2].Formula:C59H89N17O14Molecular weight:1260.443D-Monophosphoryl Lipid A-5 triethylamine
3D-Monophosphoryl Lipid A-5 (3D-MPLA-5) triethylamine is a TLR agonist that acts as an adjuvant for vaccines, enhancing their immunogenicity.Formula:C88H170N3O20PMolecular weight:1621.27Brain Natriuretic Peptide-45, mouse
CAS:Mouse BNP-45, a heart-derived peptide, lowers blood pressure and increases sodium excretion.(Iso)-Samixogrel
CAS:(Iso)-Samixogrel shows activity against Carbonic anhydrase and Cyclooxygenase 2.Formula:C25H25ClN2O4SPurity:98.85%Color and Shape:SolidMolecular weight:484.99Benzquinamide
CAS:<p>Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer</p>Formula:C22H32N2O5Purity:94.86%Color and Shape:SolidMolecular weight:404.5Urocortin II, human TFA
hUcn II, a CRF family member, targets CRF2 receptor, has time-linked stress regulation effects, showing mild motor suppression and delayed anxiolytic action.Formula:C196H340F3N63O56SPurity:98%Color and Shape:SolidMolecular weight:4564.3Gastrin-Releasing Peptide, human
CAS:Gastrin-releasing peptide, released by vagal fibers, stimulates stomach G cells to secrete gastrin, affecting acid secretion and gut motility.Formula:C130H204N38O31S2Purity:98%Color and Shape:SolidMolecular weight:2859.38L-770644
CAS:L-770644 is an agonist of B3 adrenergic receptor.Formula:C30H37N7O4SColor and Shape:SolidMolecular weight:591.72pCPA methyl ester hydrochloride
CAS:<p>pCPA methyl ester HCl inhibits tryptophan hydroxylase, 5-HT synthesis, crosses blood-brain barrier, lowers central 5-HT.</p>Formula:C10H13Cl2NO2Purity:99.73% - 99.88%Color and Shape:SolidMolecular weight:250.12Sphinganine 1-phosphate
CAS:Sphinganine 1-phosphate has protects kidney and liver through activation of the S1P1 receptor in mice and acts as an agonist for S1P4 in Homo sapien.Formula:C18H40NO5PColor and Shape:SolidMolecular weight:381.49ACTH (1-14) (TFA)
ACTH (1-14) (TFA) is a regulatory fragment of adrenocorticotropin, specifically involved in the control of cortisol and androgen synthesis [1].Formula:C79H110F3N21O22SMolecular weight:1794.9Adrenocorticotropic Hormone (ACTH) (1-10), human
CAS:ACTH (1-10), human: a weak α-MSH mimic at high doses (100-1000 nM), derived from adrenocorticotropin.Formula:C59H78N16O16SPurity:98%Color and Shape:SolidMolecular weight:1299.41Pasireotide (diaspartate)
CAS:Pasireotide diaspartate (SOM230) has high agonist activity at sst1/2/3/5, less at sst4; it's antiproliferative and proapoptotic.Formula:C66H80N12O17Color and Shape:SolidMolecular weight:1313.41Substance P(1-7)
CAS:Substance P(1-7) is a bioactive metabolite of tachykinin SP with anti-inflammatory and analgesic properties.Formula:C41H65N13O10Purity:98%Color and Shape:SolidMolecular weight:900.04Idazoxan
CAS:Idazoxan is an alpha2 receptor antagonist that also exhibits activity at imidazoline [I1] and [I2] receptors, playing a role in modulating dopamine release.Formula:C11H12N2O2Molecular weight:204.23ACTH (1-17)
CAS:ACTH (1-17), a potent MC1 receptor agonist with a Ki of 0.21 nM, is a variant of corticotropin from the pituitary gland.Formula:C95H145N29O23SPurity:98%Color and Shape:SolidMolecular weight:2093.41Neuropeptide Y (22-36)
CAS:Neuropeptide Y (22-36) is a 15-amino acid fragment of NPY, which is abundant in the mammalian brain and involved in multiple physiological functions.Formula:C85H139N29O21Purity:98%Color and Shape:SolidMolecular weight:1903.19Atriopeptin III (rat)
CAS:Atriopeptin III (rat) (ANP 127-150), a 24-amino acid atrial peptide, functions as a powerful vasodilator and natriuretic/diuretic agent, enhancing renalFormula:C107H165N35O34S2Molecular weight:2549.8Ro 23-7014
CAS:Ro 23-7014, a new thiazepinone Ca2+ channel antagonist, has high affinity for peripheral (Type A) receptors.Formula:C48H63N9O16S4Purity:98%Color and Shape:SolidMolecular weight:1150.32[18F]-Labeled L-dopa precursor
CAS:[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].Formula:C35H36N2O7Color and Shape:SolidMolecular weight:596.67MRS 2957 triethylammonium salt
CAS:MRS 2957 triethylammonium salt is a P2Y6 agonist.Formula:C19H28N5O20P3Purity:98%Color and Shape:SolidMolecular weight:739.37Prostaglandin E2 isopropyl ester
CAS:PGE2 isopropyl ester, a lipophilic prodrug of PGE2, gains solubility in lipids and activates upon in vivo hydrolysis.Formula:C23H38O5Color and Shape:SolidMolecular weight:394.552Olanzapine Lactam Impurity
CAS:Olanzapine lactam impurity, found in olanzapine, forms under heat or oxidative stress.Formula:C17H20N4O2Color and Shape:SolidMolecular weight:312.3735-trans Latanoprost
CAS:Latanoprost, an F-series prostaglandin analog for ocular hypertension, has a 5-trans isomer used as an analytical standard.Formula:C26H40O5Color and Shape:SolidMolecular weight:432.601Motilin, canine
CAS:Motilin canine, a 22-amino acid peptide, functions as a robust gastrointestinal smooth muscle contraction agonist.Formula:C120H194N36O34Purity:98%Color and Shape:SolidMolecular weight:2685.05Methylsolfonyl 25(S)-Δ7-dafachronic acid
Methylsulfonyl 25(S)-Δ7-dafachronic acid (compound 3) is a selective ssDAF-12 agonist with an IC50 value of 0.41 μM. It exhibits low cytotoxicity in HepG2 cells, with an IC50 value greater than 200 μM. Methylsulfonyl 25(S)-Δ7-dafachronic acid is applicable in the study of parasitic diseases.Formula:C28H45NO4SMolecular weight:491.30693Tocrifluor T1117
CAS:Fluorescent form of AM 251, CB1 receptor antagonistFormula:C56H53Cl2N7O5Purity:98%Color and Shape:SolidMolecular weight:974.97N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formula:C19H22N6O4Color and Shape:SolidMolecular weight:398.42Uperolein
CAS:Uperolein, a physalaemin-like endecapeptide derived from the skin of Uperoleia rugosa and Uperoleia marmorata, exhibits spasmodic activity on theFormula:C57H79N13O16SMolecular weight:1234.38GIP/GLP-1 dual receptor agonist-1
CAS:Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.Color and Shape:SolidMK-0493 HCl
CAS:MK-0493 is a novel, potent, and selective agonist for melanocortin receptor 4 (MC4R).Formula:C30H39Cl2F2N3O2Color and Shape:SolidMolecular weight:582.55ANP (1-30), frog
CAS:ANP (1-30), frog, a peptide fragment sourced from atrial natriuretic peptide of frog origin, exhibits natriuretic, diuretic, and vasorelaxant properties.Formula:C131H217N49O41S4Molecular weight:3262.69LCKLSL
CAS:LCKLSL, an N-terminal hexapeptide, inhibits AnxA2 and tPA binding, reduces plasmin, and exhibits anti-angiogenic effects.Formula:C30H57N7O8SMolecular weight:675.89Anaritide
CAS:Anaritide, a synthetic form of atrial natriuretic peptide (ANP) composed of 25 amino acids, enhances the glomerular filtration rate by dilating afferent arterioles and constricting efferent arterioles. It is utilized for studying its effects on patients with acute tubular necrosis, with a focus on improving dialysis-free survival rates.Formula:C112H175N39O35S3Molecular weight:2724.02Prolactin-Releasing Peptide (1-31), bovine
Prolactin-Releasing Peptide (1-31), bovine, is a fragment of prolactin-releasing peptide (PrRP).Formula:C44H80N14O15Molecular weight:1044.59276Oxopurpureine
CAS:Oxopurpureine, classified as an oxoaporphine compound, functions to inhibit plant pathogens.Formula:C21H19NO6Molecular weight:381.38CCK (27-33) (non-sulfated)
CAS:CCK (27-33), a non-sulfated peptide, inhibits [3H]naloxone binding (IC50=4uM) and guinea pig ileum contractions (IC50=17uM), reversed by naloxone.Formula:C45H57N9O10S2Molecular weight:948.12(Leu31,Pro34)-Peptide YY (human)
CAS:(Leu31,Pro34)-Peptide YY (human) is a derivative of Peptide YY, acting as a potent and selective Y1 receptor agonist with a dissociation constant (KD) of 1.0 nMFormula:C195H296N54O56Molecular weight:4292.75Tiaspirone hydrochloride
CAS:Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity and influences the electrophysiological activity of dopaminergic neurons.Formula:C24H33ClN4O2SPurity:99.87%Color and Shape:SoildMolecular weight:477.06[D-Phe2,6, Pro3]-LH-RH
CAS:[D-Phe2,6, Pro3]-LH-RH is a potent antagonist of luteinizing hormone-releasing hormone (LHRH).Formula:C59H80N14O13Molecular weight:1193.35Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27)
CAS:Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP(1-7)-GRF(8-27) is a selective antagonist [1] for the vasoactive intestinal peptide 1 (VIP 1) receptor.Formula:C150H246N44O38Molecular weight:3273.8315(S)-Latanoprost
CAS:15(S)-Latanoprost, a latanoprost analog with inverted hydroxyl at C-15, has an IC50 of 24 nM and reduces IOP by 1 mmHg at 3 μg.Formula:C26H40O5Color and Shape:SolidMolecular weight:432.59Contulakin G
CAS:Contulakin G: O-glycosylated neurotensin, weak neurotensin receptor agonist, strong antinociceptive.Formula:C88H140N20O37Molecular weight:2070.17Lamprey LH-RH I
CAS:Lamprey LH-RH I triggers ovulation and raises steroid levels in lamprey, inactive in other species.Formula:C58H79N15O15Molecular weight:1226.34(D-His(Bzl)6)-LHRH (1-7) (free acid)
CAS:(D-His(Bzl)6)-LHRH (1-7) free acid is a synthetic peptide derived from luteinizing hormone-releasing hormone (LHRH). It achieves enhanced stability and biological activity through the introduction of non-natural amino acid residues at specific positions within the LHRH molecule. This modification extends the drug's half-life in the body, reduces its rate of rapid metabolism and clearance, and subsequently increases its efficacy in inhibiting cell proliferation.Formula:C53H62N12O11Molecular weight:1043.13O-Desmethyl-N-deschlorobenzoyl Indomethacin
CAS:O-Desmethyl-N-deschlorobenzoyl indomethacin, a metabolite of indomethacin, reduces HL-60 cell viability and aids in synthesizing PGD2 receptor antagonists.Formula:C11H11NO3Color and Shape:SolidMolecular weight:205.213[D-p-Cl-Phe6,Leu17]-VIP
CAS:Selective vasoactive intestinal peptide (VIP) receptor antagonist (IC50 = 125.8 nM). Displays no activity on glucagon, secretin or GRF receptors.Formula:C148H239ClN44O42Purity:98%Color and Shape:SolidMolecular weight:3342.24Metaterol
CAS:Metaterol is a bioactive chemical.Formula:C11H17NO2Color and Shape:SolidMolecular weight:195.2582N-0500 HCl
CAS:N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.Formula:C15H22ClNO2Purity:98.85% - 99.54%Color and Shape:SolidMolecular weight:283.79CB2R/FAAH modulator-3
CAS:CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.Formula:C22H31NO2Purity:99.81%Color and Shape:SoildMolecular weight:341.49Secretin, canine TFA
Secretin, canine TFA, is an endocrine hormone that stimulates the secretion of pancreatic fluid rich in bicarbonate. Additionally, Secretin, canine TFA, can regulate the primary cell functions and paracellular permeability of gastric monolayer cells through an Src kinase-dependent pathway.Color and Shape:Odour SolidVVZ-149
VVZ-149 is an antagonist of both serotonin receptor 2A (5HT2A) and glycine transporter type 2 (GlyT2), with potential anti-nociceptive activity.Color and Shape:SolidSB236057
CAS:SB236057: potent selective inverse agonist at 5-HT autoreceptors; increases brain 5-HT; teratogen causing musculoskeletal defects in rodents.Formula:C33H34N4O3Purity:98%Color and Shape:SolidMolecular weight:534.65Neuromedin S (human)
CAS:Neuromedin S (human) is a 33-amino acid neuropeptide identified as an endogenous ligand for the orphan G-protein coupled receptor (GPCR) FM-4/TGR-1, acting onN-desmethyl Zolmitriptan
CAS:DZT, an active metabolite of zolmitriptan, agonizes 5-HT1B/D receptors; contracts human cerebral arteries (EC50=100nM).Formula:C15H19N3O2Color and Shape:SolidMolecular weight:273.33Norisoboldine hydrochloride
CAS:<p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>Formula:C18H20ClNO4Color and Shape:SolidMolecular weight:349.812,3-dinor Thromboxane B1
CAS:TXB2 released from platelets becomes 11-dehydro and 2,3-dinor TXB2. Rats excrete 2,3-dinor TXB1, a reliable thromboxane biosynthesis marker.Formula:C18H32O6Color and Shape:SolidMolecular weight:344.448SR 142948 TFA
SR 142948 TFA is an orally active, selective non-peptide neurotensin receptor (NT) antagonist, displaying IC50 values of 1.19 nM in h-NTR1-CHO cells, 0.32 nM in HT-29 cells, and 3.96 nM in adult rat brain. In HT-29 cells, it counteracts NT-induced inositol monophosphate formation with an IC50 of 3.9 nM. It blocks NT-induced hypothermia, analgesia, and turning behavior in vivo and can cross the blood-brain barrier, making it useful for research in psychiatric disorders.Color and Shape:Odour SolidRhazimine
CAS:Rhazimine is an indole alkaloid. It is a dual inhibitor of arachidonic acid metabolism and platelet activating factor-induced platelet aggregation.Formula:C21H22N2O3Color and Shape:SolidMolecular weight:350.418ZM 253270
CAS:ZM 253270 is an nonpeptide neurokinin A antagonist.Formula:C22H26ClN7O3Purity:98%Color and Shape:SolidMolecular weight:471.95S33084
CAS:S33084 is a potent, selective and competitive antagonist of dopamine D(3)-receptors.Formula:C29H29N3O2Purity:98%Color and Shape:SolidMolecular weight:451.56HGS101
HGS101 is a fully humanized CCR5 monoclonal antibody that exhibits high affinity for CCR5. It binds to the second extracellular loop (ECL-2) and functions as a signaling antagonist. HGS101 restores the inhibitory effect of Maraviroc in Maraviroc-resistant HIV-1 infected PBMCs. In an uninfected simian immunodeficiency virus model of rhesus monkeys, HGS101 shows anti-HIV activity by inhibiting CCR5 signaling.Color and Shape:Odour LiquidLP-20
CAS:LP-20 is a bioactive chemical.Formula:C17H20N2OColor and Shape:SolidMolecular weight:268.35Prostaglandin F2α methyl ester
CAS:Prostaglandin F2α methyl ester is a highly lipid-soluble PGF2α analog used to maintain low intraocular pressure.Formula:C21H36O5Color and Shape:SolidMolecular weight:368.51Cannabinol methyl ether
CAS:Cannabinol methyl ether, a phytocannabinoid, serves as an analytical reference standard. This compound can be obtained through isolation from Cannabis plants, derived from cannabinol, or synthesized. The physiological and toxicological properties of cannabinol methyl ether remain unknown. It is designed exclusively for research and forensic applications.Formula:C22H28O2Color and Shape:SolidMolecular weight:324.5Methimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Formula:C10H19Br2N3Color and Shape:SolidMolecular weight:341.091Cetirizine Impurity C
CAS:Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.Formula:C21H25ClN2O3Color and Shape:SolidMolecular weight:388.89Oxyntomodulin
CAS:GLP-1 analog modulates appetite, boosts metabolism, and curbs gastric acid. Increases cAMP, mildly stimulates glucagon receptor.Formula:C192H295N59O60SPurity:98%Color and Shape:SolidMolecular weight:4421.86Prolactin Releasing Peptide (1-31), human acetate
Prolactin Releasing Peptide (1-31), human (acetate), is a potent GPR10 ligand with high affinity, eliciting prolactin secretion.Formula:C162H26N56O44SMolecular weight:3724.17GLP-1(7-37)
CAS:GLP-1 (7-37) is a truncated, bioactive form of GLP-1 that is the product of proglucagon processing in intestinal endocrine L cells.Formula:C151H228N40O47Purity:98%Color and Shape:SolidMolecular weight:3355.67(S)-Osanetant
CAS:(S)-Osanetant, an S-enantiomer, is a selective NK3 antagonist with potential for treating schizophrenia and has anxiolytic and antidepressant effects.Formula:C35H41Cl2N3O2Color and Shape:SolidMolecular weight:606.62L-703606 oxalate hydrate
L-703606 oxalate hydrate is an effective, selective NK1 receptor antagonist. It is utilized in research related to gastric acid secretion.Prostaglandin F2α 1,11-lactone
CAS:Prostaglandin F2α 1,11-lactone (PGF2α 1,11-lactone) is a lipid-soluble prodrug of Prostaglandin F2α and can be used in studies about treating glaucoma.Formula:C20H32O4Purity:98%Color and Shape:SolidMolecular weight:336.47Zovaglutide
CAS:Zovaglutide is a GLP-1 receptor agonist that is utilized in diabetes research.Color and Shape:Solid[Des-His1,Glu9]-Glucagon amide
CAS:Glucagon blocker with pA2 of 7.2; no agonist effect. Boosts insulin; prevents glucagon-driven hyperglycemia in rabbits and diabetic rats.Formula:C148H221N41O47SPurity:98%Color and Shape:SolidMolecular weight:3358.68ARC 239 dihydrochloride
CAS:ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).Formula:C24H31Cl2N3O3Purity:99.72%Color and Shape:SolidMolecular weight:480.43Rp-dUTPαS tetrasodium
Rp-dUTPαS (tetrasodium) is an isomer of the sulfur-containing nucleotide dUTP-α-S and acts as an agonist of the purinergic P2Y2 receptor. It selectively induces the accumulation of inositol phosphates in P2Y2-expressing 1321N1 cells with an EC50 of 12.5 μM.Color and Shape:Odour SolidAM-0466
CAS:AM-0466 has a wide range of applications in life science related research.Formula:C27H19F3N4O4SColor and Shape:SolidMolecular weight:552.52Human follicular gonadotropin releasing peptide
CAS:Human Follicular Gonadotropin Releasing Peptide (hF-GRP) is a hormonal peptide that, in vitro, can induce the secretion of pituitary luteinizing hormone (LH)Formula:C68H94N22O27Molecular weight:1651.61Cannabigerorcinic Acid
CAS:Cannabigerorcinic acid, structurally akin to recognized phytocannabinoids, serves as an analytical reference standard designed for research and forensic purposes.Formula:C18H24O4Color and Shape:SolidMolecular weight:304.386Syk Inhibitor II hydrochloride
CAS:<p>Syk signaling is key in lupus. Syk inhibitors reduce inflammation and sepsis severity in FcgRIIb-/- mice, lowering cytokines and organ damage.</p>Formula:C14H16ClF3N6OPurity:99.05%Color and Shape:SolidMolecular weight:376.77NK3R-IN-2
NK3R-IN-2 is an orally active NK3R inhibitor with an IC50 of 330.50 nM against human NK3R. It can penetrate the blood-brain barrier and exhibits excellent NK3R binding affinity in CHO-K1 cells (IC50= 87.31 nM). NK3R-IN-2 effectively suppresses luteinizing hormone (LH) levels and is applicable for research on hormone-related diseases.Color and Shape:Odour Solid
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