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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • Amylin (8-37), rat
    Targetmol
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    Amylin (8-37), rat

    CAS:
    <p>Amylin (8-37), rat, an analog of IAPP, blocks insulin's effects on muscle glucose uptake and glycogen storage.</p>
    Formula:C140H227N43O43
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3200.61

    Ref: TM-TP1233

  • Thromboxane B1
    Targetmol
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    Thromboxane B1

    CAS:
    <p>Thromboxane B1 (TXB1) is a lipid eicosanoid, part of the TXB family, involved in blood clotting.</p>
    Formula:C20H36O6
    Color and Shape:Solid
    Molecular weight:372.5

    Ref: TM-T73855

  • NESS 0327
    Targetmol
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    NESS 0327

    CAS:
    <p>NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.</p>
    Formula:C24H23Cl3N4O
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:489.82

    Ref: TM-T22114

  • Protease-Activated Receptor-1 antagonist 2
    Targetmol
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    Protease-Activated Receptor-1 antagonist 2

    CAS:
    <p>Orally active PAR-1 antagonist with 7 nM IC50; potential for CVD research.</p>
    Formula:C24H23F2N3O2
    Color and Shape:Solid
    Molecular weight:423.46

    Ref: TM-T74266

  • Agaridoxin
    Targetmol
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    Agaridoxin

    CAS:
    <p>Agaridoxin is a mushroom metabolite.</p>
    Formula:C11H14N2O5
    Color and Shape:Solid
    Molecular weight:254.242

    Ref: TM-T29709

  • Xaliproden
    Targetmol
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    Xaliproden

    CAS:
    Xaliproden is a biochemical.
    Formula:C24H22F3N
    Color and Shape:Solid
    Molecular weight:381.43

    Ref: TM-T35152

  • [Leu31,Pro34]-Neuropeptide Y(human,rat)
    Targetmol
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    [Leu31,Pro34]-Neuropeptide Y(human,rat)

    CAS:
    <p>High affinity neuropeptide Y Y1 receptor agonist (Ki = 0.39 nM). Also shows affinity for Y4 and Y5 receptors.</p>
    Formula:C189H284N54O56S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4241

    Ref: TM-TP1985

  • LY83583
    Targetmol
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    LY83583

    CAS:
    <p>LY83583 is a soluble guanylate cyclase competitive inhibitor with IC50 of 2 µM.</p>
    Formula:C15H10N2O2
    Purity:99.54% - 99.80%
    Color and Shape:Solid
    Molecular weight:250.25

    Ref: TM-T21576

  • CymitQuimica logo
    Targetmol
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    Anti-TSHR Antibody (M22)

    <p>Anti-TSHR Antibody (M22) is a humanized IgG1 monoclonal antibody targeting the thyroid-stimulating hormone receptor (TSHR). This antibody is capable of inhibiting the interaction between TSH and TSHR.</p>
    Color and Shape:Odour Liquid

    Ref: TM-T9901A-942

  • Fabesetron
    Targetmol
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    Fabesetron

    CAS:
    <p>Fabesetron (FK1052): oral dual antagonist for 5-HT3/5-HT4 receptors. Aids in managing acute and delayed chemo-induced emesis.</p>
    Formula:C18H19N3O
    Color and Shape:Solid
    Molecular weight:293.37

    Ref: TM-T38692

  • Dipivefrin
    Targetmol
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    Dipivefrin

    CAS:
    <p>Dipivefrin is a prodrug of epinephrine, and is used to treat open-angle glaucoma.</p>
    Formula:C19H29NO5
    Color and Shape:Solid
    Molecular weight:351.44

    Ref: TM-T0103L

  • Pellotine
    Targetmol
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    Pellotine

    CAS:
    <p>Pellotine is an alkaloid isolated from Lophophora. It acts as an inverse agonist of the 5-HT7 receptor (5-HT7 receptor), with an EC50 of 291 nM. Pellotine shows strong affinity for the 5-HT1DR and 5-HT6R, with Ki values of 117 nM and 170 nM, respectively. Additionally, Pellotine reduces intracellular cAMP levels, thereby decreasing neuronal excitability and neurotransmitter release.</p>
    Formula:C13H19NO3
    Color and Shape:Solid
    Molecular weight:237.295

    Ref: TM-TN9164

  • 5-MeO-pyr-T
    Targetmol
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    5-MeO-pyr-T

    CAS:
    <p>5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.</p>
    Formula:C15H20N2O
    Color and Shape:Solid
    Molecular weight:244.33

    Ref: TM-T203568

  • Enuvaptan
    Targetmol
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    Enuvaptan

    CAS:
    <p>Enuvaptan is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.</p>
    Formula:C21H15ClF6N8O3
    Color and Shape:Solid
    Molecular weight:576.84

    Ref: TM-T39611

  • CymitQuimica logo
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    (R)-Zevaquenabant

    <p>(R)-Zevaquenabant ((R)-MRI-1867) is the enantiomer of Zevaquenabant. Zevaquenabant ((S)-MRI-1867) is a peripherally restricted, orally bioavailable dual antagonist of the cannabinoid CB1 receptor and inducible nitric oxide synthase (iNOS). It is beneficial in improving chronic kidney disease (CKD) caused by obesity.</p>
    Color and Shape:Odour Solid

    Ref: TM-TYD-02102

  • Guanylin(human)
    Targetmol
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    Guanylin(human)

    CAS:
    Peptide that activates gut guanylyl cyclase, secreted by GI mucosa, regulates water and electrolytes in gut and kidneys.
    Formula:C58H87N15O21S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1458.65

    Ref: TM-TP2034

  • Mabuterol free base
    Targetmol
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    Mabuterol free base

    CAS:
    <p>Mabuterol: selective β2 agonist, inhibits isoprenaline, affects rat uterus and rabbit jejunum, alters intestinal propulsion.</p>
    Formula:C13H18ClF3N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:310.74

    Ref: TM-T27970

  • Bromchlorbuterol hydrochloride
    Targetmol
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    Bromchlorbuterol hydrochloride

    CAS:
    <p>Bromchlorbuterol HCl, a potent β-agonist, is used to study lung diseases like asthma.</p>
    Formula:C12H19BrCl2N2O
    Color and Shape:Solid
    Molecular weight:358.1

    Ref: TM-T40896

  • TRV045
    Targetmol
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    TRV045

    CAS:
    <p>TRV045 is a selective agonist of the sphingosine-1-phosphate (S1P) subtype 1 receptor and does not impact lymphocyte trafficking. It possesses antiepileptic properties.</p>
    Formula:C18H18N4O3
    Color and Shape:Solid
    Molecular weight:338.36

    Ref: TM-T203071

  • ABT 724 trihydrochloride
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    ABT 724 trihydrochloride

    CAS:
    <p>ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.</p>
    Formula:C17H22Cl3N5
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:402.75

    Ref: TM-T22019

  • GR231118
    Targetmol
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    GR231118

    CAS:
    <p>Potent NPY Y1 antagonist &amp; Y4 agonist; inhibits rat appetite; binds to NPFF receptors (Ki: 43-73 nM).</p>
    Formula:C110H170N34O24
    Purity:98%
    Color and Shape:Lyophilized Powder
    Molecular weight:2352.77

    Ref: TM-TP2022

  • Sauvagine
    Targetmol
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    Sauvagine

    CAS:
    CRF receptor agonist; Ki: 9.4 nM (hCRF-R1), 9.9 nM (rCRF-R2a), 3.8 nM (mCRF-R2b) for 125I-[D-Tyr1]astressin binding inhibition.
    Formula:C202H346N56O63S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4599.35

    Ref: TM-TP2121

  • Mosliciguat
    Targetmol
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    Mosliciguat

    CAS:
    <p>Mosliciguat is a guanylate cyclase activator.</p>
    Formula:C41H36ClF3N2O5
    Color and Shape:Solid
    Molecular weight:729.19

    Ref: TM-T39723

  • (Rac)-Norcisapride
    Targetmol
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    (Rac)-Norcisapride

    CAS:
    <p>Norcisapride, a 5-HT3 and 5-HT4 agonist, treats GI, orofacial, and ENT disorders.</p>
    Formula:C14H20ClN3O3
    Purity:99.32%
    Color and Shape:Soild
    Molecular weight:313.78

    Ref: TM-T68116L

  • Bradykinin (1-7)
    Targetmol
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    Bradykinin (1-7)

    CAS:
    <p>Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.</p>
    Formula:C35H52N10O9
    Purity:98%
    Color and Shape:White Lyophilized Powder
    Molecular weight:756.85

    Ref: TM-TP1210

  • Lys-Bradykinin
    Targetmol
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    Lys-Bradykinin

    CAS:
    <p>Endogenous bradykinin receptor agonist</p>
    Formula:C56H85N17O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1188.38

    Ref: TM-TP2268

  • Cortistatin 14, human, rat acetate
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    Cortistatin 14, human, rat acetate

    Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows anticonvulsive, neuroprotective effects and
    Formula:C80H112N18O19S2
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:1693.98

    Ref: TM-TP1188L

  • ALEPH hydrochloride
    Targetmol
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    ALEPH hydrochloride

    CAS:
    <p>ALEPH (hydrochloride) acts as a partial agonist of h5-HT2A and h5-HT2B receptors, with EC50 values of 10.3 nM and 19.2 nM, respectively. It can induce head twitch responses in mice, with an ED50 of 0.80 mg/kg.</p>
    Formula:C12H20ClNO2S
    Color and Shape:Solid
    Molecular weight:277.81

    Ref: TM-T203157

  • CB1R agonist 1
    Targetmol
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    CB1R agonist 1

    <p>CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.</p>
    Formula:C20H18F3N3O3S
    Color and Shape:Solid
    Molecular weight:437.435

    Ref: TM-T206337

  • IRL-1038 acetate
    Targetmol
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    IRL-1038 acetate

    <p>IRL-1038 acetate is a potent ETB endothelin receptor antagonist.</p>
    Formula:C70H96N14O17S2
    Purity:97.51%
    Color and Shape:Soild
    Molecular weight:1469.73

    Ref: TM-TP2262L

  • Ki16198
    Targetmol
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    Ki16198

    CAS:
    <p>Ki16198, a methyl ester derivative of Ki16425, blocks LPA1/3, weak on LPA2; inactive on LPA4/5/6. Ki values: 0.34 μM (LPA1), 0.93 μM (LPA3).</p>
    Formula:C24H25ClN2O5S
    Purity:98.09%
    Color and Shape:Solid
    Molecular weight:488.98

    Ref: TM-T6347

  • Antisauvagine-30
    Targetmol
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    Antisauvagine-30

    CAS:
    <p>CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells &amp; stress-related responses in mice.</p>
    Formula:C161H274N48O46S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3650.29

    Ref: TM-TP2091

  • 15-keto-17-phenyl trinor Prostaglandin F2α
    Targetmol
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    15-keto-17-phenyl trinor Prostaglandin F2α

    CAS:
    <p>Bimatoprost is an F-series prostaglandin (PG) analog which has been approved for use as an ocular hypotensive drug.</p>
    Formula:C23H30O5
    Color and Shape:Solid
    Molecular weight:386.488

    Ref: TM-T37934

  • Cianopramine hydrochloride
    Targetmol
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    Cianopramine hydrochloride

    CAS:
    <p>Cianopramine hydrochloride is a bio-active chemical.</p>
    Formula:C20H24ClN3
    Color and Shape:Solid
    Molecular weight:341.88

    Ref: TM-T30929

  • [D-Phe12]-Bombesin
    Targetmol
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    [D-Phe12]-Bombesin

    CAS:
    <p>Bombesin receptor antagonist</p>
    Formula:C74H112N22O18S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1629.88

    Ref: TM-TP2239

  • [bAla8]-Neurokinin A(4-10)
    Targetmol
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    [bAla8]-Neurokinin A(4-10)

    CAS:
    [bAla8]-Neurokinin A(4-10) is a neurokinin 2 (NK2) receptor agonist.
    Formula:C35H56N8O10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:780.94

    Ref: TM-TP1100

  • allo-Yohimbine
    Targetmol
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    allo-Yohimbine

    CAS:
    <p>allo-Yohimbine is a biochemical.</p>
    Formula:C21H26N2O3
    Color and Shape:Solid
    Molecular weight:354.44

    Ref: TM-T29884

  • Secretin, porcine
    Targetmol
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    Secretin, porcine

    CAS:
    Porcine secretin: 27-amino acid peptide for diagnosing pancreatic dysfunction and gastrinoma, stimulates bicarbonate fluid.
    Formula:C130H220N44O41·xC2H4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:N/A

    Ref: TM-TP1048

  • SC 31391
    Targetmol
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    SC 31391

    CAS:
    <p>SC 31391 is a PGE1 analog.</p>
    Formula:C24H32O6
    Color and Shape:Solid
    Molecular weight:416.51

    Ref: TM-T34550

  • M40
    Targetmol
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    M40

    CAS:
    <p>Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat</p>
    Formula:C94H145N23O24
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1981.33

    Ref: TM-TP1992

  • Adrenocorticotropic Hormone (ACTH) (1-39), rat
    Targetmol
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    Adrenocorticotropic Hormone (ACTH) (1-39), rat

    CAS:
    ACTH (1-39), rat: potent MC2 agonist, forms fragments in vitro, isolated by HPLC, characterized by amino acids and NH2-terminus.
    Formula:C210H315N57O57S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4582.23

    Ref: TM-TP1249

  • Blue FPG-A trisodium
    Targetmol
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    Blue FPG-A trisodium

    CAS:
    <p>Blue FPG-A trisodium is a P2X1 &amp; P2Y1 receptor antagonist, IC50: 35.5 μM &amp; 2.6 μM, related to RB2.</p>
    Formula:C29H17ClN7Na3O11S3
    Color and Shape:Solid
    Molecular weight:840.1

    Ref: TM-T75347

  • Thielavin A
    Targetmol
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    Thielavin A

    CAS:
    <p>Thielavin A, from T. terricola, inhibits COX and glucose-6-phosphatase; non-competitive α-glucosidase inhibitor.</p>
    Formula:C29H30O10
    Color and Shape:Solid
    Molecular weight:538.549

    Ref: TM-T37774

  • CymitQuimica logo
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    HDAC6-IN-49

    <p>HDAC6-IN-49 (Compound 3) is an inhibitor of HDAC, with IC50 values of 0.012 and 0.735 µM against HDAC6 and HDAC1, respectively. Additionally, it inhibits MAO-B, cholinesterase (ChE), histamine receptor (H3R), and serotonin 6 receptor (5-HT6R). HDAC6-IN-49 exhibits neuroprotective effects in SH-SY5Y cells and enhances cognitive functions and motor abilities in fruit fly models of Parkinson's disease and C. elegans models of Alzheimer's disease.</p>
    Color and Shape:Odour Solid

    Ref: TM-T200554

  • Ethylpropyltryptamine
    Targetmol
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    Ethylpropyltryptamine

    CAS:
    <p>Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.</p>
    Formula:C15H22N2
    Color and Shape:Solid
    Molecular weight:230.35

    Ref: TM-T203137

  • Neuropeptide S(Mouse)
    Targetmol
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    Neuropeptide S(Mouse)

    CAS:
    <p>Endogenous NPSR agonist, EC50 = 3 nM. Boosts Ca2+ levels, activity, wakefulness, reduces anxiety in mice.</p>
    Formula:C93H156N34O27
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2182.47

    Ref: TM-TP1981

  • M1145
    Targetmol
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    M1145

    CAS:
    <p>Potent GAL2 agonist with EC50 = 38 nM; Ki: 6.55 nM (GAL2), 497 nM (GAL3), 587 nM (GAL1); enhances galanin signaling.</p>
    Formula:C128H205N37O32
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2774.26

    Ref: TM-TP1991

  • (Ala13)-Apelin-13
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    (Ala13)-Apelin-13

    CAS:
    (Ala13)-Apelin-13 is a useful organic compound for research related to life sciences. The catalog number is T35374 and the CAS number is 568565-11-7.
    Formula:C63H107N23O16S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1474.75

    Ref: TM-T35374

  • 2-Methyl-N,N-dimethyltryptamine
    Targetmol
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    2-Methyl-N,N-dimethyltryptamine

    CAS:
    <p>2-Methyl-N,N-dimethyltryptamine (2,N,N-TMT, compound 15) exhibits binding affinity for the serotonin (5-HT) receptor, with a pA2 value of 6.04. It plays a significant role in neurological disease research.</p>
    Formula:C13H18N2
    Color and Shape:Solid
    Molecular weight:202.3

    Ref: TM-T203691

  • Neurokinin B
    Targetmol
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    Neurokinin B

    CAS:
    <p>NKB, a tachykinin peptide, impacts human functions like gonadotropin-releasing hormone secretion.</p>
    Formula:C55H79N13O14S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1210.42

    Ref: TM-TP1363

  • Mini Gastrin I, human
    Targetmol
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    Mini Gastrin I, human

    CAS:
    <p>Mini Gastrin I, human, is a truncated form of the human gastrin peptide, encompassing amino acids 5-17 of the original sequence.</p>
    Formula:C74H99N15O26S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1646.73

    Ref: TM-TP1821

  • UCM 549
    Targetmol
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    UCM 549

    CAS:
    <p>UCM 549 is a bioactive chemical.</p>
    Formula:C19H21NO2
    Color and Shape:Solid
    Molecular weight:295.38

    Ref: TM-T34983

  • CymitQuimica logo
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    Orexin A (human, rat, mouse) (TFA)

    Endogenous orexin receptor agonist with Ki of 20 nM (OX1) and 38 nM (OX2), promotes feeding, may regulate sleep-wake cycle.
    Formula:C154H244N47F3O46S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3675.12

    Ref: TM-TP1550

  • Urocortin III, mouse
    Targetmol
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    Urocortin III, mouse

    CAS:
    <p>Mouse UcnIII, linked to stress behaviors, mainly occurs in the brain and rises in the hypothalamus post-restraint.</p>
    Formula:C186H312N52O52S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4172.97

    Ref: TM-TP1649

  • GLP-1 receptor agonist 8
    Targetmol
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    GLP-1 receptor agonist 8

    CAS:
    <p>GLP-1 receptor agonist 8, potent for diabetes and obesity research, may also study NAFLD.</p>
    Formula:C34H36ClFN6O4
    Color and Shape:Solid
    Molecular weight:647.14

    Ref: TM-T74132

  • tetranor-PGJM
    Targetmol
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    tetranor-PGJM

    CAS:
    <p>Tetranor-PGJM is a metabolite of prostaglandin D2 and is associated with the anti-inflammatory effects of curcumin.</p>
    Formula:C16H22O6
    Color and Shape:Solid
    Molecular weight:310.346

    Ref: TM-T38307

  • 4-Hydroxy MET
    Targetmol
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    4-Hydroxy MET

    CAS:
    4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.
    Formula:C13H18N2O
    Color and Shape:Solid
    Molecular weight:218.3

    Ref: TM-T203151

  • CymitQuimica logo
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    AdTx1

    <p>Selective non-competitive α1A adrenoceptor antagonist with Ki of 0.35 nM; inactive on other GPCRs; affects phenylephrine actions.</p>
    Formula:C310H481N87O100S8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:7283.22

    Ref: TM-TP2086

  • CymitQuimica logo
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    Eloralintide sodium

    <p>Eloralintide sodium (LY-3841136 sodium) is an AMYR (amylin receptor) agonist applicable for studying type 2 diabetes and obesity.</p>
    Formula:C201H319N49O65S2·xNa
    Purity:98.66%
    Color and Shape:Solid
    Molecular weight:4526.1 (free base)

    Ref: TM-TP3220

  • GR 94800
    Targetmol
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    GR 94800

    CAS:
    <p>Potent and selective tachykinin NK2 receptor antagonist</p>
    Formula:C49H61N9O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:904.082

    Ref: TM-T22811

  • Tienoxolol FA
    Targetmol
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    Tienoxolol FA

    <p>Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.</p>
    Formula:C22H30N2O7S
    Purity:97.05% - 98.85%
    Color and Shape:Soild
    Molecular weight:466.55

    Ref: TM-T68161L

  • Galantide
    Targetmol
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    Galantide

    CAS:
    <p>Galantide is a reversible and non-specific antagonist of galanin receptor.</p>
    Formula:C104H151N25O26S
    Purity:98%
    Color and Shape:White Lyophilised Solid
    Molecular weight:2199.53

    Ref: TM-T15368

  • CymitQuimica logo
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    P2Y6R antagonist 1

    <p>P2Y6R antagonist 1 (compound 5ab) is a selective, orally active antagonist of P2Y6R, featuring an IC50 value of 19.6 nM. This compound also exhibits anti-inflammatory properties.</p>
    Color and Shape:Odour Solid

    Ref: TM-T200515

  • GRK-IN-1
    Targetmol
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    GRK-IN-1

    CAS:
    <p>4-Amino-5-(bromomethyl)-2-methylpyrimidine used in vitamin B1 analogs and esters synthesis.</p>
    Formula:C6H10Br3N3
    Color and Shape:Solid
    Molecular weight:363.879

    Ref: TM-T35723

  • 19(S)-HETE
    Targetmol
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    19(S)-HETE

    CAS:
    <p>19-HETE, a CYP450 arachidonic acid metabolite from kidneys, consists of 70% (S) and 30% (R) isomers and dilates renal vessels.</p>
    Formula:C20H32O3
    Color and Shape:Solid
    Molecular weight:320.473

    Ref: TM-T35850

  • Propranolol hydrochloride
    Targetmol
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    Propranolol hydrochloride

    CAS:
    <p>Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverse</p>
    Formula:C16H22ClNO2
    Purity:99.94% - >99.99%
    Color and Shape:White Or Almost White Powder White Powder
    Molecular weight:295.80

    Ref: TM-T0812

  • SSTR4 agonist-1
    Targetmol
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    SSTR4 agonist-1

    CAS:
    <p>SSTR4agonist-1 (Compound 47) is a selective agonist of the somatostatin receptor 4 (SSTR4), with an EC50 of 4.7 nM. It has a half-life of over 130 minutes in human liver microsomes.</p>
    Formula:C16H23N3O2
    Color and Shape:Solid
    Molecular weight:289.37

    Ref: TM-T203033

  • CymitQuimica logo
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    PAR650097

    <p>PAR650097 is a humanized monoclonal antibody targeting PAR2, used in migraine research.</p>
    Purity:96.67% (SEC-HPLC) - 98.83% (SEC-HPLC)
    Color and Shape:Liquid
    Molecular weight:145.5kDa

    Ref: TM-T77402

  • CymitQuimica logo
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    Dulaglutide

    CAS:
    <p>Dulaglutide (LY2189265) is a GLP-1 receptor agonist for studying type 2 diabetes mellitus (T2DM).</p>
    Color and Shape:Solid

    Ref: TM-T75718

  • Sibenadet hydrochloride
    Targetmol
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    Sibenadet hydrochloride

    CAS:
    <p>Sibenadet, a D2/beta2-agonist, is potential useful for the treatment of symptoms of chronic obstructive pulmonary disease.</p>
    Formula:C22H29ClN2O5S2
    Color and Shape:Solid
    Molecular weight:501.06

    Ref: TM-T28774

  • [D-Phe12,Leu14]-Bombesin
    Targetmol
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    [D-Phe12,Leu14]-Bombesin

    CAS:
    <p>Bombesin receptor blocker; stops binding in rat brain (IC50=2 μM), hinders amylase release (IC50=4 μM), reduces appetite suppression in vivo.</p>
    Formula:C77H113F3N22O20
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1724.9

    Ref: TM-TP1916

  • MrgprX2 antagonist-4
    Targetmol
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    MrgprX2 antagonist-4

    CAS:
    <p>MrgprX2 antagonist-4, from patent US20210128561A1, inhibits MrgprX2 receptor; useful for skin inflammation studies.</p>
    Formula:C16H19N3O
    Color and Shape:Solid
    Molecular weight:269.348

    Ref: TM-T40268

  • Piperulin A
    Targetmol
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    Piperulin A

    CAS:
    <p>Piperulin A effectively inhibits platelet-activating factor receptor (PAFR) by specifically blocking its binding to isolated rabbit platelet plasma membranes,</p>
    Formula:C23H28O6
    Color and Shape:Solid
    Molecular weight:400.46

    Ref: TM-T79950

  • RF9 acetate
    Targetmol
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    RF9 acetate

    <p>RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.</p>
    Formula:C28H42N6O5
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:542.67

    Ref: TM-T16738L

  • Cortistatin-8 acetate
    Targetmol
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    Cortistatin-8 acetate

    <p>Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.</p>
    Formula:C49H72N12O11S2
    Purity:99.01%
    Color and Shape:Soild
    Molecular weight:1069.3

    Ref: TM-TP2236L

  • TAK-615
    Targetmol
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    TAK-615

    CAS:
    <p>TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of LPA1 receptors.</p>
    Formula:C25H22FNO4
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:419.44

    Ref: TM-T9699

  • ABT-702
    Targetmol
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    ABT-702

    CAS:
    <p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>
    Formula:C22H19BrN6O
    Purity:99.57%
    Color and Shape:Soild
    Molecular weight:463.33

    Ref: TM-T4668L

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    AMTG-DA1

    <p>AMTG-DA1 is a ligand for the gastrin-releasing peptide receptor (GRPR), and it can be utilized in cancer research.</p>
    Formula:C101H149IN22O25
    Color and Shape:Solid
    Molecular weight:2197.0109

    Ref: TM-T207222

  • GR 64349
    Targetmol
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    GR 64349

    CAS:
    <p>Potent NK2 agonist, EC50=3.7 nM in rat colon; &gt;1000x selectivity over NK1, &gt;300x over NK3; effective in vivo.</p>
    Formula:C42H68N10O11S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:921.12

    Ref: TM-TP2023

  • Phenylethanolamine A
    Targetmol
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    Phenylethanolamine A

    CAS:
    <p>Phenylethanolamine A is a β-adrenergic agonist and a byproduct of the Ractopamine synthesis process.</p>
    Formula:C19H24N2O4
    Color and Shape:Solid
    Molecular weight:344.40

    Ref: TM-T38741

  • Lobeline sulfate
    Targetmol
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    Lobeline sulfate

    CAS:
    <p>Lobeline sulfate, an alkaloid like nicotine, aids in smoking cessation, insomnia, and respiratory issues. Less potent on nicotinic receptors.</p>
    Formula:C22H29NO6S
    Purity:98%
    Color and Shape:White Powder
    Molecular weight:435.54

    Ref: TM-T22357

  • 1,8-Cineole
    Targetmol
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    1,8-Cineole

    CAS:
    <p>Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.</p>
    Formula:C10H18O
    Purity:97.44% - 97.44%
    Color and Shape:Solid
    Molecular weight:154.25

    Ref: TM-T1714

  • L-threo Lysosphingomyelin (d18:1)
    Targetmol
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    L-threo Lysosphingomyelin (d18:1)

    CAS:
    <p>L-threo Lysosphingomyelin, a natural S1P receptor agonist, has EC50s: 19.3 nM (hS1P1), 131.8 nM (hS1P3), 313.3 nM (hS1P2).</p>
    Formula:C23H49N2O5P
    Color and Shape:Solid
    Molecular weight:464.62

    Ref: TM-T38452

  • PZ-128
    Targetmol
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    PZ-128

    CAS:
    PZ-128, a PAR1 antagonist, is used potentially for the treatment of thrombosis.
    Formula:C55H99N13O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1086.46

    Ref: TM-T28477

  • [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
    Targetmol
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    [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P

    CAS:
    <p>Broad-spectrum inverse agonist; potent at ghrelin receptor (EC50=5.2 nM); blocks other neuropeptide receptors; induces apoptosis; inhibits tumor growth.</p>
    Formula:C79H109N19O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1516.85

    Ref: TM-TP1931

  • HCGRP-(8-37)
    Targetmol
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    HCGRP-(8-37)

    CAS:
    Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonist
    Formula:C139H230N44O38
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3125.59

    Ref: TM-TP1134

  • PG106
    Targetmol
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    PG106

    CAS:
    <p>Selective hMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5 receptors.</p>
    Formula:C51H69N13O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1008.19

    Ref: TM-TP1952

  • Hydroxybupropion
    Targetmol
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    Hydroxybupropion

    CAS:
    <p>Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).</p>
    Formula:C13H18ClNO2
    Purity:99.73%
    Color and Shape:Off-White Solid
    Molecular weight:255.74

    Ref: TM-T11588

  • AR-C126313
    Targetmol
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    AR-C126313

    CAS:
    <p>AR-C126313 is a thiouracil derivative.</p>
    Formula:C28H23N7O3S
    Color and Shape:Solid
    Molecular weight:537.59

    Ref: TM-T30120

  • ELA-21 (human)
    Targetmol
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    ELA-21 (human)

    CAS:
    <p>Apelin receptor agonist with high affinity for normal/PAH hearts (pKi 9.31/9.46). Blocks cAMP, promotes β-arrestin in vitro. Part of ELA-32.</p>
    Formula:C112H184N40O25S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2587.12

    Ref: TM-TP2096

  • MK-7246 S enantiomer
    Targetmol
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    MK-7246 S enantiomer

    MK-7246 S enantiomer is a potent and selective CRTH2 antagonist.
    Formula:C21H21FN2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:416.47

    Ref: TM-T12067

  • 11-deoxy Prostaglandin E1
    Targetmol
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    11-deoxy Prostaglandin E1

    CAS:
    <p>11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and cause</p>
    Formula:C20H34O4
    Color and Shape:Solid
    Molecular weight:338.48

    Ref: TM-T36770

  • SB234551
    Targetmol
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    SB234551

    CAS:
    <p>SB234551 is a selective antagonist of endothelin ETA receptor.</p>
    Formula:C34H34N2O9
    Color and Shape:Solid
    Molecular weight:614.64

    Ref: TM-T28683

  • PSB 0777 ammonium salt
    Targetmol
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    PSB 0777 ammonium salt

    CAS:
    <p>adenosine A2A receptor full agonist</p>
    Formula:C18H24N6O7S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.55

    Ref: TM-T23196

  • Secretin (28-54), human
    Targetmol
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    Secretin (28-54), human

    CAS:
    Secretin (28-54), human, is a 27-amino acid residue peptide with a C-terminal amidation, acting on human secretin receptors.
    Formula:C130H220N44O40
    Purity:98%
    Color and Shape:Powder
    Molecular weight:3039.46

    Ref: TM-TP1136

  • Sch 202596
    Targetmol
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    Sch 202596

    CAS:
    <p>Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.</p>
    Formula:C25H22Cl2O12
    Color and Shape:Solid
    Molecular weight:585.34

    Ref: TM-T28705

  • SB 201146
    Targetmol
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    SB 201146

    CAS:
    <p>SB 201146 is a leukotriene B4 antagonist with high affinity.</p>
    Formula:C30H35LiN2O5S
    Color and Shape:Solid
    Molecular weight:542.61

    Ref: TM-T28667

  • Navafenterol saccharinate
    Targetmol
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    Navafenterol saccharinate

    CAS:
    <p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>
    Formula:C45H47N7O9S3
    Color and Shape:Solid
    Molecular weight:926.09

    Ref: TM-T30265

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    Pancreatic polypeptide TFA

    <p>Pancreatic polypeptide TFA acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.</p>
    Color and Shape:Odour Solid

    Ref: TM-TP2887

  • (+)-Cloprostenol
    Targetmol
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    (+)-Cloprostenol

    CAS:
    <p>(+)-Cloprostenol is a analogue of prostaglandin F2α (PGF2α), and is selective prostaglandin receptor agonistic.</p>
    Formula:C22H29ClO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:424.92

    Ref: TM-T13461