GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 18 more subcategories

Found 5378 products of "GPCR/G-Protein"

Purity (%)

100

products per page.

+ Info
Perphenazine
CAS:
- 58-39-9
Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
Formula:C₂₁H₂₆ClN₃OS
Purity:99.3% - 99.99%
Color and Shape:Solid
Molecular weight:403.97
Ref: TM-T1090
+ Info
PF-610355 HCl
PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.
Formula:C₁₉H₂₂ClN₇O₆
Purity:97.97%
Color and Shape:Solid
Molecular weight:479.87
Ref: TM-T16509L
+ Info
AZ084
CAS:
- 929300-19-6
AZ084 is a potent, selective, allosteric, and oral active CCR8 antagonist (Ki: 0.9 nM). It has the potential to treat asthma.
Formula:C₂₆H₃₄N₄O₂
Purity:97.12%
Color and Shape:Solid
Molecular weight:434.57
Ref: TM-T10425
+ Info
Ranitidine Hydrochloride
CAS:
- 66357-59-3
Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.
Formula:C₁₃H₂₃ClN₄O₃S
Purity:99.30% - 99.49%
Color and Shape:Solid
Molecular weight:350.86
Ref: TM-T0865
+ Info
YNT-185
CAS:
- 1804978-81-1
YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,
Formula:C₃₃H₃₇N₅O₅S
Purity:99.67%
Color and Shape:Solid
Molecular weight:615.74
Ref: TM-T39229
+ Info
CCR2-RA-[R]
CAS:
- 512177-83-2
CCR2-RA-[R] is a C-C chemokine receptor type 2 (CCR2) allosteric antagonist (IC50: 103 nM).
Formula:C₁₈H₁₉ClFNO₃
Purity:99.7%
Color and Shape:Solid
Molecular weight:351.8
Ref: TM-T14900
+ Info
Urocortin (rat) acetate
Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.
Purity:97.76%
Color and Shape:Soild
Ref: TM-TP1020L
+ Info
Cloperastine hydrochloride
CAS:
- 14984-68-0
Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.
Formula:C₂₀H₂₅Cl₂NO
Purity:97.74% - 99.42%
Color and Shape:Solid
Molecular weight:366.33
Ref: TM-T0723
+ Info
ML604086
CAS:
- 850330-18-6
ML604086 suppresses CCL1 mediated chemotaxis and enhances intracellular Ca2 concentrations.
Formula:C₂₇H₃₂N₄O₄S
Purity:99.91%
Color and Shape:Solid
Molecular weight:508.63
Ref: TM-T16111
+ Info
Ramelteon
CAS:
- 196597-26-9
Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.
Formula:C₁₆H₂₁NO₂
Purity:97.21% - 99.92%
Color and Shape:Crystalline Solid
Molecular weight:259.34
Ref: TM-T1463
+ Info
Benztropine mesylate
CAS:
- 132-17-2
Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON
Formula:C₂₁H₂₅NO·CH₄SO₃
Purity:98.41% - 99.96%
Color and Shape:White Crystalline Powder; Odourless Or Almost Odourless
Molecular weight:403.53
Ref: TM-T1336
+ Info
Risperidone
CAS:
- 106266-06-2
Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
Formula:C₂₃H₂₇FN₄O₂
Purity:99.73%
Color and Shape:Crystalline Solid
Molecular weight:410.48
Ref: TM-T0351
+ Info
Balovaptan
CAS:
- 1228088-30-9
Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.
Formula:C₂₂H₂₄ClN₅O
Purity:99.88%
Color and Shape:Solid
Molecular weight:409.91
Ref: TM-T14494
+ Info
Crotedumab
CAS:
- 1452387-69-7
Crotedumab (REGN1193) is a humanized antibody targeting GCGR, which reduces fasting blood glucose and improves glucose tolerance, used in diabetes research.
Purity:>95%
Color and Shape:Liquid
Ref: TM-T76862
+ Info
Terfenadine
CAS:
- 50679-08-8
Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.
Formula:C₃₂H₄₁NO₂
Purity:98.76% - 99.75%
Color and Shape:Solid
Molecular weight:471.67
Ref: TM-T1266
+ Info
p-MPPI hydrochloride
CAS:
- 220643-77-6
p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.
Formula:C₂₅H₂₈ClIN₄O₂
Purity:99.95%
Color and Shape:Solid
Molecular weight:578.87
Ref: TM-T16421
+ Info
hGPR91 antagonist 1
CAS:
- 1314796-00-3
hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
Formula:C₃₁H₂₃F₄N₃O
Purity:98.89%
Color and Shape:Solid
Molecular weight:529.53
Ref: TM-T11560
+ Info
Cefaclor monohydrate
CAS:
- 70356-03-5
Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.
Formula:C₁₅H₁₆ClN₃O₅S
Purity:97.36% - 99.9%
Color and Shape:White Crystaling Powder
Molecular weight:385.82
Ref: TM-T1495
+ Info
Triflupromazine hydrochloride
CAS:
- 1098-60-8
Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.
Formula:C₁₈H₂₀ClF₃N₂S
Purity:99.76% - 99.82%
Color and Shape:Crystals
Molecular weight:388.88
Ref: TM-T0302
+ Info
Droperidol
CAS:
- 548-73-2
Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.
Formula:C₂₂H₂₂FN₃O₂
Purity:97.16% - 98%
Color and Shape:Solid
Molecular weight:379.43
Ref: TM-T0990