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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5696 products of "GPCR/G-Protein"

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  • Bradykinin (acetate)
    Targetmol
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    Bradykinin (acetate)

    CAS:
    <p>Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.</p>
    Formula:C52H77N15O13
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1120.26

    Ref: TM-T21610

  • Cariprazine hydrochloride
    Targetmol
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    Cariprazine hydrochloride

    CAS:
    <p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>
    Formula:C21H33Cl3N4O
    Purity:99.78% - >99.99%
    Color and Shape:Solid
    Molecular weight:463.87

    Ref: TM-T8382

  • Ditolylguanidine
    Targetmol
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    Ditolylguanidine

    CAS:
    Ditolylguanidine (Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor).
    Formula:C15H17N3
    Purity:98.42%
    Color and Shape:White To Pinkish Solid Powder
    Molecular weight:239.32

    Ref: TM-T5969

  • Midodrine
    Targetmol
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    Midodrine

    CAS:
    <p>Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.</p>
    Formula:C12H18N2O4
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:254.28

    Ref: TM-T22369

  • 1-[(5-methylisoxazol-3-yl)methyl]piperazine
    Targetmol
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    1-[(5-methylisoxazol-3-yl)methyl]piperazine

    CAS:
    <p>1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.</p>
    Formula:C9H15N3O
    Purity:95%
    Color and Shape:Solid
    Molecular weight:181.23

    Ref: TM-T8582

  • VKGILS-NH2 Acetate
    Targetmol
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    VKGILS-NH2 Acetate

    <p>VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.</p>
    Formula:C30H58N8O9
    Purity:98.83%
    Color and Shape:Solid
    Molecular weight:674.83

    Ref: TM-T21699L

  • Hydroxyzine dihydrochloride
    Targetmol
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    Hydroxyzine dihydrochloride

    CAS:
    <p>Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.</p>
    Formula:C21H27ClN2O2·2HCl
    Purity:99.46% - 99.79%
    Color and Shape:Oil Powder
    Molecular weight:447.83

    Ref: TM-T2200

  • Dapagliflozin ((2S)-1,2-propanediol, hydrate)
    Targetmol
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    Dapagliflozin ((2S)-1,2-propanediol, hydrate)

    CAS:
    <p>Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal sodium-glucose co-</p>
    Formula:C24H35ClO9
    Purity:99.88% - 99.94%
    Color and Shape:Solid
    Molecular weight:502.98

    Ref: TM-T4460

  • Pridopidine
    Targetmol
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    Pridopidine

    CAS:
    Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.
    Formula:C15H23NO2S
    Purity:95.2% - 99.89%
    Color and Shape:Solid
    Molecular weight:281.41

    Ref: TM-T7352

  • lumateperone Tosylate
    Targetmol
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    lumateperone Tosylate

    CAS:
    <p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>
    Formula:C31H36FN3O4S
    Purity:95.83% - 99.95%
    Color and Shape:Solid
    Molecular weight:565.7

    Ref: TM-TQ0084

  • Peptide YY (PYY) (3-36), human
    Targetmol
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    Peptide YY (PYY) (3-36), human

    CAS:
    <p>Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.</p>
    Formula:C176H272N52O54
    Purity:97.76%
    Color and Shape:Solid
    Molecular weight:3980.42

    Ref: TM-TP1059

  • Doxazosin
    Targetmol
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    Doxazosin

    CAS:
    <p>Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.</p>
    Formula:C23H25N5O5
    Purity:99.47% - 99.87%
    Color and Shape:Solid
    Molecular weight:451.48

    Ref: TM-T22316

  • Ropinirole hydrochloride
    Targetmol
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    Ropinirole hydrochloride

    CAS:
    <p>Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.</p>
    Formula:C16H24N2O·HCl
    Purity:99.87% - 99.98%
    Color and Shape:Off-White Solid
    Molecular weight:296.84

    Ref: TM-T2592

  • D3-βArr
    Targetmol
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    D3-βArr

    CAS:
    <p>D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct</p>
    Formula:C20H23N5
    Purity:98.82%
    Color and Shape:Solid
    Molecular weight:333.43

    Ref: TM-T5383

  • Reboxetine mesylate
    Targetmol
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    Reboxetine mesylate

    CAS:
    <p>Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).</p>
    Formula:C19H23NO3·CH4O3S
    Purity:99.18% - 99.87%
    Color and Shape:Tan Or Off-White Cyrstalline Solid
    Molecular weight:409.5

    Ref: TM-T6963

  • Anisotropine Methylbromide
    Targetmol
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    Anisotropine Methylbromide

    CAS:
    Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.
    Formula:C17H32BrNO2
    Purity:99.73%
    Color and Shape:Crystals From Acetone Solid
    Molecular weight:362.35

    Ref: TM-T4981

  • ABT-702 dihydrochloride
    Targetmol
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    ABT-702 dihydrochloride

    CAS:
    ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.
    Formula:C22H21BrCl2N6O
    Purity:98.42% - 98.98%
    Color and Shape:Solid
    Molecular weight:536.25

    Ref: TM-T4668

  • Derenofylline
    Targetmol
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    Derenofylline

    CAS:
    <p>Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)</p>
    Formula:C18H20N4O
    Purity:98.09%
    Color and Shape:Solid
    Molecular weight:308.38

    Ref: TM-T8312

  • Org 27569
    Targetmol
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    Org 27569

    CAS:
    <p>Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity and</p>
    Formula:C24H28ClN3O
    Purity:>99.99% - ≥95%
    Color and Shape:Solid
    Molecular weight:409.95

    Ref: TM-T2635

  • CAY10526
    Targetmol
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    CAY10526

    CAS:
    CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.
    Formula:C12H7BrO3S
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:311.15

    Ref: TM-T23861