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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5696 products of "GPCR/G-Protein"

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  • Dazoxiben
    Targetmol
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    Dazoxiben

    CAS:
    <p>Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthase</p>
    Formula:C12H13ClN2O3
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:268.7

    Ref: TM-T7968

  • CCG-50014
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    CCG-50014

    CAS:
    <p>CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.</p>
    Formula:C16H13FN2O2S
    Purity:98.53%
    Color and Shape:Solid
    Molecular weight:316.35

    Ref: TM-T6434

  • Ralmitaront
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    Ralmitaront

    CAS:
    <p>Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).</p>
    Formula:C17H22N4O2
    Purity:99.71% - 99.79%
    Color and Shape:Solid
    Molecular weight:314.38

    Ref: TM-T9183

  • TCS-OX2-29
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    TCS-OX2-29

    CAS:
    TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.
    Formula:C23H31N3O3
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:397.51

    Ref: TM-T4965

  • Rolapitant hydrochloride hydrate
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    Rolapitant hydrochloride hydrate

    CAS:
    Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.
    Formula:C25H29ClF6N2O3
    Color and Shape:Solid
    Molecular weight:554.95

    Ref: TM-T68371

  • Eptapirone
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    Eptapirone

    CAS:
    <p>Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.</p>
    Formula:C16H23N7O2
    Purity:99.39% - 99.65%
    Color and Shape:Solid
    Molecular weight:345.4

    Ref: TM-T3179

  • ESI-09
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    ESI-09

    CAS:
    ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.
    Formula:C16H15ClN4O2
    Purity:97.24% - 99.57%
    Color and Shape:Solid
    Molecular weight:330.77

    Ref: TM-T2244

  • Decloxizine dihydrochloride
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    Decloxizine dihydrochloride

    CAS:
    <p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>
    Formula:C21H28N2O2·2ClH
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:413.39

    Ref: TM-T5495

  • PF-06882961 Tris
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    PF-06882961 Tris

    CAS:
    <p>PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>
    Formula:C35H41FN6O7
    Purity:98.74% - 99.79%
    Color and Shape:Solid
    Molecular weight:676.7

    Ref: TM-T8876

  • Almotriptan
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    Almotriptan

    CAS:
    Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.
    Formula:C17H25N3O2S
    Purity:99.85%
    Color and Shape:Light Yellow Or White Power
    Molecular weight:335.46

    Ref: TM-T21231

  • Elagolix sodium
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    Elagolix sodium

    CAS:
    <p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>
    Formula:C32H29F5N3NaO5
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:653.57

    Ref: TM-T5031

  • Ritanserin
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    Ritanserin

    CAS:
    Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.
    Formula:C27H25F2N3OS
    Purity:99.77% - 99.89%
    Color and Shape:Solid
    Molecular weight:477.57

    Ref: TM-T16759

  • Bimatoprost
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    Bimatoprost

    CAS:
    <p>Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular</p>
    Formula:C25H37NO4
    Purity:98% - >99.99%
    Color and Shape:Crystalline Solid
    Molecular weight:415.57

    Ref: TM-T2538

  • BMY 7378 dihydrochloride
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    BMY 7378 dihydrochloride

    CAS:
    <p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>
    Formula:C22H33Cl2N3O3
    Purity:97.32% - 99.08%
    Color and Shape:Solid
    Molecular weight:458.42

    Ref: TM-T3046

  • 5-Hydroxy-1-methylhydantoin
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    5-Hydroxy-1-methylhydantoin

    CAS:
    5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.
    Formula:C4H6N2O3
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:130.1

    Ref: TM-T28222

  • Chlorpheniramine
    Targetmol
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    Chlorpheniramine

    CAS:
    <p>Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.</p>
    Formula:C16H19ClN2
    Color and Shape:Solid
    Molecular weight:274.79

    Ref: TM-T60498

  • Neuromedin N acetate(92169-45-4 free base)
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    Neuromedin N acetate(92169-45-4 free base)

    <p>Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct</p>
    Formula:C40H67N7O10
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:805.9

    Ref: TM-TP1085L

  • [Lys5,MeLeu9,Nle10]-NKA(4-10)
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    [Lys5,MeLeu9,Nle10]-NKA(4-10)

    CAS:
    Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
    Formula:C39H65N9O9
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:803.99

    Ref: TM-TP1883

  • Dolasetron
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    Dolasetron

    CAS:
    <p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>
    Formula:C19H20N2O3
    Purity:99.84% - 99.86%
    Color and Shape:White Powder
    Molecular weight:324.37

    Ref: TM-T4568

  • Ursodeoxycholic acid sodium
    Targetmol
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    Ursodeoxycholic acid sodium

    CAS:
    <p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>
    Formula:C24H40NaO4
    Purity:99.66% - 99.96%
    Color and Shape:Solid
    Molecular weight:415.56

    Ref: TM-T29078