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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5745 products of "GPCR/G-Protein"

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  • Promazine hydrochloride

    CAS:
    Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.
    Formula:C17H21ClN2S
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:320.88
  • p-MPPI hydrochloride

    CAS:
    <p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>
    Formula:C25H28ClIN4O2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:578.87
  • Spiperone

    CAS:
    Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.
    Formula:C23H26FN3O2
    Purity:99.34% - 99.91%
    Color and Shape:Solid
    Molecular weight:395.47
  • Protriptyline hydrochloride

    CAS:
    <p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>
    Formula:C19H21N·HCl
    Purity:98.54% - 99.98%
    Color and Shape:Solid
    Molecular weight:299.84
  • Desipramine hydrochloride

    CAS:
    Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.
    Formula:C18H23ClN2
    Purity:99.58% - 99.94%
    Color and Shape:White To Off-White Powder
    Molecular weight:302.842
  • Sertraline hydrochloride

    CAS:
    <p>Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.</p>
    Formula:C17H18Cl3N
    Purity:99.12% - 99.89%
    Color and Shape:Solid Powder
    Molecular weight:342.691
  • Dipivefrin hydrochloride

    CAS:
    <p>Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.</p>
    Formula:C19H27NO5·HCl
    Purity:99.22% - 99.92%
    Color and Shape:Less Gas With A Sweet Odor Colorless Gas With A Sweet Odor
    Molecular weight:387.9
  • Itopride hydrochloride

    CAS:
    Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.
    Formula:C20H27ClN2O4
    Purity:99.59%
    Color and Shape:White Or Pale Brownish Crystal
    Molecular weight:394.9
  • Pimethixene

    CAS:
    <p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 &amp; muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>
    Formula:C19H19NS
    Purity:97.50%
    Color and Shape:Solid
    Molecular weight:293.43
  • Paliperidone

    CAS:
    <p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>
    Formula:C23H27FN4O3
    Purity:95% - 99.08%
    Color and Shape:Off White To Light Orange Coloured Solid
    Molecular weight:426.48
  • α-CGRP, rat

    CAS:
    Endogenous neuropeptide, potent vasodilator
    Formula:C162H262N50O52S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3806.25
  • Guanylin TFA (mouse,rat)


    <p>Guanylin (mouse, rat) TFA is a peptide composed of 15 amino acids and acts as an activator of intestinal guanylate cyclase. This compound is utilized in research related to diarrhea.</p>
    Formula:C60H90N16O22S4·xC2HF3O2
    Color and Shape:Solid
    Molecular weight:1515.71 (free base)
  • β-CGRP, human

    CAS:
    <p>β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascular</p>
    Formula:C162H267N51O48S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3793.41
  • Amylin (8-37), rat

    CAS:
    Amylin (8-37), rat, an analog of IAPP, blocks insulin's effects on muscle glucose uptake and glycogen storage.
    Formula:C140H227N43O43
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3200.61
  • Methapyrilene hydrochloride

    CAS:
    <p>Methapyrilene hydrochloride is a biochemical.</p>
    Formula:C14H20ClN3S
    Color and Shape:Liquid Solution) 5 5 (Ntp 1992)
    Molecular weight:297.85
  • IRL-1620

    CAS:
    <p>IRL-1620 is an effective and selective agonist of endothelin receptor type B (ETB) (Ki: 16 pM).</p>
    Formula:C86H117N17O27
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1820.974
  • KwFwLL-NH2

    CAS:
    KwFwLL-NH2 is a hexapeptide that serves as a ligand for the ghrelin receptor (ghrelin receptor). This compound acts as a specific inverse agonist for the ghrelin receptor, exhibiting moderate potency (EC50=45.6 nM).
    Formula:C49H66N10O6
    Color and Shape:Solid
    Molecular weight:891.11
  • Glucagon receptor antagonists-1

    CAS:
    Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.
    Formula:C29H34FNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:447.58
  • Prazobind

    CAS:
    <p>Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.</p>
    Formula:C23H27N5O3
    Color and Shape:Solid
    Molecular weight:421.501
  • [D-Phe12,Leu14]-Bombesin

    CAS:
    <p>Bombesin receptor blocker; stops binding in rat brain (IC50=2 μM), hinders amylase release (IC50=4 μM), reduces appetite suppression in vivo.</p>
    Formula:C77H113F3N22O20
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1724.9