
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(993 products)
- Adenosine Receptor(246 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(212 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(182 products)
- Hedgehog/Smoothened(47 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(310 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5745 products of "GPCR/G-Protein"
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Promazine hydrochloride
CAS:Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Formula:C17H21ClN2SPurity:99.90%Color and Shape:SolidMolecular weight:320.88p-MPPI hydrochloride
CAS:<p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>Formula:C25H28ClIN4O2Purity:99.95%Color and Shape:SolidMolecular weight:578.87Spiperone
CAS:Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.Formula:C23H26FN3O2Purity:99.34% - 99.91%Color and Shape:SolidMolecular weight:395.47Protriptyline hydrochloride
CAS:<p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>Formula:C19H21N·HClPurity:98.54% - 99.98%Color and Shape:SolidMolecular weight:299.84Desipramine hydrochloride
CAS:Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.Formula:C18H23ClN2Purity:99.58% - 99.94%Color and Shape:White To Off-White PowderMolecular weight:302.842Sertraline hydrochloride
CAS:<p>Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.</p>Formula:C17H18Cl3NPurity:99.12% - 99.89%Color and Shape:Solid PowderMolecular weight:342.691Dipivefrin hydrochloride
CAS:<p>Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.</p>Formula:C19H27NO5·HClPurity:99.22% - 99.92%Color and Shape:Less Gas With A Sweet Odor Colorless Gas With A Sweet OdorMolecular weight:387.9Itopride hydrochloride
CAS:Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.Formula:C20H27ClN2O4Purity:99.59%Color and Shape:White Or Pale Brownish CrystalMolecular weight:394.9Pimethixene
CAS:<p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>Formula:C19H19NSPurity:97.50%Color and Shape:SolidMolecular weight:293.43Paliperidone
CAS:<p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>Formula:C23H27FN4O3Purity:95% - 99.08%Color and Shape:Off White To Light Orange Coloured SolidMolecular weight:426.48α-CGRP, rat
CAS:Endogenous neuropeptide, potent vasodilatorFormula:C162H262N50O52S2Purity:98%Color and Shape:SolidMolecular weight:3806.25Guanylin TFA (mouse,rat)
<p>Guanylin (mouse, rat) TFA is a peptide composed of 15 amino acids and acts as an activator of intestinal guanylate cyclase. This compound is utilized in research related to diarrhea.</p>Formula:C60H90N16O22S4·xC2HF3O2Color and Shape:SolidMolecular weight:1515.71 (free base)β-CGRP, human
CAS:<p>β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascular</p>Formula:C162H267N51O48S3Purity:98%Color and Shape:SolidMolecular weight:3793.41Amylin (8-37), rat
CAS:Amylin (8-37), rat, an analog of IAPP, blocks insulin's effects on muscle glucose uptake and glycogen storage.Formula:C140H227N43O43Purity:98%Color and Shape:SolidMolecular weight:3200.61Methapyrilene hydrochloride
CAS:<p>Methapyrilene hydrochloride is a biochemical.</p>Formula:C14H20ClN3SColor and Shape:Liquid Solution) 5 5 (Ntp 1992)Molecular weight:297.85IRL-1620
CAS:<p>IRL-1620 is an effective and selective agonist of endothelin receptor type B (ETB) (Ki: 16 pM).</p>Formula:C86H117N17O27Purity:98%Color and Shape:SolidMolecular weight:1820.974KwFwLL-NH2
CAS:KwFwLL-NH2 is a hexapeptide that serves as a ligand for the ghrelin receptor (ghrelin receptor). This compound acts as a specific inverse agonist for the ghrelin receptor, exhibiting moderate potency (EC50=45.6 nM).Formula:C49H66N10O6Color and Shape:SolidMolecular weight:891.11Glucagon receptor antagonists-1
CAS:Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.Formula:C29H34FNO2Purity:98%Color and Shape:SolidMolecular weight:447.58Prazobind
CAS:<p>Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.</p>Formula:C23H27N5O3Color and Shape:SolidMolecular weight:421.501[D-Phe12,Leu14]-Bombesin
CAS:<p>Bombesin receptor blocker; stops binding in rat brain (IC50=2 μM), hinders amylase release (IC50=4 μM), reduces appetite suppression in vivo.</p>Formula:C77H113F3N22O20Purity:98%Color and Shape:SolidMolecular weight:1724.9

