GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Levosalbutamol Hydrochloride
CAS:Levosalbutamol Hydrochloride is a β2-adrenergic receptor agonist. It is used to treat asthma and chronic obstructive pulmonary disease.Formula:C13H22ClNO3Purity:98%Color and Shape:SolidMolecular weight:275.775-HT3 antagonist 5
CAS:5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.Formula:C16H13N3O2Purity:99.84%Color and Shape:SolidMolecular weight:279.29Emedastine Difumarate
CAS:Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.Formula:C25H34N4O9Color and Shape:SolidMolecular weight:534.56Antazoline phosphate
CAS:Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.Formula:C17H22N3O4PPurity:98%Color and Shape:CoaMolecular weight:363.35rac-Propranolol-d7
CAS:Rac-Propranolol-d7 is the deuterated form of Rac-Propranolol. Propranolol is a β-adrenergic receptor antagonist that inhibits β1AR.Formula:C16H14D7NO2Color and Shape:SolidMolecular weight:266.39Timapiprant sodium
CAS:Timapiprant sodium: potent DP2 antagonist; inhibits mast cell activation; displaces [3H]PGD2, Ki=3-13 nM.Formula:C21H17FN2NaO2Purity:98%Color and Shape:SolidMolecular weight:371.367Diphenylpyraline
CAS:Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.Formula:C19H23NOColor and Shape:SolidMolecular weight:281.39Eticlopride hydrochloride
CAS:Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).Formula:C17H25ClN2O3·HClPurity:98%Color and Shape:SolidMolecular weight:377.31SBI-810 hydrochloride
CAS:SBI-810 hydrochloride is a β-arrestin-2 (βarr2)-biased allosteric modulator of NTSR1 (neurotensin receptor 1), exerting analgesic effects.Formula:C27H35ClN4O2Purity:99.42%Color and Shape:SolidMolecular weight:483.05Trimethobenzamide
CAS:Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.Formula:C21H28N2O5Color and Shape:SolidMolecular weight:388.46Fexofenadine-d6
CAS:Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.Formula:C32H39NO4Purity:98%Color and Shape:SolidMolecular weight:507.69SB-200646A
CAS:SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.Formula:C15H15ClN4OPurity:98%Color and Shape:SolidMolecular weight:302.76YNT-185 dihydrochloride
CAS:Potent OX2 agonist (EC50=28nM); 100x selective over OX1; prompts wakefulness, counters cataplexy in mice.Formula:C33H39Cl2N5O5SColor and Shape:SolidMolecular weight:688.67LY223982
CAS:LY223982 is an effective and specific inhibitor of the leukotriene B4 receptor (IC50: 13.2 nM). It also can against [3H]LTB4 binding to LTB4 receptor.Formula:C30H30O7Purity:99.86%Color and Shape:SolidMolecular weight:502.56MK-761 TFA
MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.Formula:C15H20F3N3O4Color and Shape:SolidMolecular weight:363.332GR79236
CAS:GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Formula:C15H21N5O5Color and Shape:SolidMolecular weight:351.36Tiapride-d3
Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.Formula:C15H21D3N2O4SColor and Shape:SolidMolecular weight:331.45Allura Red AC (Standard)
CAS:Allura Red AC (Standard) is the standard substance of Allura Red AC, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Allura Red AC (CI 16035) is a very important food azo dye used in the food, pharmaceutical, paper, cosmetic and textile industries.Allura Red AC promotes susceptibility to experimental colitis via mouse intestinal serotonin.Formula:C18H14N2Na2O8S2Color and Shape:Dark Maroon Solid PowderMolecular weight:496.42Endothelin-3 (Rat,Human) (TFA)
Endothelin-3 (Rat, Human) (TFA) is a 21-amino acid vasoactive peptide of endothelial origi, an agonist for the endothelin receptor type B (EDNRB).Formula:C123H169F3N26O35S4·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:2757.07 (free base)Fipexide hydrochloride
CAS:Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Formula:C20H22Cl2N2O4Color and Shape:SolidMolecular weight:425.31Spiroxatrine
CAS:Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.Formula:C22H25N3O3Purity:99.94%Color and Shape:SolidMolecular weight:379.45(R)-Praziquantel-d11
CAS:(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:323.47Fedovapagon
CAS:Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.Formula:C27H34N4O3Purity:99.46%Color and Shape:SolidMolecular weight:462.58SANT 2
CAS:SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.Formula:C26H26ClN3O4Purity:99.23%Color and Shape:SolidMolecular weight:479.96Cimbuterol-d9
CAS:Cimbuterol-d9 is a deuterated compound of Cimbuterol.Formula:C13H10D9N3OPurity:99.22%Color and Shape:SolidMolecular weight:242.37Calcium-Sensing Receptor Antagonists I
CAS:Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium.Formula:C23H24N2O2Color and Shape:SolidMolecular weight:360.45β2AR/M-receptor agonist-2
CAS:β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).Formula:C36H49ClN4O7SColor and Shape:SolidMolecular weight:717.31Dapagliflozin impurity
CAS:Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.Formula:C21H25ClO7Color and Shape:SolidMolecular weight:424.87SB-674042
CAS:SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is used in the treatment of depression.Formula:C24H21FN4O2SPurity:99.87% - 99.9%Color and Shape:SolidMolecular weight:448.51Diacetolol D7
CAS:Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.Formula:C16H24N2O4Purity:98%Color and Shape:SolidMolecular weight:315.42Hydroxyzine dihydrochloride-d4
CAS:Hydroxyzine dihydrochloride-d4 is a deuterated compound of Hydroxyzine dihydrochloride.Formula:C21H25D4Cl3N2O2Color and Shape:SolidMolecular weight:451.85Piribedil D8
CAS:Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.Formula:C16H18N4O2Purity:98%Color and Shape:SolidMolecular weight:306.39Setiptiline maleate
CAS:Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.Formula:C23H23NO4Purity:99.94%Color and Shape:SolidMolecular weight:377.43LUF5771
CAS:LUF5771: potent allosteric recLH & Org 43553 inhibitor, partial LH receptor activator with low efficacy.Formula:C24H23NO2Color and Shape:SolidMolecular weight:357.44SYL-4
CAS:SYL-4 is a potential P2Y12 receptor antagonist with a Ki value of 7.35 ± 1.72 for use in synthetic dyes.Formula:C20H15N3O5SPurity:95.76%Color and Shape:SoildMolecular weight:409.42Agomelatine (L(+)-Tartaric acid)
CAS:Agomelatine (L(+)-Tartaric acid) is an MT1/MT2 agonist and selective 5-HT2C antagonist, supporting melatonergic and serotonergic signaling studies in neuroscience.Formula:C19H23NO8Purity:99.79%Color and Shape:SolidMolecular weight:393.39SB-277011 hydrochloride
CAS:SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.Formula:C28H31ClN4OPurity:98.54%Color and Shape:SolidMolecular weight:475.03Cefaclor
CAS:Cefaclor (Panoral) is a cephalosporin antibiotic.Formula:C15H14ClN3O4SPurity:99.03% - 99.98%Color and Shape:SolidMolecular weight:367.81Lecirelin
CAS:Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.Formula:C59H84N16O12Color and Shape:SolidMolecular weight:1209.4Nefazodone
CAS:Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.Formula:C25H32ClN5O2Purity:99.85%Color and Shape:White To Off-White Crystalline PowderMolecular weight:470.01Ref: TM-T21451
2mg42.00€5mg60.00€10mg87.00€25mg177.00€50mg276.00€100mg422.00€200mg604.00€1mL*10mM (DMSO)95.00€Zilpaterol-d7
CAS:Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.Formula:C14H12D7N3O2Color and Shape:SolidMolecular weight:268.36Haloperidol (D4')
CAS:Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.Formula:C21H23ClFNO2Purity:98%Color and Shape:SolidMolecular weight:379.89Nadolol-d9
CAS:Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.
Formula:C17H27NO4Purity:98%Color and Shape:SolidMolecular weight:318.46Lanreotide
CAS:Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Formula:C54H69N11O10S2Color and Shape:SolidMolecular weight:1096.32Pimozide-d4
CAS:Pimozide D4 is a deuterium labeled Pimozide.Formula:C28H29F2N3OPurity:98%Color and Shape:SolidMolecular weight:465.57ST-836 hydrochloride
CAS:ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .Formula:C23H35ClN4OSPurity:98%Color and Shape:SolidMolecular weight:451.07(S)-ZINC-3573
CAS:(S)-ZINC 3573 is a negative control for (R)-ZINC 3573. (S)-ZINC 3573 displays no activity at MRGPRX2 at concentrations below 100 μM.Formula:C18H21N5Color and Shape:SolidMolecular weight:307.401L-798106
CAS:L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.Formula:C27H22BrNO4SPurity:98.97%Color and Shape:SolidMolecular weight:536.44Sumatriptan
CAS:Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.Formula:C14H21N3O2SPurity:99.93%Color and Shape:White To Off-White Crystalline PowderMolecular weight:295.4SB-649868
CAS:SB-649868 (GSK649868) is a potent and selective orally active antagonist of orexin(pKi =9.4 and 9.5 at the OX1 and OX2 receptor, respectively).Formula:C26H24FN3O3SPurity:99.53%Color and Shape:SolidMolecular weight:477.55Ref: TM-T5498
2mg37.00€5mg74.00€10mg116.00€25mg239.00€50mg386.00€100mg620.00€200mg832.00€1mL*10mM (DMSO)90.00€
