GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(993 products)
- Adenosine Receptor(246 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(212 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(182 products)
- Hedgehog/Smoothened(47 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(310 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5745 products of "GPCR/G-Protein"
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Methyldopa
CAS:Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFormula:C10H13NO4Purity:98.95% - 99.86%Color and Shape:Less Or Almost Colorless Crystals Or White To Yellowish-White FineMolecular weight:211.21Diphenylpyraline hydrochloride
CAS:Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.Formula:C19H23NO·HClPurity:98.72%Color and Shape:SolidMolecular weight:317.85JHU 75528
CAS:JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can be used to study the cannabinoid system in schizophrenic patients.Formula:C23H21Cl2N5O2Purity:99.79%Color and Shape:SolidMolecular weight:470.35Amiselimod hydrochloride
CAS:<p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>Formula:C19H31ClF3NO3Purity:99.55%Color and Shape:SolidMolecular weight:413.9Alverine citrate
CAS:<p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>Formula:C26H35NO7Purity:98.53% - 99.43%Color and Shape:CoaMolecular weight:473.57Terfenadine
CAS:Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Formula:C32H41NO2Purity:98.76% - 99.75%Color and Shape:SolidMolecular weight:471.67Filorexant
CAS:Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).Formula:C24H25FN4O2Purity:98.88%Color and Shape:SolidMolecular weight:420.48CYM 50769
CAS:<p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>Formula:C24H17ClN2O3Purity:98% - 99.08%Color and Shape:SolidMolecular weight:416.86Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formula:C9H10Cl3N3Purity:99.16% - 99.86%Color and Shape:SolidMolecular weight:266.55Triflupromazine hydrochloride
CAS:Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.Formula:C18H20ClF3N2SPurity:99.76% - 99.82%Color and Shape:CrystalsMolecular weight:388.88Tropisetron hydrochloride
CAS:<p>Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.</p>Formula:C17H21ClN2O2Purity:99.72% - 99.83%Color and Shape:SolidMolecular weight:320.82Naluzotan hydrochloride
CAS:<p>Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.</p>Formula:C23H39ClN4O3SPurity:99.96%Color and Shape:SolidMolecular weight:487.1Ondansetron hydrochloride dihydrate
CAS:<p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>Formula:C18H19N3O·HCl·2H2OPurity:99.92%Color and Shape:White Crystal PowderMolecular weight:365.86Rimonabant
CAS:<p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>Formula:C22H21Cl3N4OPurity:98% - 99.91%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:463.79Antazoline hydrochloride
CAS:Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenousFormula:C17H19N3·HClPurity:98% - 99.53%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:301.82Ticlopidine hydrochloride
CAS:<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Formula:C14H15Cl2NSPurity:99.85% - >99.99%Color and Shape:White PowderMolecular weight:300.25Proglumide
CAS:Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal motility.Formula:C18H26N2O4Purity:99.4% - 99.45%Color and Shape:White Crystalline PowderMolecular weight:334.41Alosetron hydrochloride
CAS:Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.Formula:C17H19ClN4OPurity:99.90%Color and Shape:Off-White PowderMolecular weight:330.81Trazodone hydrochloride
CAS:<p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>Formula:C19H23Cl2N5OPurity:99.5% - 99.52%Color and Shape:SolidMolecular weight:408.33Seganserin
CAS:<p>Seganserin, a 5-HT2 antagonist, negates fluoxetine and quipazine's effects on hyperphagia, depression, and pain.</p>Formula:C29H27F2N3OPurity:99.22%Color and Shape:SolidMolecular weight:471.54
