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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5938 products of "GPCR/G-Protein"

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  • Pamabrom

    CAS:
    Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.
    Formula:C11H18BrN5O3
    Purity:99.84% - >99.99%
    Color and Shape:Coa
    Molecular weight:348.2
  • Atomoxetine hydrochloride

    CAS:
    Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.
    Formula:C17H22ClNO
    Purity:99.86%
    Color and Shape:White Solid
    Molecular weight:291.82
  • Acebutolol hydrochloride

    CAS:
    <p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension &amp; ventricular arrhythmias.</p>
    Formula:C18H29ClN2O4
    Purity:99.92% - >99.99%
    Color and Shape:White Or Slightly Off-White Crystalline Powder Solid
    Molecular weight:372.89
  • Ezlopitant

    CAS:
    <p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>
    Formula:C31H38N2O
    Purity:97.49%
    Color and Shape:Solid
    Molecular weight:454.65
  • Agomelatine

    CAS:
    Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.
    Formula:C15H17NO2
    Purity:99.92%
    Color and Shape:White Solid
    Molecular weight:243.3
  • Metoclopramide hydrochloride

    CAS:
    Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.
    Formula:C14H22ClN3O2·HCl
    Purity:99.99%
    Color and Shape:White To Off-White Powder
    Molecular weight:336.26
  • Doxylamine succinate

    CAS:
    Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.
    Formula:C21H28N2O5
    Purity:99.61%
    Color and Shape:5 1 (Ntp 1992)
    Molecular weight:388.46
  • Ziprasidone hydrochloride monohydrate

    CAS:
    Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic
    Formula:C21H21ClN4OS·HCl·H2O
    Purity:98% - 99.83%
    Color and Shape:Off-White Powder
    Molecular weight:467.12
  • Traxanox

    CAS:
    Traxanox: oral diuretic, boosts phagocytosis in mice/rats, reverses antibody production inhibition in BALB/c mice.
    Formula:C13H6ClN5O2
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:299.67
  • YT 146

    CAS:
    YT 146 is a biochemical.
    Formula:C18H25N5O4
    Purity:98.81% - 99.25%
    Color and Shape:Solid
    Molecular weight:375.42
  • Tolamolol

    CAS:
    Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in the
    Formula:C19H24N2O4
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:344.4
  • Tolazoline hydrochloride

    CAS:
    Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary
    Formula:C10H13ClN2
    Purity:99.67%
    Color and Shape:Pale Yellow Crystalline Solid
    Molecular weight:196.68
  • Lamotrigine

    CAS:
    Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.
    Formula:C9H7Cl2N5
    Purity:99.76% - 99.95%
    Color and Shape:White To Pale Cream-Colored Powder Crystals From Isopropanol Solid
    Molecular weight:256.09
  • ONC206

    CAS:
    ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and
    Formula:C23H22F2N4O
    Purity:99.38% - 99.81%
    Color and Shape:Solid
    Molecular weight:408.44
  • UCM-1306

    CAS:
    <p>UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.</p>
    Formula:C14H14FNO2S
    Purity:99.98%
    Color and Shape:Soild
    Molecular weight:279.33
  • Balovaptan

    CAS:
    Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.
    Formula:C22H24ClN5O
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:409.91
  • ML604086

    CAS:
    ML604086 suppresses CCL1 mediated chemotaxis and enhances intracellular Ca2 concentrations.
    Formula:C27H32N4O4S
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:508.63
  • (-)-GSK598809 hydrochloride

    CAS:
    <p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>
    Formula:C22H24ClF4N5OS
    Purity:98.36%
    Color and Shape:Soild
    Molecular weight:517.97
  • Tiapride hydrochloride

    CAS:
    <p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>
    Formula:C15H24N2O4S·HCl
    Purity:99.4% - 99.77%
    Color and Shape:Solid
    Molecular weight:364.89
  • GR 103691

    CAS:
    GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).
    Formula:C30H35N3O3
    Purity:98.94% - 99.29%
    Color and Shape:Solid
    Molecular weight:485.62