GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(993 products)
- Adenosine Receptor(246 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(212 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(182 products)
- Hedgehog/Smoothened(47 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(310 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5745 products of "GPCR/G-Protein"
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Indacaterol maleate
CAS:<p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>Formula:C28H32N2O7Purity:99.03% - 99.67%Color and Shape:SolidMolecular weight:508.56Linaclotide
CAS:Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.Formula:C59H79N15O21S6Purity:97.93% - 98.71%Color and Shape:SolidMolecular weight:1526.74Cinnarizine
CAS:<p>Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.</p>Formula:C26H28N2Purity:99.94%Color and Shape:SolidMolecular weight:368.51Granisetron hydrochloride
CAS:<p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>Formula:C18H25ClN4OPurity:99.88% - 99.93%Color and Shape:White To Off-White Crystalline SolidMolecular weight:348.87Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Formula:C19H26ClNO2Purity:99.35%Color and Shape:SolidMolecular weight:335.87Dynarrestin
CAS:Dynarrestin inhibits cytoplasmic dynein 1/2, preventing microtubule sliding without affecting ATP hydrolysis or ciliogenesis.Formula:C22H23F2N3O2SPurity:99.64%Color and Shape:SolidMolecular weight:431.5Dopexamine hydrochloride
CAS:Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.Formula:C22H34Cl2N2O2Purity:98.55%Color and Shape:SolidMolecular weight:429.42Monatepil 2maleate
Monatepil 2maleate is an orally active Ca2+-channel antagonist and ACAT inhibitor with alpha(1)-adrenergic receptor blocking activity and antiarrhythmic properties that inhibit vasoconstriction.Monatepil 2maleate may be used to study atherosclerosis.Formula:C32H34FN3O5SPurity:98%Color and Shape:SolidMolecular weight:591.69Brompheniramine maleate
CAS:<p>Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.</p>Formula:C16H19BrN2·C4H4O4Purity:99.80%Color and Shape:Crystal PowderMolecular weight:435.31Ciliobrevin D
CAS:Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.Formula:C17H8Cl3N3O2Purity:98.09%Color and Shape:SolidMolecular weight:392.622-Bromo-6-methoxynaphthalene
CAS:2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.Formula:C11H9BrOPurity:98.51%Color and Shape:White To Off-White PowderMolecular weight:237.09Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formula:C22H22FN3O3Purity:99.19% - 99.73%Color and Shape:SolidMolecular weight:395.43Prucalopride
CAS:<p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.</p>Formula:C18H26ClN3O3Purity:>99.99%Color and Shape:SolidMolecular weight:367.87CD80-IN-3
CAS:<p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>Formula:C17H10FN3O3Purity:98.08%Color and Shape:SolidMolecular weight:323.28Venlafaxine hydrochloride
CAS:<p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>Formula:C17H28ClNO2Purity:97.32% - 99.86%Color and Shape:White Crystalline PowderMolecular weight:313.86ML-180
CAS:<p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>Formula:C20H25ClN4O2Purity:99.74%Color and Shape:SolidMolecular weight:388.89Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formula:C18H18ClNS·HClPurity:99.76%Color and Shape:White PowderMolecular weight:352.32N6-Ethyladenosine
CAS:N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).Formula:C12H17N5O4Purity:99.96%Color and Shape:SolidMolecular weight:295.29Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Formula:C19H21N3OPurity:99.44% - 99.84%Color and Shape:SolidMolecular weight:307.39Paliperidone
CAS:<p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>Formula:C23H27FN4O3Purity:95% - 99.08%Color and Shape:Off White To Light Orange Coloured SolidMolecular weight:426.48
