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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5938 products of "GPCR/G-Protein"

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  • Procaterol hydrochloride hydrate

    CAS:
    Short-acting β2-adrenergic receptor agonist used to treat asthma.
    Formula:C32H48Cl2N4O7
    Purity:99.71% - 99.97%
    Color and Shape:Solid
    Molecular weight:671.65
  • CGP 71683 (free base)

    CAS:
    CGP 71683 (free base) is a potent and highly selective non-peptide antagonist of the NPY Y(5) receptor in the study of obesity.
    Formula:C26H29N5O2S
    Color and Shape:Solid
    Molecular weight:475.61
  • Mini Gastrin I, human acetate


    Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.
    Formula:C76H103N15O28S
    Purity:99.35% - 99.82%
    Color and Shape:Solid
    Molecular weight:1706.78
  • Moxilubant

    CAS:
    Moxilubant, a small molecule, blocks LTB4R to treat immune, skin, and joint disorders, may help in psoriasis and rheumatoid arthritis research.
    Formula:C26H37N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:455.59
  • Etelcalcetide hydrochloride

    CAS:
    Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.
    Formula:C38H73N21O10S2HCl
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1353.33
  • Adoprazine hydrochloride

    CAS:
    Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.
    Formula:C24H25ClFN3O2
    Color and Shape:Solid
    Molecular weight:441.93
  • SK609

    CAS:
    SK609: selective dopamine D3 agonist; enhances impaired paw function, corrects asymmetry in hemiparkinson rats.
    Formula:C10H14ClN
    Color and Shape:Solid
    Molecular weight:183.68
  • Valbenazine dihydrochloride

    CAS:
    Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.
    Formula:C24H40Cl2N2O4
    Color and Shape:Solid
    Molecular weight:491.49
  • Pizuglanstat

    CAS:
    Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.
    Formula:C27H36N6O4
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:508.61
  • Selexipag

    CAS:
    Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.
    Formula:C26H32N4O4S
    Purity:99.98% - >99.99%
    Color and Shape:Solid
    Molecular weight:496.62
  • Betahistine EP Impurity C

    CAS:
    Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.
    Formula:C15H19N3
    Purity:≥95%
    Color and Shape:Solid
    Molecular weight:241.33
  • Aplindore

    CAS:
    Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.
    Formula:C18H18N2O3
    Color and Shape:Solid
    Molecular weight:310.35
  • NAV-2729

    CAS:
    NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.
    Formula:C25H17ClN4O3
    Purity:98.83% - 98.91%
    Color and Shape:Solid
    Molecular weight:456.88
  • Escitalopram Oxalate

    CAS:
    <p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>
    Formula:C22H23FN2O5
    Purity:97.39% - 99.73%
    Color and Shape:White Solid
    Molecular weight:414.43
  • Methiothepin mesylate

    CAS:
    Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.
    Formula:C21H28N2O3S3
    Purity:98% - 99.92%
    Color and Shape:Solid
    Molecular weight:452.65
  • Isoetharine mesylate salt

    CAS:
    Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.
    Formula:C14H25NO6S
    Purity:99.35% - 99.75%
    Color and Shape:Solid
    Molecular weight:335.42
  • Ataciguat

    CAS:
    Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.
    Formula:C21H19Cl2N3O6S3
    Purity:99.09%
    Color and Shape:Solid
    Molecular weight:576.49
  • Dimethocaine

    CAS:
    Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.
    Formula:C16H26N2O2
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:278.39
  • Rotundine

    CAS:
    Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.
    Formula:C21H25NO4
    Purity:99.8% - 99.91%
    Color and Shape:Off-White Solid
    Molecular weight:355.43
  • N-Acetylhistamine acetate


    N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
    Formula:C9H15N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:213.23