
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,020 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(60 products)
- CXCR(157 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(442 products)
- Endothelin Receptor(83 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(32 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(322 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5938 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Procaterol hydrochloride hydrate
CAS:Short-acting β2-adrenergic receptor agonist used to treat asthma.Formula:C32H48Cl2N4O7Purity:99.71% - 99.97%Color and Shape:SolidMolecular weight:671.65CGP 71683 (free base)
CAS:CGP 71683 (free base) is a potent and highly selective non-peptide antagonist of the NPY Y(5) receptor in the study of obesity.Formula:C26H29N5O2SColor and Shape:SolidMolecular weight:475.61Mini Gastrin I, human acetate
Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.Formula:C76H103N15O28SPurity:99.35% - 99.82%Color and Shape:SolidMolecular weight:1706.78Moxilubant
CAS:Moxilubant, a small molecule, blocks LTB4R to treat immune, skin, and joint disorders, may help in psoriasis and rheumatoid arthritis research.Formula:C26H37N3O4Purity:98%Color and Shape:SolidMolecular weight:455.59Etelcalcetide hydrochloride
CAS:Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.Formula:C38H73N21O10S2HClPurity:>99.99%Color and Shape:SolidMolecular weight:1353.33Adoprazine hydrochloride
CAS:Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.Formula:C24H25ClFN3O2Color and Shape:SolidMolecular weight:441.93SK609
CAS:SK609: selective dopamine D3 agonist; enhances impaired paw function, corrects asymmetry in hemiparkinson rats.Formula:C10H14ClNColor and Shape:SolidMolecular weight:183.68Valbenazine dihydrochloride
CAS:Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.Formula:C24H40Cl2N2O4Color and Shape:SolidMolecular weight:491.49Pizuglanstat
CAS:Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.Formula:C27H36N6O4Purity:99.62%Color and Shape:SolidMolecular weight:508.61Selexipag
CAS:Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.Formula:C26H32N4O4SPurity:99.98% - >99.99%Color and Shape:SolidMolecular weight:496.62Betahistine EP Impurity C
CAS:Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formula:C15H19N3Purity:≥95%Color and Shape:SolidMolecular weight:241.33Aplindore
CAS:Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.Formula:C18H18N2O3Color and Shape:SolidMolecular weight:310.35NAV-2729
CAS:NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.Formula:C25H17ClN4O3Purity:98.83% - 98.91%Color and Shape:SolidMolecular weight:456.88Escitalopram Oxalate
CAS:<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Formula:C22H23FN2O5Purity:97.39% - 99.73%Color and Shape:White SolidMolecular weight:414.43Methiothepin mesylate
CAS:Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.Formula:C21H28N2O3S3Purity:98% - 99.92%Color and Shape:SolidMolecular weight:452.65Isoetharine mesylate salt
CAS:Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.Formula:C14H25NO6SPurity:99.35% - 99.75%Color and Shape:SolidMolecular weight:335.42Ataciguat
CAS:Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.Formula:C21H19Cl2N3O6S3Purity:99.09%Color and Shape:SolidMolecular weight:576.49Dimethocaine
CAS:Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Formula:C16H26N2O2Purity:99.52%Color and Shape:SolidMolecular weight:278.39Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formula:C21H25NO4Purity:99.8% - 99.91%Color and Shape:Off-White SolidMolecular weight:355.43N-Acetylhistamine acetate
N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.Formula:C9H15N3O3Purity:98%Color and Shape:SolidMolecular weight:213.23
