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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5962 products of "GPCR/G-Protein"

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  • LP-211
    Targetmol
    + Info

    LP-211

    CAS:
    LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.
    Formula:C30H34N4O
    Purity:98.65%
    Color and Shape:Solid
    Molecular weight:466.62

    Ref: TM-T5387

  • Oxyntomodulin acetate
    Targetmol
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    Oxyntomodulin acetate

    Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
    Purity:99.24%
    Color and Shape:Liquid
    Molecular weight:N/A

    Ref: TM-TP1976L

  • Samelisant dihydrochloride
    Targetmol
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    Samelisant dihydrochloride

    CAS:
    SUVN-G3031: H3 receptor antagonist; may treat cognitive issues, ADHD, epilepsy, sleep, obesity, schizophrenia, eating disorders, pain.
    Formula:C21H33Cl2N3O3
    Color and Shape:Solid
    Molecular weight:446.41

    Ref: TM-T34752

  • S1RA hydrochloride
    Targetmol
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    S1RA hydrochloride

    CAS:
    S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki >
    Formula:C20H24ClN3O2
    Purity:98% - 99.84%
    Color and Shape:Solid
    Molecular weight:373.87

    Ref: TM-T4229

  • Trazodone
    Targetmol
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    Trazodone

    CAS:
    Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.
    Formula:C19H22ClN5O
    Purity:99.79% - 99.92%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:371.86

    Ref: TM-T22442

  • Ciproxifan maleate
    Targetmol
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    Ciproxifan maleate

    CAS:
    <p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>
    Formula:C20H22N2O6
    Purity:99.39%
    Color and Shape:Solid
    Molecular weight:386.4

    Ref: TM-T2004

  • SBI-553
    Targetmol
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    SBI-553

    CAS:
    SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).
    Formula:C26H31FN4O2
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:450.55

    Ref: TM-T16860

  • BIM-23190 aceate
    Targetmol
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    BIM-23190 aceate

    <p>BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.</p>
    Formula:C59H83N13O14S2
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:1262.5

    Ref: TM-T39262L

  • Epinastine hydrochloride
    Targetmol
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    Epinastine hydrochloride

    CAS:
    Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
    Formula:C16H15N3·HCl
    Purity:99.26% - 99.62%
    Color and Shape:White Solid
    Molecular weight:285.77

    Ref: TM-T6488

  • RVD-Hpα acetate(1193362-76-3 free base)
    Targetmol
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    RVD-Hpα acetate(1193362-76-3 free base)

    RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.
    Formula:C67H109N19O19
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:1484.71

    Ref: TM-TP1939L1

  • Lurasidone
    Targetmol
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    Lurasidone

    CAS:
    Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6
    Formula:C28H36N4O2S
    Purity:99.78% - 99.91%
    Color and Shape:Solid
    Molecular weight:492.68

    Ref: TM-T21337

  • AZD4635
    Targetmol
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    AZD4635

    CAS:
    AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).
    Formula:C15H11ClFN5
    Purity:99.15% - 99.90%
    Color and Shape:Solid
    Molecular weight:315.73

    Ref: TM-T4265

  • AM095
    Targetmol
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    AM095

    CAS:
    AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.
    Formula:C27H23N2NaO5
    Purity:98.87%
    Color and Shape:Solid
    Molecular weight:478.47

    Ref: TM-T2000

  • Cyclopiazonic acid
    Targetmol
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    Cyclopiazonic acid

    CAS:
    Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.
    Formula:C20H20N2O3
    Purity:99.27% - 99.80%
    Color and Shape:Solid
    Molecular weight:336.38

    Ref: TM-T15027

  • BWX 46 Acetate
    Targetmol
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    BWX 46 Acetate

    BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.
    Formula:C118H190N36O30S2
    Purity:96.86%
    Color and Shape:Solid
    Molecular weight:2657.12

    Ref: TM-T21611L

  • SB756050
    Targetmol
    + Info

    SB756050

    CAS:
    SB756050 is a specific TGR5 agonist.
    Formula:C21H28N2O8S2
    Purity:98.78% - >99.99%
    Color and Shape:Solid
    Molecular weight:500.59

    Ref: TM-T4352

  • Alizapride
    Targetmol
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    Alizapride

    CAS:
    Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].
    Formula:C16H21N5O2
    Color and Shape:Solid
    Molecular weight:315.37

    Ref: TM-T60813

  • Milveterol
    Targetmol
    + Info

    Milveterol

    CAS:
    Milveterol is a long-acting β(2)-adrenoceptor agonist.
    Formula:C25H29N3O4
    Color and Shape:Solid
    Molecular weight:435.52

    Ref: TM-T68930

  • 1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
    Targetmol
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    1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID

    CAS:
    <p>1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.</p>
    Formula:C13H13NO5
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:263.25

    Ref: TM-T8913

  • Diclofensine hydrochloride
    Targetmol
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    Diclofensine hydrochloride

    CAS:
    Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。
    Formula:C17H18Cl3NO
    Purity:98.86% - 99.93%
    Color and Shape:Solid
    Molecular weight:358.69

    Ref: TM-T7745