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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5965 products of "GPCR/G-Protein"

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  • ENMD-1068 HBr

    CAS:
    ENMD-1068 HBr is a novel Proteinase-Activated Receptor 2 antagonist.
    Formula:C15H30BrN3O2
    Color and Shape:Solid
    Molecular weight:364.32
  • Paltusotine

    CAS:
    Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.
    Formula:C27H22F2N4O
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:456.49
  • JNJ-5207852

    CAS:
    JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
    Formula:C20H32N2O
    Purity:97.19%
    Color and Shape:Solid
    Molecular weight:316.48
  • ML 10302

    CAS:
    ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.
    Formula:C15H21ClN2O3
    Color and Shape:Solid
    Molecular weight:312.79
  • Moxisylyte

    CAS:
    Moxisylyte (thymoxamine) treats erectile dysfunction, Reynaud's syndrome, and reverses eye mydriasis; it's an α1-adrenergic blocker.
    Formula:C16H25NO3
    Color and Shape:Solid
    Molecular weight:279.37
  • SLF1081851 TFA

    CAS:
    SLF1081851 (TFA) inhibits Spns2, IC50 at 1.93 μM for S1P release, crucial for development and immunity.
    Formula:C23H34F3N3O3
    Color and Shape:Solid
    Molecular weight:457.538
  • Bunazosin

    CAS:
    Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].
    Formula:C19H27N5O3
    Color and Shape:Solid
    Molecular weight:373.45
  • Haloperidol hydrochloride

    CAS:
    Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.
    Formula:C21H24Cl2FNO2
    Color and Shape:Solid
    Molecular weight:412.33
  • Dimethocaine

    CAS:
    Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.
    Formula:C16H26N2O2
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:278.39
  • Ataciguat

    CAS:
    Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.
    Formula:C21H19Cl2N3O6S3
    Purity:99.09%
    Color and Shape:Solid
    Molecular weight:576.49
  • Isoetharine mesylate salt

    CAS:
    Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.
    Formula:C14H25NO6S
    Purity:99.35% - 99.75%
    Color and Shape:Solid
    Molecular weight:335.42
  • Isoxsuprine Free Base

    CAS:
    Isoxsuprine Free Base relaxes uterine/vascular muscles, dilates arteries, treats peripheral vascular disease, and premature labor.
    Formula:C18H23NO3
    Color and Shape:Solid
    Molecular weight:301.38
  • Pemirolast

    CAS:
    Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.
    Formula:C10H8N6O
    Color and Shape:Solid
    Molecular weight:228.21
  • H4 Receptor antagonist 1

    CAS:
    H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
    Formula:C16H17ClN4O
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:316.79
  • Fabomotizole

    CAS:
    Fabomotizole (Obenoxazine) is an anxiolytic drug; produces anxiolytic and neuroprotective effects without any sedative or muscle relaxant actions.
    Formula:C15H21N3O2S
    Purity:99.4%
    Color and Shape:Solid
    Molecular weight:307.41
  • N-Cbz-DL-tryptophan

    CAS:
    N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.
    Formula:C19H18N2O4
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:338.36
  • Ganirelix Acetate

    CAS:
    Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
    Formula:C82H117ClN18O15
    Purity:96.05%
    Color and Shape:Solid
    Molecular weight:1630.4
  • RU 24969 free base

    CAS:
    <p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>
    Formula:C14H16N2O
    Purity:97.38%
    Color and Shape:Solid
    Molecular weight:228.29
  • BD 1008 dihydrobromide

    CAS:
    <p>BD 1008 dihydrobromide: selective σ1 receptor antagonist (Ki=2 nM), high σ1 and moderate σ2 affinity.</p>
    Formula:C15H24Br2Cl2N2
    Purity:97.81%
    Color and Shape:Solid
    Molecular weight:463.08
  • Lys-[Des-Arg9]Bradykinin,TFA


    Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2
    Formula:C54H75F6N13O15
    Purity:97.35%
    Color and Shape:Solid
    Molecular weight:1260.24