
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(441 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5965 products of "GPCR/G-Protein"
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ENMD-1068 HBr
CAS:ENMD-1068 HBr is a novel Proteinase-Activated Receptor 2 antagonist.Formula:C15H30BrN3O2Color and Shape:SolidMolecular weight:364.32Paltusotine
CAS:Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Formula:C27H22F2N4OPurity:99.91%Color and Shape:SolidMolecular weight:456.49JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Formula:C20H32N2OPurity:97.19%Color and Shape:SolidMolecular weight:316.48ML 10302
CAS:ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.Formula:C15H21ClN2O3Color and Shape:SolidMolecular weight:312.79Moxisylyte
CAS:Moxisylyte (thymoxamine) treats erectile dysfunction, Reynaud's syndrome, and reverses eye mydriasis; it's an α1-adrenergic blocker.Formula:C16H25NO3Color and Shape:SolidMolecular weight:279.37SLF1081851 TFA
CAS:SLF1081851 (TFA) inhibits Spns2, IC50 at 1.93 μM for S1P release, crucial for development and immunity.Formula:C23H34F3N3O3Color and Shape:SolidMolecular weight:457.538Bunazosin
CAS:Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].Formula:C19H27N5O3Color and Shape:SolidMolecular weight:373.45Haloperidol hydrochloride
CAS:Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.Formula:C21H24Cl2FNO2Color and Shape:SolidMolecular weight:412.33Dimethocaine
CAS:Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Formula:C16H26N2O2Purity:99.52%Color and Shape:SolidMolecular weight:278.39Ataciguat
CAS:Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.Formula:C21H19Cl2N3O6S3Purity:99.09%Color and Shape:SolidMolecular weight:576.49Isoetharine mesylate salt
CAS:Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.Formula:C14H25NO6SPurity:99.35% - 99.75%Color and Shape:SolidMolecular weight:335.42Isoxsuprine Free Base
CAS:Isoxsuprine Free Base relaxes uterine/vascular muscles, dilates arteries, treats peripheral vascular disease, and premature labor.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formula:C10H8N6OColor and Shape:SolidMolecular weight:228.21H4 Receptor antagonist 1
CAS:H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formula:C16H17ClN4OPurity:98.81%Color and Shape:SolidMolecular weight:316.79Fabomotizole
CAS:Fabomotizole (Obenoxazine) is an anxiolytic drug; produces anxiolytic and neuroprotective effects without any sedative or muscle relaxant actions.Formula:C15H21N3O2SPurity:99.4%Color and Shape:SolidMolecular weight:307.41N-Cbz-DL-tryptophan
CAS:N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.Formula:C19H18N2O4Purity:99.97%Color and Shape:SolidMolecular weight:338.36Ganirelix Acetate
CAS:Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFormula:C82H117ClN18O15Purity:96.05%Color and Shape:SolidMolecular weight:1630.4RU 24969 free base
CAS:<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Formula:C14H16N2OPurity:97.38%Color and Shape:SolidMolecular weight:228.29BD 1008 dihydrobromide
CAS:<p>BD 1008 dihydrobromide: selective σ1 receptor antagonist (Ki=2 nM), high σ1 and moderate σ2 affinity.</p>Formula:C15H24Br2Cl2N2Purity:97.81%Color and Shape:SolidMolecular weight:463.08Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2Formula:C54H75F6N13O15Purity:97.35%Color and Shape:SolidMolecular weight:1260.24
