GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,025 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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11-deoxy Prostaglandin E2
CAS:11-deoxy PGE2 is a synthetic PGE2 analog, a potent bronchoconstrictor, 5-30x stronger than PGF2α on human respiratory muscles.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47Dabelotine, (R)-
CAS:Dabelotine, (R)- is the R-isomer of Dabelotine. Dabelotine is an adrenergic agonist used in the study of dementia.Formula:C15H22N2O2Color and Shape:SolidMolecular weight:262.3516-phenoxy tetranor Prostaglandin F2α
CAS:16-phenoxy PGF2α is a metabolically stable analog of PGF2α. It binds to the FP receptor on ovine luteal cells with much greater affinity (440%) than PGF2α.Formula:C22H30O6Color and Shape:SolidMolecular weight:390.47GR 94800
CAS:Potent and selective tachykinin NK2 receptor antagonistFormula:C49H61N9O8Purity:98%Color and Shape:SolidMolecular weight:904.0824-Hydroxy MET
CAS:4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.Formula:C13H18N2OColor and Shape:SolidMolecular weight:218.3PSB 0777 ammonium salt
CAS:adenosine A2A receptor full agonistFormula:C18H24N6O7S2Purity:98%Color and Shape:SolidMolecular weight:500.55des-Gln14-Ghrelin
CAS:Endogenous rat ghrelin gene variant binds GHS-R1a; strong Ca2+ release (EC50=2.4 nM); boosts GH secretion in vivo.Formula:C142H237N43O40Purity:98%Color and Shape:SolidMolecular weight:3186.7GRK-IN-1
CAS:4-Amino-5-(bromomethyl)-2-methylpyrimidine used in vitamin B1 analogs and esters synthesis.
Formula:C6H10Br3N3Color and Shape:SolidMolecular weight:363.879RFRP-1(human)
CAS:Endogenous NPFF agonist with EC50 of 0.0011 nM (NPFF2) and 29 nM (NPFF1); reduces cardiac function and raises prolactin in rats. GnIH homolog.Formula:C67H101N19O14SPurity:98%Color and Shape:SolidMolecular weight:1428.72Eloralintide sodium
Eloralintide sodium (LY-3841136 sodium) is an AMYR (amylin receptor) agonist applicable for studying type 2 diabetes and obesity.Formula:C201H319N49O65S2·xNaPurity:98.66%Color and Shape:SolidMolecular weight:4526.1 (free base)Tienoxolol FA
Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.Formula:C22H30N2O7SPurity:97.05% - 98.53%Color and Shape:SoildMolecular weight:466.551a,1b-dihomo Prostaglandin E1
CAS:1a,1b-dihomo Prostaglandin E1 is a class of prostaglandin compounds.Formula:C22H38O5Color and Shape:SolidMolecular weight:382.541Enuvaptan
CAS:Enuvaptan is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.Formula:C21H15ClF6N8O3Color and Shape:SolidMolecular weight:576.84Pentagastrin meglumine
CAS:Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.Formula:C44H66N8O14SColor and Shape:SolidMolecular weight:963.11GLP-1R agonist 15
CAS:GLP-1R agonist 15 (Compound 101) is a GLP-1 receptor agonist [1] .Formula:C46H47FN8O7SColor and Shape:SolidMolecular weight:874.98Protease-Activated Receptor-1 antagonist 2
CAS:Orally active PAR-1 antagonist with 7 nM IC50; potential for CVD research.Formula:C24H23F2N3O2Color and Shape:SolidMolecular weight:423.46Albenatide
CAS:Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.
Formula:C26H47N7O9SPurity:98%Color and Shape:SolidMolecular weight:633.76(−)-6α-hydroxy Cannabidiol
CAS:(−)-6α-Hydroxy Cannabidiol, an analytical reference standard and a phytocannabinoid metabolite, serves primarily as a metabolite of cannabidiol (CBD). This product is designed for use in research and forensic applications.Formula:C21H30O3Color and Shape:SolidMolecular weight:330.46NSC380324
NSC380324 is a P2Y12 receptor antagonist with antiplatelet properties, which can be employed in research on atherosclerotic cardiovascular diseases.Formula:C31H24N4O4Color and Shape:SolidMolecular weight:516.55TAK-615
CAS:TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of LPA1 receptors.Formula:C25H22FNO4Purity:99.73%Color and Shape:SolidMolecular weight:419.44Ref: TM-T9699
1mg72.00€5mg160.00€1mL*10mM (DMSO)172.00€10mg245.00€25mg405.00€50mg572.00€100mg772.00€500mg1,539.00€
