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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • Palonosetron hydrochloride

    CAS:
    <p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>
    Formula:C19H24N2O·HCl
    Purity:99.84% - 99.92%
    Color and Shape:White Solid
    Molecular weight:332.87
  • Levodropropizine

    CAS:
    <p>Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.</p>
    Formula:C13H20N2O2
    Purity:99.87% - 99.93%
    Color and Shape:White Or Off White Crystalline Powder
    Molecular weight:236.31
  • Dimenhydrinate

    CAS:
    Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.
    Formula:C24H28ClN5O3
    Purity:99.57% - 99.77%
    Color and Shape:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Molecular weight:469.96
  • Clonidine hydrochloride

    CAS:
    Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
    Formula:C9H10Cl3N3
    Purity:99.16% - 99.86%
    Color and Shape:Solid
    Molecular weight:266.55
  • Dexpramipexole dihydrochloride

    CAS:
    <p>Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine</p>
    Formula:C10H19Cl2N3S
    Purity:99.75% - 99.88%
    Color and Shape:Solid
    Molecular weight:284.25
  • Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Formula:C22H21Cl3N4O
    Purity:98% - 99.91%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:463.79
  • KGA-2727

    CAS:
    <p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>
    Formula:C26H40N4O8
    Purity:98.46%
    Color and Shape:Solid
    Molecular weight:536.62
  • Cetirizine dihydrochloride

    CAS:
    Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.
    Formula:C21H27Cl3N2O3
    Purity:99.4% - 99.97%
    Color and Shape:Solid
    Molecular weight:461.81
  • Alverine citrate

    CAS:
    <p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>
    Formula:C26H35NO7
    Purity:98.53% - 99.43%
    Color and Shape:Coa
    Molecular weight:473.57
  • Promazine hydrochloride

    CAS:
    Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.
    Formula:C17H21ClN2S
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:320.88
  • Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Formula:C19H25F3N2O6
    Purity:99.92% - 99.94%
    Color and Shape:White Crystalline Powder
    Molecular weight:434.41
  • Silodosin

    CAS:
    Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
    Formula:C25H32F3N3O4
    Purity:99.282% - 99.76%
    Color and Shape:Colorless To Pink Solid
    Molecular weight:495.53
  • Metaproterenol hemisulfate

    CAS:
    <p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>
    Formula:C11H17NO3·5H2O4S
    Purity:98.53% - 99.74%
    Color and Shape:Solid
    Molecular weight:260.3
  • Cyproheptadine hydrochloride sesquihydrate

    CAS:
    <p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>
    Formula:C21H24ClNO
    Purity:99.77% - >99.99%
    Color and Shape:White To Slightly Yellowish Crystalline Solid
    Molecular weight:341.88
  • Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Formula:C28H32N2O7
    Purity:99.03% - 99.67%
    Color and Shape:Solid
    Molecular weight:508.56
  • 2-Bromo-6-methoxynaphthalene

    CAS:
    <p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>
    Formula:C11H9BrO
    Purity:98.51%
    Color and Shape:White To Off-White Powder
    Molecular weight:237.09
  • Terlipressin Acetate

    CAS:
    <p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>
    Formula:C56H82N16O19S2
    Purity:98.50% - 99.69%
    Color and Shape:Solid
    Molecular weight:1347.5
  • Dopexamine hydrochloride

    CAS:
    <p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>
    Formula:C22H34Cl2N2O2
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:429.42
  • Ketanserin

    CAS:
    Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.
    Formula:C22H22FN3O3
    Purity:99.19% - 99.73%
    Color and Shape:Solid
    Molecular weight:395.43
  • Glycerol phenylbutyrate

    CAS:
    Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).
    Formula:C33H38O6
    Purity:98.54% - 99.74%
    Color and Shape:Solid
    Molecular weight:530.65