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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • ML-180
    Targetmol
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    ML-180

    CAS:
    <p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>
    Formula:C20H25ClN4O2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:388.89

    Ref: TM-T12075

  • PF-06882961
    Targetmol
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    PF-06882961

    CAS:
    PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Formula:C31H30FN5O4
    Purity:97.19% - 99.56%
    Color and Shape:Solid
    Molecular weight:555.6

    Ref: TM-T12431

  • Fluparoxan hydrochloride
    Targetmol
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    Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H11ClFNO2
    Purity:99.98%
    Color and Shape:Soild
    Molecular weight:231.65

    Ref: TM-T77565

  • Phenothiazine
    Targetmol
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    Phenothiazine

    CAS:
    <p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>
    Formula:C12H9NS
    Purity:99.95%
    Color and Shape:Yellow Solid Pellets
    Molecular weight:199.27

    Ref: TM-T0776

  • JNJ-18038683
    Targetmol
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    JNJ-18038683

    CAS:
    <p>JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.</p>
    Formula:C26H28ClN3O7
    Purity:97.29%
    Color and Shape:Solid
    Molecular weight:529.97

    Ref: TM-T11720

  • Desipramine hydrochloride
    Targetmol
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    Desipramine hydrochloride

    CAS:
    Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.
    Formula:C18H23ClN2
    Purity:99.58% - 99.94%
    Color and Shape:White To Off-White Powder
    Molecular weight:302.842

    Ref: TM-T0991

  • Levosulpiride
    Targetmol
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    Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Formula:C15H23N3O4S
    Purity:98.20% - 99.88%
    Color and Shape:White Crystalline Powder
    Molecular weight:341.43

    Ref: TM-T1211

  • Zolmitriptan
    Targetmol
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    Zolmitriptan

    CAS:
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Formula:C16H21N3O2
    Purity:99.69% - 99.91%
    Color and Shape:White Or Kind Of White Powder
    Molecular weight:287.36

    Ref: TM-T1092

  • PF429242 dihydrochloride
    Targetmol
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    PF429242 dihydrochloride

    CAS:
    <p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>
    Formula:C25H37Cl2N3O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:482.49

    Ref: TM-T12437

  • Urapidil hydrochloride
    Targetmol
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    Urapidil hydrochloride

    CAS:
    <p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>
    Formula:C20H29N5O3·HCl
    Purity:99.58%
    Color and Shape:White Or Off-White Crystalline Powder
    Molecular weight:423.94

    Ref: TM-T0088

  • Cetirizine dihydrochloride
    Targetmol
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    Cetirizine dihydrochloride

    CAS:
    Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.
    Formula:C21H27Cl3N2O3
    Purity:99.4% - 99.97%
    Color and Shape:Solid
    Molecular weight:461.81

    Ref: TM-T0089

  • Ezlopitant
    Targetmol
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    Ezlopitant

    CAS:
    <p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>
    Formula:C31H38N2O
    Purity:97.49%
    Color and Shape:Solid
    Molecular weight:454.65

    Ref: TM-T68068

  • PF-610355 HCl
    Targetmol
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    PF-610355 HCl

    <p>PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.</p>
    Formula:C19H22ClN7O6
    Purity:97.97%
    Color and Shape:Solid
    Molecular weight:479.87

    Ref: TM-T16509L

  • Granisetron hydrochloride
    Targetmol
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    Granisetron hydrochloride

    CAS:
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Formula:C18H25ClN4O
    Purity:99.88% - 99.93%
    Color and Shape:White To Off-White Crystalline Solid
    Molecular weight:348.87

    Ref: TM-T1042

  • Olinciguat
    Targetmol
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    Olinciguat

    CAS:
    <p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>
    Formula:C21H16F5N7O3
    Purity:99.33% - 99.71%
    Color and Shape:Solid
    Molecular weight:509.39

    Ref: TM-T16383

  • NF-56-EJ40 hydrochloride
    Targetmol
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    NF-56-EJ40 hydrochloride

    CAS:
    <p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>
    Formula:C27H31Cl2N3O3
    Purity:99.33%
    Color and Shape:Soild
    Molecular weight:516.46

    Ref: TM-T12216L

  • Quetiapine
    Targetmol
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    Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Formula:C21H25N3O2S
    Purity:99.14% - 99.63%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:383.51

    Ref: TM-T0162

  • Naftopidil
    Targetmol
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    Naftopidil

    CAS:
    <p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>
    Formula:C24H28N2O3
    Purity:99.60% - 99.97%
    Color and Shape:White Crystalline Powder
    Molecular weight:392.49

    Ref: TM-T0696

  • Aripiprazole
    Targetmol
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    Aripiprazole

    CAS:
    Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.
    Formula:C23H27Cl2N3O2
    Purity:99.43% - 99.62%
    Color and Shape:Colourless Flake Crystalline Solid
    Molecular weight:448.39

    Ref: TM-T1566

  • (±) Clopidogrel hydrogen sulfate
    Targetmol
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    (±) Clopidogrel hydrogen sulfate

    CAS:
    <p>(±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clots</p>
    Formula:C16H16ClNO2S·H2SO4
    Purity:98.67% - 99.04%
    Color and Shape:Colorless To Light Yellow Liquid
    Molecular weight:419.9

    Ref: TM-T0182L2