GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Lisuride maleate
CAS:Lisuride maleate is a non-selective dopamine agonist and G-protein-biased 5-HT2A receptor agonist capable of blocking prolactin release.Formula:C24H30N4O5Purity:99.85%Color and Shape:SolidMolecular weight:454.52Ref: TM-T8775
1mg204.00€5mg627.00€1mL*10mM (DMSO)627.00€10mg898.00€25mg1,346.00€50mg1,745.00€100mg2,382.00€Neuropeptide W-23 (human) (TFA)
Neuropeptide W-23 (human) (NPW-23) TFA, representing the active form of Neuropeptide W, functions as an endogenous agonist for both NPBW1 (GPR7) and NPBW2 (GPR8Color and Shape:Odour SolidTecastemizole
CAS:Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.Formula:C19H21FN4Purity:99.70%Color and Shape:SolidMolecular weight:324.4Ref: TM-T26253
1mg54.00€5mg118.00€1mL*10mM (DMSO)131.00€10mg168.00€25mg288.00€50mg414.00€100mg583.00€500mg1,161.00€Acetyl-(D-Arg2)-GRF (1-29) amide (human)
CAS:Acetyl-(D-Arg2)-GRF (1-29) amide (human) serves as an antagonist to growth hormone-releasing factor (GRF) and inhibits growth hormone (GH) secretion, withFormula:C154H255N47O43SMolecular weight:3485.03Benzoquinamide hydrochloride
CAS:Benzoquinamide hydrochloride (3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride) is an antiemeticFormula:C22H33ClN2O5Purity:97.13% - 99.56%Color and Shape:SolidMolecular weight:440.96Phenoxybenzamine
CAS:Phenoxybenzamine blocks α-1 receptors, potentially reducing neuroinflammation post brain trauma.Formula:C18H22ClNOPurity:98%Color and Shape:Crystals From Petroleum Ether SolidMolecular weight:303.83Apelin-17(human, bovine)
CAS:Endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).Formula:C96H156N34O20SPurity:98%Color and Shape:SolidMolecular weight:2138.56AP 811
CAS:AP 811: Selective NPR3 antagonist, Ki of 0.48 nM, >20,000x selective over NPR1, blocks ANP-induced pump stimulation.Formula:C46H66N12O8Color and Shape:SolidMolecular weight:915.11γ-Glu-Abu TFA
Gamma-Glu-AbuTFA is the TFA salt form of Gamma-Glu-Abu. This compound acts as an agonist for the calcium sensing receptor (CaSR), activating CaSR in HEK-293 cells with an EC50 of 0.21 μM.Formula:C11H17F3N2O7Color and Shape:SolidMolecular weight:346.26LM11A-31
CAS:LM11A-31 is a useful organic compound for research related to life sciences. The catalog number is T35365 and the CAS number is 289475-77-0.Formula:C12H25N3O2Purity:98%Color and Shape:SolidMolecular weight:243.351V-0219 hydrochloride
V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.
Formula:C20H26ClF3N4O2Purity:99.97%Color and Shape:SoildMolecular weight:446.89BAY-747
CAS:BAY-747: oral, brain-penetrant sGC stimulator; improves rat memory, cognition, lowers blood pressure, aids Duchenne muscular dystrophy.Formula:C22H26F2N4O2Color and Shape:SolidMolecular weight:416.46Pirepemat
CAS:Pirepemat (IRL752) is a cortical-preferring catecholamine agent that enhances cognition. It is utilized in the investigation of Parkinson's disease.Formula:C11H13F2NOColor and Shape:SolidMolecular weight:213.22BMS-604992 dihydrochloride
CAS:BMS-604992 dihydrochloride is a selective GHSR agonist with high affinity (Ki=2.3 nM) and potent activity (EC50=0.4 nM), stimulating rodent appetite.Formula:C24H33Cl2N7O5Color and Shape:SolidMolecular weight:570.47[D-p-Cl-Phe6,Leu17]-VIP
CAS:Selective vasoactive intestinal peptide (VIP) receptor antagonist (IC50 = 125.8 nM). Displays no activity on glucagon, secretin or GRF receptors.Formula:C148H239ClN44O42Purity:98%Color and Shape:SolidMolecular weight:3342.24RF9 acetate
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.Formula:C28H42N6O5Purity:99.77%Color and Shape:SolidMolecular weight:542.67Ref: TM-T16738L
1mg65.00€5mg125.00€1mL*10mM (DMSO)167.00€10mg182.00€25mg325.00€50mg467.00€100mg645.00€200mg868.00€O-Desmethyl-N-deschlorobenzoyl Indomethacin
CAS:O-Desmethyl-N-deschlorobenzoyl indomethacin, a metabolite of indomethacin, reduces HL-60 cell viability and aids in synthesizing PGD2 receptor antagonists.Formula:C11H11NO3Color and Shape:SolidMolecular weight:205.213Fasitibant chloride
CAS:Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.
Formula:C36H49Cl3N6O6SColor and Shape:SolidMolecular weight:800.23N-0500 HCl
CAS:N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.Formula:C15H22ClNO2Purity:98.85% - 99.54%Color and Shape:SolidMolecular weight:283.79[Lys8, Lys9]-Neurotensin (8-13)
CAS:[JMV438] is a Neurotensin analog, analgesic via NTS1/NTS2 activation, with K i of 0.33 nM (hNTS1) and 0.95 nM (hNTS2).Formula:C38H64N8O8Molecular weight:760.978
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