Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
Subcategories of "Chromatin/Epigenetics"
Found 2592 products of "Chromatin/Epigenetics"
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EML 425
CAS:EML 425 is a potent and selective inhibitor of CREB binding protein (CBP)/p300 (IC50s: 2.9 and 1.1 μM, respectively).Formula:C27H24N2O4Purity:97.6%Color and Shape:SolidMolecular weight:440.49Ref: TM-T15216
5mg42.00€10mg67.00€25mg129.00€50mg187.00€100mg276.00€200mg391.00€1mL*10mM (DMSO)46.00€EBI-2511
CAS:EBI-2511 is a highly potent and orally active inhibitor of EZH2 (IC50: 6 nM in Pfeffiera cell lines).Formula:C34H48N4O4Purity:99.74%Color and Shape:SolidMolecular weight:576.77Brepocitinib P-Tosylate
CAS:Brepocitinib P-Tosylate (PF-06700841 P-Tosylate) is a potent dual inhibitor of Janus kinase 1 (JAK1) and TYK2 (IC50s of 17 nM and 23 nM, respectively).Formula:C25H29F2N7O4SPurity:99.82% - 99.97%Color and Shape:SolidMolecular weight:561.6BVT948
CAS:BVT948 is a protein tyrosine phosphatase (PTP) inhibitor.It can also inhibit lysine methyltransferase SETD8 (KMT5A) and several cytochrome P450 (P450) isoforms.Formula:C14H11NO3Purity:98.87%Color and Shape:SolidMolecular weight:241.24Ref: TM-T14841
1mg38.00€2mg49.00€5mg80.00€10mg104.00€25mg157.00€50mg210.00€100mg338.00€1mL*10mM (DMSO)88.00€Hydroxycitric acid tripotassium hydrate
CAS:Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) effectively inhibits HIF, has antioxidation, anti-inflammation, and anti-tumor effects.Formula:C6H7K3O8Purity:99.85%Color and Shape:White Solid CrystallineMolecular weight:324.41Chloramphenicol
CAS:Chloramphenicol (Chloromycetin) is a broad-spectrum antibiotic that inhibits the biosynthesis of bacterial proteins. Cost-effective and quality-assured.
Formula:C11H12Cl2N2O5Purity:99.6% - 99.84%Color and Shape:Needles Or Elongated Plates From Water Or Ethylene Dichloride SolidMolecular weight:323.13Diflunisal
CAS:Diflunisal (Dolobid) is a cyclooxygenase (COX) Inhibitor, used as an anti-inflammatory analgesic.Formula:C13H8F2O3Purity:98.92% - 99.42%Color and Shape:SolidMolecular weight:250.20Tulmimetostat
CAS:Tulmimetostat (CPI-0209) is an orally active EZH1/EZH2 inhibitor.Tulmimetostat has antitumor activity and is used in the study of ovarian cancer and advancedFormula:C28H36ClN3O5SPurity:98.04% - 99.872%Color and Shape:SolidMolecular weight:562.12Albendazole
CAS:Albendazole (SKF-62979) is used as a drug indicated for the treatment of a variety of worm infestations.Formula:C12H15N3O2SPurity:98.21% - 98.76%Color and Shape:Colorless Crystals SolidMolecular weight:265.33mTOR/HDAC-IN-1 HCl
mTOR/HDAC-IN-1 HCl，a dual inhibitor of mTOR and HDAC with potential anti-inflammatory, anti-proliferative, autophagic and apoptosis-inducing effects for cancerFormula:C23H24ClN11O3Purity:99.56%Color and Shape:SoildMolecular weight:537.96Niraparib (R-enantiomer)
CAS:Niraparib R-enantiomer (MK 4827 R-enantiomer) is an inhibitor of PARP1(IC50 of 2.4 nM).
Formula:C19H20N4OPurity:99.83%Color and Shape:SolidMolecular weight:320.39Flufenamic acid
CAS:Flufenamic acid (Arlef) is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties.Formula:C14H10F3NO2Purity:98.68%Color and Shape:White To Light Yellow Crystalline PowderMolecular weight:281.23AES-135
CAS:AES-135 is a potent HDAC inhibitor, inhibits HDAC3, HDAC6, HDAC11 (IC50s: 654, 190, and 636 nM) with anti-tumor activity.Formula:C33H29F6N3O5SPurity:97.72%Color and Shape:SolidMolecular weight:693.66Ref: TM-T10255
1mg79.00€5mg152.00€10mg250.00€25mg424.00€50mg583.00€100mg803.00€1mL*10mM (DMSO)225.00€PBIT
CAS:PBIT is a JARID1 inhibitor with IC50: 3 μM for JARID1B, 6 μM for JARID1A, and 4.9 μM for JARID1C.Formula:C14H11NOSPurity:99.61% - 99.83%Color and Shape:SolidMolecular weight:241.31Ref: TM-T16435
1mg35.00€2mg50.00€5mg75.00€10mg105.00€25mg215.00€50mg340.00€100mg550.00€200mg780.00€1mL*10mM (DMSO)84.00€Bufexamac
CAS:Bufexamac (Bufexamic acid) is a COX inhibitor for IFN-α release with anti-inflammatory, analgesic, and antipyretic action.Formula:C12H17NO3Purity:99.73%Color and Shape:Acicular CrystalMolecular weight:223.27SMARCA-BD ligand 1 for Protac
CAS:SMARCA-BD ligand 1 for Protac is a compound capable of binding to SMARCA2, the BAF ATPase subunit, based on the Protac technology for degrading SMARCA2Formula:C14H17N5OPurity:99.93%Color and Shape:SolidMolecular weight:271.32Nicotinamide riboside
CAS:Nicotinamide riboside increases NAD[+] levels and activates SIRT1 and SIRT3, culminating in enhanced oxidative metabolism and protection against high fat diet-
Formula:C11H15N2O5Purity:98.82% - 99.58%Color and Shape:SolidMolecular weight:255.25TAK-901
CAS:TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid Metaplasia, and Advanced Solid Tumors, among othersFormula:C28H32N4O3SPurity:99.02% - 99.59%Color and Shape:SolidMolecular weight:504.64Ref: TM-T2709
1mg35.00€5mg70.00€10mg104.00€25mg202.00€50mg329.00€100mg525.00€200mg748.00€1mL*10mM (DMSO)79.00€Indoprofen
CAS:Indoprofen ((±)-Indoprofe) is a non-steroidal anti-inflammatory drug.Formula:C17H15NO3Purity:99.34%Color and Shape:SolidMolecular weight:281.31N-(3-Aminopropyl)cyclohexylamine
CAS:N-(3-Aminopropyl)cyclohexylamine inhibits spermine synthase; used in neuro disease research.Formula:C9H20N2Purity:98.05% - 98.82%Color and Shape:Pale Yellow Clear LiquidMolecular weight:156.2685Curcumin
CAS:Curcumin (Natural Yellow 3) is a phenolic natural product, an inhibitor of histone acetyltransferase p300/CREB (IC50=25 μM) with specificity.Formula:C21H20O6Purity:95% - 98.98%Color and Shape:Orange-Yellow Crystal Powder; Gives Brownish-Red Color With Alkali; Light-Yellow Color With Acids Physical Description Orange-Yellow Needles (Ntp 1992)Molecular weight:368.38Delcasertib
CAS:Delcasertib (KAI-9803) is a potent and selective inhibitor of δ-protein kinase C (δPKC).Formula:C120H199N45O34S2Purity:99.96%Color and Shape:SolidMolecular weight:2880.28Ref: TM-T11740
1mg192.00€5mg485.00€10mg700.00€25mg1,063.00€50mg1,459.00€100mg1,963.00€1mL*10mM (DMSO)1,603.00€T-3775440 hydrochloride
CAS:T-3775440 hydrochloride is an irreversible inhibitor of lysine-specific histone demethylase (LSD1)(IC50 : 2.1 nM).Formula:C18H23ClN4OPurity:99.88%Color and Shape:SolidMolecular weight:346.85Ref: TM-T13055
1mg92.00€2mg118.00€5mg192.00€10mg289.00€25mg485.00€50mg663.00€100mg893.00€1mL*10mM (DMSO)212.00€PT-1
CAS:PT-1 is an AMPKα1 activator that dose-dependently activates AMPK α1394, α1335, and α2398 and enhances AMPK phosphorylation.Formula:C23H16ClN3O6SPurity:99.62%Color and Shape:SolidMolecular weight:497.91MC3482
CAS:MC3482 is a specific inhibitor of sirtuin5 (SIRT5).Formula:C33H38N4O8Purity:98% - 99.90%Color and Shape:SoildMolecular weight:618.68Ref: TM-T11962
1mg50.00€2mg71.00€5mg105.00€10mg170.00€25mg268.00€50mg423.00€100mg685.00€500mg1,378.00€Abexinostat
CAS:Abexinostat (PCI-24781) is a pan-HDAC inhibitor, strongest on HDAC1; less so on HDACs 2, 3, 6, 10. Very select for HDAC8. In Phase 1/2 trials.Formula:C21H23N3O5Purity:98.19% - 98.43%Color and Shape:SolidMolecular weight:397.42PKC β pseudosubstrate acetate
PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) is a selective cell-permeable inhibitor of PKC.Purity:95.42%Color and Shape:SoildYPX-C-05
CAS:YPX-C-05, an isohydroxamic acid derivative, is an HDAC inhibitor with vasodilatory and antihypertensive activity.CAS 번호134608-84-5Formula:C21H19N3O4Purity:98.09%Color and Shape:SoildMolecular weight:377.39Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formula:C21H24ClNOPurity:99.77% - >99.99%Color and Shape:White To Slightly Yellowish Crystalline SolidMolecular weight:341.88Citric acid trilithium salt tetrahydrate
CAS:Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) , the active component of Lithium, is a medicine used in the therapy ofFormula:C6H13Li3O11Purity:99.88%Color and Shape:White Crystalline PowderMolecular weight:281.98N-Desmethyltamoxifen hydrochloride
CAS:N-Desmethyltamoxifen hydrochloride is the major tamoxifen metabolite in humans.Formula:C25H28ClNOPurity:99.15%Color and Shape:SolidMolecular weight:393.95iso-Azalansta
CAS:(2R,4S)-Azalanstat (Iso-Azalansta) is a selective heme oxygenase (HO) inhibitor that is used in the study of cardiovascular disease.Formula:C22H24ClN3O2SPurity:99.53% - 99.89%Color and Shape:SoildMolecular weight:429.96PT2399
CAS:PT2399, an oral HIF-2 inhibitor, blocks HIF-2α/1β dimerization, showing strong in vivo antitumor effects.Formula:C17H10F5NO4SPurity:98.8% - 99.45%Color and Shape:SolidMolecular weight:419.32Ref: TM-T12675L
1mg88.00€5mg212.00€10mg318.00€25mg575.00€50mg848.00€100mg1,189.00€1mL*10mM (DMSO)233.00€(R)-CR8
CAS:(R)-CR8 ((R)-Isomer) is a potent and selective CDK inhibitor.
Formula:C24H29N7OPurity:98.41%Color and Shape:SolidMolecular weight:431.53Chitosan oligosaccharide
CAS:Chitosan oligosaccharide (COS) is an oligomer of β-(1→4)-linked D-glucosamine.Formula:C12H24N2O9Purity:98%Color and Shape:SolidMolecular weight:340.327DC-05
CAS:DC-05 is an inhibitor of DNA methyltransferase 1 (DNMT1) (IC50 and a Kd: 10.3 μM and 1.09 μM, respectively).Formula:C25H25N3OPurity:98.95%Color and Shape:SolidMolecular weight:383.49Ref: TM-T15080
1mg66.00€5mg145.00€10mg236.00€25mg515.00€50mg858.00€100mg1,251.00€200mg1,684.00€1mL*10mM (DMSO)158.00€WDR5-IN-6
CAS:WDR5-IN-6 is a WDR5 inhibitor targeting the WBM locus.WDR5-IN-6 is highly synergistic with OICR-9429, a WDR5 inhibitor that targets the WIN locus.WDR5-IN-6Formula:C13H8Cl2N2O2SPurity:99.69%Color and Shape:SoildMolecular weight:327.19EHP-101
CAS:EHP-101 is a PPARγ/CB2 dual agonist with anti-inflammatory properties, inhibits fat formation, and combats diet-related obesity.Formula:C28H35NO3Purity:98.36%Color and Shape:SolidMolecular weight:433.58Ref: TM-T13289
1mg107.00€5mg227.00€10mg378.00€25mg620.00€50mg868.00€100mg1,169.00€1mL*10mM (DMSO)250.00€Hydralazine hydrochloride
CAS:Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.Formula:C8H9ClN4Purity:99.85% - 99.86%Color and Shape:Yellow Crystals White Crystalline SolidMolecular weight:196.64Diperodon hydrochloride
CAS:Diperodon hydrochloride (Diperocaine) is a local anesthetic that can be broken down by serolytic enzymes to produce local anesthetic effects.Formula:C22H28ClN3O4Purity:99.91%Color and Shape:SolidMolecular weight:433.93Nefiracetam
CAS:Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Formula:C14H18N2O2Purity:97.37%Color and Shape:White To Off-White Crystalline PowderMolecular weight:246.3Miglitol
CAS:Miglitol (BAY1099) is an alpha-Glucosidase Inhibitor with antihyperglycemic activity.Formula:C8H17NO5Purity:99.75% - 99.88%Color and Shape:White To Pale-Yellow Powder SolidMolecular weight:207.22NI-42
CAS:NI-42, a BRPFs inhibitor: IC50(BRPF1/2/3)=7.9/48/260 nM, Kd(BRPF1/2/3)=40/210/940 nM; selective for class IV BRDs.Formula:C18H15N3O3SPurity:99.18%Color and Shape:SolidMolecular weight:353.39CBP/p300-IN-3
CAS:CBP/p300-IN-3 (P300/CBP-IN-3) is an inhibitor of p300/CBP histone acetyltransferase.Formula:C24H29N7OPurity:97.38% - 98.08%Color and Shape:SolidMolecular weight:431.53Ref: TM-T12345
1mg87.00€5mg177.00€10mg295.00€25mg532.00€50mg767.00€100mg1,063.00€500mg2,115.00€1mL*10mM (DMSO)203.00€Phenelzine sulfate
CAS:Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.Formula:C8H14N2O4SPurity:98.38% - 99.83%Color and Shape:SolidMolecular weight:234.27MS31 trihydrochloride (2366264-12-0 free base)
MS31 trihydrochloride (2366264-12-0 free base) is a potent, highly affinity and selective fragment-like methyllysine reader protein spindlin 1 (SPIN1) inhibitorFormula:C20H30Cl3N3O2Purity:99.69%Color and Shape:SolidMolecular weight:450.83Ref: TM-T12111L
1mg185.00€5mg369.00€10mg542.00€25mg867.00€50mg1,153.00€100mg1,584.00€1mL*10mM (DMSO)379.00€Tinengotinib
CAS:Tinengotinib is a multikinase inhibitor that targets a series of kinases , including Aurora kinases A/B, JAK1/2, FGFR1/2/3, VEGFRs, and many other kinases.Formula:C20H19ClN6OPurity:99.05%Color and Shape:SolidMolecular weight:394.86BRM/BRG1 ATP Inhibitor-1
CAS:BRM/BRG1 ATP Inhibitor-1 is an allosteric dual Brahma homolog (BRM)/SWI/SNF related matrix-associated actin-dependent regulator of chromatin subfamily A memberFormula:C11H9F3N4O2SPurity:98.17% - 99.84%Color and Shape:SolidMolecular weight:318.27Ref: TM-T10616
1mg167.00€5mg409.00€10mg615.00€25mg1,063.00€50mg1,558.00€100mg2,187.00€1mL*10mM (DMSO)442.00€Safingol hydrochloride
CAS:Safingol hydrochloride (L-threo-dihydrosphingosine hydrochloride) is a PKC-specific inhibitor that inhibits PKC and PI3k and induces cancer cell death.Formula:C18H40ClNO2Purity:99.39% - 99.71%Color and Shape:SoildMolecular weight:337.969Acetaminophen
CAS:Acetaminophen: pain reliever, fever reducer; mild anti-inflammatory. Risks: liver, kidney damage, blood cell effects.Formula:C8H9NO2Purity:99.85% - 99.99%Color and Shape:Colourless Solid CrystallineMolecular weight:151.16BMS-986158
CAS:BMS-986158: BET inhibitor, IC50 of 6.6 nM in SCLC, 5 nM in TNBC cells.Formula:C30H33N5O2Purity:98.78%Color and Shape:SolidMolecular weight:495.62Ref: TM-T14685
1mg87.00€5mg259.00€10mg465.00€25mg745.00€50mg1,026.00€100mg1,388.00€1mL*10mM (DMSO)283.00€BRD-6929
CAS:BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.Formula:C19H17N3O2SPurity:98.01% - 99.05%Color and Shape:SolidMolecular weight:351.42Ref: TM-T10603
5mg48.00€10mg86.00€25mg166.00€50mg289.00€100mg419.00€200mg587.00€1mL*10mM (DMSO)49.00€LIN28 inhibitor LI71
CAS:LIN28 inhibitor LI71 is a potent and cell-permeable LIN28 inhibitor, which abolishes LIN28-mediated oligouridylation with an IC50 of 7 uM.Formula:C21H21NO3Purity:95.88%Color and Shape:SolidMolecular weight:335.4Ref: TM-T11850
1mg107.00€5mg255.00€10mg414.00€25mg745.00€50mg1,063.00€100mg1,459.00€1mL*10mM (DMSO)341.00€BRD 4354
CAS:BRD 4354 is an inhibitor of HDAC5 and HDAC9. For HDAC5 and HDAC9, the IC50s values are 0.85 and 1.88 μM, respectively.Formula:C21H23ClN4OPurity:99.86%Color and Shape:SolidMolecular weight:382.89Ref: TM-T10602L
1mg34.00€2mg44.00€5mg66.00€10mg92.00€25mg178.00€50mg308.00€100mg512.00€500mg1,071.00€1mL*10mM (DMSO)73.00€ODM-207
CAS:ODM-207 (BET-IN-4) is a potent BRD4 inhibitor.Formula:C22H21N3O3Purity:99.75%Color and Shape:SolidMolecular weight:375.42Ref: TM-T10521
1mg44.00€5mg92.00€10mg133.00€25mg235.00€50mg339.00€100mg480.00€200mg660.00€1mL*10mM (DMSO)90.00€Fenbendazole
CAS:Fenbendazole (Fenbendazol) is an antinematodal benzimidazole used in veterinary medicine.Formula:C15H13N3O2SPurity:99.74%Color and Shape:White To Yellowish PowderMolecular weight:299.351-Naphthohydroxamic acid
CAS:1-Naphthohydroxamic acid (Compound 2) is a potent and selective HDAC8 inhibitor with an IC50 of 14 μM, and it is more selectively for HDAC8 than class I HDAC1Formula:C11H9NO2Purity:99.19%Color and Shape:SolidMolecular weight:187.19Ref: TM-T13996
5mg33.00€10mg60.00€25mg108.00€50mg200.00€100mg299.00€200mg430.00€1mL*10mM (DMSO)38.00€SIRT-IN-2
CAS:SIRT-IN-2 is a potent SIRT1/2/3 inhibitor(IC50s of 4, 1, 7 μM, respectively).Formula:C15H21N5O3S2Purity:98.26%Color and Shape:SolidMolecular weight:383.49Ref: TM-T12919
1mg92.00€5mg215.00€10mg344.00€25mg587.00€50mg803.00€100mg1,099.00€200mg1,468.00€1mL*10mM (DMSO)236.00€A-3 hydrochloride
CAS:A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.Formula:C12H14Cl2N2O2SPurity:99.32%Color and Shape:SolidMolecular weight:321.22Ref: TM-T14069
1mg34.00€5mg63.00€10mg90.00€25mg161.00€50mg260.00€100mg416.00€500mg888.00€1mL*10mM (DMSO)95.00€Histone Acetyltransferase Inhibitor II
CAS:Histone Acetyltransferase Inhibitor II is a selective and cell permeable inhibitor of p300 histone acetyltransferase(IC50 : 5 μM).with anti-acetylase activityFormula:C20H16Br2O3Purity:97.13%Color and Shape:SolidMolecular weight:464.15Ilginatinib
CAS:Ilginatinib (NS-018) is a highly active and orally bioavailable inhibitor of JAK2.Formula:C21H20FN7Purity:98.4% - 99.01%Color and Shape:SolidMolecular weight:389.43Ref: TM-T12266
1mg64.00€5mg138.00€10mg187.00€25mg273.00€50mg393.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)133.00€Deferoxamine Mesylate
CAS:Deferoxamine Mesylate (DFOM) is an iron chelator and iron death inhibitor.Formula:C26H52N6O11SPurity:94.68% - 99.8%Color and Shape:SolidMolecular weight:656.79Ilginatinib hydrochloride
CAS:Ilginatinib hydrochloride (NS-018 hydrochloride) is a highly active and orally bioavailable inhibitor of JAK2.Formula:C21H21ClFN7Purity:99.55%Color and Shape:SolidMolecular weight:425.89Ref: TM-T12266L2
1mg70.00€5mg150.00€10mg215.00€25mg358.00€50mg517.00€100mg707.00€200mg973.00€1mL*10mM (DMSO)166.00€TRIM24/BRPF1-IN-2
CAS:TRIM24/BRPF1-IN-2 is a TRIM24/BRPF1 dual inhibitor with anticancer activity that inhibits the proliferation of prostate cancer cells.Formula:C20H22N2O4SPurity:98.69% - 99.13%Color and Shape:SoildMolecular weight:386.47FIDAS-5
CAS:FIDAS-5 is an orally active methionine adenosyltransferase 2A (MAT2A) inhibitor with an IC50 of 2.1 μM. Cost-effective and quality-assured.Formula:C15H13ClFNPurity:98.3% - 99.17%Color and Shape:SolidMolecular weight:261.72Ref: TM-T11285
1mg59.00€2mg85.00€5mg116.00€10mg187.00€25mg331.00€50mg512.00€100mg740.00€500mg1,415.00€Uzansertib phosphate
CAS:Uzansertib phosphate (INCB053914 phosphate) is an orally active, ATP-competitive inhibitor of pan-PIM kinase, inhibiting PIM1, PIM2 and PIM3.Formula:C26H29F3N5O7PPurity:99.75% - 99.79%Color and Shape:SolidMolecular weight:611.51Levetiracetam
CAS:Levetiracetam (SIB-S1) is a relatively unique anticonvulsant that is typically used in combination with other antiepileptic medications for partial onsetFormula:C8H14N2O2Purity:99.67% - 99.86%Color and Shape:White Crystalline PowderMolecular weight:170.21MS402
CAS:MS402 is a novel BD1-selective BET BrD inhibitor.Formula:C20H19ClN2O3Purity:99.72%Color and Shape:SolidMolecular weight:370.83Minocycline hydrochloride
CAS:Minocycline HCl: tetracycline antibiotic, treats bacterial infections and acne, may cause acute or chronic hepatitis.Formula:C23H28ClN3O7Purity:99.28% - >99.99%Color and Shape:Bright Yellow-Orange Amorphous Solid Crystalline YellowMolecular weight:493.94MAK683
CAS:MAK683 is an inhibitor of embryonic ectoderm development (EED) (IC50s: 59, 89, 26 nM in EED Alphascreen binding, LC-MS and ELISA assay).Formula:C20H17FN6OPurity:98.25% - 99.92%Color and Shape:SolidMolecular weight:376.39Ref: TM-T15201
1mg52.00€5mg107.00€10mg188.00€25mg411.00€50mg607.00€100mg847.00€500mg1,758.00€1mL*10mM (DMSO)95.00€A-485
CAS:A-485 is a p300/CBP histone acetyltransferase (HAT) inhibitor that inhibits p300 and CBP. A-485 has antitumor effects. Cost effective and quality assured.Formula:C25H24F4N4O5Purity:98.01% - 99.44%Color and Shape:SolidMolecular weight:536.48Ref: TM-T14073
1mg88.00€5mg159.00€10mg273.00€25mg339.00€50mg404.00€100mg698.00€1mL*10mM (DMSO)187.00€Miltefosine
CAS:Miltefosine (HePC), effective oral drug for both visceral and cutaneous leishmaniasis, in clinical trials worldwide.Formula:C21H46NO4PPurity:98% - 99.94%Color and Shape:White To Off-White PowderMolecular weight:407.57Amifostine
CAS:Amifostine (Ethyol) anhydrous is a cytoprotective agent, acts as a free radical scavenging activity.Formula:C5H15N2O3PSPurity:99.59%Color and Shape:White SolidMolecular weight:214.22L-2-Hydroxyglutaric acid disodium
CAS:L-2-Hydroxyglutaric acid disodium may affect epigenetics and contribute to renal cancer, inhibiting Mi-CK (Km 2.52 mM, Ki 11.13 mM).Formula:C5H6Na2O5Purity:99.92%Color and Shape:SolidMolecular weight:192.08ZEN-3694
CAS:ZEN-3694 (ZEN 3694) is a bromo-structural domain extra-terminal inhibitor (BETi) with activity in androgen signaling inhibitor (ASI) resistance models and canFormula:C19H19N5OPurity:98.94% - 99.76%Color and Shape:SolidMolecular weight:333.39Oltipraz
CAS:Oltipraz (RP 35972) is a synthetic dithiolethione with potential chemopreventive and anti-angiogenic properties.Formula:C8H6N2S3Purity:98.79% - 99.77%Color and Shape:SolidMolecular weight:226.34ZL0580
CAS:ZL0580 suppresses HIV by blocking Tat activation, halting transcription, and promoting repressive chromatin at the HIV promoter.Formula:C25H23F3N4O4SPurity:99.70%Color and Shape:SolidMolecular weight:532.53NU6140
CAS:NU6140 is a selective inhibitor of CDK2-cyclin A (IC50, 0.41 μM).Formula:C23H30N6O2Purity:98.33%Color and Shape:SolidMolecular weight:422.52Ref: TM-T16359
2mg39.00€5mg60.00€10mg92.00€25mg177.00€50mg285.00€100mg414.00€200mg580.00€1mL*10mM (DMSO)67.00€VTP50469
CAS:VTP50469 is a highly selective and orally active small molecule inhibitor of the Menin-MLL protein-protein interaction.Cost-effective and quality-assured.Formula:C32H47FN6O4SPurity:98.31% - 99.55%Color and Shape:SolidMolecular weight:630.82Ref: TM-T13336
1mg164.00€5mg334.00€10mg401.00€25mg560.00€50mg715.00€100mg964.00€1mL*10mM (DMSO)465.00€Glucosamine hydrochloride
CAS:Glucosamine hydrochloride (Chitosamine hydrochloride) is commonly used as a treatment for osteoarthritis, although its acceptance as a medical therapy varies.Formula:C6H13NO5·HClPurity:99.77%Color and Shape:White Solid CrystallineMolecular weight:215.63N6-Cyclohexyladenosine
CAS:N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.Formula:C16H23N5O4Purity:99.92% - 99.98%Color and Shape:SolidMolecular weight:349.38GNE-781
CAS:GNE-781: potent CBP inhibitor (IC50: 0.94 nM), also targets BRET/BRD4(1) (IC50: 6.2/5100 nM).Formula:C27H33F2N7O2Purity:99.25% - 99.64%Color and Shape:SolidMolecular weight:525.59Ref: TM-T15405
1mg138.00€5mg298.00€10mg485.00€25mg808.00€50mg1,093.00€100mg1,483.00€1mL*10mM (DMSO)343.00€SNDX-5613
CAS:Revumenib (SNDX-5613) is a potent and selective oral inhibitor of menin-KMT2A interaction.Cost-effective and quality-assured.Formula:C32H47FN6O4SPurity:99.12% - 99.74%Color and Shape:SolidMolecular weight:630.82Ref: TM-T12943
1mg73.00€2mg97.00€5mg160.00€10mg274.00€25mg542.00€50mg778.00€100mg1,074.00€1mL*10mM (DMSO)217.00€Tranylcypromine (2-PCPA) hydrochloride
CAS:Tranylcypromine (2-PCPA) HCl, a MAO inhibitor, treats major, dysthymic, and atypical depression.Formula:C9H11N·HClPurity:99.48% - 99.86%Color and Shape:SolidMolecular weight:169.66Pulrodemstat benzenesulfonate
CAS:Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally inhibitor of lysine specific demethylase-1 (LSD1) with anticancer effect.Formula:C30H29F2N5O5SPurity:97.67%Color and Shape:SolidMolecular weight:609.64Ref: TM-T11882
1mg60.00€2mg86.00€5mg124.00€10mg188.00€25mg329.00€50mg490.00€100mg710.00€1mL*10mM (DMSO)170.00€Bendazol
CAS:Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.
Formula:C14H12N2Purity:98.7% - 99.87%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:208.26A-395
CAS:A-395 blocks PRC2 (EZH2-EED-SUZ12) interactions, strongly inhibiting the complex with an IC50 of 18 nM.
Formula:C26H35FN4O2SPurity:98.43%Color and Shape:SolidMolecular weight:486.65Lin28-let-7a antagonist 1
CAS:Lin28-let-7a antagonist 1, with an IC50 of 4.03 μM for Lin28A-let-7a-1 interaction，and shows a clear antagonistic effect against the Lin28-let-7a interaction.Formula:C31H29N5O7Purity:99.44%Color and Shape:SolidMolecular weight:583.59Ref: TM-T11851
1mg96.00€5mg205.00€10mg313.00€25mg562.00€50mg845.00€100mg1,243.00€1mL*10mM (DMSO)266.00€Ilginatinib maleate
CAS:Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:C25H24FN7O4Purity:99.74% - 99.82%Color and Shape:SolidMolecular weight:505.5Delgocitinib
CAS:Delgocitinib is a potent JAK inhibitor (IC50: 2.8-58 nM), treats inflammatory diseases, and is the first topical drug for atopic dermatitis.Formula:C16H18N6OPurity:99.95%Color and Shape:SolidMolecular weight:310.35Ref: TM-T15096
1mg160.00€5mg295.00€10mg462.00€25mg879.00€50mg1,341.00€100mg1,953.00€200mg2,628.00€1mL*10mM (DMSO)330.00€5-Azacytidine
CAS:5-Azacytidine (Ladakamycin) is a cytidine nucleoside analog, a DNA methylation inhibitor with specificity.Formula:C8H12N4O5Purity:98% - 99.79%Color and Shape:Crystals From Methanol Physical Description White Crystalline Powder (Ntp 1992)Molecular weight:244.2Gusacitinib
CAS:Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 nM).Formula:C24H28N8O2Purity:98.06% - 99.94%Color and Shape:SolidMolecular weight:460.53Ref: TM-T14331
1mg39.00€5mg84.00€10mg116.00€25mg178.00€50mg333.00€100mg495.00€200mg710.00€1mL*10mM (DMSO)110.00€MAT2A inhibitor 2
CAS:MAT2A inhibitor 2 is an inhibitor of methionine adenosyltransferase 2A (MAT2A).Formula:C18H24ClN3O3Purity:99.52%Color and Shape:SolidMolecular weight:365.85Golidocitinib
CAS:Golidocitinib (AZD4205) is a selective JAK1 inhibitor (IC50: 73 nM) and weakly inhibits JAK2/JAK3 (IC50: >14.7, >30 μM).Formula:C25H31N9O2Purity:98.87% - 99.88%Color and Shape:SolidMolecular weight:489.57Centrinone
CAS:Centrinone (LCR-263) (LCR-263) is a reversible inhibitor of polo-like kinase 4 (PLK4; Ki:0.16 nM).Formula:C26H25F2N7O6S2Purity:98.76%Color and Shape:SolidMolecular weight:633.65JAK2 Inhibitor V
CAS:JAK2 Inhibitor V (JAK2 Inhibitor V Z3) is a novel specific inhibitor of Jak2, inhibiting Jak2-V617F and Jak2-WT autophosphorylation in a dose-dependent manner.Formula:C23H24N2OPurity:98.36% - 99.15%Color and Shape:SolidMolecular weight:344.45Ref: TM-T3042
2mg37.00€5mg54.00€10mg80.00€25mg148.00€50mg259.00€100mg477.00€500mg1,063.00€1mL*10mM (DMSO)59.00€MK8722
CAS:MK8722 is an effective and systemic activator of pan-AMPK.Formula:C24H20ClN3O4Purity:98.08% - 99.8800%Color and Shape:SolidMolecular weight:449.89Ref: TM-T16099
1mg34.00€2mg49.00€5mg74.00€10mg113.00€25mg215.00€50mg396.00€100mg585.00€1mL*10mM (DMSO)82.00€MS417
CAS:MS417 (GTPL7512) is an inhibitor of BET-specific BRD4(BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively), with weakFormula:C20H19ClN4O2SPurity:99.87%Color and Shape:SolidMolecular weight:414.91L002
CAS:L002 is a potent inhibitor of acetyltransferase p300 with an IC50 of 1.98 μM, blocking histone and p53 acetylation, and may treat cardiac hypertrophy.Formula:C15H15NO5SPurity:98.59%Color and Shape:SolidMolecular weight:321.35SYP-5
CAS:SYP-5 is a novel inhibitor of HIF-1, suppresses tumor cells invasion and angiogenesis.Formula:C18H16O3SPurity:98.31%Color and Shape:SolidMolecular weight:312.38
