Metabolism
Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.
Subcategories of "Metabolism"
- AhR(41 products)
- Aminopeptidase(67 products)
- CETP(18 products)
- Carbonic Anhydrase(178 products)
- Casein Kinase(130 products)
- DHFR(33 products)
- Decarboxylase(4 products)
- Dehydrogenase(271 products)
- FAAH(64 products)
- FXR(58 products)
- Factor Xa(80 products)
- Fatty Acid Synthase(33 products)
- Ferroptosis(215 products)
- GR(3 products)
- GSNOR(3 products)
- Glucokinase(54 products)
- HIF/HIF Prolyl-Hydroxylase(142 products)
- HMG-CoA Reductase(33 products)
- Hydroxylase(30 products)
- IDO(82 products)
- LDL(8 products)
- Lipase(98 products)
- Lipid(58 products)
- Lipoxygenase(124 products)
- MAO(87 products)
- MPO(2 products)
- NAMPT(36 products)
- P450(6 products)
- PAI-1(25 products)
- PDE(166 products)
- PED(1 products)
- PKM(15 products)
- PPAR(164 products)
- Phospholipase(82 products)
- ROR(42 products)
- Retinoid Receptor(29 products)
- SGK(11 products)
- Thioredoxin(12 products)
- Transferase(30 products)
- Transporter(42 products)
- UGT(4 products)
- Xanthine Oxidase (XO) Inhibitors(9 products)
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Found 8626 products of "Metabolism"
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CL 242817
CAS:<p>CL 242817 is an inhibitor of angiotensin converting enzyme (ACE).</p>Formula:C18H21NO5SColor and Shape:SolidMolecular weight:363.43(±)-γ-Tocopherol
CAS:<p>(±)-γ-Tocopherol is a form of vitamin E with antioxidant and anti-inflammatory properties.</p>Formula:C28H48O2Color and Shape:SolidMolecular weight:416.68Factor VII-IN-1
CAS:<p>Factor VII-IN-1 (example 43) is an effective Factor VII (FVII) inhibitor (IC50=1.1 μM) with anticoagulant properties.</p>Formula:C15H10BrNO3Purity:99.19%Color and Shape:SolidMolecular weight:332.15Nampt-IN-7
CAS:<p>Nampt-IN-7 (GF8) inhibits NAMPT (IC50: 7.31 μM) and kills HepG2 cells (IC50: 24.28 μM).</p>Formula:C20H21N5O3Color and Shape:SolidMolecular weight:379.41DGAT1-IN-3
CAS:<p>DGAT1-IN-3: a potent, selective DGAT-1 inhibitor (IC50: 38 nM human, 120 nM rat), oral, for obesity and dyslipidemia research.</p>Formula:C20H19F3N4O3Color and Shape:SolidMolecular weight:420.39CP-532623
CAS:<p>CP-532623, a close structural analog of Torcetrapib, is a CETP inhibitor with highly lipophilic properties. It elevates high-density lipoprotein cholesterol.</p>Formula:C27H27F9N2O3Purity:98%Color and Shape:SolidMolecular weight:598.5CD 1530
CAS:<p>CD 1530 is an ARγ agonist (Kd:150 nM) with potential anticancer activity for the study of oral carcinogenesis.</p>Formula:C27H26O3Purity:98.13%Color and Shape:SolidMolecular weight:398.49JMS-053
CAS:<p>JMS-053 is a phosphatase DUSP3 inhibitor that inhibits CDC25B and prevents VEGF from disrupting the microvascular endothelial barrier.</p>Formula:C13H8N2O2SPurity:≥98.0%Color and Shape:SolidMolecular weight:256.28Epostane
CAS:<p>Epostane is a 3β-hydroxysteroid dehydrogenase inhibitor that blocks the biosynthesis of progesterone and pregnenolone.Cost-effective and quality-assured.</p>Formula:C22H31NO3Purity:>99.99%Color and Shape:SolidMolecular weight:357.4911β-HSD1-IN-6
CAS:<p>11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs).</p>Formula:C21H19ClN4OColor and Shape:SolidMolecular weight:378.86AMP-Deoxynojirimycin
CAS:<p>AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.</p>Formula:C22H39NO5Purity:>99.99%Color and Shape:SolidMolecular weight:397.5514(S)-HDHA
CAS:<p>DHA is an ω-3 important for development and therapy for inflammation and cancer; its derivative, 14(S)-HDHA, aids in reducing inflammation.</p>Formula:C22H32O3Color and Shape:SolidMolecular weight:344.49hCAIX/XII-IN-4
CAS:<p>hCAIX/XII-IN-4 inhibits CAIX/XII with Ki: 4.5 nM (CAXII), 23.6 nM (CAIX), and >10000 nM (CAI/CAII).</p>Formula:C20H16N2O5Color and Shape:SolidMolecular weight:364.35Carbonic anhydrase inhibitor 11
CAS:<p>Potent carbonic anhydrase inhibitor VI targets CA II, IX, XII with Ki: 40, 39, 900 nM respectively.</p>Formula:C19H15F3N4O3S2Color and Shape:SolidMolecular weight:468.47PTP1B-IN-15
CAS:<p>PTP1B-IN-15 is a potent and selective protein tyrosine phosphatase 1B (PTP1B) inhibitor that has shown research potential in type II diabetes and obesity.</p>Formula:C19H17Br2NO5SColor and Shape:SolidMolecular weight:531.22(S)-Bromoenol lactone
CAS:<p>(S)-BEL, a chiral inhibitor of iPLA2β, blocks vasopressin-induced arachidonate release in A10 cells; IC50 = 2μM.</p>Formula:C16H13BrO2Color and Shape:SolidMolecular weight:317.18URB-694
CAS:<p>URB-694 is a fatty acid amide hydrolase (FAAH) inhibitor.</p>Formula:C19H21NO3Color and Shape:SolidMolecular weight:311.37Nitrefazole
CAS:<p>Nitrefazole: a 4-nitroimidazole, inhibits ALDH enzyme crucial for alcohol metabolism, has potent, durable effects.</p>Formula:C10H8N4O4Color and Shape:SolidMolecular weight:248.19DTP348
CAS:<p>DTP348: Oral carbonic anhydrase IX inhibitor & hypoxic cell radiosensitizer with sulfamide & 5-nitroimidazole components.</p>Formula:C6H11N5O4SColor and Shape:SolidMolecular weight:249.25Oxythiamine diphosphate
CAS:<p>Oxythiamine diphosphate is a competitivethiamine pyrophosphate inhibitor(Ki of 30 nM).</p>Formula:C12H17N3O8P2SPurity:98%Color and Shape:SolidMolecular weight:425.29CM39
CAS:<p>CM39 inhibits ALDH, linked to cancer stem-like cells & chemoresistance.</p>Formula:C19H15FN4OSColor and Shape:SolidMolecular weight:366.41ICI 211965
CAS:<p>ICI 211965 is a selective and orally potent of 5-Lipoxygenase (5-LPO).</p>Formula:C24H23NO2SPurity:98%Color and Shape:SolidMolecular weight:389.51SCH-42354
CAS:<p>SCH-42354: potent oral NEP inhibitor, activates ANP & leu-enkephalin, has anti-hypertensive properties, IC50s of 8.3 & 10.0 nM.</p>Formula:C16H23NO3S2Color and Shape:SolidMolecular weight:341.49CYP1B1-IN-3
CAS:<p>CYP1B1-IN-3: strong CYP1B1 inhibitor (IC50: 6.6 nM); weak on CYP1A1/CYP1A2; hinders cell migration, invasion; blocks P-gp, AKT/ERK, FAK/SRC, EMT.</p>Formula:C20H16FN3O2S2Color and Shape:SolidMolecular weight:413.49ACC1/2-IN-2
CAS:<p>PF-3: potent ACC1/2 inhibitor; IC50: 22 nM (ACC1), 48 nM (ACC2); anti-cancer research potential.</p>Formula:C24H25N3O3Color and Shape:SolidMolecular weight:403.47GSK376501A
CAS:<p>GSK376501A is a selective and effective modulator of peroxisome proliferator-activated receptor γ (PPARγ) for the study of type 2 diabetes.</p>Formula:C32H37NO6Purity:>99.99%Color and Shape:SolidMolecular weight:531.64Protizinic acid
CAS:<p>Protizinic acid is an oral NSAID with anti-inflammatory and antipyretic properties, inhibiting PLA2 at IC50 of 210μM.</p>Formula:C17H17NO3SColor and Shape:SolidMolecular weight:315.39F-1394
CAS:<p>F-1394 is an ACAT inhibitor that reduces atherosclerosis and neointimal thickening without changing serum cholesterol.</p>Formula:C33H61N3O6Color and Shape:SolidMolecular weight:595.85KCN1
CAS:<p>KCN1: a synthetic sulfonamide, nanomolar HIF inhibitor with preclinical anti-glioma and anti-pancreatic cancer effects.</p>Formula:C26H27NO5SColor and Shape:SolidMolecular weight:465.56FXR agonist 4
<p>FXR agonist 4: EC50 of 1.05μM, treats hyperlipidemia, steatosis, insulin resistance, inflammation in DIO mice, for NAFLD research.</p>Formula:C21H28ClN3OColor and Shape:SolidMolecular weight:373.92RORγt modulator 2
CAS:RORγt modulator 2 is a modulator of retinol-related orphan receptor γt (RORyt) (IC50<50 nM) and can be used in the study of RORγt-mediated diseases such as painFormula:C28H29ClN2O4SColor and Shape:SolidMolecular weight:525.06CK2-IN-6
CAS:<p>CK2-IN-6: Potent CK2 inhibitor for cancer, inflammation, pain, and immune research.</p>Formula:C19H16ClN7O2Color and Shape:SolidMolecular weight:409.83CYP3A4-IN-1
CAS:<p>CYP3A4-IN-1 is a potent inhibitor of cytochrome P450 3A4 (CYP3A4) (IC50: 0.085 μM).</p>Formula:C31H37N5O3SColor and Shape:SolidMolecular weight:559.72TK-642
CAS:<p>TK-642 is a potent and selective SHP2 inhibitor with oral activity, based on pyrazole and pyrazine structures (IC50 = 2.7 nmol/L). It effectively inhibits the proliferation of esophageal carcinoma cells and induces apoptosis, making it useful for studying esophageal cancer.</p>Formula:C17H20ClN7SColor and Shape:SolidMolecular weight:389.91PKR activator 2
CAS:PKR activator 2 is a potent activator of pyruvate kinase-R (PKR).Formula:C18H16N8OSPurity:98%Color and Shape:SolidMolecular weight:392.44BKIDC-1553
CAS:<p>BKIDC-1553, an orally active antiglycolytic agent and bumped kinase inhibitor-derived compound, has a predicted half-life of approximately 17 hours in humans. It inhibits CYP2C8 and Angiotensin Converting Enzyme, making it suitable for cancer research [1].</p>Formula:C22H23N5O2Color and Shape:SolidMolecular weight:389.45OMDM-3
CAS:<p>OMDM-3 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 16.6 μM).</p>Formula:C29H43NO3Purity:98%Color and Shape:SolidMolecular weight:453.66JNJ-42165279 dihydrochloride
CAS:<p>JNJ-42165279 (dihydrochloride) is an FAAH inhibitor with IC50 values of 70 nM for hFAAH and 313 nM for rFAAH, respectively [1].</p>Formula:C18H19Cl3F2N4O3Color and Shape:SolidMolecular weight:483.72Phosphodiesterase-IN-1
CAS:<p>Phosphodiesterase-IN-1 (Compound 7), a phosphodiesterase (PDE) inhibitor, exhibits anti-Plasmodium and antiproliferative activities. It effectively inhibits P. falciparum (strain 3D7) with an IC 50 value of 0.64 μM [1].</p>Formula:C15H15FN4OColor and Shape:SolidMolecular weight:286.3HIF-1/2α-IN-2
CAS:<p>HIF-1/2α-IN-2 is a potent inhibitor of HIF-1/2α, which effectively reduces the levels of HIF-1/2α.</p>Formula:C16H11FN4O2SColor and Shape:SolidMolecular weight:342.35IDH2R140Q-IN-1
CAS:<p>IDH2R140Q-IN-1 is a potent inhibitor of IDH2R140Q (IC50: 6.1 nM) and can be used in studies of acute myeloid leukemia.</p>Formula:C22H20F6N6Color and Shape:SolidMolecular weight:482.42FAAH-IN-5
CAS:<p>FAAH-IN-5 (Compound 7) selectively, irreversibly inhibits FAAH (IC50: 10.5 nM) with low PAMPA permeability.</p>Formula:C21H19N3O6SColor and Shape:SolidMolecular weight:441.46IDO-IN-14
CAS:<p>IDO-IN-14 is an IDO inhibitor (IC50: 0.6928 nM).</p>Formula:C23H23ClN4O2Color and Shape:SolidMolecular weight:422.917β,27-dihydroxy Cholesterol
CAS:<p>7β,27-dihydroxy Cholesterol is an oxysterol and agonist of retinoic acid receptor-related orphan receptor γ (RORγ) and RORγt.</p>Formula:C27H46O3Color and Shape:SolidMolecular weight:418.65ACC1/2-IN-1
CAS:<p>ACC1/2-IN-1 is a potent inhibitor of ACC1/2 and acts on ACC1 (IC50: 98.06 nM) and ACC2 (IC50: 29.43 nM). ACC1/2-IN-1 can be used in cancer research.</p>Formula:C34H32N4O4Color and Shape:SolidMolecular weight:560.642-TEDC
CAS:<p>2-TEDC: Potent LOX inhibitor, blocks 5-LOX, 12-LOX, 15-LOX (IC50: 0.09, 0.013, 0.5 μM); aids atherosclerosis research.</p>Formula:C16H13NO4SPurity:99.75%Color and Shape:SolidMolecular weight:315.34IDO1-IN-17
CAS:<p>IDO1-IN-17 (I-4) is an IDO1 inhibitor, with an IC 50 of 0.44 μM in hela cells .</p>Formula:C28H32BrClFN5O2Color and Shape:SolidMolecular weight:604.94Carbonic anhydrase inhibitor 13
CAS:<p>Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).</p>Formula:C17H15N5O3S2Color and Shape:SolidMolecular weight:401.46hCAIX-IN-6
CAS:<p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>Formula:C18H12N2O4SColor and Shape:SolidMolecular weight:352.36Eggmanone
CAS:<p>EGM1: potent PDE4D3 inhibitor, IC50=72 nM, 40-50x selectivity over other PDEs, activates PKA, blocks Hh.</p>Formula:C20H20N2O2S3Color and Shape:SolidMolecular weight:416.58α-Glucosidase-IN-8
CAS:<p>α-Glucosidase-IN-8 (Compound 4k) is a potent, competitive inhibitor of α-glucosidase. It displays an impressive IC50 value of 0.18 μg/mL [1].</p>Formula:C19H20FN3O2Color and Shape:SolidMolecular weight:341.38Glucokinase activator 3
CAS:<p>Glucokinase activator 3: potent GK activator, AC50=38 nM, potential for type 2 diabetes research.</p>Formula:C26H33N2O9PS2Color and Shape:SolidMolecular weight:612.65Clethodim
CAS:<p>Clethodim is a selective herbicide inhibiting acetyl-CoA carboxylase, effective on grasses with low environmental persistence and moderate toxicity to wildlife.</p>Formula:C17H26ClNO3SPurity:99.99%Color and Shape:Light Yellow LiquidMolecular weight:359.91α-Glucosidase-IN-10
CAS:<p>α-Glucosidase-IN-10 (compound 13) is a potent inhibitor of α-glucosidase (IC50: 92.7 μM). α-Glucosidase-IN-10 can be used to study type II diabetes.</p>Formula:C21H15BrN4O2SColor and Shape:SolidMolecular weight:467.34TUPS
CAS:<p>TUPS is a selective soluble epoxide hydrolase inhibitor which protects against isoprenaline-induced cardiac hypertrophy.</p>Formula:C14H18F3N3O4SColor and Shape:SolidMolecular weight:381.37AX 048
CAS:<p>Group IVA cPLA2 inhibitor AX 048 halts arachidonic acid release, preventing prostaglandin production, with XI(50) of 0.022 and ED50 of 1.2 mg/kg.</p>Formula:C22H41NO4Color and Shape:SolidMolecular weight:383.57Xanthine oxidoreductase-IN-2
CAS:<p>Xanthine oxidoreductase-IN-2 inhibits XOR with 7.2 nM IC50 and shows hypouricemic effects in mice.</p>Formula:C21H19N3O2Color and Shape:SolidMolecular weight:345.39AMG-7980
CAS:<p>AMG-7980 is a highly specific phosphodiesterase 10A ligand. It shows a good uptake in the striatum.</p>Formula:C19H22N4O2Purity:98%Color and Shape:SolidMolecular weight:338.4ATX inhibitor 11
CAS:<p>ATX inhibitor 11 blocks autotaxin (IC50: 2.7 nM), reduces fibrosis and α-SMA in mice. Useful for lung fibrosis studies.</p>Formula:C32H35N5O6Color and Shape:SolidMolecular weight:585.65UK-414,495
CAS:<p>UK-414,495 is a potent, selective inhibitor of the neutral endopeptidase, the enzyme normally serves to break down the neuropeptide VIP.</p>Formula:C16H25N3O3SColor and Shape:SolidMolecular weight:339.45BI-4924
CAS:BI-4924 is a PHGDH inhibitor that disrupts serine biosynthesis by intracellular trapping and can be used to study metabolic disorders.Formula:C21H20Cl2N2O6SPurity:99.55%Color and Shape:SolidMolecular weight:499.36mIDH1-IN-1
CAS:<p>mIDH1-IN-1 is a selective mIDH1 inhibitor (IC50: 961.5 nM), blocks 2-HG production, and hinders IDH1 mutant cell growth (IC50: 41.8 nM).</p>Formula:C25H27N3O5Color and Shape:SolidMolecular weight:449.5Enpp-1-IN-5
CAS:<p>Enpp-1-IN-5 is a potent enpp-1 inhibitor with potential in cancer and infectious disease research.</p>Formula:C17H26N6O4SColor and Shape:SolidMolecular weight:410.49GGsTop
CAS:<p>GGsTop (Nahlsgen) is a GGT inhibitor with anti-aging activity.</p>Formula:C13H18NO7PPurity:98.96%Color and Shape:SolidMolecular weight:331.26CAY10485
CAS:<p>CAY10485 blocks human ACAT-1 & ACAT-2 (IC50: 95 & 81 μM) and hinders oxidation of LDL by 91% at 2 μM, possibly impacting atherosclerosis development.</p>Formula:C27H27NO7Color and Shape:SolidMolecular weight:477.51IDO-IN-11
CAS:<p>IDO-IN-11 is an indoleamine-2,3-dioxygenase (IDO) inhibitor with IC50s of 0.18 μM (Kinase) and 0.014 μM (Hela Cell).</p>Formula:C19H23BrFN7O4SPurity:98%Color and Shape:SolidMolecular weight:544.4IACS-8968 R-enantiomer
CAS:<p>IACS-8968 R-enantiomer is the R-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).</p>Formula:C17H18F3N5O2Purity:98%Color and Shape:SolidMolecular weight:381.35SGK1 inhibitor
CAS:<p>SGK1 inhibitor targets SGK1/2 over SGK3, blocks GSK3β phosphorylation, lowers HCC1954 cell viability with BYL719, and reduces tumor growth in mice.</p>Formula:C17H12Cl2N6O2SColor and Shape:SolidMolecular weight:435.29MitoTEMPO hydrate
CAS:<p>MitoTEMPO, a mitochondria-targeted antioxidant, scavenges superoxide and alkyl radicals supporting potential therapy for mitochondrial dysfunction.</p>Formula:C29H35N2O2P·Cl·H2OColor and Shape:SolidMolecular weight:528.04Deltazinone
CAS:<p>Deltazinone selectively inhibits PDEδ with low cytotoxicity, mimicking PDEδ knockdown in human pancreatic cancer cells.</p>Formula:C27H31N5O2Purity:98%Color and Shape:SolidMolecular weight:457.57Quinethazone
CAS:<p>Quinethazone is a thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels.</p>Formula:C10H12ClN3O3SColor and Shape:Fibrous Crystals From 50% Acetone Physical Description Fibrous Crystals Or White Powder (Ntp 1992)Molecular weight:289.74sEH inhibitor-14
CAS:<p>sEH inhibitor-14, a benzoxazolone-5-urea analogue, acts as an efficient soluble Epoxide Hydrolase (sEH) inhibitor, demonstrating significant activity with an</p>Formula:C16H12F3N3O4Color and Shape:SoildMolecular weight:367.28Andolast
CAS:<p>Andolast (CR-2039) is an anti-allergic for asthma and COPD, inhibiting IgE synthesis and improving airflow.</p>Formula:C15H11N9OColor and Shape:SolidMolecular weight:333.31Oxagrelate
CAS:<p>Oxagrelate inhibits cAMP phosphodiesterase and reduces platelet aggregation by collagen and ADP.</p>Formula:C14H16N2O4Color and Shape:SolidMolecular weight:276.29PDE5-IN-4
CAS:<p>PDE5-IN-4, a phosphodiesterase 5 (PDE5) inhibitor, is utilized in research concerning acute myocardial infarction and reperfusion-related damage,</p>Formula:C21H27N5O5SColor and Shape:SolidMolecular weight:461.53JTP-4819
CAS:<p>JTP-4819: potent PEP inhibitor, may treat Alzheimer's, boosts brain peptides and acetylcholine, aiding memory.</p>Formula:C19H25N3O4Color and Shape:SolidMolecular weight:359.42AMG-221
CAS:<p>AMG-221: potent 11β-HSD1 inhibitor, lowers glucose & insulin, reduces obesity in mice.</p>Formula:C14H22N2OSPurity:98%Color and Shape:SolidMolecular weight:266.4Boc-Glu(OBzl)-OSu
CAS:<p>Boc-Glu(OBzl)-OSu can be used for the synthesis of solid phase peptides containing benzyl glutamate residues.</p>Formula:C21H26N2O8Color and Shape:SolidMolecular weight:434.44HS79
CAS:<p>HS-79, a Fasnall enantiomer, selectively inhibits FASN with an IC50 of 1.57 μM, blocking tritiated acetate lipid incorporation.</p>Formula:C19H22N4SPurity:98%Color and Shape:SolidMolecular weight:338.47Hydroxychlorodenafil
CAS:<p>Hydroxychlorodenafil is a derivative of the phosphodiesterase 5 (PDE5) inhibitor sildenafil.</p>Formula:C19H23ClN4O3Color and Shape:SolidMolecular weight:390.86Lp-PLA2-IN-3
CAS:<p>Lp-PLA2-IN-3: Potent oral inhibitor of human Lp-PLA2 with a 14 nM IC50.</p>Formula:C20H13ClF3N3O3SPurity:99.65%Color and Shape:SolidMolecular weight:467.85Sch 34826
CAS:<p>Sch 34826 is a potent, selective neutral endopeptidase inhibitor.</p>Formula:C27H34N2O7Purity:98%Color and Shape:SolidMolecular weight:498.57Glycogen phosphorylase-IN-1
CAS:<p>Glycogen phosphorylase-IN-1 is an hlGPa inhibitor that can be used in the study of type 2 diabetes and canine lupus.</p>Formula:C17H15ClF2N4O4Purity:97.98% - 98.15%Color and Shape:SolidMolecular weight:412.78sEH inhibitor-3
CAS:<p>sEH inhibitor-3 is an orally available, selective and potent inhibitor of sEH for cancer research.</p>Formula:C19H23F4N3O4Purity:98%Color and Shape:SolidMolecular weight:433.4Senazodan hydrochloride
CAS:<p>Senazodan hydrochloride (Senazodan HCl) is a Ca2+ sensitizer and phosphodiesterase 3 (PDE3) inhibitor used in the study of cardiovascular diseases.</p>Formula:C15H15ClN4OPurity:99.93%Color and Shape:SolidMolecular weight:302.76NPD-1335
CAS:<p>NPD1335: potent TbrPDEB1 inhibitor, submicromolar efficacy, low toxicity, raises cAMP, disrupts cell cycle, kills T. brucei.</p>Formula:C28H29N3O3Purity:98%Color and Shape:SolidMolecular weight:455.55BI-135585
CAS:<p>BI-135585 is an orally active, selective and potent inhibitor of human 11β-hydroxysteroid dehydrogenase-1 (HSD1) for the study of type 2 diabetes.</p>Formula:C28H32N2O4Purity:99.45% - 99.57%Color and Shape:SolidMolecular weight:460.57α-Amylase/α-Glucosidase-IN-2
CAS:α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μMFormula:C22H16ClN5Color and Shape:SolidMolecular weight:385.85D-threo-PPMP hydrochloride
CAS:<p>D-threo-PPMP inhibits GlyCer synthetase; active enantiomer; reduces MDCK cell growth by 70% at 20 μM.</p>Formula:C29H51ClN2O3Color and Shape:SolidMolecular weight:511.196-Hydroxyluteolin
CAS:<p>6-Hydroxyluteolin, a flavonoid compound extracted from Salvia amarissima Ortega, inhibits aldose reductase (AR) and has antimicrobial activity.</p>Formula:C15H10O7Purity:99.69%Color and Shape:SolidMolecular weight:302.24Xanthine oxidase-IN-5
CAS:<p>Xanthine oxidase-IN-5: oral XO inhibitor, IC50 = 0.70 μM, LE = 0.33, LLE = 3.41, reduces uric acid in rats.</p>Formula:C18H16FN3O3Color and Shape:SolidMolecular weight:341.34ICI 153110
CAS:<p>ICI 153110: Oral phosphodiesterase inhibitor for treating congestive heart failure, has inotropic, vasodilator effects.</p>Formula:C11H11N3OPurity:98%Color and Shape:SolidMolecular weight:201.22hCAIX-IN-8
CAS:<p>hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.</p>Formula:C19H16N4O6Color and Shape:SolidMolecular weight:396.35PRRSV/CD163-IN-1
CAS:<p>PRRSV/CD163-IN-1 blocks PRRSV GP2a/GP4 and CD163-SRCR5, aiding PRRS research.</p>Formula:C25H24FN5O5S2Color and Shape:SolidMolecular weight:557.62Xanthine oxidase-IN-4
CAS:<p>Xanthine oxidase-IN-4: an oral XO inhibitor with 0.039 μM IC50, useful for hyperuricemia/gout research.</p>Formula:C15H13N5O2Color and Shape:SolidMolecular weight:295.3DP00477
CAS:<p>DP00477, a potent inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1), exhibits an inhibitory concentration (IC50) of 7.0 µM.</p>Formula:C17H11ClF3N3OSColor and Shape:SolidMolecular weight:397.8PDE4-IN-11
CAS:<p>PDE4-IN-11: Potent PDE4 inhibitor with strong bronchodilatory and anti-inflammatory effects for airway disease research.</p>Formula:C21H19FN2O2Color and Shape:SolidMolecular weight:350.39ENPP1 inhibitor 43
CAS:<p>ENPP1 inhibitor 43 is a novel small molecule for cancer immunotherapy.</p>Formula:C16H18N6O3SColor and Shape:SolidMolecular weight:374.42MY33-3 hydrochloride
CAS:<p>MY33-3 HCl: Inhibits RPTPβ/ζ (IC50~0.1μM), PTP-1B (IC50~0.7μM), curbs alcohol intake, fights neuroinflammation and memory issues.</p>Formula:C16H14ClF6NS2Color and Shape:SolidMolecular weight:433.86hCAXII-IN-1
CAS:<p>hCAXII-IN-1 selectively inhibits HCA IX/XII, promising for new cancer drug development.</p>Formula:C20H17NO5Color and Shape:SolidMolecular weight:351.35
