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Metabolism

Metabolism

Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.

Subcategories of "Metabolism"

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Found 8626 products of "Metabolism"

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  • KCN1

    CAS:
    <p>KCN1: a synthetic sulfonamide, nanomolar HIF inhibitor with preclinical anti-glioma and anti-pancreatic cancer effects.</p>
    Formula:C26H27NO5S
    Color and Shape:Solid
    Molecular weight:465.56
  • LAZABEMIDE

    CAS:
    <p>Lazabemide (Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and &gt; 100 μM for MAO-B and MAO-A respectively).</p>
    Formula:C8H10ClN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:199.64
  • F-1394

    CAS:
    <p>F-1394 is an ACAT inhibitor that reduces atherosclerosis and neointimal thickening without changing serum cholesterol.</p>
    Formula:C33H61N3O6
    Color and Shape:Solid
    Molecular weight:595.85
  • CYP1B1-IN-3

    CAS:
    <p>CYP1B1-IN-3: strong CYP1B1 inhibitor (IC50: 6.6 nM); weak on CYP1A1/CYP1A2; hinders cell migration, invasion; blocks P-gp, AKT/ERK, FAK/SRC, EMT.</p>
    Formula:C20H16FN3O2S2
    Color and Shape:Solid
    Molecular weight:413.49
  • Acetyltrialanine

    CAS:
    <p>Acetyltrialanine is a dipeptide compound that binds at two sites on the Tb+3-pancreatic elastase complex and can be used as a nitrogen source.</p>
    Formula:C11H19N3O5
    Purity:99.53%
    Color and Shape:White Powder
    Molecular weight:273.29
  • JBP485

    CAS:
    <p>JBP485 is an inhibitor of renal transporters OAT1 and OAT3. JBP485 is an antihepatitis agent as a substrate for intestinal PEPT1.</p>
    Formula:C8H12N2O4
    Color and Shape:Solid
    Molecular weight:200.19
  • PGAM1-IN-1

    CAS:
    <p>PGAM1-IN-1 is an inhibitor of phosphoglycerate mutase 1 ( PGAM1 ) with an IC 50 of 6.4 μM [1].</p>
    Formula:C19H11ClFNO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.81
  • hCAIX/XII-IN-3

    CAS:
    <p>Compound 6q inhibits hCAIX/CAXII; K i : hCAI &gt;10000 nM, hCAII &gt;10000 nM, hCAIX 66.2 nM, hCAXII 4.4 nM.</p>
    Formula:C20H13F3N2O4
    Color and Shape:Solid
    Molecular weight:402.32
  • YCT529 free acid

    CAS:
    <p>YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .</p>
    Formula:C29H25NO3
    Color and Shape:Solid
    Molecular weight:435.51
  • hDHODH-IN-9

    CAS:
    <p>hDHODH-IN-9 is a potent hDHODH inhibitor, IC50=0.34 μM, toxic to MCF-7/A375 cells, promising for cancer research.</p>
    Formula:C21H21NO4
    Color and Shape:Solid
    Molecular weight:351.4
  • CM39

    CAS:
    <p>CM39 inhibits ALDH, linked to cancer stem-like cells &amp; chemoresistance.</p>
    Formula:C19H15FN4OS
    Color and Shape:Solid
    Molecular weight:366.41
  • Oxythiamine diphosphate

    CAS:
    <p>Oxythiamine diphosphate is a competitivethiamine pyrophosphate inhibitor(Ki of 30 nM).</p>
    Formula:C12H17N3O8P2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.29
  • hCAIX/XII-IN-6


    <p>hCAIX/XII-IN-6: Oral carbonic anhydrase inhibitor, targets hCA I/II/IV/IX/XII, aids rheumatoid arthritis research. Ki: 6697/2950/4093/4.1/7.7 nM.</p>
    Formula:C26H23N3O6S4
    Color and Shape:Solid
    Molecular weight:601.74
  • hCAI/II-IN-3

    CAS:
    <p>"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."</p>
    Formula:C16H18N4O4S2
    Color and Shape:Solid
    Molecular weight:394.47
  • Prolyl Endopeptidase Inhibitor 1

    CAS:
    <p>Prolyl Endopeptidase Inhibitor 1 is a potent inhibitor of prolyl endopeptidase (PEP; PE)(Ki : 15 nM) , has anti-amnesic effect.</p>
    Formula:C15H24N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:296.36
  • DTP348

    CAS:
    <p>DTP348: Oral carbonic anhydrase IX inhibitor &amp; hypoxic cell radiosensitizer with sulfamide &amp; 5-nitroimidazole components.</p>
    Formula:C6H11N5O4S
    Color and Shape:Solid
    Molecular weight:249.25
  • Sp-cAMPS

    CAS:
    <p>Rp-cAMPS TEA salt is a cAMP-dependent protein kinase (PKA) activator.</p>
    Formula:C10H12N5O5PS
    Color and Shape:Solid
    Molecular weight:345.27
  • Nitrefazole

    CAS:
    <p>Nitrefazole: a 4-nitroimidazole, inhibits ALDH enzyme crucial for alcohol metabolism, has potent, durable effects.</p>
    Formula:C10H8N4O4
    Color and Shape:Solid
    Molecular weight:248.19
  • hCAII-IN-2

    CAS:
    <p>hCAII-IN-2 inhibits human carbonic anhydrases I, II, IX, XII with Ki values of 261.4, 3.8, 19.6, 45.2 nM respectively.</p>
    Formula:C25H18ClN5O4S
    Color and Shape:Solid
    Molecular weight:519.96
  • URB-694

    CAS:
    <p>URB-694 is a fatty acid amide hydrolase (FAAH) inhibitor.</p>
    Formula:C19H21NO3
    Color and Shape:Solid
    Molecular weight:311.37
  • UKI-1

    CAS:
    <p>UKI-1 is a urokinase-type plasminogen activator system synthetic inhibitor.</p>
    Formula:C32H47N5O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:613.81
  • 11β-HSD1-IN-6

    CAS:
    <p>11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs).</p>
    Formula:C21H19ClN4O
    Color and Shape:Solid
    Molecular weight:378.86
  • CAY10761

    CAS:
    <p>CAY10761 inhibits ENPP1 (IC50: 467 μM human, 429 μM snake), mushroom tyrosinase (Ki: 1.9 μM), and urease from different sources (IC50: 0.093-&lt;0.125 mM).</p>
    Formula:C7H8N4O2S2
    Color and Shape:Solid
    Molecular weight:244.29
  • FR-221647

    CAS:
    <p>FR-221647: non-nucleoside adenosine deaminase blocker, moderate efficacy, better pharmacokinetics than EHNA/Pentostatin.</p>
    Formula:C14H17N3O2
    Color and Shape:Solid
    Molecular weight:259.3
  • JMS-053

    CAS:
    <p>JMS-053 is a phosphatase DUSP3 inhibitor that inhibits CDC25B and prevents VEGF from disrupting the microvascular endothelial barrier.</p>
    Formula:C13H8N2O2S
    Purity:≥98.0%
    Color and Shape:Solid
    Molecular weight:256.28
  • Genz-669178

    CAS:
    <p>Genz-669178 is a wild-type inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH).</p>
    Formula:C17H14N4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:322.38
  • 11β-HSD1-IN-10

    CAS:
    <p>11β-HSD1-IN-10, a potent inhibitor of 11β-HSD1 with an IC50 value of 1.8 µM for humans, is suitable for research into obesity, hyperglycemia, and cognitive</p>
    Formula:C16H10F3NO2
    Color and Shape:Solid
    Molecular weight:305.25
  • Indolapril hydrochloride

    CAS:
    <p>Indolapril hydrochloride is a nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity.</p>
    Formula:C24H35ClN2O5
    Color and Shape:Solid
    Molecular weight:467
  • (±)-γ-Tocopherol

    CAS:
    <p>(±)-γ-Tocopherol is a form of vitamin E with antioxidant and anti-inflammatory properties.</p>
    Formula:C28H48O2
    Color and Shape:Solid
    Molecular weight:416.68
  • CD 1530

    CAS:
    <p>CD 1530 is an ARγ agonist (Kd:150 nM) with potential anticancer activity for the study of oral carcinogenesis.</p>
    Formula:C27H26O3
    Purity:98.13%
    Color and Shape:Solid
    Molecular weight:398.49
  • IQA

    CAS:
    <p>IQA is a casein kinase 2 (CK2) inhibitor.</p>
    Formula:C17H12N2O3
    Color and Shape:Solid
    Molecular weight:292.29
  • Factor VII-IN-1

    CAS:
    <p>Factor VII-IN-1 (example 43) is an effective Factor VII (FVII) inhibitor (IC50=1.1 μM) with anticoagulant properties.</p>
    Formula:C15H10BrNO3
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:332.15
  • Dacisteine

    CAS:
    <p>Dacisteine (N,S-Diacetyl-L-cysteine) is an inhibitor of New Delhi metallo-beta-lactamase-1 (NDM-1, IC50 = 1000 μM).</p>
    Formula:C7H11NO4S
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:205.23
  • Tyrphostin AG 1112

    CAS:
    <p>Tyrphostin AG 1112 is a Bcr-Abl kinase blocker. It can activate the terminal differentiation of K562 cells and the purging of Ph+ cells.</p>
    Formula:C15H10N6
    Color and Shape:Solid
    Molecular weight:274.28
  • Win-62005

    CAS:
    <p>Win-62005 is an inhibitor of cyclic AMP phosphodiesterase III (PDE III)(Kis: 25 and 26 nM for rat heart and canine aorta).</p>
    Formula:C12H10N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:226.23
  • 103D5R

    CAS:
    <p>103D5R selectively inhibits hif-1α, reducing its levels in hypoxia or with cobalt ions, dose- and time-dependently.</p>
    Formula:C20H21N3O2
    Color and Shape:Solid
    Molecular weight:335.4
  • BN-82685

    CAS:
    <p>BN-82685, a quinone-based CDC25 inhibitor, shows in vitro and in vivo efficacy, suggesting potential as an anticancer therapy.</p>
    Formula:C12H15N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:265.33
  • hCAI/II-IN-2

    CAS:
    <p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>
    Formula:C12H12N4O5S2
    Color and Shape:Solid
    Molecular weight:356.38
  • IM176OUT05

    CAS:
    <p>IM176OUT05 activates stem cell metabolism with hair regrowth-promoting effects.</p>
    Formula:C11H17N5
    Color and Shape:Solid
    Molecular weight:219.29
  • FASN-IN-4

    CAS:
    <p>FAS-IN-1 is a potent inhibitor of Fatty acid synthase (FAS) wtih IC50 of 10 nM.</p>
    Formula:C26H27N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:477.58
  • L 656224

    CAS:
    <p>L 656224 is a 5-LO inhibitor.</p>
    Formula:C20H21ClO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:344.83
  • Methyl-3β-hydroxycholenate

    CAS:
    <p>Methyl-3β-hydroxycholenate (Methyl 3beta-hydroxychol-5-enoate) is a modulator of RORγ.</p>
    Formula:C25H40O3
    Purity:98.78%
    Color and Shape:Solid
    Molecular weight:388.58
  • K134

    CAS:
    <p>K134 is an inhibitor of phosphodiesterase 3. The IC50s of K134 for PDE3A, PDE3B, PDE5, PDE2 and PDE4 are 0.1, 0.28, 12.1, &gt;300 and &gt;300 μM, respectively.</p>
    Formula:C22H29N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.48
  • 2-Hydroxy atorvastatin calcium salt

    CAS:
    <p>2-Hydroxy atorvastatin calcium salt is a hydroxy metabolite of Atorvastatin calcium salt which is a potent HMG-CoA reductase inhibitor (IC50 = 8 nM).</p>
    Formula:C33H34FN2O60·5Ca
    Purity:97.06%
    Color and Shape:Solid
    Molecular weight:593.68
  • CL67

    CAS:
    <p>CL67 is a hypoxia-inducible factor pathway inhibitor. It acts by binding to a G-quadruplex higher-order structure in the HIF promoter sequence in vitro.</p>
    Formula:C38H42N10O2
    Color and Shape:Solid
    Molecular weight:670.81
  • (RS)-Eflucimibe

    CAS:
    <p>Eflucimibe is an ACAT inhibitor.</p>
    Formula:C29H43NO2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:469.72
  • SK-216

    CAS:
    <p>SK-216,PAI-1 inhibitor. Reduces tumor angiogenesis. Inhibits VEGF-induced endothelial cell migration. Alleviates pulmonary fibrosis.</p>
    Formula:C29H29NNa2O6
    Purity:98.29%
    Color and Shape:Solid
    Molecular weight:533.52
  • (-)-Ketoconazole

    CAS:
    <p>(-)-Ketoconazole is a potential mitochondrial CYP24A1 inhibitor and has antifungal activity against Aspergillus fumigatus.</p>
    Formula:C26H28Cl2N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.43
  • SRPKIN-1

    CAS:
    <p>SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).</p>
    Formula:C27H21FN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.53
  • PKM2 activator 5

    CAS:
    <p>PKM2 activator 5 is a novel and potent PKM2 activator (AC50: 0.316 µM) with potential anticancer activity for the study of cancer metabolism-related diseases.</p>
    Formula:C18H19FN2O6S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:442.48
  • CS-722 Free base

    CAS:
    <p>CS-722 Free base: synthetic muscle relaxant; inhibits spinal reflex and sodium/calcium currents affecting synaptic activity.</p>
    Formula:C16H19ClN2O4
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:338.79
  • IDO-IN-3

    CAS:
    <p>IDO-IN-3 is a potent indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 290 nM).</p>
    Formula:C11H12BrFN6O2
    Color and Shape:Solid
    Molecular weight:359.15
  • Rovazolac

    CAS:
    <p>Rovazolac (ALX-101) is a liver x receptor (LXR) modulator used in the study of immune system disorders and atopic dermatitis.</p>
    Formula:C21H19F3N2O4S
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:452.45
  • ALDH1A1-IN-2

    CAS:
    <p>ALDH1A1-IN-2 is an aldehyde dehydrogenase 1a1 inhibitor with anticancer activity.ALDH1A1-IN-2 may be used in the study of breast cancer, inflammation or obesity</p>
    Formula:C25H23ClN4O3S
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:494.99
  • BAY 73-6691

    CAS:
    <p>BAY 73-6691 is an inhibitor of brain penetrant PDE9A.</p>
    Formula:C15H12ClF3N4O
    Color and Shape:Solid
    Molecular weight:356.73
  • GSK2945

    CAS:
    <p>GSK2945, a specific Rev-erbα antagonist, boosts CYP7A1 and cholesterol metabolism. EC50: 21.5 μM (mouse), 20.8 μM (human).</p>
    Formula:C20H18Cl2N2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:421.34
  • 8-CSC

    CAS:
    <p>8-CSC: hMAO-B inhibitor (Ki: 235 nM, baboon liver) &amp; A2A receptor affinity (Ki: 36 nM, rat brain).</p>
    Formula:C16H15ClN4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:330.77
  • TP-004

    CAS:
    <p>TP-004 is a potent and reversible methionine aminopeptidase 2 (MetAP2) inhibitor (IC50: 6 nM).</p>
    Formula:C17H16F3N5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.34
  • Succinyladenosine

    CAS:
    <p>Succinyladenosine, a marker for ASL deficiency, is made by dephosphorylating S-AMP with 5-nucleotidase.</p>
    Formula:C14H17N5O8
    Color and Shape:Solid
    Molecular weight:383.317
  • SCH-351591

    CAS:
    <p>SCH-351591 is an orally active inhibitor of phosphodiesterase 4.</p>
    Formula:C17H10Cl2F3N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.18
  • Gcase activator 3

    CAS:
    <p>Gcase activator 3 is a glucocerebrosidase (GCase) activator that enhances GBA1 mutant fibroblast lysosomal GCase activity.</p>
    Formula:C23H20N4O2
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:384.43
  • PDE9-IN-1

    CAS:
    <p>PDE9-IN-1 is a selective and orally bioavailable Inhibitor of PDE9A(IC50 of 8.7 nM).</p>
    Formula:C17H23FN6O2
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:362.4
  • HSL-IN-1

    CAS:
    <p>HSL-IN-1 is an HSL inhibitor that significantly reduces the reactive metabolite load and reduces the release of free fatty acids from stored fat.</p>
    Formula:C19H13BClF3N2O4
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:436.58
  • Nebicapone

    CAS:
    <p>Nebicapone, a reversible COMT inhibitor, reduces L-DOPA breakdown, aiding Parkinson's treatment.</p>
    Formula:C14H11NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:273.24
  • CAY10487

    CAS:
    <p>CAY10487 reduces aortic fatty streaks in high-cholesterol rabbits by 37.4% and inhibits LDL oxidation by 75% at 2μM, without altering lipids or ACAT activity.</p>
    Formula:C13H15NO5
    Color and Shape:Solid
    Molecular weight:265.26
  • Camylofin Hydrochloride

    CAS:
    <p>Camylofin HCl is an antispasmodic used in labor treatment and is also used to deliver drug therapy for ulcerative colinitis.</p>
    Formula:C19H33ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.94
  • PGAM1-IN-2

    CAS:
    <p>PGAM1-IN-2 is an inhibitor of phosphoglycerate mutase 1 ( PGAM1 ) with an IC 50 of 2.1 μM [1].</p>
    Formula:C25H16N2O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:488.47
  • Otamixaban

    CAS:
    <p>Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.</p>
    Formula:C25H26N4O4
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:446.5
  • OMDM-2

    CAS:
    <p>OMDM-2 is a metabolically stable and selective inhibitor of anandamide cellular uptake (ACU), exhibiting a Ki value of 3.0 μM in RBL-2H3 cells.</p>
    Formula:C27H45NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.65
  • ML-262

    CAS:
    <p>ML-262 is an effective inhibitor of hepatic lipid droplet formation and is used in studies of non-alcoholic fatty liver disease.</p>
    Formula:C27H32N2O4S
    Color and Shape:Solid
    Molecular weight:480.62
  • Epiroprim

    CAS:
    <p>Epiroprim (Ro11-8958) is a selective dihydrofolate reductase (DHFR) inhibitor with antibacterial activity, inhibiting Staphylococcus and Streptococcus.</p>
    Formula:C19H23N5O2
    Purity:99.68% - >99.99%
    Color and Shape:Solid
    Molecular weight:353.42
  • Enpp-1-IN-13

    CAS:
    <p>Enpp-1-IN-13 inhibits ENPP1 (IC50: 1.29 μM) &amp; ENPP3 (IC50: 20.2 μM) with anticancer properties.</p>
    Formula:C28H22ClN5OS
    Color and Shape:Solid
    Molecular weight:512.03
  • Spiraprilat

    CAS:
    <p>Spiraprilat is an ACE inhibitor. It also is an active metabolite of spirapril.</p>
    Formula:C20H26N2O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.56
  • sPLA2-X Inhibitor 31

    CAS:
    <p>sPLA2-X Inhibitor 31 targets sPLA2-X with IC50: 26 nM; less effective on sPLA2-IIa (310 nM), sPLA2-V (2230 nM).</p>
    Formula:C19H15F3N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.33
  • MRL-871

    CAS:
    <p>MRL-871 is a selective RORγt allosteric inhibitor, reducing IL-17a mRNA production in EL4 cells, interacting with PPARgamma in partial agonistic binding modes.</p>
    Formula:C22H12ClF3N2O3
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:444.79
  • S07-2010

    CAS:
    <p>S07-2010 is a pan-Aldo-Keto Reductase 1C3 (AKR1C3) inhibitor with potential anti-cancer activity, inducing apoptosis in A549/DDP cells.</p>
    Formula:C19H21N3O3S
    Purity:98.13%
    Color and Shape:Solid
    Molecular weight:371.45
  • AGN 191701

    CAS:
    <p>AGN 191701 is an agonist of the Retinoid X receptor.</p>
    Formula:C23H28O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.53
  • AHR-15010

    CAS:
    <p>AHR-15010 is a novel anti-arthritic agent.</p>
    Formula:C10H16N2O8S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.37
  • 2'-O-Methyladenosine

    CAS:
    <p>2'-O-Methyladenosine, a methylated adenine residue is found in the urine of normals and adenosine deaminase deficient patients.</p>
    Formula:C11H15N5O4
    Purity:99.89%
    Color and Shape:White Solid
    Molecular weight:281.27
  • IMB-XMA0038

    CAS:
    <p>IMB-XMA0038 is a Mycobacterium tuberculosis aspartate semialdehyde dehydrogenase inhibitor with antimicrobial activity for use in tuberculosis research.</p>
    Formula:C11H10N4O6
    Purity:98.94% - 99.96%
    Color and Shape:Solid
    Molecular weight:294.22
  • THR-0921

    CAS:
    <p>THR-0921 (CLX-0921) is a peroxisome proliferator-activated receptor (PPAR) agonist that can be used to study cardiovascular and metabolic diseases.</p>
    Formula:C28H25NO7S
    Purity:100% - 99.83%
    Color and Shape:Solid
    Molecular weight:519.57
  • BI-135585

    CAS:
    <p>BI-135585 is an orally active, selective and potent inhibitor of human 11β-hydroxysteroid dehydrogenase-1 (HSD1) for the study of type 2 diabetes.</p>
    Formula:C28H32N2O4
    Purity:99.45% - 99.57%
    Color and Shape:Solid
    Molecular weight:460.57
  • sEH inhibitor-3

    CAS:
    <p>sEH inhibitor-3 is an orally available, selective and potent inhibitor of sEH for cancer research.</p>
    Formula:C19H23F4N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.4
  • Glycogen phosphorylase-IN-1

    CAS:
    <p>Glycogen phosphorylase-IN-1 is an hlGPa inhibitor that can be used in the study of type 2 diabetes and canine lupus.</p>
    Formula:C17H15ClF2N4O4
    Purity:97.98% - 98.15%
    Color and Shape:Solid
    Molecular weight:412.78
  • MDK-4823

    CAS:
    <p>MDK-4823 (LMPTP inhibitor1) blocks LMPTP, fighting insulin resistance and diabetes in obesity.</p>
    Formula:C28H36N4O
    Color and Shape:Solid
    Molecular weight:444.61
  • Enpp-1-IN-8

    CAS:
    <p>Enpp-1-IN-8: potent inhibitor of enpp-1, an enzyme breaking down various nucleotide bonds; potential in cancer/infectious disease research.</p>
    Formula:C19H26N6O4S
    Color and Shape:Solid
    Molecular weight:434.51
  • FAAH-IN-7


    <p>FAAH-IN-7: Reversible FAAH inhibitor, IC50=8.29 nM, reduces oxidative stress, neuroprotective in neuroinflammation.</p>
    Formula:C26H29N3O4
    Color and Shape:Solid
    Molecular weight:447.53
  • Delapril

    CAS:
    <p>Delapril is an ACE inhibitor. It blocks the conversion of angiotensin I to angiotensin II.</p>
    Formula:C26H32N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:452.54
  • Isospaglumate sodium

    CAS:
    <p>Isospaglumate sodium is the sodium salt of isospaglumate which is an antiallergic agent.</p>
    Formula:C11H16N2NaO8
    Color and Shape:Solid
    Molecular weight:327.245
  • OSMI-3

    CAS:
    <p>OSMI-3 is a potent and cell-permeable inhibitor of O-GlcNAc transferase (OGT) for the study of cancer and cardiovascular disease.</p>
    Formula:C32H35N3O9S2
    Purity:99.03% - 99.08%
    Color and Shape:Solid
    Molecular weight:669.77
  • HIF-1α-IN-3

    CAS:
    <p>HIF-1α-IN-3, also known as Compound (S)-3f, is a hypoxia-selective inhibitor of HIF-1α. It exhibits potent antiestrogenic activity [1].</p>
    Formula:C19H17N5O2
    Color and Shape:Solid
    Molecular weight:347.37
  • Agn 190727

    CAS:
    <p>Agn 190727 is a retonoic acid receptor that can induce retinoid-induced hypertriglyceridemia.</p>
    Formula:C20H22O2
    Color and Shape:Solid
    Molecular weight:294.39
  • α-Glucosidase-IN-2

    CAS:
    <p>α-Glucosidase-IN-2 (compound 5d) is a potent inhibitor of α-Glucosidase, exhibiting an inhibitory concentration (IC50) of 9.48 μM, and functions as an</p>
    Formula:C17H11N3O2S2
    Color and Shape:Solid
    Molecular weight:353.42
  • JNJ-42314415

    CAS:
    <p>JNJ-42314415 is a potent, specific, and centrally active inhibitor of PDE10A.</p>
    Formula:C19H23N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.42
  • hCAIX-IN-3

    CAS:
    <p>hCAII-IN-3 (7e) selectively inhibits CA II/IX with Kis of 124.2/30.5 nM, showing promise for cancer treatment.</p>
    Formula:C21H21BrN6O4S
    Color and Shape:Solid
    Molecular weight:533.4
  • α-Glycosidase-IN-1

    CAS:
    <p>α-Glycosidase-IN-1 (compound MZ7) is a potent inhibitor of α-GLY (α-glycosidase) (IC50: 44.72 nM, Ki: 44.74 nM).</p>
    Formula:C21H19N9O6S2
    Color and Shape:Solid
    Molecular weight:557.56
  • Glucosylceramide synthase-IN-1

    CAS:
    <p>Potent oral GCS inhibitor T-036, crosses BBB, targets human (IC50: 31 nM) and mouse GCS (IC50: 51 nM), for Gaucher disease research.</p>
    Formula:C24H20F4N2O3
    Color and Shape:Solid
    Molecular weight:460.42
  • 9(R)-HODE

    CAS:
    <p>9(R)-HODE, a linoleic acid product, is made by some human/bovine endothelial cells, but its function and forming enzyme are unknown.</p>
    Formula:C18H32O3
    Color and Shape:Solid
    Molecular weight:296.44
  • ATX inhibitor 8

    CAS:
    <p>ATX inhibitor 8 is an inhibitor of the autocrine motor factor Autotaxin (ATX).</p>
    Formula:C28H26N10O
    Color and Shape:Solid
    Molecular weight:518.57
  • FTase-IN-1

    CAS:
    <p>FTase-IN-1, a potent FTase inhibitor, has an IC50 of 0.35 μM with strong antitumor activity and cytotoxicity.</p>
    Formula:C23H16N2O2S
    Color and Shape:Solid
    Molecular weight:384.45