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Metabolism

Metabolism

Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.

Subcategories of "Metabolism"

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Found 8626 products of "Metabolism"

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  • DU717

    CAS:
    <p>DU717 is an antihypertensive agent.</p>
    Formula:C12H15ClN4O2S
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:314.79
  • BI 689648

    CAS:
    <p>BI 689648 is a highly selective inhibitor of aldosterone synthase(CYP11B1 and CYP11B2 with IC50s of 310 and 2.1 nM, respectively).</p>
    Formula:C16H18N4O2
    Color and Shape:Solid
    Molecular weight:298.34
  • CGP-28014

    CAS:
    <p>CGP-28014 inhibits COMT, boosts renal dopamine &amp; DOPAC excretion, lowers HVA, no effect on renal sodium.</p>
    Formula:C12H19N3O
    Color and Shape:Solid
    Molecular weight:221.3
  • 3-Oxo-hop-22(29)-ene

    CAS:
    <p>3-Oxo-hop-22(29)-ene inhibits yeast α-glucosidase, moderately affects T. cruzi and L. mexicana, and has slight anti-inflammatory activity.</p>
    Formula:C30H48O
    Color and Shape:Solid
    Molecular weight:424.7
  • LEO 39652

    CAS:
    <p>LEO 39652: Dual-soft PDE4 inhibitor, IC50s: PDE4A/B: 1.2 nM, PDE4C: 3.0 nM, PDE4D: 3.8 nM; TNF-α IC50: 6.0 nM; for Atopic dermatitis research.</p>
    Formula:C23H23N3O5
    Color and Shape:Solid
    Molecular weight:421.45
  • IDO-IN-16

    CAS:
    <p>IDO-IN-16 (compound 5) is an IDO inhibitor (IC50: 36 nM).</p>
    Formula:C22H21F3N4O
    Color and Shape:Solid
    Molecular weight:414.42
  • ME-143

    CAS:
    <p>ME-143, a 2nd-gen NADH oxidase inhibitor, blocks WNT/β-catenin pathway, active against various cancers in vitro/vivo.</p>
    Formula:C21H18O4
    Color and Shape:Solid
    Molecular weight:334.37
  • AMPD2 inhibitor 2


    <p>AMPD2 inhibitor 2: strong h/mAMPD2 blocker, IC50s: 0.1/0.28μM. Potentially assesses AMPD2's role in high-fat diet mice.</p>
    Formula:C26H27F2N3O3
    Color and Shape:Solid
    Molecular weight:467.51
  • BMS-351

    CAS:
    <p>BMS-351: potent, selective CYP17A1 inhibitor, promising for prostate cancer, minimal side effects.</p>
    Formula:C15H12F3N3
    Color and Shape:Solid
    Molecular weight:291.27
  • IDO/TDO-IN-1

    CAS:
    <p>IDO/TDO-IN-1 is an orally active dual indoleamine-2,3-dioxygenase (IDO) and tryptophan 2,3-dioxygenase (TDO) inhibitor (IC50s: 9.7 and 47 nM).</p>
    Formula:C25H24FN5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:413.49
  • Nampt-IN-7

    CAS:
    <p>Nampt-IN-7 (GF8) inhibits NAMPT (IC50: 7.31 μM) and kills HepG2 cells (IC50: 24.28 μM).</p>
    Formula:C20H21N5O3
    Color and Shape:Solid
    Molecular weight:379.41
  • DGAT1-IN-3

    CAS:
    <p>DGAT1-IN-3: a potent, selective DGAT-1 inhibitor (IC50: 38 nM human, 120 nM rat), oral, for obesity and dyslipidemia research.</p>
    Formula:C20H19F3N4O3
    Color and Shape:Solid
    Molecular weight:420.39
  • hCAIX/XII-IN-4

    CAS:
    <p>hCAIX/XII-IN-4 inhibits CAIX/XII with Ki: 4.5 nM (CAXII), 23.6 nM (CAIX), and &gt;10000 nM (CAI/CAII).</p>
    Formula:C20H16N2O5
    Color and Shape:Solid
    Molecular weight:364.35
  • Carbonic anhydrase inhibitor 11

    CAS:
    <p>Potent carbonic anhydrase inhibitor VI targets CA II, IX, XII with Ki: 40, 39, 900 nM respectively.</p>
    Formula:C19H15F3N4O3S2
    Color and Shape:Solid
    Molecular weight:468.47
  • SCD1 inhibitor-1

    CAS:
    SCD1 inhibitor-1 is a potent and liver-selective inhibitor of stearoyl-CoA desaturase-1 (SCD1).
    Formula:C21H23N3NaO3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:452.54
  • PTP1B-IN-15

    CAS:
    <p>PTP1B-IN-15 is a potent and selective protein tyrosine phosphatase 1B (PTP1B) inhibitor that has shown research potential in type II diabetes and obesity.</p>
    Formula:C19H17Br2NO5S
    Color and Shape:Solid
    Molecular weight:531.22
  • Senazodan

    CAS:
    <p>Senazodan is a sensitiser of Ca2+, and shows inhibition effect on PDE III.</p>
    Formula:C15H14N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:266.3
  • (S)-Bromoenol lactone

    CAS:
    <p>(S)-BEL, a chiral inhibitor of iPLA2β, blocks vasopressin-induced arachidonate release in A10 cells; IC50 = 2μM.</p>
    Formula:C16H13BrO2
    Color and Shape:Solid
    Molecular weight:317.18
  • Pteropterin

    CAS:
    <p>Pteropterin is an antineoplastic agent.</p>
    Formula:C29H33N9O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:699.63
  • PAT-048

    CAS:
    <p>PAT-048 is an effective and selective autotaxin inhibitor.</p>
    Formula:C22H18ClF2N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:461.91
  • CYP1B1-IN-3

    CAS:
    <p>CYP1B1-IN-3: strong CYP1B1 inhibitor (IC50: 6.6 nM); weak on CYP1A1/CYP1A2; hinders cell migration, invasion; blocks P-gp, AKT/ERK, FAK/SRC, EMT.</p>
    Formula:C20H16FN3O2S2
    Color and Shape:Solid
    Molecular weight:413.49
  • FXR agonist 4


    <p>FXR agonist 4: EC50 of 1.05μM, treats hyperlipidemia, steatosis, insulin resistance, inflammation in DIO mice, for NAFLD research.</p>
    Formula:C21H28ClN3O
    Color and Shape:Solid
    Molecular weight:373.92
  • Risotilide

    CAS:
    <p>Risotilide is a voltage-dependent potassium channel inhibitor. It can prolong cardiac action potentials and refractory periods.</p>
    Formula:C15H27N3O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.52
  • NC1153

    CAS:
    <p>NC1153 blocks IL-2/JAK3/STAT5a/b, aids allograft survival, reduces toxicities.</p>
    Formula:C18H38Cl2N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:369.42
  • Alitame

    CAS:
    <p>Alitame is a high-intensity sweetener and sugar substitute widely used in biochemical experiments and drug synthesis research.</p>
    Formula:C14H25N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.43
  • MAO-B Inhibitor 58

    CAS:
    <p>MAO-B inhibitor 58 is an effective, selective, and reversible inhibitor of monoamine oxidase B.</p>
    Formula:C14H9Cl2N3
    Color and Shape:Solid
    Molecular weight:290.15
  • DCYM21

    CAS:
    <p>DCYM21: Menin-MLL inhibitor, halts leukemia cell growth with MLL changes, causing arrest and differentiation.</p>
    Formula:C26H33ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:409.01
  • LTV-1

    CAS:
    LTV-1 has the potential for autoimmunity treatment. LTV-1 is a potent lymphoid tyrosine phosphatase (LYP) inhibitor in T cells with an IC50 of 508 nM.
    Formula:C26H20N2O5S
    Color and Shape:Solid
    Molecular weight:472.51
  • Muristerone A

    CAS:
    <p>Muristerone A is a phytoecdysteroid analog of ecdysone and a potent ecdysteroid receptor agonist with a K d of 1 nM [1].</p>
    Formula:C27H44O8
    Color and Shape:Solid
    Molecular weight:496.63
  • 7β,27-dihydroxy Cholesterol

    CAS:
    <p>7β,27-dihydroxy Cholesterol is an oxysterol and agonist of retinoic acid receptor-related orphan receptor γ (RORγ) and RORγt.</p>
    Formula:C27H46O3
    Color and Shape:Solid
    Molecular weight:418.65
  • ACC1/2-IN-1

    CAS:
    <p>ACC1/2-IN-1 is a potent inhibitor of ACC1/2 and acts on ACC1 (IC50: 98.06 nM) and ACC2 (IC50: 29.43 nM). ACC1/2-IN-1 can be used in cancer research.</p>
    Formula:C34H32N4O4
    Color and Shape:Solid
    Molecular weight:560.64
  • α-Glucosidase-IN-10

    CAS:
    <p>α-Glucosidase-IN-10 (compound 13) is a potent inhibitor of α-glucosidase (IC50: 92.7 μM). α-Glucosidase-IN-10 can be used to study type II diabetes.</p>
    Formula:C21H15BrN4O2S
    Color and Shape:Solid
    Molecular weight:467.34
  • TUPS

    CAS:
    <p>TUPS is a selective soluble epoxide hydrolase inhibitor which protects against isoprenaline-induced cardiac hypertrophy.</p>
    Formula:C14H18F3N3O4S
    Color and Shape:Solid
    Molecular weight:381.37
  • Sermetacin

    CAS:
    <p>Sermetacin is an anti-inflammatory agent.</p>
    Formula:C22H21ClN2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:444.86
  • AX 048

    CAS:
    <p>Group IVA cPLA2 inhibitor AX 048 halts arachidonic acid release, preventing prostaglandin production, with XI(50) of 0.022 and ED50 of 1.2 mg/kg.</p>
    Formula:C22H41NO4
    Color and Shape:Solid
    Molecular weight:383.57
  • CYP11B2-IN-1

    CAS:
    <p>CYP11B2-IN-1 是一种有效的选择性 CYP11B2 抑制剂,对 CYP11B2 和 CYP11B1 的 IC50 分别为 2.3 nM 和 142 nM。</p>
    Formula:C18H18FN3O
    Purity:99.79% - 99.89%
    Color and Shape:Solid
    Molecular weight:311.35
  • JTP-4819

    CAS:
    <p>JTP-4819: potent PEP inhibitor, may treat Alzheimer's, boosts brain peptides and acetylcholine, aiding memory.</p>
    Formula:C19H25N3O4
    Color and Shape:Solid
    Molecular weight:359.42
  • AMG-221

    CAS:
    <p>AMG-221: potent 11β-HSD1 inhibitor, lowers glucose &amp; insulin, reduces obesity in mice.</p>
    Formula:C14H22N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:266.4
  • Boc-Glu(OBzl)-OSu

    CAS:
    <p>Boc-Glu(OBzl)-OSu can be used for the synthesis of solid phase peptides containing benzyl glutamate residues.</p>
    Formula:C21H26N2O8
    Color and Shape:Solid
    Molecular weight:434.44
  • α-Amylase/α-Glucosidase-IN-2

    CAS:
    α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μM
    Formula:C22H16ClN5
    Color and Shape:Solid
    Molecular weight:385.85
  • Nampt-IN-9

    CAS:
    <p>Nampt-IN-9 (Compound 8) is a potent inhibitor of NAMPT with anticancer properties.Nampt-IN-9 can be used to study ductal adenocarcinoma of the pancreas.</p>
    Formula:C26H33N3O4
    Color and Shape:Solid
    Molecular weight:451.56
  • p-Synephrine

    CAS:
    <p>p-Synephrine is a natural product for research related to life sciences. The catalog number is T8265 and the CAS number is 614-35-7.</p>
    Formula:C9H13NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:167.21
  • IACS-8968 R-enantiomer

    CAS:
    <p>IACS-8968 R-enantiomer is the R-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and &lt;5 for TDO).</p>
    Formula:C17H18F3N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:381.35
  • α-Glucosidase-IN-4

    CAS:
    <p>α-Glucosidase-IN-4 is a potent α-glucosidase inhibitor with antihypertensive and hypoglycemic activity.</p>
    Formula:C19H14O4
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:306.31
  • IDO1-IN-15

    CAS:
    <p>IDO1-IN-15 is an effective IDO1 inhibitor with IC50 of 127 nM. The potency of IDO1-IN-15 against IDO1 enzyme is comparable with Epacadostat in vitro.</p>
    Formula:C13H14BrFN6O3
    Color and Shape:Solid
    Molecular weight:401.19
  • CG-707

    CAS:
    <p>CG-707 is an inhibitor of PRL-3 that acts by blocking the migration and invasion of metastatic cancer cells.</p>
    Formula:C20H17NO3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.48
  • S 12340

    CAS:
    <p>S 12340 is a potent inhibitor of the oxidative modification of low-density lipoprotein.</p>
    Formula:C24H38N2O3S
    Color and Shape:Solid
    Molecular weight:434.64
  • (R)-DNMDP

    CAS:
    <p>(R)-DNMDP is a potent and selective cancer cytotoxic agent that directly binds PDE3A and has an EC50 500-fold lower than that of (S)-DNMDP against HeLa.</p>
    Formula:C15H20N4O3
    Color and Shape:Solid
    Molecular weight:304.34
  • hCAIX-IN-14

    CAS:
    hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .
    Formula:C11H17ClN6O2S
    Color and Shape:Solid
    Molecular weight:332.81
  • MSPG

    CAS:
    <p>mGlu receptor antagonist</p>
    Formula:C9H11NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:245.25
  • CDP 840 hydrochloride

    CAS:
    <p>CDP-840 (GR259653X), a potent oral PDE IV inhibitor, curbs early and late phase bronchoconstriction in squirrel monkeys.</p>
    Formula:C25H27NO2
    Color and Shape:Solid
    Molecular weight:373.49
  • ATX inhibitor 8

    CAS:
    <p>ATX inhibitor 8 is an inhibitor of the autocrine motor factor Autotaxin (ATX).</p>
    Formula:C28H26N10O
    Color and Shape:Solid
    Molecular weight:518.57
  • FAAH-IN-7


    <p>FAAH-IN-7: Reversible FAAH inhibitor, IC50=8.29 nM, reduces oxidative stress, neuroprotective in neuroinflammation.</p>
    Formula:C26H29N3O4
    Color and Shape:Solid
    Molecular weight:447.53
  • Enpp-1-IN-8

    CAS:
    <p>Enpp-1-IN-8: potent inhibitor of enpp-1, an enzyme breaking down various nucleotide bonds; potential in cancer/infectious disease research.</p>
    Formula:C19H26N6O4S
    Color and Shape:Solid
    Molecular weight:434.51
  • MDK-4823

    CAS:
    <p>MDK-4823 (LMPTP inhibitor1) blocks LMPTP, fighting insulin resistance and diabetes in obesity.</p>
    Formula:C28H36N4O
    Color and Shape:Solid
    Molecular weight:444.61
  • TDP1 Inhibitor-2

    CAS:
    <p>TDP1 Inhibitor-2 strongly blocks TDP1 (IC50: 99 nM) &amp; treats SCAN1 (IC50: 3.5 μM).</p>
    Formula:C25H14Cl2O5
    Color and Shape:Solid
    Molecular weight:465.28
  • hACC2-IN-1

    CAS:
    <p>hACC2-IN-1 is a potent inhibitor of acetyl coenzyme A carboxylase 2 (ACC2) with an IC50 value of 2.5 μM for hACC2. hACC2-IN-1 has potential for obesity studies.</p>
    Formula:C23H32N2O4S
    Color and Shape:Solid
    Molecular weight:432.58
  • S32826 disodium

    CAS:
    <p>autotaxin inhibitor</p>
    Formula:C21H36NNa2O4P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:443.47
  • AZD-3289

    CAS:
    <p>AZD-3289, a potent BACE1 inhibitor, is used potentially for the treatment of Alzheimer's disease.</p>
    Formula:C24H14F5N5
    Color and Shape:Solid
    Molecular weight:467.39
  • Metyltetraprole

    CAS:
    <p>Metyltetraprole: potent fungicide, effective against Zymoseptoria, low EC50 (0.002 ppm), inhibits respiratory chain.</p>
    Formula:C19H17ClN6O2
    Color and Shape:Solid
    Molecular weight:396.83
  • α-Glucosidase-IN-9

    CAS:
    <p>α-Glucosidase-IN-9 (compound 7) is a highly potent α-glucosidase inhibitor with an IC50 of 55.6 μM, making it suitable for type II diabetes research [1].</p>
    Formula:C19H12N4OS
    Color and Shape:Solid
    Molecular weight:344.39
  • α-Amylase-IN-2

    CAS:
    α-Glucosidase-IN-3, an oxime ester derivative of oleanolic acid (OA), exhibits inhibitory activity against α-glucosidase (IC50 = 1.28 µM) and α-amylase (IC50 =
    Formula:C39H52BrNO4
    Color and Shape:Solid
    Molecular weight:678.74
  • HIF-PHD-IN-2

    CAS:
    <p>HIF-PHD-IN-2 (compound 25) is a highly effective PHD inhibitor, displaying IC50 values below 100 nM for PHD1, PHD2, and PHD3 [1].</p>
    Formula:C17H15N5O3S
    Color and Shape:Solid
    Molecular weight:369.4
  • Nebicapone

    CAS:
    <p>Nebicapone, a reversible COMT inhibitor, reduces L-DOPA breakdown, aiding Parkinson's treatment.</p>
    Formula:C14H11NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:273.24
  • trans-Ned 19

    CAS:
    <p>trans-Ned 19 blocks NAADP and TPC, hindering calcium signaling and aorta relaxation at low histamine levels.</p>
    Formula:C30H31FN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:514.59
  • SQ-31765

    CAS:
    <p>SQ-31765 is a blocker of benzazepine calcium channel.</p>
    Formula:C24H27F3N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:464.48
  • CAY10487

    CAS:
    <p>CAY10487 reduces aortic fatty streaks in high-cholesterol rabbits by 37.4% and inhibits LDL oxidation by 75% at 2μM, without altering lipids or ACAT activity.</p>
    Formula:C13H15NO5
    Color and Shape:Solid
    Molecular weight:265.26
  • tHGA

    CAS:
    <p>tHGA is a potent inhibitor of lipoxygenase.</p>
    Formula:C18H24O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:304.38
  • (Rac)-3′-Hydroxy simvastatin

    CAS:
    <p>(Rac)-3′-Hydroxy Simvastatin, a metabolite of Simvastatin, acts as a competitive inhibitor of HMG-CoA reductase, demonstrating a K i value of 0.2 nM.</p>
    Formula:C25H38O6
    Color and Shape:Solid
    Molecular weight:434.57
  • HX-600

    CAS:
    <p>HX-600 is a synthetic agonist for the RXR-Nurr1 heterodimer complex. HX-600 prevents ischemia-induced neuronal damage.</p>
    Formula:C29H30N2O2
    Color and Shape:Solid
    Molecular weight:438.56
  • SAHO

    CAS:
    <p>SAHO is a methyl donor cleaved by SAM enzymes into adenosylhomocysteine and thioadenosine derivatives.</p>
    Formula:C14H20N6O6S
    Color and Shape:Solid
    Molecular weight:400.41
  • Enpp-1-IN-13

    CAS:
    <p>Enpp-1-IN-13 inhibits ENPP1 (IC50: 1.29 μM) &amp; ENPP3 (IC50: 20.2 μM) with anticancer properties.</p>
    Formula:C28H22ClN5OS
    Color and Shape:Solid
    Molecular weight:512.03
  • YC-001

    CAS:
    <p>YC-001: inverse agonist/antagonist for rod opsin, prevents light-induced retinal degeneration.</p>
    Formula:C12H7ClO2S2
    Color and Shape:Solid
    Molecular weight:282.77
  • Ipenoxazone

    CAS:
    <p>Ipenoxazone is an effective and centrally acting muscle relaxant.</p>
    Formula:C22H34N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:358.52
  • SAR127303

    CAS:
    <p>SAR127303 is an effective covalent inhibitor of MAGL. SAR127303 behaves as a selective and competitive inhibitor of mouse and human MAGL.</p>
    Formula:C16H17ClF6N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:482.83
  • IHVR-19029

    CAS:
    <p>IHVR-19029: ER α-glucosidases I/II inhibitor, IC50 0.48μM; halts Ebola, Dengue, Rift Valley fever virus replication.</p>
    Formula:C23H45N3O5
    Color and Shape:Solid
    Molecular weight:443.62
  • ALDH3A1-IN-2

    CAS:
    <p>ALDH3A1-IN-2 is a potent inhibitor targeting ALDH3A1 (IC50=1.29µM), potentially useful in cancer research.</p>
    Formula:C11H14N2O3
    Color and Shape:Solid
    Molecular weight:222.24
  • ARI-3531

    CAS:
    <p>ARI-3531 is a selective prolyl endopeptidase inhibitor.</p>
    Formula:C15H22BN3O4
    Color and Shape:Solid
    Molecular weight:319.16
  • AChE/hCA I/II-IN-1

    CAS:
    <p>Compound 6: Potent inhibitor for AChE, Hca I &amp; II with IC50s of 22.21, 60.79, 66.64 nM, useful in glaucoma, Alzheimer's, diabetes research.</p>
    Formula:C15H13N3S
    Color and Shape:Solid
    Molecular weight:267.35
  • sEH inhibitor-6

    CAS:
    <p>sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].</p>
    Formula:C21H14ClN3O2
    Color and Shape:Solid
    Molecular weight:375.81
  • Oncrasin-72

    CAS:
    Oncrasin-72 is an analog of oncrasin-1. It has antitumor activity mediated by JNK activation and STAT3 inhibition.
    Formula:C16H14ClNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:271.74
  • N-Acetylserine

    CAS:
    <p>N-Acetylserine (N-Acetyl-L-serine) serves as the physiological inducer of cysteine biosynthesis by binding to the CysB apoprotein and stimulating cysJIH</p>
    Formula:C5H9NO4
    Purity:99.28%
    Color and Shape:Solid
    Molecular weight:147.13
  • Izumerogant

    CAS:
    <p>Izumerogant is an inverse agonist of the retinoid-related orphan receptor-gamma (RORγ).</p>
    Formula:C22H18ClF4N5O2
    Color and Shape:Solid
    Molecular weight:495.86
  • YCT529 free acid

    CAS:
    <p>YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .</p>
    Formula:C29H25NO3
    Color and Shape:Solid
    Molecular weight:435.51
  • hCAI/II-IN-3

    CAS:
    <p>"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."</p>
    Formula:C16H18N4O4S2
    Color and Shape:Solid
    Molecular weight:394.47
  • iGP-5

    CAS:
    <p>iGP-5 is a cell-permeable mitochondrial sn-Glycerol 3-phosphate dehydrogenase (mGPDH) inhibitor.</p>
    Formula:C21H17N3O3
    Color and Shape:Solid
    Molecular weight:359.38
  • hCAXII-IN-3

    CAS:
    <p>hCAXII-IN-3 (Compound 6o) is a selective inhibitor of human carbonic anhydrase XII (hCAXII) (Ki: 10.0 nM).</p>
    Formula:C26H20BrN5O3S
    Color and Shape:Solid
    Molecular weight:562.44
  • Enpp-1-IN-9

    CAS:
    <p>Enpp-1-IN-9 inhibits ENPP1, cleaves numerous bonds in nucleotides/sugars; may advance cancer/infectious disease research.</p>
    Formula:C17H24N4O5S
    Color and Shape:Solid
    Molecular weight:396.46
  • FCE 28654

    CAS:
    <p>FCE 28654 is a water-soluble acyl-CoA inhibitor.</p>
    Formula:C25H35N2O7P
    Color and Shape:Solid
    Molecular weight:506.53
  • SCD1 Inhibitor

    CAS:
    <p>SCD1 Inhibitor is a novel stearoyl-CoA desaturase1 (SCD1) inhibitor.</p>
    Formula:C21H20F3N3O3
    Color and Shape:Solid
    Molecular weight:419.4
  • hCAIX-IN-5

    CAS:
    <p>hCAIX-IN-5 was a selective hCAIX inhibitor, inhibiting hCAI, hCAII, hCAIV, and hCAIX with Ki values of &gt;10000, &gt;10000, 130.7, and 829.1 nM, respectively.</p>
    Formula:C18H12FNO3
    Purity:99.26%
    Color and Shape:Solid
    Molecular weight:309.29
  • OMDM-4

    CAS:
    <p>OMDM-4 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 17.7 μM).</p>
    Formula:C29H43NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.66
  • Asterriquinol D dimethyl ether

    CAS:
    <p>Asterriquinol D dimethyl ether inhibits mouse myeloma (IC50: 28 μg/mL) and Tritrichomonas foetus.</p>
    Formula:C26H24N2O4
    Color and Shape:Solid
    Molecular weight:428.48
  • PF 04671536 hydrochloride

    CAS:
    <p>Potent PDE8B/8A inhibitor; IC50: PDE8B-1.3nM, PDE8A-1.9nM; selective over other PDEs; enhances insulin secretion; orally bioavailable.</p>
    Formula:C14H19ClN8OS
    Color and Shape:Solid
    Molecular weight:382.87
  • TAK 21d

    CAS:
    <p>Potent FAAH inhibitor</p>
    Formula:C19H17F2N7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:397.38
  • Nampt activator-3

    CAS:
    <p>NAMPT activator-3: a NAT derivative, EC50 of 2.6 μM, KD 132 nM, protects cells, prevents FK866 toxicity, and is neuroprotective in CIPN mice.</p>
    Formula:C19H20N2O3
    Color and Shape:Solid
    Molecular weight:324.37
  • hDHODH-IN-11

    CAS:
    <p>hDHODH-IN-11: potent hDHODH inhibitor, IC50 7.2 nM, low cytotoxicity, for AML research.</p>
    Formula:C24H23N3O3
    Color and Shape:Solid
    Molecular weight:401.46
  • LY 269415

    CAS:
    <p>LY 269415 is an anti-inflammatory agent with antioxidant properties in vitro and could be beneficial as therapeutic agents in inflammatory arthritis.</p>
    Formula:C19H28N2O2S
    Color and Shape:Solid
    Molecular weight:348.5
  • TPN729MA

    CAS:
    <p>TPN729MA, a potent PDE5 inhibitor, IC50: 2.28 nM, targets erectile dysfunction research.</p>
    Formula:C29H40N6O8S
    Color and Shape:Solid
    Molecular weight:632.73
  • SR1555 HCl

    CAS:
    <p>SR1555: A selective RORγ inverse agonist, hinders TH17 cells, key in autoimmune diseases like RA and MS.</p>
    Formula:C22H22F6N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:460.41