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Metabolism

Metabolism

Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.

Subcategories of "Metabolism"

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Found 8626 products of "Metabolism"

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  • Genz-669178

    CAS:
    <p>Genz-669178 is a wild-type inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH).</p>
    Formula:C17H14N4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:322.38
  • Trandolaprilat

    CAS:
    <p>Trandolaprilat is an inhibitor of non-sulfhydryl angiotensin-converting enzyme.</p>
    Formula:C22H30N2O5
    Color and Shape:Pale Yellow Solid
    Molecular weight:402.48
  • BMS 740808

    CAS:
    <p>BMS-740808 is a highly effective and selective factor X inhibitor.</p>
    Formula:C31H27F3N6O3
    Color and Shape:Solid
    Molecular weight:588.58
  • TMCB

    CAS:
    <p>CK2 and ERK8 inhibitor</p>
    Formula:C11H9Br4N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:534.82
  • Liarozole dihydrochloride

    CAS:
    <p>Liarozole dihydrochloride, an oral CYP450 inhibitor, blocks estrogen and androgens, targeting prostate cancer and skin disorders.</p>
    Formula:C17H15Cl3N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:381.69
  • Cycloguanil

    CAS:
    <p>Cycloguanil is an antimalarial.</p>
    Formula:C11H14ClN5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:251.72
  • UK51656

    CAS:
    <p>UK51656 is an antagonist of calcium (IC50: 4 nM).</p>
    Formula:C22H28ClN3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:465.93
  • IM176OUT05

    CAS:
    <p>IM176OUT05 activates stem cell metabolism with hair regrowth-promoting effects.</p>
    Formula:C11H17N5
    Color and Shape:Solid
    Molecular weight:219.29
  • α-Glucosidase-IN-20

    CAS:
    <p>α-Glucosidase-IN-20 (Compound 3B) is a highly effective and orally active inhibitor of α-glucosidase.</p>
    Formula:C23H21NOS
    Color and Shape:Solid
    Molecular weight:359.48
  • Rosuvastatin lactone

    CAS:
    <p>Tilavonemab (ABBV-8E12) is a monoclonal antibody that binds to the N-terminus of the human microtubule-associated protein tau.</p>
    Formula:C22H26FN3O5S
    Color and Shape:Solid
    Molecular weight:463.52
  • SR1555 HCl

    CAS:
    <p>SR1555: A selective RORγ inverse agonist, hinders TH17 cells, key in autoimmune diseases like RA and MS.</p>
    Formula:C22H22F6N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:460.41
  • L-Xylulose

    CAS:
    <p>L-Xylulose: a rare sugar, key in metabolism, α-glucosidase inhibitor, lowers glucose, precursor to antiviral drug components.</p>
    Formula:C5H10O5
    Color and Shape:Solid
    Molecular weight:150.13
  • DHODH-IN-21

    CAS:
    <p>DHODH-IN-21, orally active DHODH blocker with 1.1 nM IC50, shows anticancer activity, potential for AML research.</p>
    Formula:C20H19ClF4N6O4
    Color and Shape:Solid
    Molecular weight:518.85
  • RORγt inverse agonist 30

    CAS:
    <p>RORγt inverse agonist 30 (Compound 1) is a potent RORγt inverse agonist (IC50: 46 nM).</p>
    Formula:C24H31N3O3S
    Color and Shape:Solid
    Molecular weight:441.59
  • HIF-PHD-IN-2

    CAS:
    <p>HIF-PHD-IN-2 (compound 25) is a highly effective PHD inhibitor, displaying IC50 values below 100 nM for PHD1, PHD2, and PHD3 [1].</p>
    Formula:C17H15N5O3S
    Color and Shape:Solid
    Molecular weight:369.4
  • Desfluoro-atorvastatin

    CAS:
    <p>Desfluoro-atorvastatin is an impurity of atorvastatin, an oral HMG-CoA reductase inhibitor that lowers blood lipids.</p>
    Formula:C33H36N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:540.65
  • KM04416

    CAS:
    <p>KM04416 is a GPD2 inhibitor that inhibits LUAD progression by modulating immune cell infiltration.</p>
    Formula:C12H11NO3S
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:249.29
  • α-Amylase-IN-2

    CAS:
    <p>α-Glucosidase-IN-3, an oxime ester derivative of oleanolic acid (OA), exhibits inhibitory activity against α-glucosidase (IC50 = 1.28 µM) and α-amylase (IC50 =</p>
    Formula:C39H52BrNO4
    Color and Shape:Solid
    Molecular weight:678.74
  • Afegostat D-Tartrate

    CAS:
    <p>Afegostat D-Tartrate: pharmacological chaperone, reversibly binds acid-β-glucosidase in ER with high affinity.</p>
    Formula:C10H19NO9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.26
  • RYL-552

    CAS:
    <p>RYL-552 is a potent inhibitor of PfNDH2.</p>
    Formula:C24H17F4NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:427.39
  • Indolapril hydrochloride

    CAS:
    <p>Indolapril hydrochloride is a nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity.</p>
    Formula:C24H35ClN2O5
    Color and Shape:Solid
    Molecular weight:467
  • α-Glucosidase-IN-9

    CAS:
    <p>α-Glucosidase-IN-9 (compound 7) is a highly potent α-glucosidase inhibitor with an IC50 of 55.6 μM, making it suitable for type II diabetes research [1].</p>
    Formula:C19H12N4OS
    Color and Shape:Solid
    Molecular weight:344.39
  • Metyltetraprole

    CAS:
    <p>Metyltetraprole: potent fungicide, effective against Zymoseptoria, low EC50 (0.002 ppm), inhibits respiratory chain.</p>
    Formula:C19H17ClN6O2
    Color and Shape:Solid
    Molecular weight:396.83
  • XEN103

    CAS:
    <p>XEN103 is a potent and selective Stearoyl-CoA Desaturase-1 inhibitor.</p>
    Formula:C22H23F4N5O2
    Color and Shape:Solid
    Molecular weight:465.44
  • Delapril

    CAS:
    <p>Delapril is an ACE inhibitor. It blocks the conversion of angiotensin I to angiotensin II.</p>
    Formula:C26H32N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:452.54
  • IDO-IN-12

    CAS:
    <p>IDO-IN-12 is an inhibitor of indoleamine 2,3-dioxygenase (IDO).</p>
    Formula:C13H11BrFN5O3S
    Purity:99.727%
    Color and Shape:Solid
    Molecular weight:416.23
  • GKA-71

    CAS:
    <p>GKA-71 is an effective glucokinase activator (GKA).</p>
    Formula:C21H23N3O6S2
    Color and Shape:Solid
    Molecular weight:477.55
  • ML368

    CAS:
    <p>ML368 is a selective inhibitor of CYP3A4.</p>
    Formula:C26H18N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.46
  • JNJ-61803534

    CAS:
    <p>JNJ-61803534: RORγt inverse agonist, IC50=9.6 nM, oral, anti-inflammatory, reduces IL-17A in T cells.</p>
    Formula:C23H23Cl2F6N3O4S
    Color and Shape:Solid
    Molecular weight:622.41
  • Umbralisib tosylate

    CAS:
    <p>Umbralisib tosylate, an oral PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), shows promise for CLL research.</p>
    Formula:C38H32F3N5O6S
    Color and Shape:Solid
    Molecular weight:743.75
  • (R)-Lercanidipine hydrochloride

    CAS:
    <p>(R)-Lercanidipine hydrochloride is the R-enantiomer of Lercanidipine. (R)-lercanidipine hydrochloride is a blocker of calcium channel.</p>
    Formula:C36H42ClN3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:648.2
  • hCAIX-IN-3

    CAS:
    <p>hCAII-IN-3 (7e) selectively inhibits CA II/IX with Kis of 124.2/30.5 nM, showing promise for cancer treatment.</p>
    Formula:C21H21BrN6O4S
    Color and Shape:Solid
    Molecular weight:533.4
  • Saterinone hydrochloride

    CAS:
    <p>Saterinone hydrochloride is an inhibitor of phosphodiesterase III (PDE III).</p>
    Formula:C27H31ClN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:511.01
  • JTV-519

    CAS:
    <p>K201 (JTV-519) is a Ca2+-dependent blocker and prevents abnormal Ca(2+) leak from the sarcoplasmic reticulum in the ischemic heart and skeletal muscle (SkM) by</p>
    Formula:C25H33ClN2O2S
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:461.06
  • PKM2 activator 4

    CAS:
    <p>PKM2 Activator 4, a chemical compound, functions as an activator of PKM2 with an activation concentration (AC 50) ranging from 1 to 10 μM.</p>
    Formula:C16H16N2O4S
    Color and Shape:Solid
    Molecular weight:332.37
  • α-Glucosidase-IN-21

    CAS:
    <p>α-Glucosidase-IN-21 (Compound 2B) is a highly potent and orally bioavailable inhibitor of α-glucosidase.</p>
    Formula:C24H23NO2S
    Color and Shape:Solid
    Molecular weight:389.51
  • 3,3-Dimethyl-1-butanol

    CAS:
    <p>3,3-Dimethyl-1-butanol (DMB) inhibits TMA/TMAO and affects p65 NF-κB, TGF-β1/Smad3 signaling; potential for CVD treatment.</p>
    Formula:C6H14O
    Color and Shape:Solid
    Molecular weight:102.17
  • Fexarine

    CAS:
    <p>Fexarine is a potent, selective agonist of farnesoid X receptor.</p>
    Formula:C31H31NO5
    Color and Shape:Solid
    Molecular weight:497.58
  • hCA IX-IN-2


    <p>hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferative</p>
    Formula:C23H24N2O4STe
    Color and Shape:Solid
    Molecular weight:552.11
  • PDE-9 inhibitor

    CAS:
    <p>PDE-9 inhibitor is used for treatment neurodegenerative diseases.</p>
    Formula:C22H27N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.48
  • GK187

    CAS:
    <p>GK187 is a selective and potent Group VIA calcium-independent phospholipase A2 (GVIA iPLA2) inhibitor, used in the study of neurological disorders.</p>
    Formula:C14H15F5O2
    Color and Shape:Solid
    Molecular weight:310.26
  • EP6

    CAS:
    <p>EP6 blocks 5-LO, key in the AA cascade, reducing leukotrienes to curb inflammation and allergies.</p>
    Formula:C24H30N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:390.52
  • THR-0921

    CAS:
    <p>THR-0921 (CLX-0921) is a peroxisome proliferator-activated receptor (PPAR) agonist that can be used to study cardiovascular and metabolic diseases.</p>
    Formula:C28H25NO7S
    Purity:100% - 99.83%
    Color and Shape:Solid
    Molecular weight:519.57
  • 24(S),25-Epoxycholesterol

    CAS:
    <p>24(S),25-Epoxycholesterol is an oxysterol agonist of the liver X receptor.</p>
    Formula:C27H44O2
    Color and Shape:Solid
    Molecular weight:400.64
  • ATX inhibitor 19

    CAS:
    <p>ATX inhibitor 19 is a potent inhibitor of ATX (IC50: 156 nM).</p>
    Formula:C28H33ClN6O2S
    Color and Shape:Solid
    Molecular weight:553.12
  • Theodrenaline

    CAS:
    <p>Theodrenaline is a cardiac stimulant, also acts as an agent of anti-hypotensive together with cafedrine.</p>
    Formula:C17H21N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:375.38
  • FCE 28654

    CAS:
    <p>FCE 28654 is a water-soluble acyl-CoA inhibitor.</p>
    Formula:C25H35N2O7P
    Color and Shape:Solid
    Molecular weight:506.53
  • IMB-XMA0038

    CAS:
    <p>IMB-XMA0038 is a Mycobacterium tuberculosis aspartate semialdehyde dehydrogenase inhibitor with antimicrobial activity for use in tuberculosis research.</p>
    Formula:C11H10N4O6
    Purity:98.94% - 99.96%
    Color and Shape:Solid
    Molecular weight:294.22
  • MY33-3 hydrochloride

    CAS:
    <p>MY33-3 HCl: Inhibits RPTPβ/ζ (IC50~0.1μM), PTP-1B (IC50~0.7μM), curbs alcohol intake, fights neuroinflammation and memory issues.</p>
    Formula:C16H14ClF6NS2
    Color and Shape:Solid
    Molecular weight:433.86
  • TC-E 5008

    CAS:
    <p>TC-E 5008 is a selective inhibitor of mutant isocitrate dehydrogenase 1 (mIDH1).</p>
    Formula:C13H13NO2
    Color and Shape:Solid
    Molecular weight:215.25
  • hCAXII-IN-3

    CAS:
    <p>hCAXII-IN-3 (Compound 6o) is a selective inhibitor of human carbonic anhydrase XII (hCAXII) (Ki: 10.0 nM).</p>
    Formula:C26H20BrN5O3S
    Color and Shape:Solid
    Molecular weight:562.44
  • PDE10-IN-5

    CAS:
    <p>PDE10-IN-5 is a phosphodiesterase 10 (PDE 10) inhibitor that can be used to study certain central nervous system disorders.</p>
    Formula:C26H19F3N4O
    Color and Shape:Solid
    Molecular weight:460.45
  • hDHODH-IN-9

    CAS:
    <p>hDHODH-IN-9 is a potent hDHODH inhibitor, IC50=0.34 μM, toxic to MCF-7/A375 cells, promising for cancer research.</p>
    Formula:C21H21NO4
    Color and Shape:Solid
    Molecular weight:351.4
  • PDE4-IN-11

    CAS:
    <p>PDE4-IN-11: Potent PDE4 inhibitor with strong bronchodilatory and anti-inflammatory effects for airway disease research.</p>
    Formula:C21H19FN2O2
    Color and Shape:Solid
    Molecular weight:350.39
  • Phortress free base

    CAS:
    <p>Phortress free base is a P450 CYP1A1-activated antitumor prodrug with antitumor activity.</p>
    Formula:C20H23FN4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.49
  • AVE5688

    CAS:
    <p>AVE5688 is an inhibitor of glycogen phosphorylase (GP, IC50s: 430 nM and 915 nM; Kds: 170 nM and 530 nM for rmGPb and rmGPa).</p>
    Formula:C16H8ClF5N2O5
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:438.69
  • DP00477

    CAS:
    <p>DP00477, a potent inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1), exhibits an inhibitory concentration (IC50) of 7.0 µM.</p>
    Formula:C17H11ClF3N3OS
    Color and Shape:Solid
    Molecular weight:397.8
  • TFB-TBOA

    CAS:
    <p>glial glutamate transporter EAAT1 and EAAT2 inhibitor</p>
    Formula:C19H17F3N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:426.34
  • ML299

    CAS:
    <p>ML299 (VU0463568) is a dual PLD1/2 inhibitor (PLD1 and PLD2, IC50 of 6 nM, 20 nM, respectively).</p>
    Formula:C23H26BrFN4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.38
  • D-threo-PPMP hydrochloride

    CAS:
    <p>D-threo-PPMP inhibits GlyCer synthetase; active enantiomer; reduces MDCK cell growth by 70% at 20 μM.</p>
    Formula:C29H51ClN2O3
    Color and Shape:Solid
    Molecular weight:511.19
  • FTase-IN-1

    CAS:
    <p>FTase-IN-1, a potent FTase inhibitor, has an IC50 of 0.35 μM with strong antitumor activity and cytotoxicity.</p>
    Formula:C23H16N2O2S
    Color and Shape:Solid
    Molecular weight:384.45
  • NPD-1335

    CAS:
    <p>NPD1335: potent TbrPDEB1 inhibitor, submicromolar efficacy, low toxicity, raises cAMP, disrupts cell cycle, kills T. brucei.</p>
    Formula:C28H29N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:455.55
  • DSHN

    CAS:
    <p>DSHN activates SHP, boosting its mRNA and protecting it from ubiquitination and degradation.</p>
    Formula:C15H17NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:323.36
  • LEI-106

    CAS:
    <p>LEI-106 is an effective dual inhibitor of DAGL-α and ABHD6, with Ki values of 0.7 and 0.8 μM respectively, for obesity and metabolic syndrome research.</p>
    Formula:C26H27NO6S
    Color and Shape:Solid
    Molecular weight:481.56
  • Sch 34826

    CAS:
    <p>Sch 34826 is a potent, selective neutral endopeptidase inhibitor.</p>
    Formula:C27H34N2O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.57
  • PDE5-IN-4

    CAS:
    <p>PDE5-IN-4, a phosphodiesterase 5 (PDE5) inhibitor, is utilized in research concerning acute myocardial infarction and reperfusion-related damage,</p>
    Formula:C21H27N5O5S
    Color and Shape:Solid
    Molecular weight:461.53
  • Phenylthiazolylthiourea

    CAS:
    <p>Phenylthiazolylthiourea ia a dopamine-beta-hydroxylase inhibitor.</p>
    Formula:C10H9N3S2
    Color and Shape:Solid
    Molecular weight:235.33
  • Oxagrelate

    CAS:
    <p>Oxagrelate inhibits cAMP phosphodiesterase and reduces platelet aggregation by collagen and ADP.</p>
    Formula:C14H16N2O4
    Color and Shape:Solid
    Molecular weight:276.29
  • Quinethazone

    CAS:
    <p>Quinethazone is a thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels.</p>
    Formula:C10H12ClN3O3S
    Color and Shape:Fibrous Crystals From 50% Acetone Physical Description Fibrous Crystals Or White Powder (Ntp 1992)
    Molecular weight:289.74
  • Deltazinone

    CAS:
    <p>Deltazinone selectively inhibits PDEδ with low cytotoxicity, mimicking PDEδ knockdown in human pancreatic cancer cells.</p>
    Formula:C27H31N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.57
  • SGK1 inhibitor

    CAS:
    <p>SGK1 inhibitor targets SGK1/2 over SGK3, blocks GSK3β phosphorylation, lowers HCC1954 cell viability with BYL719, and reduces tumor growth in mice.</p>
    Formula:C17H12Cl2N6O2S
    Color and Shape:Solid
    Molecular weight:435.29
  • CAY10485

    CAS:
    <p>CAY10485 blocks human ACAT-1 &amp; ACAT-2 (IC50: 95 &amp; 81 μM) and hinders oxidation of LDL by 91% at 2 μM, possibly impacting atherosclerosis development.</p>
    Formula:C27H27NO7
    Color and Shape:Solid
    Molecular weight:477.51
  • Afegostat

    CAS:
    <p>Afegostat is a pharmacological chaperone that specifically and reversibly binds acid-β-glucosidase (GCase) in the endoplasmic reticulum with high affinity.</p>
    Formula:C6H13NO3
    Purity:98%
    Color and Shape:Yellow Low-Melting Solid
    Molecular weight:147.17
  • KT185

    CAS:
    <p>KT185 is an orally-bioavailable and brain-penetrant ABHD6 inhibitor (IC50: 0.21 nM in Neuro2A cells).</p>
    Formula:C32H33N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:519.64
  • PF-06471553

    CAS:
    <p>PF-06471553 is an effective and selective inhibitor of monoacylglycerol acyltransferase 3 (IC50: 92 nM).</p>
    Formula:C23H25N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:467.54
  • (R)-Bromoenol lactone

    CAS:
    <p>(R)-Bromoenol lactone (BEL) irreversibly inhibits iPLA2γ with 0.6 μM IC50, not affecting iPLA2β unless at 20-30 μM doses.</p>
    Formula:C16H13BrO2
    Color and Shape:Solid
    Molecular weight:317.18
  • (R)-DNMDP

    CAS:
    <p>(R)-DNMDP is a potent and selective cancer cytotoxic agent that directly binds PDE3A and has an EC50 500-fold lower than that of (S)-DNMDP against HeLa.</p>
    Formula:C15H20N4O3
    Color and Shape:Solid
    Molecular weight:304.34
  • Benserazide

    CAS:
    <p>Benserazide blocks dopa decarboxylase; paired with levodopa for Parkinson's to boost CNS dopamine levels and lower dosage.</p>
    Formula:C10H15N3O5
    Color and Shape:Solid
    Molecular weight:257.24
  • K134

    CAS:
    <p>K134 is an inhibitor of phosphodiesterase 3. The IC50s of K134 for PDE3A, PDE3B, PDE5, PDE2 and PDE4 are 0.1, 0.28, 12.1, &gt;300 and &gt;300 μM, respectively.</p>
    Formula:C22H29N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.48
  • L 669262

    CAS:
    <p>L 669262 is a potent inhibitor of HMG-CoA reductase.</p>
    Formula:C25H36O6
    Color and Shape:Solid
    Molecular weight:432.55
  • Abiraterone metabolite 1

    CAS:
    <p>Abiraterone metabolite 1, a derivative of abiraterone, inhibits CYP17A1, halts androgen formation, aiding in prostate cancer treatment.</p>
    Formula:C24H33NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.52
  • CG-707

    CAS:
    <p>CG-707 is an inhibitor of PRL-3 that acts by blocking the migration and invasion of metastatic cancer cells.</p>
    Formula:C20H17NO3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.48
  • SK-216

    CAS:
    <p>SK-216,PAI-1 inhibitor. Reduces tumor angiogenesis. Inhibits VEGF-induced endothelial cell migration. Alleviates pulmonary fibrosis.</p>
    Formula:C29H29NNa2O6
    Purity:98.29%
    Color and Shape:Solid
    Molecular weight:533.52
  • CS-722 Free base

    CAS:
    <p>CS-722 Free base: synthetic muscle relaxant; inhibits spinal reflex and sodium/calcium currents affecting synaptic activity.</p>
    Formula:C16H19ClN2O4
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:338.79
  • Benproperine

    CAS:
    <p>Benproperine is a bioactive molecule with antineoplastic properties.</p>
    Formula:C21H27NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:309.45
  • IACS-8968 S-enantiomer

    CAS:
    <p>IACS-8968 S-enantiomer is the S-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and &lt;5 for TDO).</p>
    Formula:C17H18F3N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:381.35
  • UCM 765

    CAS:
    <p>UCM 765 is a partial agonist of melatonin MT(2) receptor.</p>
    Formula:C17H20N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:284.35
  • Incadronate Disodium

    CAS:
    <p>Incadronate Disodium: halts bone loss, limits macrophage migration and inflammation, and induces cancer cell apoptosis in vitro.</p>
    Formula:C8H19NNaO6P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:310.178
  • YM758 Phosphate

    CAS:
    <p>YM758 Phosphate, a current channel inhibitor, selectively lowers a heart beat and decreases oxygen consumption of heart muscle.</p>
    Formula:C26H35FN3O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:567.54
  • 12(S)-HpETE

    CAS:
    <p>12(S)-HpETE activates human blood leukocyte 5-LOE and mediates induction of c-fos and c-jun, activation of AP-1, and endothelium-dependent vasoconstriction.</p>
    Formula:C20H32O4
    Color and Shape:Solid
    Molecular weight:336.47
  • CL67

    CAS:
    <p>CL67 is a hypoxia-inducible factor pathway inhibitor. It acts by binding to a G-quadruplex higher-order structure in the HIF promoter sequence in vitro.</p>
    Formula:C38H42N10O2
    Color and Shape:Solid
    Molecular weight:670.81
  • Muristerone A

    CAS:
    <p>Muristerone A is a phytoecdysteroid analog of ecdysone and a potent ecdysteroid receptor agonist with a K d of 1 nM [1].</p>
    Formula:C27H44O8
    Color and Shape:Solid
    Molecular weight:496.63
  • NBD-125

    CAS:
    <p>NBD-125 (B-12) is a berberine analogue. NBD-125 is an RXRα activator. The IC50 value of NBD-125 in KM12C cell is 31.10 μM [1].</p>
    Formula:C19H18ClNO2
    Color and Shape:Solid
    Molecular weight:327.81
  • MAO-B Inhibitor 58

    CAS:
    <p>MAO-B inhibitor 58 is an effective, selective, and reversible inhibitor of monoamine oxidase B.</p>
    Formula:C14H9Cl2N3
    Color and Shape:Solid
    Molecular weight:290.15
  • MAGL-IN-1

    CAS:
    <p>MAGL-IN-1 is a selective and potent monoacylglycerol lipase (MAGL) inhibitor with an IC50 of 80 nM.</p>
    Formula:C22H24FNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:369.43
  • 7ETMC

    CAS:
    <p>7ETMC inhibits Human Cytochrome P450s 1A1/1A2 with IC50: 0.46/0.50 μM; not effective on P450s 2A6/2B1 even at 50 μM.</p>
    Formula:C14H12O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:212.24
  • Gallopamil hydrochloride

    CAS:
    <p>Gallopamil hydrochloride (Methoxyverapamil hydrochloride) is an antagonist of phenylalkylamine calcium.</p>
    Formula:C28H41ClN2O5
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:521.09
  • 8-CSC

    CAS:
    <p>8-CSC: hMAO-B inhibitor (Ki: 235 nM, baboon liver) &amp; A2A receptor affinity (Ki: 36 nM, rat brain).</p>
    Formula:C16H15ClN4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:330.77
  • PSN-GK1

    CAS:
    <p>PSN-GK1 is a potent activator of glucokinase (EC50: 0.13 μM).</p>
    Formula:C20H23FN2O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.54
  • TA-7552

    CAS:
    <p>TA-7552 is a potent agent of cholesterol-lowering.</p>
    Formula:C25H26O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:486.47
  • BMS270394

    CAS:
    <p>BMS270394 is a RARγ agonist used in the study of breast cancer and skin diseases.</p>
    Formula:C23H26FNO4
    Color and Shape:Solid
    Molecular weight:399.46
  • BFE-37

    CAS:
    <p>BFE-37 is a partial agonist of beta-adrenergic.</p>
    Formula:C16H23NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:277.36
  • PF-4191834

    CAS:
    <p>PF-4191834: Non-iron, non-redox 5-LOX inhibitor, IC50 = 229 nM, 300x selective over 12/15-LOX, inactive on COX enzymes.</p>
    Formula:C22H23N3O2S
    Purity:99.83% - 99.98%
    Color and Shape:Solid
    Molecular weight:393.5
  • PMPMEase-IN L-28

    CAS:
    <p>PMPMEase-IN L-28 is a novel inhibitor of prenylated methylated protein methylesterase.</p>
    Formula:C17H29FO2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.54
  • Ethylene thiourea

    CAS:
    <p>Ethylene thiourea (NCIC03372) is a pesticide used in fruit and vegetable production.</p>
    Formula:C3H6N2S
    Purity:≥98%
    Color and Shape:Needles Prisms From Alcohol Or Amyl Alcohol
    Molecular weight:102.16
  • Pteropterin

    CAS:
    <p>Pteropterin is an antineoplastic agent.</p>
    Formula:C29H33N9O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:699.63
  • Alitame

    CAS:
    <p>Alitame is a high-intensity sweetener and sugar substitute widely used in biochemical experiments and drug synthesis research.</p>
    Formula:C14H25N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.43
  • DCYM21

    CAS:
    <p>DCYM21: Menin-MLL inhibitor, halts leukemia cell growth with MLL changes, causing arrest and differentiation.</p>
    Formula:C26H33ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:409.01
  • Camylofin Hydrochloride

    CAS:
    <p>Camylofin HCl is an antispasmodic used in labor treatment and is also used to deliver drug therapy for ulcerative colinitis.</p>
    Formula:C19H33ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.94
  • Pirbuterol hydrochloride

    CAS:
    <p>Pirbuterol hydrochloride is a bronchodilator.</p>
    Formula:C12H21ClN2O3
    Color and Shape:Solid
    Molecular weight:276.76
  • Pegnivacogin

    CAS:
    <p>Pegnivacogin is a coagulation factor IXa RNA aptamer inhibitor.</p>
    Formula:C20H40N3O11P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:529.52
  • D-4418

    CAS:
    <p>D-4418, a PDE4 inhibitor in development, targets asthma and COPD as an anti-inflammatory treatment.</p>
    Formula:C16H11Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.18
  • LP8

    CAS:
    <p>LP8 is a novel inhibitor of Trypanosoma cruzi CYP51.</p>
    Formula:C16H19N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:349.4
  • KC-12615

    CAS:
    <p>KC-12615 is an inhibitior of endopeptidase.</p>
    Formula:C29H34N2O6
    Color and Shape:Solid
    Molecular weight:506.59
  • Leucinal

    CAS:
    <p>Leucinal inhibits the activity of brain aminopeptidase and potentiates analgesia induced by leu-enkephalen.</p>
    Formula:C6H13NO
    Color and Shape:Solid
    Molecular weight:115.17
  • Texasin

    CAS:
    <p>Texasin is a selective inhibitor of human leukocyte 5-lipoxygenase.</p>
    Formula:C16H12O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:284.26
  • AZD-3289

    CAS:
    <p>AZD-3289, a potent BACE1 inhibitor, is used potentially for the treatment of Alzheimer's disease.</p>
    Formula:C24H14F5N5
    Color and Shape:Solid
    Molecular weight:467.39
  • tHGA

    CAS:
    <p>tHGA is a potent inhibitor of lipoxygenase.</p>
    Formula:C18H24O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:304.38
  • JNJ-40413269

    CAS:
    <p>JNJ-40413269 inhibits FAAH, engages central targets, and is effective in rat neuropathic pain.</p>
    Formula:C19H15ClF3N3O
    Color and Shape:Solid
    Molecular weight:393.79
  • Radamide

    CAS:
    <p>Radamide is an inhibitor of Grp94.</p>
    Formula:C18H18ClNO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.79
  • Amiquinsin

    CAS:
    <p>Amiquinsin is a drug with hypotensive effect.</p>
    Formula:C11H12N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:204.23
  • Dexecadotril

    CAS:
    <p>Dexecadotril is a powerful and selective neprilysin inhibitor. It behaves as a prodrug of the enantiomer of thiorphan.</p>
    Formula:C21H23NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.48
  • MJN228

    CAS:
    <p>MJN228 is a NUCB1 inhibitor that blocks AEA-DA probe labeling of endogenous NUCB1 in Neuro2a cells and can be used to study metabolic disorders.</p>
    Formula:C20H20N4O3
    Purity:98.42%
    Color and Shape:Solid
    Molecular weight:364.4
  • ZM223

    CAS:
    <p>ZM223 is an inhibitor of NEDD8 activating enzyme (NAE).</p>
    Formula:C23H17F3N4O2S2
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:502.53
  • Indoleacetyl phenylalanine

    CAS:
    <p>Indoleacetyl phenylalanine is an indole-acetyl-amino acid involved in regulating auxin activity.</p>
    Formula:C19H18N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:322.36
  • OH-Ubenimex

    CAS:
    <p>OH-Ubenimex is an orally active aminopeptidase inhibitor that has an immunomodulating action.</p>
    Formula:C16H24N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.37
  • BVT-116429

    CAS:
    <p>BVT-116429 is an inhibitor of 11β-HSD1.</p>
    Formula:C13H12F4N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:320.31
  • LB42908

    CAS:
    <p>LB42908 is a highly potent Ras farnesyltransferase inhibitor(IC(50)=0.9 nM against H-Ras and 2.4 nM against K-Ras) with potential anticancer activity.</p>
    Formula:C32H31N5O3
    Color and Shape:Solid
    Molecular weight:533.62
  • Langkamide

    CAS:
    <p>Langkamide is a HIF-2 inhibitor with EC₅₀ values of 14.0 uM.</p>
    Formula:C16H17NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:303.31
  • sEH-IN-12

    CAS:
    <p>sEH-IN-12 is an effective inhibitor of the enzyme soluble epoxide hydrolase (sEH).</p>
    Formula:C25H29N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.53
  • Benzpiperylone

    CAS:
    <p>Benzpiperylone is a synthetic anti-inflammatory drug. It also has anti-inflammatory activity.</p>
    Formula:C22H25N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:347.45
  • Noreximide

    CAS:
    <p>Noreximide is an agent of sedative.</p>
    Formula:C9H9NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:163.17
  • Rev 6207

    CAS:
    <p>Rev 6207 is a non-sulfhydryl ACE-inhibitor.</p>
    Formula:C21H31N3O5
    Color and Shape:Solid
    Molecular weight:405.49
  • DBC

    CAS:
    <p>DBC is a halogenated hydrocarbon, widely used in biochemical experiments and drug synthesis research.</p>
    Formula:C20H13N
    Purity:99.76%
    Color and Shape:Needles From Ethanol 7H-Dibenzo(C G)Carbazole Is A Crystalline Solid
    Molecular weight:267.32
  • BAY 59-9435

    CAS:
    <p>HSL-IN-2 is a selective inhibitor of Hormone Sensitive Lipase (HSL; IC50: 0.023 μM).</p>
    Formula:C14H22N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:266.34
  • Pinoxepin HCl

    CAS:
    <p>Pinoxepin HCl is an antipsychotic.</p>
    Formula:C23H29Cl3N2O2
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:471.85
  • Nebicapone

    CAS:
    <p>Nebicapone, a reversible COMT inhibitor, reduces L-DOPA breakdown, aiding Parkinson's treatment.</p>
    Formula:C14H11NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:273.24
  • CR4056

    CAS:
    <p>CR4056 (6-(1H-imidazol-1-yl)-2-phenylquinazoline) is a selective inhibitor of MAO-A with IC50 of 202.7 nM and a ligand of I2-imidazoline receptor with IC50 of</p>
    Formula:C17H12N4
    Purity:98.73%
    Color and Shape:Solid
    Molecular weight:272.3
  • CX08005

    CAS:
    <p>CX08005 inhibits PTP1B, cuts liver fat, and improves microcirculation in NAFLD.</p>
    Formula:C28H39NO4
    Purity:≥98%
    Color and Shape:Solid
    Molecular weight:453.61
  • A-1293201

    CAS:
    <p>A-1293201 is a potent and selective NAMPT inhibitor.</p>
    Formula:C21H23N3O3
    Color and Shape:Solid
    Molecular weight:365.43
  • VU0155056

    CAS:
    <p>VU0155056 is a dual PLD1/2 inhibitor with IC50 &lt; 1 µM in cellular assays, inhibits breast cancer cell invasion.</p>
    Formula:C25H26N4O2
    Purity:98.6% - 99.15%
    Color and Shape:Solid
    Molecular weight:414.5
  • FABP4/5-IN-5

    CAS:
    <p>FABP4/5-IN-5 (compound D9) serves as a potent inhibitor of both FABP 4 and FABP 5, demonstrating IC50 values of 4.68 μM and 10.72 μM, respectively. It is notably effective in addressing metabolic disorders such as diabetes mellitus [1].</p>
    Formula:C23H14ClF2NO4S
    Color and Shape:Solid
    Molecular weight:473.88
  • RO6806051

    CAS:
    RO6806051 (compound 12) is a potent dual inhibitor of fatty acid binding proteins 4 and 5 (FABP4 and FABP5), exhibiting excellent selectivity and absorption, distribution, metabolism, and excretion (eADME) properties.
    Formula:C21H19ClN6
    Color and Shape:Solid
    Molecular weight:390.87
  • CAY10762

    CAS:
    <p>CAY10762, a MAGL inhibitor (IC50=34.1 nM), curbs H2O2-induced LDH in Neuro2a cells and boosts 2-AG in mouse brains at 10 mg/kg.</p>
    Formula:C15H13NOS
    Color and Shape:Solid
    Molecular weight:255.33
  • McN3716

    CAS:
    <p>McN3716 is a carnitine palmitoyltransferase I (CPT-1) inhibitor for the study of metabolic diseases.</p>
    Formula:C18H34O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:298.46
  • BBMP

    CAS:
    <p>BBMP is an inhibitor of mitochondrial permeability transition pore.</p>
    Formula:C12H11BrN2O3S
    Color and Shape:Solid
    Molecular weight:343.2
  • LY367385

    CAS:
    <p>LY367385 is a highly effective and selective mGluR1a antagonist.</p>
    Formula:C10H11NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:209.2
  • AVE-8134

    CAS:
    <p>AVE-8134 is an agonist of PPARα. For human and rodent PPARα receptor, the EC50 values are 100 and 3000 nM, respectively.</p>
    Formula:C22H23NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:381.42
  • N-(α-Linolenoyl) Tyrosine

    CAS:
    <p>Certain chronic neurologic disorders, such as Parkinson's disease, are caused by an insufficiency of the neurotransmitter dopamine secondary to the degeneration</p>
    Formula:C27H39NO4
    Color and Shape:Solid
    Molecular weight:441.6
  • Teludipine hydrochloride

    CAS:
    <p>Teludipine hydrochloride is a blocker of lipophilic calcium channel.</p>
    Formula:C28H39ClN2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:535.07
  • IDO-IN-6

    CAS:
    <p>IDO-IN-6 is an indoleamine 2,3-dioxygenase (IDO) inhibitor.</p>
    Formula:C18H21FN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:316.37
  • UCK2 Inhibitor-2

    CAS:
    <p>UCK2 Inhibitor-2 is a non-competitive inhibitor of uridine-cytidine kinase 2 (UCK2) with IC50=3.8 µM that inhibits UCK2-mediated nucleoside recycling in cells.</p>
    Formula:C28H23N3O4S
    Purity:98.76% - 99.25%
    Color and Shape:Solid
    Molecular weight:497.57
  • ATX inhibitor 5

    CAS:
    <p>ATX inhibitor 5: potent, oral autotaxin blocker, IC50 15.3 nM, curbs CCl4 liver fibrosis.</p>
    Formula:C22H18ClF3N6O
    Purity:98.77%
    Color and Shape:Solid
    Molecular weight:474.87
  • MAO-IN-1

    CAS:
    <p>MAO-IN-1 is a potent monoamine oxidase B (MAO B) inhibitor (IC50: 20 nM) for the study of neurologically related diseases.</p>
    Formula:C17H19ClO4
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:322.78
  • LYS006

    CAS:
    <p>LYS006 is a highly efficient and selective LTA4H (leukotriene A4 hydrolase) inhibitor,for neutrophil-driven inflammatory diseases ulcerative colitis.</p>
    Formula:C16H14ClFN6O3
    Purity:99.33%
    Color and Shape:Soild
    Molecular weight:392.77
  • (-)-L-threo-PDMP (hydrochloride)

    CAS:
    <p>(-)-L-threo-PDMP boosts ganglioside production, enhances neurite and synapse growth, and aids memory post-ischemia at 40 mg/kg/day.</p>
    Formula:C23H39ClN2O3
    Color and Shape:Solid
    Molecular weight:427.03
  • ACAT-IN-1 cis isomer

    CAS:
    <p>ACAT-IN-1 cis isomer is a potent ACAT inhibitor (IC50: 100 nM) for the study of immune system-related diseases.</p>
    Formula:C29H25NO2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:419.51
  • PGAM1-IN-1

    CAS:
    <p>PGAM1-IN-1 is an inhibitor of phosphoglycerate mutase 1 ( PGAM1 ) with an IC 50 of 6.4 μM [1].</p>
    Formula:C19H11ClFNO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.81
  • Tanogitran

    CAS:
    <p>Tanogitran, a coagulation factor Xa inhibitor, is used potentially for the treatment of septic shock.</p>
    Formula:C25H31N7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:477.56
  • Prenyl-IN-1

    CAS:
    <p>Prenyl-IN-1 inhibits prenylation selectively, counters oxidative stress in Parkinson's.</p>
    Formula:C28H24ClN5O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:497.98
  • HZ52

    CAS:
    <p>HZ52: Potent reversible 5-LO inhibitor; IC50 0.7 μM; blocks LTs in human leukocytes.</p>
    Formula:C24H26ClN3O2S
    Color and Shape:Solid
    Molecular weight:456
  • ATX inhibitor 20

    CAS:
    <p>ATX inhibitor 20 is a potent inhibitor of ATX (IC50: 2.3 nM).</p>
    Formula:C31H34FN5O3
    Color and Shape:Solid
    Molecular weight:543.63
  • Factor VII-IN-1

    CAS:
    <p>Factor VII-IN-1 (example 43) is an effective Factor VII (FVII) inhibitor (IC50=1.1 μM) with anticoagulant properties.</p>
    Formula:C15H10BrNO3
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:332.15
  • CAY10486

    CAS:
    <p>CAY10486 blocks ACAT-1/2, which form cholesterol esters, potentially reducing atherosclerosis; inhibits LDL oxidation. IC50 ~60μM; 28% effect at 3μM.</p>
    Formula:C19H19NO4
    Color and Shape:Solid
    Molecular weight:325.36
  • Valibose

    CAS:
    <p>Valibose, α-glucosidase inhibitor, improves glucose/lipid metabolism, lowers serum BUN/NAG, reduces kidney weight index.</p>
    Formula:C10H21NO6
    Color and Shape:Solid
    Molecular weight:251.28
  • Epostane

    CAS:
    <p>Epostane is a 3β-hydroxysteroid dehydrogenase inhibitor that blocks the biosynthesis of progesterone and pregnenolone.Cost-effective and quality-assured.</p>
    Formula:C22H31NO3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:357.49
  • Mesopram

    CAS:
    <p>PDE4 inhibitor, orally active</p>
    Formula:C14H19NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:265.3
  • AMP-Deoxynojirimycin

    CAS:
    <p>AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.</p>
    Formula:C22H39NO5
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:397.55
  • ML-148

    CAS:
    <p>ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM).</p>
    Formula:C20H21N3O
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:319.4
  • MRL-871

    CAS:
    <p>MRL-871 is a selective RORγt allosteric inhibitor, reducing IL-17a mRNA production in EL4 cells, interacting with PPARgamma in partial agonistic binding modes.</p>
    Formula:C22H12ClF3N2O3
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:444.79
  • CD2665

    CAS:
    <p>CD2665 is an orally active antagonist of retinoic acid receptor (RAR). For RARγ and RARβ, the Kis are 110 nM and 306 nM.</p>
    Formula:C31H34O5
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:486.6
  • CFG920

    CAS:
    <p>CFG920 is an oral CYP17 inhibitor that may reduce androgen production and inhibit growth of androgen-dependent tumors.</p>
    Formula:C14H13ClN4O
    Color and Shape:Solid
    Molecular weight:288.73
  • S07-2010

    CAS:
    <p>S07-2010 is a pan-Aldo-Keto Reductase 1C3 (AKR1C3) inhibitor with potential anti-cancer activity, inducing apoptosis in A549/DDP cells.</p>
    Formula:C19H21N3O3S
    Purity:98.13%
    Color and Shape:Solid
    Molecular weight:371.45
  • 4-Desmethyl Istradefylline

    CAS:
    <p>4-Desmethyl Istradefylline: a metabolite of Istradefylline, a strong, selective oral adenosine A2A receptor blocker, Ki 2.2 nM, used in Parkinson's.</p>
    Formula:C19H22N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.40
  • (R)-Irsenontrine

    CAS:
    <p>(R)-Irsenontrine (R-E2027), R-enantiomer, is a potent PDE9 inhibitor, IC50 = 0.041 μM, for neurological disease research.</p>
    Formula:C22H22N4O3
    Color and Shape:Solid
    Molecular weight:390.44
  • L-5-BromoTryptophan

    CAS:
    <p>L-5-BromoTryptophan (5-BrW) is an analog of the tryptophan (Trp) effector and inhibits the gelation of hemoglobin S.</p>
    Formula:C11H11BrN2O2
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:283.12
  • SU 10603

    CAS:
    <p>SU 10603 is a specific inhibitor of 17α-hydroxylase (also known as CYP17A1 and P450c17) used to study steroid hormone synthesis.</p>
    Formula:C15H12ClNO
    Purity:99.93% - 99.96%
    Color and Shape:Solid
    Molecular weight:257.72
  • 7-Biopterin

    CAS:
    <p>7-Biopterin, a 7-substituted pterin, forms non-enzymatically and elevates in urine of hyperphenylalaninemics with PCBD mutations.</p>
    Formula:C9H11N5O3
    Color and Shape:Solid
    Molecular weight:237.22
  • Dibefurin

    CAS:
    <p>Dibefurin blocks calcineurin, a calcium-dependent enzyme, reducing T lymphocyte activation.</p>
    Formula:C18H16O8
    Color and Shape:Solid
    Molecular weight:360.31
  • TM6089

    CAS:
    <p>TM6089 is an inhibitor of Prolyl Hydroxylase that stimulates HIF activity without iron chelation, induces angiogenesis, and protects organ against ischemia.</p>
    Formula:C13H14N4O3S
    Purity:99.70%
    Color and Shape:Solid
    Molecular weight:306.34
  • Enpp-1-IN-9

    CAS:
    <p>Enpp-1-IN-9 inhibits ENPP1, cleaves numerous bonds in nucleotides/sugars; may advance cancer/infectious disease research.</p>
    Formula:C17H24N4O5S
    Color and Shape:Solid
    Molecular weight:396.46
  • OHM1

    CAS:
    <p>OHM1, an analog of HIF1α CTAD, effectively inhibits the interaction between HIF1α CTAD and p300/CBP by targeting the CH1 domain with a binding affinity of 0.53</p>
    Formula:C24H42N6O5
    Color and Shape:Solid
    Molecular weight:494.63
  • Dacisteine

    CAS:
    <p>Dacisteine (N,S-Diacetyl-L-cysteine) is an inhibitor of New Delhi metallo-beta-lactamase-1 (NDM-1, IC50 = 1000 μM).</p>
    Formula:C7H11NO4S
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:205.23
  • 13(S)-HOTrE(γ)

    CAS:
    <p>13(S)-HOTrE(γ) is a metabolite and octadecatrienoic acid used as a metabolic marker, in the study of metabolic disorders and neurological diseases.</p>
    Formula:C18H30O3
    Color and Shape:Solid
    Molecular weight:294.43
  • sEH inhibitor-6

    CAS:
    <p>sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].</p>
    Formula:C21H14ClN3O2
    Color and Shape:Solid
    Molecular weight:375.81
  • TDP1 Inhibitor-2

    CAS:
    <p>TDP1 Inhibitor-2 strongly blocks TDP1 (IC50: 99 nM) &amp; treats SCAN1 (IC50: 3.5 μM).</p>
    Formula:C25H14Cl2O5
    Color and Shape:Solid
    Molecular weight:465.28
  • GW844520

    CAS:
    <p>GW844520 is a potent and selective inhibitor of the cytochrome bc1 complex of mitochondrial electron transport in P. falciparum.</p>
    Formula:C20H15ClF3NO3
    Color and Shape:Solid
    Molecular weight:409.79
  • Soluble epoxide hydrolase inhibitor

    CAS:
    <p>Soluble epoxide hydrolase inhibitor is a soluble epoxide hydrolase inhibitor (human soluble epoxide hydrolase (h-sEH) with pIC50 of 8.4).</p>
    Formula:C18H12F5N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.31
  • Acetylhydrolase-IN-1

    CAS:
    <p>Acetylhydrolase-IN-1 is an inhibitor of the esterase 1-Alkyl-2-acetylglycerophosphocholine (Alkylacetyl-GPC: acetylhydrolase).</p>
    Formula:C23H48NO7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.6
  • Kojibiose

    CAS:
    <p>Kojibiose (Kojibiose) is a disaccharide in honey. Kojibiose is a product of the caramelization of glucose.</p>
    Formula:C12H22O11
    Purity:99.933%
    Color and Shape:Solid
    Molecular weight:342.3
  • Phosphodiesterase-IN-1

    CAS:
    <p>Phosphodiesterase-IN-1 (Compound 7), a phosphodiesterase (PDE) inhibitor, exhibits anti-Plasmodium and antiproliferative activities. It effectively inhibits P. falciparum (strain 3D7) with an IC 50 value of 0.64 μM [1].</p>
    Formula:C15H15FN4O
    Color and Shape:Solid
    Molecular weight:286.3
  • L 656224

    CAS:
    <p>L 656224 is a 5-LO inhibitor.</p>
    Formula:C20H21ClO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:344.83
  • Fenleuton

    CAS:
    <p>Fenleuton is a 5-lipoxygenase inhibitor.</p>
    Formula:C17H15FN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:314.31
  • CDP 840 hydrochloride

    CAS:
    <p>CDP-840 (GR259653X), a potent oral PDE IV inhibitor, curbs early and late phase bronchoconstriction in squirrel monkeys.</p>
    Formula:C25H27NO2
    Color and Shape:Solid
    Molecular weight:373.49
  • M77976

    CAS:
    <p>M77976 inhibits PDK4 with an IC50 of 648 μM, targeting obesity and diabetes research.</p>
    Formula:C17H16N2O3
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:296.32
  • Entacapone sodium salt

    CAS:
    <p>Entacapone sodium salt, a potent peripheral COMT inhibitor (IC50=151 nM), hinders α-syn/β-amyloid aggregation and protects PC12 cells.</p>
    Formula:C14H15N3NaO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.28
  • Sp-Cyclic AMPS (sodium salt)

    CAS:
    <p>Sp-cAMPS Na salt activates PKA I/II and competitively inhibits PDE3A (Ki: 47.6 μM), also binds PDE10 GAF (EC50: 40 μM).</p>
    Formula:C10H12N5NaO5PS
    Color and Shape:Solid
    Molecular weight:367.25
  • Inolitazone dihydrochloride

    CAS:
    <p>Inolitazone dihydrochloride is an effective, high-affinity PPARγ agonist; its biological activity is dependent on PPARγ (IC50:0.8 nM) to inhibit cell growth.</p>
    Formula:C27H28Cl2N4O4S
    Color and Shape:Solid
    Molecular weight:575.51
  • SAR127303

    CAS:
    <p>SAR127303 is an effective covalent inhibitor of MAGL. SAR127303 behaves as a selective and competitive inhibitor of mouse and human MAGL.</p>
    Formula:C16H17ClF6N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:482.83
  • Niraparib metabolite M1

    CAS:
    <p>Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1) is the carboxylic acid metabolite of niraparib.</p>
    Formula:C19H19N3O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:321.37