GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(993 products)
- Adenosine Receptor(246 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(212 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(182 products)
- Hedgehog/Smoothened(47 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(310 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5745 products of "GPCR/G-Protein"
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Apraclonidine hydrochloride
CAS:<p>Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.</p>Formula:C9H11Cl3N4Purity:99.74%Color and Shape:SolidMolecular weight:281.57MRS-3777 hemioxalate
CAS:<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Formula:C17H19N5OC2H2O4Purity:97.10%Color and Shape:SolidMolecular weight:354.39WZ4141
CAS:WZ4141 is an intermediate in compound synthesis.Formula:C16H13N3O2Purity:98%Color and Shape:SolidMolecular weight:279.29Tegaserod
CAS:Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).Formula:C16H23N5OPurity:99.20% - 99.89%Color and Shape:SolidMolecular weight:301.39Neurotensin(8-13)
CAS:Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.Formula:C38H64N12O8Purity:99.95%Color and Shape:SolidMolecular weight:816.99rac-Propranolol-d7
CAS:Rac-Propranolol-d7 is the deuterated form of Rac-Propranolol. Propranolol is a β-adrenergic receptor antagonist that inhibits β1AR.Formula:C16H14D7NO2Color and Shape:SolidMolecular weight:266.39Zilpaterol-d7
CAS:<p>Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.</p>Formula:C14H12D7N3O2Color and Shape:SolidMolecular weight:268.36SB-277011 hydrochloride
CAS:<p>SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.</p>Formula:C28H31ClN4OPurity:98.54%Color and Shape:SolidMolecular weight:475.03Zagociguat
CAS:Zagociguat (CY6463) is a stimulator of guanylate cyclase that increases nitric oxide (NO) signaling and can be used in the research of neurological diseases.Formula:C16H10F4N6Purity:99.37%Color and Shape:SolidMolecular weight:362.28Hydroxyzine dihydrochloride-d4
CAS:Hydroxyzine dihydrochloride-d4 is a deuterated compound of Hydroxyzine dihydrochloride.Formula:C21H25D4Cl3N2O2Color and Shape:SolidMolecular weight:451.85TP-16
CAS:<p>TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs and enhances cytotoxic T cell-mediated tumor elimination in vivo.</p>Formula:C24H22FNO4SPurity:98.53% - 99.15%Color and Shape:SolidMolecular weight:439.5Eplivanserin (mixture)
CAS:Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,Formula:C19H21FN2O2Color and Shape:SolidMolecular weight:328.387Quetiapine-d8 Hemifumarate
CAS:Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formula:C25H21D8N3O6SColor and Shape:SolidMolecular weight:507.63GLP-1R modulator C16
CAS:GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.Formula:C21H26ClFN2O3Purity:99.6% - >99.99%Color and Shape:SolidMolecular weight:408.89LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Formula:C18H14FN5OPurity:99.03% - >99.99%Color and Shape:SolidMolecular weight:335.344-(4-Chlorobenzyl)phthalazin-1(2H)-one
CAS:4-(4-Chlorobenzyl)phthalazin-1(2H)-one is a useful organic compound for research related to life sciences. The catalog number is T67610 and the CAS number is 53242-88-9.Formula:C15H11ClN2OColor and Shape:SolidMolecular weight:270.72Setiptiline maleate
CAS:Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.Formula:C23H23NO4Purity:99.94%Color and Shape:SolidMolecular weight:377.43Piribedil D8
CAS:Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.Formula:C16H18N4O2Purity:98%Color and Shape:SolidMolecular weight:306.39Trimethobenzamide
CAS:<p>Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.</p>Formula:C21H28N2O5Color and Shape:SolidMolecular weight:388.46RU-SKI 43 Hydrochloride
CAS:RU-SKI 43 Hydrochloride is a selective Hedgehog acyltransferase inhibitor (IC50 850 nM) with reported anticancer activity in tumor biology studies.Formula:C22H31ClN2O2SPurity:98%Color and Shape:SolidMolecular weight:423.01Spiroxatrine
CAS:<p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>Formula:C22H25N3O3Purity:99.94%Color and Shape:SolidMolecular weight:379.45Fedovapagon
CAS:<p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>Formula:C27H34N4O3Purity:99.33%Color and Shape:SolidMolecular weight:462.58L 888607
CAS:L 888607 is an effective and selective CRTH2 agonist (Ki: 0.8 nM).Formula:C19H15ClFNO2SColor and Shape:SolidMolecular weight:375.84Ziprasidone D8
CAS:Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.Formula:C21H21ClN4OSPurity:98%Color and Shape:SolidMolecular weight:420.99Thiethylperazine
CAS:Thiethylperazine (Tietilperazina) is a D2 receptor and H1 receptor antagonist, and an ABCC1 activator with antimicrobial and antiemetic activity.Formula:C22H29N3S2Purity:98.72%Color and Shape:SolidMolecular weight:399.62Olanzapine D3
CAS:<p>Olanzapine D3 is the deuterium labeled Olanzapine.</p>Formula:C17H20N4SPurity:98%Color and Shape:SolidMolecular weight:315.45Ziprasidone amino acid
CAS:<p>Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.</p>Formula:C21H23ClN4O2SColor and Shape:SolidMolecular weight:430.95Calcium-Sensing Receptor Antagonists I
CAS:Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium.Formula:C23H24N2O2Color and Shape:SolidMolecular weight:360.45Levomepromazine
CAS:Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.Formula:C19H24N2OSPurity:99.15%Color and Shape:SolidMolecular weight:328.47Ivabradine-d6 hydrochloride
CAS:Ivabradine HCl: novel If inhibitor, IC50 2.9 μM; lowers heart rate. Ivabradine D6 HCl is its deuterium variant.Formula:C27H37ClN2O5Purity:98%Color and Shape:SolidMolecular weight:511.08(+)-Penbutolol
CAS:(+)-Penbutolol is an antagonist of β-adrenoceptor(IC50 of 0.74 μM). (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action.Formula:C18H29NO2Color and Shape:SolidMolecular weight:291.43SANT 2
CAS:SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.Formula:C26H26ClN3O4Purity:99.23%Color and Shape:SolidMolecular weight:479.96Cimbuterol-d9
CAS:<p>Cimbuterol-d9 is a deuterated compound of Cimbuterol.</p>Formula:C13H10D9N3OPurity:99.22%Color and Shape:SolidMolecular weight:242.37Lecirelin
CAS:Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.Formula:C59H84N16O12Color and Shape:SolidMolecular weight:1209.4Tiapride-d3
Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.Formula:C15H21D3N2O4SColor and Shape:SolidMolecular weight:331.45Brombuterol hydrochloride
CAS:Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.Formula:C12H19Br2ClN2OColor and Shape:SolidMolecular weight:402.56Methyldopate
CAS:<p>Methyldopate, an ethyl ester prodrug of methyldopa, inhibits dopamine decarboxylase to treat hypertension.</p>Formula:C12H17NO4Color and Shape:SolidMolecular weight:239.27Tetrahexyldecyl ascorbate
CAS:Tetrahexyldecyl ascorbate is a precursor of ascorbic acid, a more stable and permeable form of vitamin C. anti-hyperpigmentation antioxidant that inhibits MMP.Formula:C70H128O10Purity:98%Color and Shape:SolidMolecular weight:1129.76Propranolol-d7 hydrochloride
CAS:Propranolol D7 HCl: deuterium-labeled, nonselective βAR antagonist.Formula:C16H22ClNO2Purity:98%Color and Shape:SolidMolecular weight:302.85Metipranolol hydrochloride
CAS:Metipranolol hydrochloride is a non-selective β-adrenergic receptor blocking agent.Formula:C17H28ClNO4Purity:98%Color and Shape:SolidMolecular weight:345.86Acrivastine D7
CAS:Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.Formula:C22H24N2O2Purity:98%Color and Shape:SolidMolecular weight:355.48Bombesin
CAS:Bombesin: 14-amino acid peptide from toad skin with two mammalian homologs, neuromedin B and gastrin-releasing peptide.Formula:C71H110N24O18SColor and Shape:While Lyophilized PowderMolecular weight:1619.85GRK2 Inhibitor
CAS:GRK2 Inhibitor is an inhibitor of β-Adrenergic Receptor Kinase 1 (β ARK1).Formula:C12H9NO6Color and Shape:SolidMolecular weight:263.2Benoxathian hydrochloride
CAS:Benoxathian hydrochloride is effective α 1 Adrenaline receptor antagonist. Benoxathian hydrochloride has value in the study of anorexia.Formula:C19H24ClNO4SColor and Shape:SolidMolecular weight:397.91β2AR/M-receptor agonist-2
CAS:<p>β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).</p>Formula:C36H49ClN4O7SColor and Shape:SolidMolecular weight:717.31GLP-1 receptor agonist 2
CAS:GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C30H31ClFN5O4Color and Shape:SolidMolecular weight:580.05Ceralifimod
CAS:Ceralifimod (ONO-4641) is a potent agonist for sphingosine 1-phosphate receptors 1 and 5 (EC50s: 27.3, 334 pM for human S1P receptor 1 and 5).Formula:C27H33NO4Color and Shape:SolidMolecular weight:435.56MK-761 TFA
<p>MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.</p>Formula:C15H20F3N3O4Color and Shape:SolidMolecular weight:363.332Mozavaptan hydrochloride
CAS:Mozavaptan is a vasopressin receptor antagonist.Formula:C27H30ClN3O2Color and Shape:SolidMolecular weight:464MrgprX2 antagonist-1
CAS:MrgprX2 antagonist-1 (compound E23) is a MrgprX2 antagonist applicable to cutaneous inflammation.Formula:C15H15F5N4O2SPurity:99.80%Molecular weight:410.36Canagliflozin (Standard)
CAS:Canagliflozin (Standard) is the standard substance of Canagliflozin, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor that inhibits CHO cells expressing mSGLT2, rSGLT2, and hSGLT2 (IC50=2/3.7/4.4 nM). Canagliflozin can be used for the treatment of type II diabetes mellitus (T2DM).Formula:C24H25FO5SMolecular weight:444.52Bradykinin (1-5)
CAS:Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Formula:C27H40N8O6Color and Shape:SolidMolecular weight:572.66Cetirizine D8
CAS:Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Formula:C21H25ClN2O3Purity:98%Color and Shape:SolidMolecular weight:396.94(S)-ZINC-3573
CAS:(S)-ZINC 3573 is a negative control for (R)-ZINC 3573. (S)-ZINC 3573 displays no activity at MRGPRX2 at concentrations below 100 μM.Formula:C18H21N5Color and Shape:SolidMolecular weight:307.401Endothelin-3 (Rat,Human) (TFA)
<p>Endothelin-3 (Rat, Human) (TFA) is a 21-amino acid vasoactive peptide of endothelial origi, an agonist for the endothelin receptor type B (EDNRB).</p>Formula:C123H169F3N26O35S4·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:2757.07 (free base)SAR247799
CAS:SAR247799 is a selective and G-protein-biased S1P1 agonist that activates downstream G-protein signaling pathways more preferentially on endothelial cells.Formula:C21H16ClN3O5Color and Shape:SolidMolecular weight:425.82Timapiprant sodium
CAS:Timapiprant sodium: potent DP2 antagonist; inhibits mast cell activation; displaces [3H]PGD2, Ki=3-13 nM.Formula:C21H17FN2NaO2Purity:98%Color and Shape:SolidMolecular weight:371.367Altanserin
CAS:Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.Formula:C22H22FN3O2SColor and Shape:SolidMolecular weight:411.494-Hydroxypropranolol-d7 hydrochloride
CAS:<p>Deuterium-labeled 4-Hydroxypropranolol HCl, a Propranolol metabolite that blocks β1/β2 receptors.</p>Formula:C16H22ClNO3Purity:98%Color and Shape:SolidMolecular weight:318.85Doxepin D3 Hydrochloride
CAS:Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 andFormula:C19H22ClNOPurity:98%Color and Shape:SolidMolecular weight:318.86Emedastine Difumarate
CAS:Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.Formula:C25H34N4O9Color and Shape:SolidMolecular weight:534.56Substance P TFA
CAS:Substance P TFA is a CNS neuropeptide, serving as a neurotransmitter and modulator, targeting NK1R.Formula:C65H99F3N18O15SPurity:98%Color and Shape:SolidMolecular weight:1461.67Diacetolol D7
CAS:<p>Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.</p>Formula:C16H24N2O4Purity:98%Color and Shape:SolidMolecular weight:315.42Diphenylpyraline
CAS:<p>Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.</p>Formula:C19H23NOColor and Shape:SolidMolecular weight:281.39Doxazosin D8
CAS:Doxazosin D8, a deuterium-labeled version, is a selective AP1 adrenergic antagonist and a quinazoline derivative.Formula:C23H25N5O5Purity:98%Color and Shape:SolidMolecular weight:459.52R121919
CAS:R121919 (NBI30775) is an adrenocorticotropin-releasing factor receptor 1 (CRF1) receptor antagonist with antidepressant and anxiolytic activity.Formula:C22H32N6Purity:99.75%Color and Shape:SolidMolecular weight:380.53Tulobuterol-d9 HCl
CAS:Tulobuterol-d9 HCl is a deuterated compound of Tulobuterol HCl.Formula:C12H10D9Cl2NOMolecular weight:273.25GB-88
CAS:GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.Formula:C32H42N4O4Color and Shape:SolidMolecular weight:546.7SUN B8155
CAS:SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant human CT receptor.Formula:C14H15N3O3Purity:99.38% - 99.38%Color and Shape:SolidMolecular weight:273.29Cudarolimab
CAS:<p>Cudarolimab (IBI-101) is a fully human anti-OX40 antibody with potential immune checkpoint inhibitory and anti-tumor activity for the study of cancer.</p>Purity:97.5% (SDS-PAGE); 98.2% (SEC-HPLC) - 97.5% (SDS-PAGE); 98.2% (SEC-HPLC)Color and Shape:LiquidLevosalbutamol Hydrochloride
CAS:Levosalbutamol Hydrochloride is a β2-adrenergic receptor agonist. It is used to treat asthma and chronic obstructive pulmonary disease.Formula:C13H22ClNO3Purity:98%Color and Shape:SolidMolecular weight:275.77Flibanserin-d4
CAS:<p>Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.</p>Formula:C20H21F3N4OPurity:98%Color and Shape:SolidMolecular weight:394.43ML224
CAS:<p>ML224 (NCGC00242364) is a TSHR antagonist for the treatment of Graves' orbital disease and Graves' hyperthyroidism.</p>Formula:C31H31N3O5Purity:99.14%Color and Shape:SolidMolecular weight:525.591-Phenylbiguanide HCl
CAS:<p>Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.</p>Formula:C8H12ClN5Purity:99.31%Color and Shape:SolidMolecular weight:213.67Alosetron D3 Hydrochloride
CAS:<p>Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>Formula:C17H19ClN4OPurity:98%Color and Shape:SolidMolecular weight:333.83Dapagliflozin impurity
CAS:Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.Formula:C21H25ClO7Color and Shape:SolidMolecular weight:424.87Fexofenadine-d6
CAS:Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.Formula:C32H39NO4Purity:98%Color and Shape:SolidMolecular weight:507.69Lanreotide
CAS:Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Formula:C54H69N11O10S2Color and Shape:SolidMolecular weight:1096.32Terlipressin
CAS:Terlipressin is a potent vasoconstrictor that acts via V1 receptors on arteriolar smooth muscle cells.Formula:C52H74N16O15S2Purity:98%Color and Shape:SolidMolecular weight:1227.37Fipexide hydrochloride
CAS:Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Formula:C20H22Cl2N2O4Color and Shape:SolidMolecular weight:425.315-HT2B antagonist-1
CAS:Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.Formula:C11H14BrN5Purity:99.965%Color and Shape:SolidMolecular weight:296.17Cefaclor
CAS:Cefaclor (Panoral) is a cephalosporin antibiotic.Formula:C15H14ClN3O4SPurity:99.03% - 99.98%Color and Shape:SolidMolecular weight:367.81Antazoline phosphate
CAS:Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.Formula:C17H22N3O4PPurity:98%Color and Shape:CoaMolecular weight:363.35NBI-27914
CAS:<p>NBI-27914 is a selective and non-peptide CRFR1 (corticotropin-releasing factor receptor 1) antagonist with analgesic effects, capable of blocking CRF-induced anxiety.</p>Formula:C18H20Cl4N4Purity:99.47% - 99.64%Color and Shape:SolidMolecular weight:434.19Dehydroaripiprazole
CAS:Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.Formula:C23H25Cl2N3O2Purity:98.7%Color and Shape:SolidMolecular weight:446.37SKF-82958 hydrobromide
CAS:SKF-82958 hydrobromide is a D1/D5 receptor full agonist.Formula:C19H21BrClNO2Purity:98%Color and Shape:SolidMolecular weight:410.73Ramelteon-d5
CAS:<p>Ramelteon-d5 is a deuterated compound of Ramelteon.</p>Formula:C16H16D5NO2Color and Shape:SolidMolecular weight:264.37Clomipramine D3 hydrochloride
CAS:Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).Formula:C19H24Cl2N2Color and Shape:SolidMolecular weight:354.33Etofylline clofibrate
CAS:Etofylline clofibrate has a hypolipidemic and antithrombotic effect and it also has an agonistic interaction with intimal PGI2.Formula:C19H21ClN4O5Color and Shape:SolidMolecular weight:420.85Thioridazine
CAS:Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.Formula:C21H26N2S2Color and Shape:SolidMolecular weight:370.57Nadolol-d9
CAS:<p>Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.</p>Formula:C17H27NO4Purity:98%Color and Shape:SolidMolecular weight:318.46(R)-Praziquantel-d11
CAS:(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:323.47Vilazodone-d8
CAS:Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.Formula:C26H27N5O2Purity:98%Color and Shape:SolidMolecular weight:449.57Fluvoxamine
CAS:Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.Formula:C15H21F3N2O2Purity:99.91%Color and Shape:SolidMolecular weight:318.33JNJ-10397049
CAS:OX2 receptor antagonistFormula:C19H20Br2N2O3Color and Shape:SolidMolecular weight:484.18SB-674042
CAS:SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is used in the treatment of depression.Formula:C24H21FN4O2SPurity:99.9%Color and Shape:SolidMolecular weight:448.51Clorprenaline
CAS:Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formula:C11H16ClNOPurity:98.9%Color and Shape:SolidMolecular weight:213.7GLP-1 receptor agonist 7
CAS:GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.Formula:C31H30ClFN4O5Color and Shape:SolidMolecular weight:593.05Dexloxiglumide
CAS:Dexloxiglumide is the active enantiomer of Loxiglumide; it inhibits CCK-8-induced contractions and is a selective CCKA receptor antagonist.Formula:C21H30Cl2N2O5Color and Shape:SolidMolecular weight:461.38Cariprazine D6
CAS:<p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>Formula:C21H26D6Cl2N4OPurity:98%Color and Shape:SolidMolecular weight:433.45
