GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,003 products)
- Adenosine Receptor(247 products)
- Adrenergic Receptor(3,010 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(60 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(215 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(435 products)
- Endothelin Receptor(83 products)
- GNRH Receptor(82 products)
- GPCR19(33 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(190 products)
- Hedgehog/Smoothened(48 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(321 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5838 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
GR79236
CAS:GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Formula:C15H21N5O5Color and Shape:SolidMolecular weight:351.36LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Formula:C18H14FN5OPurity:99.03% - >99.99%Color and Shape:SolidMolecular weight:335.34JNJ-10397049
CAS:OX2 receptor antagonistFormula:C19H20Br2N2O3Color and Shape:SolidMolecular weight:484.18Omidenepag
CAS:Omidenepag (UR-7276) is an EP2 agonist and a novel topical ocular hypotensive agent.Omidenepag can be used to study glaucoma and hypertension.Formula:C23H22N6O4SPurity:99.67% - 99.77%Color and Shape:SolidMolecular weight:478.52Calcitonin (salmon)
CAS:<p>Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.</p>Formula:C145H240N44O48S2Purity:99.41% - 99.80%Color and Shape:PowderMolecular weight:3431.85Lecirelin
CAS:Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.Formula:C59H84N16O12Color and Shape:SolidMolecular weight:1209.4V-0219
CAS:V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.Formula:C20H25F3N4O2Purity:99.91%Color and Shape:SoildMolecular weight:410.43SB-200646A
CAS:SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.Formula:C15H15ClN4OPurity:98%Color and Shape:SolidMolecular weight:302.76SKF-82958 hydrobromide
CAS:SKF-82958 hydrobromide is a D1/D5 receptor full agonist.Formula:C19H21BrClNO2Purity:98%Color and Shape:SolidMolecular weight:410.73Fipexide hydrochloride
CAS:Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Formula:C20H22Cl2N2O4Color and Shape:SolidMolecular weight:425.31Clothiapine
CAS:Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Formula:C18H18ClN3SPurity:99.93%Color and Shape:SolidMolecular weight:343.87Flibanserin-d4
CAS:<p>Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.</p>Formula:C20H21F3N4OPurity:98%Color and Shape:SolidMolecular weight:394.43Asenapine
CAS:Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophreniaFormula:C17H16ClNOPurity:99.64%Color and Shape:CoaMolecular weight:285.77Scopine hydrochloride
CAS:<p>Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist.</p>Formula:C8H13NO2·HClPurity:98%Color and Shape:White PowderMolecular weight:191.66SLIGRL-NH2
CAS:SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a PAR-2 agonist that induces non-histaminergic pruritus.Formula:C29H56N10O7Purity:98.29%Color and Shape:SolidMolecular weight:656.82Endothelin-3 (Rat,Human) (TFA)
<p>Endothelin-3 (Rat, Human) (TFA) is a 21-amino acid vasoactive peptide of endothelial origi, an agonist for the endothelin receptor type B (EDNRB).</p>Formula:C123H169F3N26O35S4·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:2757.07 (free base)GLP-1R modulator C5
CAS:GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.Formula:C24H21NO3Purity:99.59%Color and Shape:SolidMolecular weight:371.43GLP-1R modulator C16
CAS:GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.Formula:C21H26ClFN2O3Purity:99.6% - >99.99%Color and Shape:SolidMolecular weight:408.89GLP-1R modulator L7-028
CAS:GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.Formula:C24H28N2O3Purity:98.76% - >99.99%Color and Shape:SolidMolecular weight:392.49GLP-1 receptor agonist 2
CAS:GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C30H31ClFN5O4Color and Shape:SolidMolecular weight:580.05Calcium-Sensing Receptor Antagonists I
CAS:Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium.Formula:C23H24N2O2Color and Shape:SolidMolecular weight:360.454-Hydroxyatomoxetine D3
CAS:<p>4-Hydroxyatomoxetine D3, a deuterium variant, is Atomoxetine's active metabolite, metabolized by CYP2D6, an adrenergic reuptake blocker.</p>Formula:C17H21NO2Purity:98%Color and Shape:SolidMolecular weight:274.37Olanzapine D3
CAS:<p>Olanzapine D3 is the deuterium labeled Olanzapine.</p>Formula:C17H20N4SPurity:98%Color and Shape:SolidMolecular weight:315.45SB-269970 hydrochloride
CAS:SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivityFormula:C18H28N2O3S·HClPurity:99.8%Color and Shape:SolidMolecular weight:388.95Ziprasidone D8
CAS:Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.Formula:C21H21ClN4OSPurity:98%Color and Shape:SolidMolecular weight:420.99TFLLR-NH2(TFA)
CAS:TFLLR-NH2 (TFA) is a selective PAR1 agonist with an EC50 of 1.9 μM. EC50: 1.9 μM (PAR1)Formula:C33H54F3N9O8Purity:98%Color and Shape:SolidMolecular weight:761.83SB-408124 Hydrochloride
CAS:SB-408124 Hydrochloride is a non-peptide OX1 receptor antagonist(Ki of 57 nM and 27 nM in both whole cell and membrane, respectively).Formula:C19H19ClF2N4OPurity:98%Color and Shape:SolidMolecular weight:392.83Trimethobenzamide
CAS:<p>Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.</p>Formula:C21H28N2O5Color and Shape:SolidMolecular weight:388.46Piribedil D8
CAS:Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.Formula:C16H18N4O2Purity:98%Color and Shape:SolidMolecular weight:306.39GSK682753A
CAS:GSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2; IC50: 53.6 nM).Formula:C23H21Cl3N2O3Color and Shape:SolidMolecular weight:479.78YNT-185 dihydrochloride
CAS:<p>Potent OX2 agonist (EC50=28nM); 100x selective over OX1; prompts wakefulness, counters cataplexy in mice.</p>Formula:C33H39Cl2N5O5SColor and Shape:SolidMolecular weight:688.67Asenapine hydrochloride
CAS:<p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>Formula:C17H17Cl2NOColor and Shape:SolidMolecular weight:322.23Haloperidol (D4')
CAS:Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.Formula:C21H23ClFNO2Purity:98%Color and Shape:SolidMolecular weight:379.89ST-836 hydrochloride
CAS:ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .Formula:C23H35ClN4OSPurity:98%Color and Shape:SolidMolecular weight:451.07Paliperidone Palmitate
CAS:Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.Formula:C39H57FN4O4Purity:98%Color and Shape:SolidMolecular weight:664.89PSB-0739
CAS:PSB-0739 Selective platelet P2Y12 receptor antagonist characterized by competitive binding with antithrombotic and platelet aggregation modulating effects.Formula:C26H17N3Na2O8S2Purity:98%Color and Shape:SolidMolecular weight:609.54Telcagepant
CAS:Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.Formula:C26H27F5N6O3Purity:98.98% - 98.98%Color and Shape:SolidMolecular weight:566.52Zagociguat
CAS:Zagociguat (CY6463) is a stimulator of guanylate cyclase that increases nitric oxide (NO) signaling and can be used in the research of neurological diseases.Formula:C16H10F4N6Purity:99.37%Color and Shape:SolidMolecular weight:362.28Diphenylpyraline
CAS:<p>Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.</p>Formula:C19H23NOColor and Shape:SolidMolecular weight:281.39Quetiapine-d4 hemifumarate
CAS:<p>Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.</p>Formula:C25H29N3O6SPurity:98%Color and Shape:White SolidMolecular weight:503.61Agomelatine-d6
CAS:Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.Formula:C15H17NO2Purity:98%Color and Shape:SolidMolecular weight:249.34Glucagon (1-29), bovine, human, porcine
CAS:Corynoxine B (Cory B) is a naturally occurring alkaloid isolated from Uncaria rhynchophylla (Miq. ) and is an autophagy inducer.Formula:C153H225N43O49SPurity:99.56% - 99.56%Color and Shape:SolidMolecular weight:3482.75Ipragliflozin (L-Proline)
CAS:Ipragliflozin is a highly potent and selective SGLT2 inhibitor with an IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6.Formula:C26H30FNO7SColor and Shape:SolidMolecular weight:519.58Sumatriptan
CAS:Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.Formula:C14H21N3O2SPurity:99.93%Color and Shape:White To Off-White Crystalline PowderMolecular weight:295.4Virodhamine
CAS:<p>Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.</p>Formula:C22H37NO2Purity:98%Color and Shape:SoildMolecular weight:347.53Alimemazine D6
CAS:Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.Formula:C18H22N2SPurity:98%Color and Shape:SolidMolecular weight:304.48Aripiprazole (D8)
CAS:Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).Formula:C23H27Cl2N3O2Purity:98%Color and Shape:SolidMolecular weight:456.44Dexloxiglumide
CAS:Dexloxiglumide is the active enantiomer of Loxiglumide; it inhibits CCK-8-induced contractions and is a selective CCKA receptor antagonist.Formula:C21H30Cl2N2O5Color and Shape:SolidMolecular weight:461.38Thiethylperazine
CAS:Thiethylperazine (Tietilperazina) is a D2 receptor and H1 receptor antagonist, and an ABCC1 activator with antimicrobial and antiemetic activity.Formula:C22H29N3S2Purity:98.72%Color and Shape:SolidMolecular weight:399.62Clorprenaline
CAS:Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formula:C11H16ClNOPurity:98.9%Color and Shape:SolidMolecular weight:213.7(R)-Praziquantel-d11
CAS:(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:323.47Nadolol-d9
CAS:<p>Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.</p>Formula:C17H27NO4Purity:98%Color and Shape:SolidMolecular weight:318.46Clencyclohexerol-d10
CAS:Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.Formula:C14H20Cl2N2O2Color and Shape:SolidMolecular weight:329.29NBI-27914
CAS:<p>NBI-27914 is a selective and non-peptide CRFR1 (corticotropin-releasing factor receptor 1) antagonist with analgesic effects, capable of blocking CRF-induced anxiety.</p>Formula:C18H20Cl4N4Purity:99.47% - 99.64%Color and Shape:SolidMolecular weight:434.19Antazoline phosphate
CAS:Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.Formula:C17H22N3O4PPurity:98%Color and Shape:CoaMolecular weight:363.35Cefaclor
CAS:Cefaclor (Panoral) is a cephalosporin antibiotic.Formula:C15H14ClN3O4SPurity:99.03% - 99.98%Color and Shape:SolidMolecular weight:367.81Terlipressin
CAS:Terlipressin is a potent vasoconstrictor that acts via V1 receptors on arteriolar smooth muscle cells.Formula:C52H74N16O15S2Purity:98%Color and Shape:SolidMolecular weight:1227.37Tiapride-d3
Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.Formula:C15H21D3N2O4SColor and Shape:SolidMolecular weight:331.45Dapagliflozin impurity
CAS:Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.Formula:C21H25ClO7Color and Shape:SolidMolecular weight:424.87Cimbuterol-d9
CAS:<p>Cimbuterol-d9 is a deuterated compound of Cimbuterol.</p>Formula:C13H10D9N3OPurity:99.22%Color and Shape:SolidMolecular weight:242.37Zilpaterol-d7
CAS:<p>Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.</p>Formula:C14H12D7N3O2Color and Shape:SolidMolecular weight:268.36R121919
CAS:R121919 (NBI30775) is an adrenocorticotropin-releasing factor receptor 1 (CRF1) receptor antagonist with antidepressant and anxiolytic activity.Formula:C22H32N6Purity:99.75%Color and Shape:SolidMolecular weight:380.53Diacetolol D7
CAS:<p>Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.</p>Formula:C16H24N2O4Purity:98%Color and Shape:SolidMolecular weight:315.42Substance P TFA
CAS:Substance P TFA is a CNS neuropeptide, serving as a neurotransmitter and modulator, targeting NK1R.Formula:C65H99F3N18O15SPurity:98%Color and Shape:SolidMolecular weight:1461.67Doxepin D3 Hydrochloride
CAS:Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 andFormula:C19H22ClNOPurity:98%Color and Shape:SolidMolecular weight:318.864-Hydroxypropranolol-d7 hydrochloride
CAS:Deuterium-labeled 4-Hydroxypropranolol HCl, a Propranolol metabolite that blocks β1/β2 receptors.Formula:C16H22ClNO3Purity:98%Color and Shape:SolidMolecular weight:318.85Altanserin
CAS:Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.Formula:C22H22FN3O2SColor and Shape:SolidMolecular weight:411.49Timapiprant sodium
CAS:Timapiprant sodium: potent DP2 antagonist; inhibits mast cell activation; displaces [3H]PGD2, Ki=3-13 nM.Formula:C21H17FN2NaO2Purity:98%Color and Shape:SolidMolecular weight:371.367(S)-ZINC-3573
CAS:(S)-ZINC 3573 is a negative control for (R)-ZINC 3573. (S)-ZINC 3573 displays no activity at MRGPRX2 at concentrations below 100 μM.Formula:C18H21N5Color and Shape:SolidMolecular weight:307.401Bradykinin (1-5)
CAS:Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Formula:C27H40N8O6Color and Shape:SolidMolecular weight:572.66SB-674042
CAS:SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is used in the treatment of depression.Formula:C24H21FN4O2SPurity:99.9%Color and Shape:SolidMolecular weight:448.51MK-761 TFA
MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.Formula:C15H20F3N3O4Color and Shape:SolidMolecular weight:363.332Ceralifimod
CAS:Ceralifimod (ONO-4641) is a potent agonist for sphingosine 1-phosphate receptors 1 and 5 (EC50s: 27.3, 334 pM for human S1P receptor 1 and 5).Formula:C27H33NO4Color and Shape:SolidMolecular weight:435.56β2AR/M-receptor agonist-2
CAS:<p>β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).</p>Formula:C36H49ClN4O7SColor and Shape:SolidMolecular weight:717.31Bombesin
CAS:Bombesin: 14-amino acid peptide from toad skin with two mammalian homologs, neuromedin B and gastrin-releasing peptide.Formula:C71H110N24O18SColor and Shape:While Lyophilized PowderMolecular weight:1619.85Docosahexaenoic acid ethyl ester
CAS:Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.Formula:C24H36O2Purity:98.35%Color and Shape:SolidMolecular weight:356.54Metipranolol hydrochloride
CAS:Metipranolol hydrochloride is a non-selective β-adrenergic receptor blocking agent.Formula:C17H28ClNO4Purity:98%Color and Shape:SolidMolecular weight:345.86Propranolol-d7 hydrochloride
CAS:Propranolol D7 HCl: deuterium-labeled, nonselective βAR antagonist.Formula:C16H22ClNO2Purity:98%Color and Shape:SolidMolecular weight:302.85Doxazosin D8
CAS:Doxazosin D8, a deuterium-labeled version, is a selective AP1 adrenergic antagonist and a quinazoline derivative.Formula:C23H25N5O5Purity:98%Color and Shape:SolidMolecular weight:459.52GB-88
CAS:GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.Formula:C32H42N4O4Color and Shape:SolidMolecular weight:546.7Tetrahexyldecyl ascorbate
CAS:Tetrahexyldecyl ascorbate is a precursor of ascorbic acid, a more stable and permeable form of vitamin C. anti-hyperpigmentation antioxidant that inhibits MMP.Formula:C70H128O10Purity:98%Color and Shape:SolidMolecular weight:1129.76Alosetron D3 Hydrochloride
CAS:<p>Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>Formula:C17H19ClN4OPurity:98%Color and Shape:SolidMolecular weight:333.83Clomipramine D3 hydrochloride
CAS:Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).Formula:C19H24Cl2N2Color and Shape:SolidMolecular weight:354.33Brombuterol hydrochloride
CAS:Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.Formula:C12H19Br2ClN2OColor and Shape:SolidMolecular weight:402.56Vilazodone-d8
CAS:Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.Formula:C26H27N5O2Purity:98%Color and Shape:SolidMolecular weight:449.57Cimetidine (Standard)
CAS:Cimetidine (Standard) is the standard substance of Cimetidine, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological actions. It inhibits GASTRIC ACID secretion, as well as PEPSIN and GASTRIN output.Formula:C10H16N6SMolecular weight:252.34(+)-Penbutolol
CAS:(+)-Penbutolol is an antagonist of β-adrenoceptor(IC50 of 0.74 μM). (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action.Formula:C18H29NO2Color and Shape:SolidMolecular weight:291.43Ivabradine-d6 hydrochloride
CAS:Ivabradine HCl: novel If inhibitor, IC50 2.9 μM; lowers heart rate. Ivabradine D6 HCl is its deuterium variant.Formula:C27H37ClN2O5Purity:98%Color and Shape:SolidMolecular weight:511.08SBI-810 hydrochloride
CAS:SBI-810 hydrochloride is a β-arrestin-2 (βarr2)-biased allosteric modulator of NTSR1 (neurotensin receptor 1), exerting analgesic effects.Formula:C27H35ClN4O2Purity:99.42%Molecular weight:483.05ML 00253764
CAS:melanocortin MC4 receptor antagonistFormula:C18H18BrFN2OColor and Shape:SolidMolecular weight:377.25Tiotidine
CAS:Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).Formula:C10H16N8S2Purity:98%Color and Shape:SolidMolecular weight:312.42RU-SKI 43 Hydrochloride
CAS:RU-SKI 43 Hydrochloride is a selective Hedgehog acyltransferase inhibitor (IC50 850 nM) with reported anticancer activity in tumor biology studies.Formula:C22H31ClN2O2SPurity:98%Color and Shape:SolidMolecular weight:423.01Dehydroaripiprazole
CAS:Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.Formula:C23H25Cl2N3O2Purity:98.7%Color and Shape:SolidMolecular weight:446.37Levosalbutamol Hydrochloride
CAS:Levosalbutamol Hydrochloride is a β2-adrenergic receptor agonist. It is used to treat asthma and chronic obstructive pulmonary disease.Formula:C13H22ClNO3Purity:98%Color and Shape:SolidMolecular weight:275.77Cudarolimab
CAS:<p>Cudarolimab (IBI-101) is a fully human anti-OX40 antibody with potential immune checkpoint inhibitory and anti-tumor activity for the study of cancer.</p>Purity:97.5% (SDS-PAGE); 98.2% (SEC-HPLC) - 97.5% (SDS-PAGE); 98.2% (SEC-HPLC)Color and Shape:LiquidCetirizine D8
CAS:Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Formula:C21H25ClN2O3Purity:98%Color and Shape:SolidMolecular weight:396.94Mozavaptan hydrochloride
CAS:Mozavaptan is a vasopressin receptor antagonist.Formula:C27H30ClN3O2Color and Shape:SolidMolecular weight:464Methyldopate
CAS:Methyldopate, an ethyl ester prodrug of methyldopa, inhibits dopamine decarboxylase to treat hypertension.Formula:C12H17NO4Color and Shape:SolidMolecular weight:239.275-HT3 antagonist 5
CAS:5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.Formula:C16H13N3O2Purity:99.84%Color and Shape:SolidMolecular weight:279.29Allura Red AC (Standard)
CAS:Allura Red AC (Standard) is the standard substance of Allura Red AC, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Allura Red AC (CI 16035) is a very important food azo dye used in the food, pharmaceutical, paper, cosmetic and textile industries.Allura Red AC promotes susceptibility to experimental colitis via mouse intestinal serotonin.Formula:C18H14N2Na2O8S2Color and Shape:Dark Maroon Solid PowderMolecular weight:496.42
