GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(985 products)
- Adenosine Receptor(244 products)
- Adrenergic Receptor(2,991 products)
- Bombesin Receptor(32 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(209 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(181 products)
- Hedgehog/Smoothened(46 products)
- Histamine Receptor(380 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(309 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5696 products of "GPCR/G-Protein"
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(E)-3,4,5-Trimethoxycinnamic acid
CAS:<p>(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.</p>Formula:C12H14O5Purity:99.83%Color and Shape:SolidMolecular weight:238.24Loxiglumide
CAS:<p>Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor.</p>Formula:C21H30Cl2N2O5Purity:97.55% - 99.81%Color and Shape:SolidMolecular weight:461.38Opaganib
CAS:<p>Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).</p>Formula:C23H25ClN2OPurity:98.86% - 99.85%Color and Shape:SolidMolecular weight:380.91BETP
CAS:<p>BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).</p>Formula:C20H17F3N2O2SPurity:98.51%Color and Shape:SolidMolecular weight:406.42Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFormula:C49H70N12O13Purity:99.93%Color and Shape:SolidMolecular weight:1035.15Preladenant
CAS:<p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine</p>Formula:C25H29N9O3Purity:98.02% - 99.68%Color and Shape:SolidMolecular weight:503.56AM1241
CAS:<p>AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.</p>Formula:C22H22IN3O3Purity:98.937% - 99.1%Color and Shape:SolidMolecular weight:503.33[Sar9] Substance P acetate(77128-75-7 free base)
<p>[Sar9]-Substance P acetate, an NK-1 receptor agonist, mimics SP's effect on progesterone metabolism.</p>Formula:C66H104N18O15SPurity:96.67%Color and Shape:SolidMolecular weight:1421.71Ponesimod
CAS:<p>Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating activity.</p>Formula:C23H25ClN2O4SPurity:99.42% - 99.96%Color and Shape:SolidMolecular weight:460.97HCGRP-(8-37) acetate
<p>HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.</p>Formula:C141H234N44O40Purity:99.29%Color and Shape:SolidMolecular weight:3185.64Ibrolipim
CAS:<p>Ibrolipim (NO-1886) attenuates high glucose-induced endothelial dysfunction in cultured human umbilical vein endothelial cells via PI3K/Akt pathway.</p>Formula:C19H20BrN2O4PPurity:98.04%Color and Shape:SolidMolecular weight:451.25Amitriptyline
CAS:<p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>Formula:C20H23NPurity:98.24% - 99.64%Color and Shape:Crystals SolidMolecular weight:277.4Siramesine
CAS:Siramesine (Lu 28-179)(Lu 28-179) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of cancer cells and to exhibit a potentFormula:C30H31FN2OPurity:98%Color and Shape:SolidMolecular weight:454.58[Sar9,Met(O2)11]-Substance P acetate
<p>[Sar9,Met(O2)11]-Substance P acetate is an NK1 agonist, raising MAP and HR equally to septide but with unique timing and behaviors.</p>Formula:C66H106N18O18SPurity:>99.99%Color and Shape:SolidMolecular weight:1471.75BD 1008 dihydrobromide
CAS:<p>BD 1008 dihydrobromide: selective σ1 receptor antagonist (Ki=2 nM), high σ1 and moderate σ2 affinity.</p>Formula:C15H24Br2Cl2N2Purity:97.81%Color and Shape:SolidMolecular weight:463.08Almotriptan
CAS:Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Formula:C17H25N3O2SPurity:99.85%Color and Shape:Light Yellow Or White PowerMolecular weight:335.46[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS:Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).Formula:C39H65N9O9Purity:>99.99%Color and Shape:SolidMolecular weight:803.99FAUC 346
CAS:FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.Formula:C24H29N3O2SPurity:99.46%Color and Shape:SolidMolecular weight:423.57Neuropeptide S (Mouse) acetate
Neuropeptide S (Mouse) acetate is a bioactive peptide.Formula:C95H160N34O29Purity:98.25%Color and Shape:SolidMolecular weight:2242.5S26131
CAS:<p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>Formula:C31H34N2O4Purity:99.77%Color and Shape:SolidMolecular weight:498.61PU02
CAS:<p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>Formula:C16H12N4SPurity:99.35%Color and Shape:SolidMolecular weight:292.36MIPS521
CAS:MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Formula:C19H10ClF6NOSPurity:99.76%Color and Shape:SolidMolecular weight:449.8ML-178
CAS:ML-178: selective S1PR4 agonist, EC50 of 46 nM; inactive on other S1P receptors at 25 μM.Formula:C13H9Br2Cl2NO2Purity:95.92%Color and Shape:SolidMolecular weight:441.93ML417
CAS:ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).Formula:C22H25N3O3Purity:98.4% - 99.42%Color and Shape:SolidMolecular weight:379.45Rizatriptan benzoate
CAS:<p>Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraine</p>Formula:C22H25N5O2Purity:99% - 99.79%Color and Shape:White To Off-White Crystalline PowderMolecular weight:391.47SB 204741
CAS:SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.Formula:C14H14N4OSPurity:99.83%Color and Shape:SolidMolecular weight:286.35Istradefylline
CAS:<p>Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.</p>Formula:C20H24N4O4Purity:98.18% - 99.95%Color and Shape:SolidMolecular weight:384.43H4 Receptor antagonist 1
CAS:H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formula:C16H17ClN4OPurity:98.81%Color and Shape:SolidMolecular weight:316.791-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
CAS:<p>1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.</p>Formula:C13H13NO5Purity:99.55%Color and Shape:SolidMolecular weight:263.25AZD4635
CAS:AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Formula:C15H11ClFN5Purity:99.15% - 99.90%Color and Shape:SolidMolecular weight:315.73RVD-Hpα acetate(1193362-76-3 free base)
<p>RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>Formula:C67H109N19O19Purity:99.87%Color and Shape:SolidMolecular weight:1484.71BIM-23190 aceate
<p>BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.</p>Formula:C59H83N13O14S2Purity:99.7%Color and Shape:SolidMolecular weight:1262.5Trazodone
CAS:<p>Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.</p>Formula:C19H22ClN5OPurity:99.79% - 99.92%Color and Shape:White To Off-White Crystalline PowderMolecular weight:371.86LP-211
CAS:LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.Formula:C30H34N4OPurity:98.65%Color and Shape:SolidMolecular weight:466.62Montelukast
CAS:<p>Montelukast (Singular), oral asthma med, linked to rare liver injury.</p>Formula:C35H36ClNO3SPurity:98.56% - >99.99%Color and Shape:SolidMolecular weight:586.18Ramosetron hydrochloride
CAS:<p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>Formula:C17H18ClN3OPurity:99.95%Color and Shape:SolidMolecular weight:315.8Harmine
CAS:Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.Formula:C13H12N2OPurity:98.29% - 99.92%Color and Shape:Off-White SolidMolecular weight:212.25(R)-Propranolol hydrochloride
CAS:(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.Formula:C16H22ClNO2Purity:98.63% - 99.01%Color and Shape:SolidMolecular weight:295.8Capromorelin Tartrate
CAS:<p>Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).</p>Formula:C32H41N5O10Purity:97.69%Color and Shape:SolidMolecular weight:655.7Vanoxerine dihydrochloride
CAS:<p>Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)</p>Formula:C28H34Cl2F2N2OPurity:98.16% - 98.35%Color and Shape:White SolidMolecular weight:523.49Pramipexole dihydrochloride hydrate
CAS:<p>Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.</p>Formula:C10H17N3S·2HCl·H2OPurity:99.68%Color and Shape:White To Off-White Crystalline PowderMolecular weight:302.26Sultopride hydrochloride
CAS:Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.Formula:C17H27ClN2O4SPurity:≥95%Color and Shape:White Or Yellowish PowderMolecular weight:390.93SHU 9119 acetate
<p>SHU 9119 acetate: hMC3R & hMC4R antagonist, hMC5R partial agonist. IC50: MC3R 0.23nM, MC4R 0.06nM, MC5R 0.09nM.</p>Formula:C56H75N15O11Purity:99.8%Color and Shape:SolidMolecular weight:1134.29TGR5 Receptor Agonist
CAS:TGR5 is a potent TGR5(GPCR19) agonist.Formula:C18H14Cl2N2O2Purity:99.77% - ≥95%Color and Shape:SolidMolecular weight:361.22Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formula:C14H22ClN3O2Purity:99.75%Color and Shape:SolidMolecular weight:299.80GR-73632
CAS:<p>Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).</p>Formula:C40H59N7O6SPurity:99.68%Color and Shape:SolidMolecular weight:766Naftopidil dihydrochloride
CAS:<p>Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.</p>Formula:C24H28N2O3·2HClPurity:99.76%Color and Shape:White SolidMolecular weight:465.415-Iodotubercidin
CAS:<p>5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.</p>Formula:C11H13IN4O4Purity:99.98%Color and Shape:Tan SolidMolecular weight:392.15Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Formula:C18H18ClNOSPurity:99.78%Color and Shape:SolidMolecular weight:331.86Exo-1
CAS:Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism of various nutrients, asFormula:C15H12FNO3Purity:99.45%Color and Shape:SolidMolecular weight:273.26Mebhydrolin
CAS:<p>Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.</p>Formula:C19H20N2Purity:99.3% - ≥98%Color and Shape:SolidMolecular weight:276.38Fexofenadine
CAS:<p>Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.</p>Formula:C32H39NO4Purity:99.35%Color and Shape:White To Off-White SolidMolecular weight:501.66Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Formula:C20H20ClF5N2OPurity:99.77%Color and Shape:SolidMolecular weight:434.83Dimemorfan phosphate
CAS:<p>Dimemorfan phosphate (3,17-dimethylmorphinan) is a sigma 1 receptor agonist. Dimemorfan phosphate is used as a potent antitussive.</p>Formula:C18H25N·H3O4PPurity:99.65%Color and Shape:SolidMolecular weight:353.4TG6-10-1
CAS:<p>TG6-10-1 is an EP2 antagonist.</p>Formula:C23H23F3N2O4Purity:99.66% - ≥95%Color and Shape:SolidMolecular weight:448.43BAR501
CAS:<p>BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。</p>Formula:C26H46O3Purity:99.29% - 99.68%Color and Shape:SolidMolecular weight:406.64ANP(1-28) Acetate (human, porcine)
CAS:<p>Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.</p>Formula:C129H207N45O41S3Purity:98.24%Color and Shape:SolidMolecular weight:3140.5ACTH 11-24 acetate(4237-93-8 free base)
CAS:ACTH 11-24 acetate is a cortisol-stimulating adrenocorticotrophin fragment and a competitive antagonist of ACTH 1-39 and 1-10.Formula:C79H138N24O18Purity:>99.99%Color and Shape:SolidMolecular weight:1712.12PEN (human) aceate
PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein ProSAAS, is an endogenous ligand of GPR83.Formula:C99H163N27O34Purity:99.25%Color and Shape:SolidMolecular weight:2275.51Bradykinin (2-9)
CAS:Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.Formula:C44H61N11O10Purity:>99.99%Color and Shape:SolidMolecular weight:904.02PAR-4 Agonist Peptide, amide TFA
CAS:<p>PAR-4 agonist peptide doesn't affect PAR-1/PAR-2; blocked by PAR-4 antagonist.</p>Formula:C36H49F3N8O9Purity:99.72%Color and Shape:SolidMolecular weight:794.824F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Formula:C22H26FNO·C2H2O4Purity:97.34%Color and Shape:SolidMolecular weight:429.49Adrenocorticotropic Hormone (ACTH) (4-10) TFA
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .Formula:C46H60F3N13O12SPurity:98.49%Color and Shape:SolidMolecular weight:1076.12Pramlintide acetate(151126-32-8 free base)
CAS:<p>Pramlintide acetate is a polypeptide analogue of human amylin. It serves as an antidiabetic agent and exhibits antineoplastic activity in colorectal cancer.</p>Formula:C173H271N51O55S2Purity:>99.99%Color and Shape:SolidMolecular weight:4009Tasimelteon
CAS:<p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>Formula:C15H19NO2Purity:98.93% - 99.93%Color and Shape:SolidMolecular weight:245.32Terazosin hydrochloride dihydrate
CAS:<p>Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).</p>Formula:C19H25N5O4·HCl·2H2OPurity:99.81%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:459.92Relenopride hydrochloride
CAS:<p>Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.</p>Formula:C24H31Cl2FN4O4Color and Shape:SolidMolecular weight:529.43Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formula:C68H87N17O15Purity:99.98%Color and Shape:SolidMolecular weight:1382.55BQ-788 sodium salt
CAS:BQ-788 sodium salt is a potent and selective antagonist of ETB receptor(ETB receptors with an IC50 of 1.2 nM in human Girrardi heart cells).Formula:C34H51N5NaO7Color and Shape:SolidMolecular weight:664.8Naluzotan
CAS:Naluzotan（PRX 00023） is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+Formula:C23H38N4O3SPurity:>99.99%Color and Shape:SolidMolecular weight:450.64Antazoline
CAS:<p>Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.</p>Formula:C17H19N3Purity:≥95%Color and Shape:White Crystalline Powder SolidMolecular weight:265.35ELA-11 (human) acetate(1784687-32-6 free base)
ELA-11: potent apelin receptor agonist, Ki=14 nM. Blocks cAMP, boosts β-arrestin. Part of ELA-32.Formula:C60H94N16O15S2Purity:99.53%Color and Shape:SolidMolecular weight:1343.61CB1 antagonist 4
CAS:TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.Formula:C30H25Cl2F3N4OSPurity:98.97%Color and Shape:SolidMolecular weight:617.51Fenspiride
CAS:<p>Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.</p>Formula:C15H20N2O2Color and Shape:SolidMolecular weight:260.33Bupranolol
CAS:Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.Formula:C14H22ClNO2Purity:97.63%Color and Shape:SolidMolecular weight:271.78Fluorogestone acetate
CAS:FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.Formula:C23H31FO5Purity:99.47%Color and Shape:CoaMolecular weight:406.49Dobutamine tartrate
CAS:Dobutamine tartrate is a cardiotonic.Formula:C22H29NO9Color and Shape:SolidMolecular weight:451.472RTICBM-189
CAS:RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Formula:C15H14Cl2N2OPurity:99.96%Color and Shape:SolidMolecular weight:309.19Afamelanotide acetate
CAS:<p>Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.</p>Formula:C80H115N21O21Purity:98% - 99.494%Color and Shape:SolidMolecular weight:1706.9Naftopidil hydrochloride
CAS:<p>Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.</p>Formula:C24H29ClN2O3Purity:99.5%Color and Shape:SolidMolecular weight:428.95Darusentan
CAS:Darusentan (Lu-135252) is a potent inhibitor of endothelin signaling and function in both large and small arteriesFormula:C22H22N2O6Purity:98.72%Color and Shape:SolidMolecular weight:410.43GRK5-IN-2
CAS:GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.Formula:C20H20N4O4Purity:99.92%Color and Shape:SolidMolecular weight:380.4NPS2390
CAS:<p>NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively)</p>Formula:C19H21N3OPurity:97.13%Color and Shape:SolidMolecular weight:307.39LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Formula:C24H27FN2O2·HClPurity:99.8%Color and Shape:SolidMolecular weight:430.94Liraglutide
CAS:<p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>Formula:C172H265N43O51Purity:97.65% - 99.04%Color and Shape:SolidMolecular weight:3751.25[Des-Arg9]-Bradykinin TFA
CAS:<p>[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.</p>Formula:C46H62F3N11O12Purity:>99.99%Color and Shape:SolidMolecular weight:1018.05MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Formula:C23H21N5O3SPurity:97.69% - 98.15%Color and Shape:SolidMolecular weight:447.51Orexin 2 Receptor Agonist
CAS:Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.Formula:C32H34N4O5SPurity:98.26% - 99.43%Color and Shape:SolidMolecular weight:586.7Metadoxine
CAS:<p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>Formula:C8H11NO3·C5H7NO3Purity:99.19%Color and Shape:Off-White PowderMolecular weight:298.29Talnetant hydrochloride
CAS:<p>Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.</p>Formula:C25H23ClN2O2Color and Shape:SolidMolecular weight:418.92PD 117519
CAS:PD 117519 (CI947) is an agonist of adenosine receptorFormula:C19H21N5O4Purity:99.98%Color and Shape:SolidMolecular weight:383.4Poloxamer 407
CAS:<p>Poloxamer 407 is a nonionic surfactant.</p>Purity:98%Color and Shape:White Crystalline PowderMolecular weight:7700(Average)Decynium 22
CAS:Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitorFormula:C23H23IN2Purity:99.92%Color and Shape:Dark Red CrystalsMolecular weight:454.35Aripiprazole monohydrate
CAS:<p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>Formula:C23H29Cl2N3O3Color and Shape:SolidMolecular weight:466.4Tandospirone hydrochloride
CAS:<p>Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.</p>Formula:C21H30ClN5O2Color and Shape:SolidMolecular weight:419.95Clozapine HCl
CAS:<p>Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.</p>Formula:C18H20Cl2N4Color and Shape:SolidMolecular weight:363.29ML-191
CAS:<p>ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.</p>Formula:C24H25N3O3Purity:99.58%Color and Shape:SolidMolecular weight:403.47Bavisant dihydrochloride hydrate
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