GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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TRAP-6 amide acetate
<p>TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].</p>Formula:C36H61N11O10Purity:98.55%Color and Shape:SolidMolecular weight:807.94EST64454 Maleic acid salt
CAS:<p>EST64454 Maleic acid salt, a σ1 receptor antagonist, is a pain treatment candidate with high solubility.</p>Formula:C22H26F2N4O6Purity:97.54%Color and Shape:SolidMolecular weight:480.46ELN-441958
CAS:<p>ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.</p>Formula:C29H29ClN4O2Purity:99.88%Color and Shape:SolidMolecular weight:501.02Metiamide
CAS:Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .Formula:C9H16N4S2Purity:97.41%Color and Shape:SolidMolecular weight:244.38Grapiprant
CAS:Grapiprant (AAT-007) is a selective EP4 receptor antagonist.Formula:C26H29N5O3SPurity:99.49% - 99.843%Color and Shape:SolidMolecular weight:491.61Darbufelone mesylate
CAS:Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).Formula:C19H28N2O5S2Purity:96.81% - 99.92%Color and Shape:SolidMolecular weight:428.57Otenabant
CAS:<p>Otenabant (CP-945598) has been investigated for the treatment of Obesity.</p>Formula:C25H25Cl2N7OPurity:99.43%Color and Shape:SolidMolecular weight:510.42GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Formula:C25H29N5OPurity:99.2%Color and Shape:SolidMolecular weight:415.53[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.Formula:C81H113N19O14Purity:97.68%Color and Shape:SolidMolecular weight:1576.91DOPEXAMINE
CAS:<p>Dopexamine is a dopaminergic agonist</p>Formula:C22H32N2O2Purity:99.42%Color and Shape:SolidMolecular weight:356.5Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Formula:C21H25ClN2O4SPurity:99.04%Color and Shape:SolidMolecular weight:436.95RS-127445 hydrochloride
CAS:<p>RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).</p>Formula:C17H17ClFN3Purity:99.48%Color and Shape:SolidMolecular weight:317.79Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Formula:C14H23BrClN3O2Color and Shape:SolidMolecular weight:380.71ML-097
CAS:ML-097 (CID-2160985) is a pan activator of Ras-related GTPasesFormula:C14H11BrO3Purity:99.12%Color and Shape:SolidMolecular weight:307.139[Lys8, Lys9]-Neurotensin (8-13) acetate
<p>[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2</p>Formula:C40H68N8O10Purity:99.31%Color and Shape:SolidMolecular weight:821.02R 396 acetate
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.Formula:C41H55N9O12Purity:99.52%Color and Shape:SolidMolecular weight:865.93SB-203186 hydrochloride
CAS:<p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>Formula:C16H20N2O2·HClPurity:99.64%Color and Shape:SolidMolecular weight:308.81Atipamezole hydrochloride
CAS:<p>Atipamezole is a synthetic α2 adrenergic receptor antagonist.</p>Formula:C14H16N2·HClPurity:99.74%Color and Shape:SolidMolecular weight:248.75PF-06882961 Tris
CAS:<p>PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>Formula:C35H41FN6O7Purity:98.74% - 99.79%Color and Shape:SolidMolecular weight:676.7CPI-444
CAS:<p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>Formula:C20H21N7O3Purity:98.78%Color and Shape:SolidMolecular weight:407.43AM281
CAS:<p>AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.</p>Formula:C21H19Cl2IN4O2Purity:98.6% - >99.99%Color and Shape:White To Off-White SolidMolecular weight:557.21Bindarit
CAS:<p>Bindarit is a selective inhibitor of monocyte chemoattractant proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.Cost-effective and quality-assured.</p>Formula:C19H20N2O3Purity:98.35% - 98.55%Color and Shape:SolidMolecular weight:324.37Tafluprost
CAS:<p>Tafluprost, a prostaglandin analog, is the selective agonist of fluoroprostaglandin (FP) receptor PGF2α.</p>Formula:C25H34F2O5Purity:97.7% - 99.67%Color and Shape:LiquidMolecular weight:452.53Hydroxyzine
CAS:<p>Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.</p>Formula:C21H27ClN2O2Purity:99.54% - ≥95%Color and Shape:Oil SolidMolecular weight:374.9GUANABENZ
CAS:<p>GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.</p>Formula:C8H8Cl2N4Purity:98.31%Color and Shape:White Solid From Acetonitrile SolidMolecular weight:231.08BPTU
CAS:<p>BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).</p>Formula:C23H22F3N3O3Purity:99.37% - 99.89%Color and Shape:SolidMolecular weight:445.43Prazosin
CAS:<p>Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.</p>Formula:C19H21N5O4Purity:99.86%Color and Shape:White To Tan Powder SolidMolecular weight:383.4ICI 89406
CAS:<p>ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.</p>Formula:C19H22N4O3Purity:99.92%Color and Shape:SolidMolecular weight:354.4MK-571 sodium
CAS:<p>MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.</p>Formula:C26H27ClN2O3S2·NaPurity:97.86% - 99.58%Color and Shape:SolidMolecular weight:537.07Betazole dihydrochloride
CAS:<p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>Formula:C5H11Cl2N3Purity:99.12%Color and Shape:SolidMolecular weight:184.067idalopirdine
CAS:Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Formula:C20H19F5N2OPurity:99.73%Color and Shape:SolidMolecular weight:398.37E7046
CAS:<p>E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.</p>Formula:C22H18F5N3O4Purity:99.86%Color and Shape:SolidMolecular weight:483.4Dobutamine hydrochloride
CAS:<p>Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.</p>Formula:C18H24ClNO3Purity:97.15% - 99.94%Color and Shape:SolidMolecular weight:337.84Phenylephrine
CAS:<p>Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).</p>Formula:C9H13NO2Purity:99.5% - 99.89%Color and Shape:SolidMolecular weight:167.21[Leu31,Pro34]-Neuropeptide Y (porcine)
CAS:<p>[Leu31,Pro34]-Neuropeptide Y (porcine), is a selective and high affinity agonist of neuropeptide Y (NPY) Y1 receptor with anxiolytic effects.</p>Formula:C190H286N54O56Purity:99.39%Color and Shape:SolidMolecular weight:4223Amylin, amide, rat acetate(124447-81-0,free base)
<p>Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 receptors and variably of AMY2 receptors.</p>Formula:C169H276N52O55S2Purity:98.93%Color and Shape:SolidMolecular weight:3980.45Piperoxan hydrochloride
CAS:<p>Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.</p>Formula:C14H20ClNO2Purity:99.61%Color and Shape:SolidMolecular weight:269.77GLP-1(7-37) acetate(106612-94-6 free base)
CAS:<p>Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.</p>Formula:C151H228N40O47Purity:98.89%Color and Shape:SolidMolecular weight:3355.67Ralinepag
CAS:Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human andFormula:C23H26ClNO5Purity:99.79% - 99.85%Color and Shape:SolidMolecular weight:431.91Procaterol hydrochloride hydrate
CAS:Short-acting β2-adrenergic receptor agonist used to treat asthma.Formula:C32H48Cl2N4O7Purity:99.71% - 99.97%Color and Shape:SolidMolecular weight:671.65Mini Gastrin I, human acetate
<p>Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.</p>Formula:C76H103N15O28SPurity:99.35% - 99.82%Color and Shape:SolidMolecular weight:1706.78Naratriptan
CAS:<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Formula:C17H25N3O2SPurity:99.08%Color and Shape:SolidMolecular weight:335.47Pizuglanstat
CAS:<p>Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.</p>Formula:C27H36N6O4Purity:99.62%Color and Shape:SolidMolecular weight:508.61Selexipag
CAS:<p>Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.</p>Formula:C26H32N4O4SPurity:99.98% - >99.99%Color and Shape:SolidMolecular weight:496.62Diclofensine hydrochloride
CAS:Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Formula:C17H18Cl3NOPurity:98.86% - 99.93%Color and Shape:SolidMolecular weight:358.69Substance P (7-11)
CAS:<p>Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .</p>Formula:C31H44N6O5SPurity:98.39%Color and Shape:SolidMolecular weight:612.78NAV-2729
CAS:<p>NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.</p>Formula:C25H17ClN4O3Purity:98.83% - 98.91%Color and Shape:SolidMolecular weight:456.88Escitalopram Oxalate
CAS:<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Formula:C22H23FN2O5Purity:97.39% - 99.73%Color and Shape:White SolidMolecular weight:414.43Pentagastrin
CAS:Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis ofFormula:C37H49N7O9SPurity:96.98% - 99.49%Color and Shape:Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water SolidMolecular weight:767.89Isoetharine mesylate salt
CAS:Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.Formula:C14H25NO6SPurity:99.35% - 99.75%Color and Shape:SolidMolecular weight:335.42Praliciguat
CAS:<p>Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.</p>Formula:C21H14F8N6O2Purity:98.82%Color and Shape:SolidMolecular weight:534.36Ataciguat
CAS:Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.Formula:C21H19Cl2N3O6S3Purity:99.09%Color and Shape:SolidMolecular weight:576.49Dimethocaine
CAS:<p>Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.</p>Formula:C16H26N2O2Purity:99.52%Color and Shape:SolidMolecular weight:278.39Ursodeoxycholic acid sodium
CAS:<p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>Formula:C24H40NaO4Purity:99.66% - 99.96%Color and Shape:SolidMolecular weight:415.56FK962
CAS:<p>FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.</p>Formula:C14H17FN2O2Purity:99.89%Color and Shape:SolidMolecular weight:264.3BMS 182874 hydrochloride
CAS:<p>BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.</p>Formula:C17H20ClN3O3SPurity:97.01%Color and Shape:SolidMolecular weight:381.88AC 187 Acetate
<p>AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.</p>Formula:C129H209N37O42Purity:99.71%Color and Shape:SolidMolecular weight:2950.26Landiolol hydrochloride
CAS:<p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>Formula:C25H40ClN3O8Purity:99.91%Color and Shape:White Crystalline PowderMolecular weight:546.05S1p receptor agonist 1
CAS:<p>S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist.</p>Formula:C23H24FN3O3Purity:99.07% - 99.9%Color and Shape:SolidMolecular weight:409.45Detomidine hydrochloride
CAS:Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.Formula:C12H14N2·HClPurity:99.97%Color and Shape:SolidMolecular weight:222.71[Pyr1]-Apelin-13
CAS:[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.Formula:C69H108N22O16SPurity:99.71%Color and Shape:SolidMolecular weight:1533.8VPC171
CAS:<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Formula:C18H12F3NOSPurity:99.78%Color and Shape:SolidMolecular weight:347.35SAX-187
CAS:<p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>Formula:C15H13ClN4O2S2Purity:97.82% - 98%Color and Shape:SolidMolecular weight:380.87GRA Ex-25
CAS:<p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>Formula:C29H36F3N3O5Purity:98.2% - 98.88%Color and Shape:SolidMolecular weight:563.61Mequitazine
CAS:Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Formula:C20H22N2SPurity:99.98%Color and Shape:SolidMolecular weight:322.47Lixisenatide acetate (320367-13-3 free base)
CAS:<p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>Formula:C215H347N61O65S·6C2H4O2Purity:98% - 99.9%Color and Shape:SolidMolecular weight:5218.88MF-766
CAS:<p>MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.</p>Formula:C27H21F3N2O3Purity:99.54% - 99.59%Color and Shape:SolidMolecular weight:478.46Chlorcyclizine
CAS:<p>CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.</p>Formula:C18H21ClN2Purity:98.75%Color and Shape:SolidMolecular weight:300.83Ranitidine
CAS:<p>Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).</p>Formula:C13H22N4O3SPurity:99.52%Color and Shape:Solid SolidMolecular weight:314.40Orexin B, rat, mouse Acetate
Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formula:C128H219N45O36SPurity:94.61%Color and Shape:SolidMolecular weight:2996.45Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formula:C25H29N3O2Purity:99.83% - 99.97%Color and Shape:SolidMolecular weight:403.52S1RA hydrochloride
CAS:<p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki ></p>Formula:C20H24ClN3O2Purity:98% - 99.84%Color and Shape:SolidMolecular weight:373.87Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Formula:C20H22N2O6Purity:99.39%Color and Shape:SolidMolecular weight:386.4AM095
CAS:AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.Formula:C27H23N2NaO5Purity:98.87%Color and Shape:SolidMolecular weight:478.47AHN 1-055 hydrochloride
CAS:<p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>Formula:C21H24ClF2NOPurity:99.89%Color and Shape:SolidMolecular weight:379.87Neurotensin(8-13) 3TFA(60482-95-3(free base))
CAS:<p>Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.</p>Formula:C40H65F3N12O10Purity:98.31%Color and Shape:SolidMolecular weight:931.03SCH 58261
CAS:SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Formula:C18H15N7OPurity:99.07% - 99.75%Color and Shape:SolidMolecular weight:345.36ACEPROMAZINE MALEATE
CAS:<p>ACEPROMAZINE MALEATE is a dopamine receptor antagonist</p>Formula:C23H26N2O5SPurity:98.87% - 99.51%Color and Shape:Off White Or Yellow Crystalline PowderMolecular weight:442.53Piboserod
CAS:<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Formula:C22H31N3O2Purity:97.21% - 99.49%Color and Shape:SolidMolecular weight:369.5L-745870 trihydrochloride
CAS:<p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>Formula:C18H22Cl4N4Purity:97.52%Color and Shape:SolidMolecular weight:436.214i
CAS:<p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>Formula:C16H12ClN3OPurity:99.49%Color and Shape:SolidMolecular weight:297.74CGP71683 hydrochloride
CAS:<p>CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).</p>Formula:C26H30ClN5O2SPurity:99.92%Color and Shape:SolidMolecular weight:512.07Perospirone
CAS:<p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>Formula:C23H30N4O2SPurity:99.23%Color and Shape:White PowderMolecular weight:426.57DAPTA
CAS:DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.Formula:C35H56N10O15Purity:>99.99%Color and Shape:SolidMolecular weight:856.88Neurokinin A(4-10) TFA(97559-35-8 free base)
<p>Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].</p>Formula:C36H55F3N8O12SPurity:>99.99%Color and Shape:SolidMolecular weight:880.93Bevantolol hydrochloride
CAS:<p>Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.</p>Formula:C20H28ClNO4Purity:99.49%Color and Shape:SolidMolecular weight:381.9Pimozide
CAS:<p>Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.</p>Formula:C28H29F2N3OPurity:99.63% - >99.99%Color and Shape:SolidMolecular weight:461.55RS 504393
CAS:RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).Formula:C25H27N3O3Purity:98.64% - 99.62%Color and Shape:SolidMolecular weight:417.5Idazoxan hydrochloride
CAS:<p>Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.</p>Formula:C11H12N2O2·HClPurity:99.42% - 99.84%Color and Shape:SolidMolecular weight:240.69Ivabradine hydrochloride
CAS:<p>Ivabradine HCl (S 16257-2) is an If inhibitor (IC50: 2.9 μM) and SA node HCN channel blocker that slows heart rate.</p>Formula:C27H37ClN2O5Purity:99% - 99.73%Color and Shape:SolidMolecular weight:505.05HPI 1
CAS:<p>HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.</p>Formula:C27H29NO6Purity:97.6%Color and Shape:SolidMolecular weight:463.52Chlorphenesin
CAS:<p>Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.</p>Formula:C9H11ClO3Purity:99.59%Color and Shape:SolidMolecular weight:202.63AZD2098
CAS:AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research.Formula:C11H9Cl2N3O3SPurity:99.80% - >99.99%Color and Shape:SolidMolecular weight:334.18C-021
CAS:C 021 dihydrochloride is a potent CCR4 antagonist.Formula:C27H41N5O2Purity:99.74% - 99.90%Color and Shape:SolidMolecular weight:467.65Tulobuterol hydrochloride
CAS:<p>Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.</p>Formula:C12H19Cl2NOPurity:99.24% - >99.99%Color and Shape:Appearance White Crystalline PowderMolecular weight:264.19Taladegib
CAS:<p>Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.</p>Formula:C26H24F4N6OPurity:98.75% - >99.99%Color and Shape:SolidMolecular weight:512.5Nitrobenzylthioinosine
CAS:<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Formula:C17H17N5O6SPurity:99.69% - 99.74%Color and Shape:Off-White SolidMolecular weight:419.41Chlorprothixene
CAS:<p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>Formula:C18H18ClNSPurity:98.77% - 99.756%Color and Shape:Pale Yellow Crystals SolidMolecular weight:315.86LY334370
CAS:<p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>Formula:C21H22FN3OPurity:99.32%Color and Shape:SolidMolecular weight:351.42Ozagrel hydrochloride
CAS:<p>Ozagrel hydrochloride (OKY-046 HCl) is a selective thromboxane A(2) synthetase inhibitor used for the improvement of postoperative cerebrovascular contraction</p>Formula:C13H12N2O2·HClPurity:99.80%Color and Shape:White Or Off White Crystalline PowderMolecular weight:264.71
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