GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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HAEGTFT acetate(926018-95-3 free base)
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.Formula:C35H51N9O14Purity:>99.99%Color and Shape:SolidMolecular weight:821.84Azaphen dihydrochloride monohydrate
CAS:Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.Formula:C16H23Cl2N5O2Purity:99.85%Color and Shape:SolidMolecular weight:388.29NPY 5RA972
CAS:NPY 5RA972 is a neuropeptide Y Y5 receptor antagonistFormula:C21H25N3O2Purity:99.02% - 99.56%Color and Shape:SolidMolecular weight:351.44SCH442416
CAS:SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).Formula:C20H19N7O2Purity:99.58%Color and Shape:SolidMolecular weight:389.41Ref: TM-T23336
1mg46.00€5mg88.00€10mg132.00€25mg266.00€50mg409.00€100mg573.00€200mg807.00€1mL*10mM (DMSO)92.00€Bunazosin
CAS:Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].Formula:C19H27N5O3Color and Shape:SolidMolecular weight:373.45dasiglucagon acetate
Dasiglucagon acetate: new, stable glucagon for hypoglycemia with better absorption and longer half-life.Formula:C154H226N38O52Purity:99.63%Color and Shape:SolidMolecular weight:3441.67Eltoprazine hydrochloride
CAS:Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formula:C12H17ClN2O2Purity:99.35%Color and Shape:SolidMolecular weight:256.73Siponimod
CAS:Siponimod (BAF312) modulates S1P1/S1P5 with EC50s of 0.39/0.98 nM; >1000x selectivity over S1P2-4.Formula:C29H35F3N2O3Purity:99.13% - 99.8%Color and Shape:SolidMolecular weight:516.59Guanfacine hydrochloride
CAS:Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.Formula:C9H10Cl3N3OPurity:99.89% - 99.91%Color and Shape:SolidMolecular weight:282.55Pridopidine
CAS:Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.Formula:C15H23NO2SPurity:95.2% - 99.89%Color and Shape:SolidMolecular weight:281.41Brexpiprazole
CAS:Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formula:C25H27N3O2SPurity:99.06% - 99.96%Color and Shape:SolidMolecular weight:433.57Ref: TM-T2306
5mg50.00€10mg63.00€25mg75.00€50mg88.00€100mg94.00€200mg140.00€500mg259.00€1mL*10mM (DMSO)To inquireClemizole
CAS:Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.Formula:C19H20ClN3Purity:98% - 99.65%Color and Shape:SolidMolecular weight:325.84Ref: TM-T1822
1mg42.00€5mg82.00€10mg101.00€25mg152.00€50mg256.00€100mg460.00€500mg973.00€1mL*10mM (DMSO)93.00€Nuciferine
CAS:Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.Formula:C19H21NO2Purity:98.76% - 99.79%Color and Shape:SolidMolecular weight:295.38Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Formula:C58H89N17O14Purity:99.86%Color and Shape:SolidMolecular weight:1248.43Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.Formula:C35H47FN10O8Purity:97.97%Color and Shape:SolidMolecular weight:754.85Taladegib
CAS:Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.Formula:C26H24F4N6OPurity:98.75% - >99.99%Color and Shape:SolidMolecular weight:512.5Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Formula:C17H17N5O6SPurity:99.69% - 99.74%Color and Shape:Off-White SolidMolecular weight:419.41Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurity:98.77% - 99.756%Color and Shape:Pale Yellow Crystals SolidMolecular weight:315.86Vortioxetine hydrobromide
CAS:Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Formula:C18H22N2S·HBrPurity:98.85% - 99.98%Color and Shape:SolidMolecular weight:379.36Taminadenant mesylate
CAS:Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Formula:C11H12BrN7O3SColor and Shape:SolidMolecular weight:402.227
