GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,998 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5960 products of "GPCR/G-Protein"
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Loxapine succinate
CAS:Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.Formula:C22H24ClN3O5Purity:99.69%Color and Shape:White To Of-White SolidMolecular weight:445.9AM095 free acid
CAS:AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).Formula:C27H24N2O5Purity:99.88%Color and Shape:SolidMolecular weight:456.49Ref: TM-T10293
1mg34.00€5mg63.00€10mg92.00€25mg170.00€50mg268.00€100mg416.00€200mg625.00€1mL*10mM (DMSO)70.00€Tropanserin
CAS:Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.Formula:C17H23NO2Purity:99.74%Color and Shape:SolidMolecular weight:273.37Aniracetam
CAS:Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.Formula:C12H13NO3Purity:99.88% - 99.89%Color and Shape:White Crystalline Or Crystalline PowdeMolecular weight:219.24Lofepramine
CAS:Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.
Formula:C26H27ClN2OPurity:98.38%Color and Shape:Crystals From Methanol Or Acetone SolidMolecular weight:418.96Isoxsuprine hydrochloride
CAS:Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.Formula:C18H24ClNO3Purity:99.38%Color and Shape:Crystals From Water SolidMolecular weight:337.84Loratadine
CAS:Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.
Formula:C22H23ClN2O2Purity:99.71% - 99.98%Color and Shape:White PowderMolecular weight:382.88ONC206
CAS:ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations andFormula:C23H22F2N4OPurity:99.38% - 99.81%Color and Shape:SolidMolecular weight:408.44Retatrutide sodium salt
Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.Purity:99.97%Color and Shape:SoildLeronlimab
CAS:Leronlimab (PRO 140), a humanized IgG4 monoclonal antibody, targets CCR5 to combat HIV and cancer.Purity:SDS-PAGE:95.0%;SEC-HPLC:99.6%Color and Shape:LiquidMolecular weight:146.66 kDaPaliperidone
CAS:Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.Formula:C23H27FN4O3Purity:95% - 99.08%Color and Shape:Off White To Light Orange Coloured SolidMolecular weight:426.48Molindone hydrochloride
CAS:Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.
Formula:C16H24N2O2·HClPurity:99% - 99.99%Color and Shape:SolidMolecular weight:312.84Ziprasidone
CAS:Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.Formula:C21H21ClN4OSPurity:99.55%Color and Shape:Tan SolidMolecular weight:412.94Olodaterol
CAS:Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptorsFormula:C21H26N2O5Purity:98.9%Color and Shape:SolidMolecular weight:386.45Fenoterol
CAS:Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.Formula:C17H21NO4Purity:98.29%Color and Shape:SolidMolecular weight:303.35AVN 322 free base
CAS:AVN 322 free base is an orally available, selective and potent 5-HT6R antagonist for the study of neuropathic system disorders such as Alzheimer's disease (AD) and schizophrenia.Formula:C17H19N5O2SPurity:99.24%Color and Shape:SolidMolecular weight:357.43Carvedilol EP IMpurity E
CAS:Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.Formula:C9H14ClNO2Purity:99.53%Color and Shape:White To Almost White Solid CrystallineMolecular weight:203.666Imidazolidinyl urea
CAS:Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.Formula:C11H16N8O8Purity:98.6%Color and Shape:White Fluid Powder With Slight Characteristic OdorMolecular weight:388.29Brefonalol HCl
Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.Formula:C22H29ClN2O2Purity:99.98%Color and Shape:SolidMolecular weight:388.93CI 169369
CAS:CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and depression.Formula:C19H21ClN2SPurity:98.97%Color and Shape:SoildMolecular weight:344.9
