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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • Citalopram hydrobromide
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    Citalopram hydrobromide

    CAS:
    <p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>
    Formula:C20H22BrFN2O
    Purity:99.81%
    Color and Shape:White Crystalline Powder
    Molecular weight:405.304

    Ref: TM-T1483

  • KGA-2727
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    KGA-2727

    CAS:
    <p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>
    Formula:C26H40N4O8
    Purity:98.46%
    Color and Shape:Solid
    Molecular weight:536.62

    Ref: TM-T15656

  • (3aR,9aR)-Fluparoxan
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    (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H10FNO2
    Purity:97.82%
    Color and Shape:Soild
    Molecular weight:195.19

    Ref: TM-T77566

  • [Leu15]-Gastrin I, human
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    [Leu15]-Gastrin I, human

    CAS:
    [Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.
    Formula:C98H126N20O31
    Purity:98.02% - 98.84%
    Color and Shape:Solid
    Molecular weight:2080.16

    Ref: TM-T8761

  • Zolmitriptan
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    Zolmitriptan

    CAS:
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Formula:C16H21N3O2
    Purity:99.69% - 99.91%
    Color and Shape:White Or Kind Of White Powder
    Molecular weight:287.36

    Ref: TM-T1092

  • Ozagrel
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    Ozagrel

    CAS:
    <p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>
    Formula:C13H12N2O2
    Purity:97.90% - 99.38%
    Color and Shape:White Powder
    Molecular weight:228.25

    Ref: TM-T6236

  • AH 6809
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    AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Formula:C17H14O5
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:298.29

    Ref: TM-T14148

  • Ketanserin
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    Ketanserin

    CAS:
    Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.
    Formula:C22H22FN3O3
    Purity:99.19% - 99.73%
    Color and Shape:Solid
    Molecular weight:395.43

    Ref: TM-T1066

  • Noradrenaline bitartrate
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    Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Formula:C12H19NO10
    Purity:99.53% - >99.99%
    Color and Shape:Solid
    Molecular weight:337.28

    Ref: TM-T0871

  • Protriptyline hydrochloride
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    Protriptyline hydrochloride

    CAS:
    <p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>
    Formula:C19H21N·HCl
    Purity:98.54% - 99.98%
    Color and Shape:Solid
    Molecular weight:299.84

    Ref: TM-T0204

  • CymitQuimica logo
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    Sonepcizumab

    CAS:
    <p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>
    Purity:SDS-PAGE:95% SEC-HPLC:98.90%
    Color and Shape:Liquid
    Molecular weight:146.43 kDa

    Ref: TM-T76828

  • Tetrabenazine
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    Tetrabenazine

    CAS:
    Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.
    Formula:C19H27NO3
    Purity:98% - 99.91%
    Color and Shape:White To Off-White White To Off-White Solid
    Molecular weight:317.42

    Ref: TM-T0719

  • Clomipramine hydrochloride
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    Clomipramine hydrochloride

    CAS:
    <p>Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.</p>
    Formula:C19H23ClN2·HCl
    Purity:99.04% - 99.47%
    Color and Shape:White To Slightly Yellow Crystalline Powder
    Molecular weight:351.31

    Ref: TM-T0255

  • Terlipressin Acetate
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    Terlipressin Acetate

    CAS:
    <p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>
    Formula:C56H82N16O19S2
    Purity:98.50% - 99.69%
    Color and Shape:Solid
    Molecular weight:1347.5

    Ref: TM-T13920L

  • (R)-Elagolix
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    (R)-Elagolix

    CAS:
    <p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>
    Formula:C32H30F5N3O5
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:631.59

    Ref: TM-T11174

  • Fluoxetine hydrochloride
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    Fluoxetine hydrochloride

    CAS:
    Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.
    Formula:C17H19ClF3NO
    Purity:99.6% - 99.98%
    Color and Shape:White To Off-White Crystalline Solid White To Off-White Powder
    Molecular weight:345.787

    Ref: TM-T0450L

  • Desipramine hydrochloride
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    Desipramine hydrochloride

    CAS:
    Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.
    Formula:C18H23ClN2
    Purity:99.58% - 99.94%
    Color and Shape:White To Off-White Powder
    Molecular weight:302.842

    Ref: TM-T0991

  • YNT-185
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    YNT-185

    CAS:
    <p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>
    Formula:C33H37N5O5S
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:615.74

    Ref: TM-T39229

  • Ziprasidone hydrochloride
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    Ziprasidone hydrochloride

    CAS:
    <p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>
    Formula:C21H22CL2N4OS
    Purity:97.97% - 99.82%
    Color and Shape:Solid
    Molecular weight:449.4

    Ref: TM-T0031L

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    Somatostatin acetate

    <p>Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for the study of cancer and neurological disorders.</p>
    Purity:99.11%
    Color and Shape:Odour Solid

    Ref: TM-TP1302L