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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5745 products of "GPCR/G-Protein"

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  • Eletriptan hydrobromide
    Targetmol
    + Info

    Eletriptan hydrobromide

    CAS:
    <p>Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D receptor.</p>
    Formula:C22H27BrN2O2S
    Purity:99.69% - 99.85%
    Color and Shape:Tan Solid
    Molecular weight:463.43

    Ref: TM-T0216

  • Pizotifen Malate
    Targetmol
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    Pizotifen Malate

    CAS:
    <p>Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based on benzocycloheptane.</p>
    Formula:C19H21NS·C4H6O5
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:429.53

    Ref: TM-T0225

  • Buflomedil hydrochloride
    Targetmol
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    Buflomedil hydrochloride

    CAS:
    Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.
    Formula:C17H26ClNO4
    Purity:99.7% - 99.91%
    Color and Shape:White Or Off-White Crystalline Powder
    Molecular weight:343.85

    Ref: TM-T0317

  • Aripiprazole Lauroxil
    Targetmol
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    Aripiprazole Lauroxil

    CAS:
    <p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>
    Formula:C36H51Cl2N3O4
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:660.71

    Ref: TM-T14319

  • Lesopitron HCl
    Targetmol
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    Lesopitron HCl

    CAS:
    <p>Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.</p>
    Formula:C15H22Cl2N6
    Purity:97.05% - 99.89%
    Color and Shape:Soild
    Molecular weight:357.28

    Ref: TM-T11839L

  • Lofepramine
    Targetmol
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    Lofepramine

    CAS:
    <p>Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.</p>
    Formula:C26H27ClN2O
    Purity:98.38%
    Color and Shape:Crystals From Methanol Or Acetone Solid
    Molecular weight:418.96

    Ref: TM-T15773

  • Flopropione
    Targetmol
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    Flopropione

    CAS:
    <p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>
    Formula:C9H10O4
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:182.17

    Ref: TM-T0525

  • CYM50308
    Targetmol
    + Info

    CYM50308

    CAS:
    <p>CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).</p>
    Formula:C20H21F2N3O2S
    Purity:99.43% - 99.77%
    Color and Shape:Solid
    Molecular weight:405.46

    Ref: TM-T15032

  • Monatepil 2maleate
    Targetmol
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    Monatepil 2maleate

    Monatepil 2maleate is an orally active Ca2+-channel antagonist and ACAT inhibitor with alpha(1)-adrenergic receptor blocking activity and antiarrhythmic properties that inhibit vasoconstriction.Monatepil 2maleate may be used to study atherosclerosis.
    Formula:C32H34FN3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:591.69

    Ref: TM-T25828L

  • Tropisetron hydrochloride
    Targetmol
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    Tropisetron hydrochloride

    CAS:
    <p>Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.</p>
    Formula:C17H21ClN2O2
    Purity:99.72% - 99.83%
    Color and Shape:Solid
    Molecular weight:320.82

    Ref: TM-T1173

  • Ebalzotan
    Targetmol
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    Ebalzotan

    CAS:
    <p>NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.</p>
    Formula:C19H30N2O2
    Purity:98.09% - 99.41%
    Color and Shape:Solid
    Molecular weight:318.45

    Ref: TM-T68059

  • Itopride hydrochloride
    Targetmol
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    Itopride hydrochloride

    CAS:
    Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.
    Formula:C20H27ClN2O4
    Purity:99.59%
    Color and Shape:White Or Pale Brownish Crystal
    Molecular weight:394.9

    Ref: TM-T1552

  • Sergliflozin A
    Targetmol
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    Sergliflozin A

    CAS:
    Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.
    Formula:C20H24O7
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:376.4

    Ref: TM-T68174

  • Naluzotan hydrochloride
    Targetmol
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    Naluzotan hydrochloride

    CAS:
    <p>Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.</p>
    Formula:C23H39ClN4O3S
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:487.1

    Ref: TM-T68113

  • Carbinoxamine Maleate Salt
    Targetmol
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    Carbinoxamine Maleate Salt

    CAS:
    <p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>
    Formula:C20H23ClN2O5
    Purity:99.97%
    Color and Shape:Off-White Solid
    Molecular weight:406.86

    Ref: TM-T2222

  • Blonanserin
    Targetmol
    + Info

    Blonanserin

    CAS:
    Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.
    Formula:C23H30FN3
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:367.5

    Ref: TM-T1180

  • Fezolinetant
    Targetmol
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    Fezolinetant

    CAS:
    <p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>
    Formula:C16H15FN6OS
    Purity:98.62% - 99.7%
    Color and Shape:Solid
    Molecular weight:358.39

    Ref: TM-T15278

  • Astemizole
    Targetmol
    + Info

    Astemizole

    CAS:
    <p>Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.</p>
    Formula:C28H31FN4O
    Purity:98.24% - 99.67%
    Color and Shape:White Crystals Solid
    Molecular weight:458.57

    Ref: TM-T1278

  • p-MPPI hydrochloride
    Targetmol
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    p-MPPI hydrochloride

    CAS:
    <p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>
    Formula:C25H28ClIN4O2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:578.87

    Ref: TM-T16421

  • Delequamine
    Targetmol
    + Info

    Delequamine

    CAS:
    Delequamine (RS 15385-197) is a TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.
    Formula:C18H26N2O3S
    Purity:99.39%
    Color and Shape:Solid
    Molecular weight:350.48

    Ref: TM-T68051