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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • Palonosetron hydrochloride

    CAS:
    <p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>
    Formula:C19H24N2O·HCl
    Purity:99.84% - 99.92%
    Color and Shape:White Solid
    Molecular weight:332.87
  • Ro 10-5824 dihydrochloride

    CAS:
    Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).
    Formula:C17H22Cl2N4
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:353.29
  • Moxisylyte hydrochloride

    CAS:
    Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
    Formula:C16H26ClNO3
    Purity:99.94% - ≥95%
    Color and Shape:Solid
    Molecular weight:315.84
  • Ziprasidone hydrochloride

    CAS:
    <p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>
    Formula:C21H22CL2N4OS
    Purity:97.97% - 99.82%
    Color and Shape:Solid
    Molecular weight:449.4
  • Vilazodone

    CAS:
    <p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>
    Formula:C26H27N5O2
    Purity:99.61%
    Color and Shape:Light Yellow Solid
    Molecular weight:441.52
  • Dopexamine hydrochloride

    CAS:
    <p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>
    Formula:C22H34Cl2N2O2
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:429.42
  • Dimenhydrinate

    CAS:
    Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.
    Formula:C24H28ClN5O3
    Purity:99.57% - 99.77%
    Color and Shape:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Molecular weight:469.96
  • Adrenalone hydrochloride

    CAS:
    Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.
    Formula:C9H11NO3·HCl
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:217.65
  • Imidazolidinyl urea

    CAS:
    <p>Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.</p>
    Formula:C11H16N8O8
    Purity:98.6%
    Color and Shape:White Fluid Powder With Slight Characteristic Odor
    Molecular weight:388.29
  • Promazine hydrochloride

    CAS:
    Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.
    Formula:C17H21ClN2S
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:320.88
  • Acebutolol hydrochloride

    CAS:
    <p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension &amp; ventricular arrhythmias.</p>
    Formula:C18H29ClN2O4
    Purity:99.92% - >99.99%
    Color and Shape:White Or Slightly Off-White Crystalline Powder Solid
    Molecular weight:372.89
  • Pizotifen

    CAS:
    <p>Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.</p>
    Formula:C19H21NS
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:295.44
  • Linaclotide

    CAS:
    <p>Linaclotide treats IBS-C &amp; chronic constipation; it's a selective guanylate cyclase C agonist.</p>
    Formula:C59H79N15O21S6
    Purity:97.93% - 98.71%
    Color and Shape:Solid
    Molecular weight:1526.74
  • MP-A08

    CAS:
    <p>MP-A08 selectively inhibits SPHK1; targets SphK1 &amp; SphK2 with Ki of 6.9 μM &amp; 27 μM, respectively.</p>
    Formula:C27H25N3O4S2
    Purity:97.44%
    Color and Shape:Solid
    Molecular weight:519.64
  • Fenspiride hydrochloride

    CAS:
    <p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>
    Formula:C15H20N2O2·HCl
    Purity:99.64% - 99.92%
    Color and Shape:Solid
    Molecular weight:296.79
  • Doxofylline

    CAS:
    <p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>
    Formula:C11H14N4O4
    Purity:99.958% - >99.99%
    Color and Shape:Solid
    Molecular weight:266.25
  • Cetirizine dihydrochloride

    CAS:
    Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.
    Formula:C21H27Cl3N2O3
    Purity:99.4% - 99.97%
    Color and Shape:Solid
    Molecular weight:461.81
  • Olinciguat

    CAS:
    <p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>
    Formula:C21H16F5N7O3
    Purity:99.33% - 99.71%
    Color and Shape:Solid
    Molecular weight:509.39
  • Roxatidine Acetate hydrochloride

    CAS:
    <p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>
    Formula:C19H29ClN2O4
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:384.9
  • Pramipexole

    CAS:
    <p>Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.</p>
    Formula:C10H17N3S
    Purity:98% - 99.96%
    Color and Shape:Solid
    Molecular weight:211.33