
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(441 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5965 products of "GPCR/G-Protein"
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BRL 54443
CAS:BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Formula:C14H18N2OPurity:98.07%Color and Shape:SolidMolecular weight:230.31Butyrophenone
CAS:<p>Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.</p>Formula:C10H12OPurity:99.84%Color and Shape:Colourless To Yellow LiquidMolecular weight:148.2Tavapadon
CAS:Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Formula:C19H16F3N3O3Purity:99.33% - 99.8%Color and Shape:SolidMolecular weight:391.34Ambrisentan
CAS:Ambrisentan, an endothelin antagonist for PAH, has a low risk of liver enzyme elevation, not linked to acute liver injury.Formula:C22H22N2O4Purity:99.65% - 99.86%Color and Shape:SolidMolecular weight:378.42Oxyntomodulin acetate
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].Purity:99.24%Color and Shape:LiquidMolecular weight:N/ASBI-553
CAS:SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).Formula:C26H31FN4O2Purity:99.33%Color and Shape:SolidMolecular weight:450.551-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
CAS:<p>1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.</p>Formula:C13H13NO5Purity:99.55%Color and Shape:SolidMolecular weight:263.254-Methylhistamine hydrochloride
CAS:<p>Compound with imidazole ring & amine group; inhibits copper enzymes, affects gene expression.</p>Formula:C6H12ClN3Purity:95%Color and Shape:SolidMolecular weight:161.633Glucagon-like peptide 1 (1-37), human acetate
Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.Purity:98%Color and Shape:LiquidMolecular weight:N/AHPI 1
CAS:HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.Formula:C27H29NO6Purity:97.6%Color and Shape:SolidMolecular weight:463.52Alimemazine hemitartrate
CAS:Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formula:C18H22N2SC4H6O6Purity:98.16% - 99.69%Color and Shape:SolidMolecular weight:448.53Piboserod hydrochloride
CAS:Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.Formula:C22H32ClN3O2Color and Shape:SolidMolecular weight:405.96Bremelanotide Acetate
CAS:<p>Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .</p>Formula:C52H72N14O12Purity:96.72% - >99.99%Color and Shape:SolidMolecular weight:1085.22Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formula:C21H25NO4Purity:99.8% - 99.91%Color and Shape:Off-White SolidMolecular weight:355.43Azepexole
CAS:Azepexole is a selective α2-adrenoceptor agonist that exhibits greater than 300-fold selectivity for the α2-adrenoceptor over the α1-adrenoceptor.Formula:C9H15N3OColor and Shape:SolidMolecular weight:181.23CGP 71683 (free base)
CAS:CGP 71683 (free base) is a potent and highly selective non-peptide antagonist of the NPY Y(5) receptor in the study of obesity.Formula:C26H29N5O2SColor and Shape:SolidMolecular weight:475.61α-MSH, amide Acetate
a-MSH, amide Acetate as an endogenous neuropeptide.Formula:C79H113N21O21SPurity:98.67%Color and Shape:SolidMolecular weight:1724.94N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formula:C17H17ClN4Purity:97.25% - 99.83%Color and Shape:Yellow Crystalline SolidMolecular weight:312.8(±)-Ibipinabant
CAS:(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formula:C23H20Cl2N4O2SPurity:99.28% - 99.83%Color and Shape:SolidMolecular weight:487.4H4 Receptor antagonist 1
CAS:H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formula:C16H17ClN4OPurity:98.81%Color and Shape:SolidMolecular weight:316.79
