GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(441 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5965 products of "GPCR/G-Protein"
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Evatanepag
CAS:<p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>Formula:C25H28N2O5SPurity:97.09%Color and Shape:SolidMolecular weight:468.57Sumatriptan succinate
CAS:Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.Formula:C18H27N3O6SPurity:97.53% - 99.51%Color and Shape:White PowderMolecular weight:413.49Terbutaline
CAS:Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterolFormula:C12H19NO3Purity:99.12%Color and Shape:SolidMolecular weight:225.3Amp579 TFA
<p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>Formula:C24H29ClF3N5O5SPurity:96.56%Color and Shape:SoildMolecular weight:592.03Luzindole
CAS:Luzindole (N-0774) is a selective melatonin receptor antagonist.Formula:C19H20N2OPurity:98.53%Color and Shape:Off-White Amorphous SolidMolecular weight:292.37SEP-363856 hydrochloride
CAS:<p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>Formula:C9H14ClNOSPurity:99.86% - 99.99%Color and Shape:SolidMolecular weight:219.73Promethazine
CAS:Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .Formula:C17H20N2SPurity:99.76%Color and Shape:CrystalsMolecular weight:284.42Orphenadrine hydrochloride
CAS:Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.Formula:C18H23NO·HClPurity:99.88%Color and Shape:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Molecular weight:305.85Dipivefrin hydrochloride
CAS:<p>Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.</p>Formula:C19H27NO5·HClPurity:99.22% - 99.92%Color and Shape:Less Gas With A Sweet Odor Colorless Gas With A Sweet OdorMolecular weight:387.9Ritodrine hydrochloride
CAS:Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.Formula:C17H21NO3·HClPurity:99% - 99.52%Color and Shape:SolidMolecular weight:323.82Naftidrofuryl oxalate
CAS:<p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>Formula:C26H35NO7Purity:97.12% - 98.38%Color and Shape:SolidMolecular weight:473.56Capeserod
CAS:<p>Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive disorders and neurological disorders.</p>Formula:C23H25ClN4O4Purity:98.10% - 99.94%Color and Shape:SolidMolecular weight:456.92Glycerol phenylbutyrate
CAS:Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).Formula:C33H38O6Purity:98.54% - 99.74%Color and Shape:SolidMolecular weight:530.65Prostaglandin E1
CAS:Alprostadil (PGE1) is a natural vasodilator that also inhibits platelets and induces bronchodilation, used in erectile dysfunction treatment.Formula:C20H34O5Purity:99.78% - >99.99%Color and Shape:SolidMolecular weight:354.48Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formula:C21H25NO·CH4SO3Purity:98.41% - 99.96%Color and Shape:White Crystalline Powder; Odourless Or Almost OdourlessMolecular weight:403.53J-113863
CAS:J-113863 is also a potent antagonist of the human CCR3 (IC50 of 0.58 nM) , but a weak antagonist of the mouse CCR3 (IC50 of 460 nM).Formula:C30H37Cl2IN2O2Purity:95.11%Color and Shape:SolidMolecular weight:655.44Alarelin Acetate
CAS:Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.Formula:C56H78N16O12Purity:99.81% - >99.99%Color and Shape:White PowderMolecular weight:1167.34Tiapride hydrochloride
CAS:<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Formula:C15H24N2O4S·HClPurity:99.4% - 99.77%Color and Shape:SolidMolecular weight:364.89EMPA
CAS:<p>EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM</p>Formula:C23H26N4O4SPurity:99.11%Color and Shape:SolidMolecular weight:454.54PF-04995274
CAS:PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.Formula:C23H32N2O6Purity:99.52%Color and Shape:SolidMolecular weight:432.51
