CymitQuimica logo
GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 19 more subcategories

Found 5965 products of "GPCR/G-Protein"

Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Sergliflozin A
    Targetmol
    + Info

    Sergliflozin A

    CAS:
    Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.
    Formula:C20H24O7
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:376.4

    Ref: TM-T68174

  • Promethazine hydrochloride
    Targetmol
    + Info

    Promethazine hydrochloride

    CAS:
    Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.
    Formula:C17H20N2S·HCl
    Purity:99.85%
    Color and Shape:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)
    Molecular weight:320.88

    Ref: TM-T0445L

  • NS-2028
    Targetmol
    + Info

    NS-2028

    CAS:
    NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.
    Formula:C9H5BrN2O3
    Purity:99.44%
    Color and Shape:A Crystalline Solid
    Molecular weight:269.05

    Ref: TM-T16344

  • Cimetidine
    Targetmol
    + Info

    Cimetidine

    CAS:
    Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.
    Formula:C10H16N6S
    Purity:99.82%
    Color and Shape:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)
    Molecular weight:252.34

    Ref: TM-T0797

  • Ketotifen fumarate
    Targetmol
    + Info

    Ketotifen fumarate

    CAS:
    Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.
    Formula:C23H23NO5S
    Purity:99.25% - 99.73%
    Color and Shape:Solid
    Molecular weight:425.50

    Ref: TM-T0994

  • Labetalol hydrochloride
    Targetmol
    + Info

    Labetalol hydrochloride

    CAS:
    Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
    Formula:C19H25ClN2O3
    Purity:99.54% - 99.85%
    Color and Shape:Solid
    Molecular weight:364.87

    Ref: TM-T0348

  • Chlorpheniramine maleate
    Targetmol
    + Info

    Chlorpheniramine maleate

    CAS:
    Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.
    Formula:C20H23ClN2O4
    Purity:99.64% - 99.98%
    Color and Shape:Odorless White Crystalline Solid Or White Powder With A Bitter Taste
    Molecular weight:390.87

    Ref: TM-T1553

  • Clopidogrel hydrogen sulfate
    Targetmol
    + Info

    Clopidogrel hydrogen sulfate

    CAS:
    Clopidogrel hydrogen sulfate is a selective P2Y12 receptor blocker that inhibits platelet adhesion and aggregation.
    Formula:C16H16ClNO2S·H2SO4
    Purity:99.57% - 99.79%
    Color and Shape:Solid
    Molecular weight:419.9

    Ref: TM-T0182L

  • Nardeterol HCl
    Targetmol
    + Info

    Nardeterol HCl

    <p>Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4</p>
    Formula:C20H25ClFN3O2
    Purity:97.72% - 98.65%
    Color and Shape:Soild
    Molecular weight:393.88

    Ref: TM-T68114L

  • Quetiapine hemifumarate
    Targetmol
    + Info

    Quetiapine hemifumarate

    CAS:
    Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.
    Formula:C46H54N6O8S2
    Purity:99.32% - >99.99%
    Color and Shape:White Crystalline Solid
    Molecular weight:883.09

    Ref: TM-T6241

  • Domperidone
    Targetmol
    + Info

    Domperidone

    CAS:
    <p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>
    Formula:C22H24ClN5O2
    Purity:98% - 99.82%
    Color and Shape:Solid
    Molecular weight:425.91

    Ref: TM-T0082

  • L-741626
    Targetmol
    + Info

    L-741626

    CAS:
    L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3
    Formula:C20H21ClN2O
    Purity:98.57%
    Color and Shape:Solid
    Molecular weight:340.85

    Ref: TM-T15686

  • Lesopitron HCl
    Targetmol
    + Info

    Lesopitron HCl

    CAS:
    <p>Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.</p>
    Formula:C15H22Cl2N6
    Purity:97.05% - 99.89%
    Color and Shape:Soild
    Molecular weight:357.28

    Ref: TM-T11839L

  • Rimonabant hydrochloride
    Targetmol
    + Info

    Rimonabant hydrochloride

    CAS:
    Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂， Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。
    Formula:C22H22Cl4N4O
    Purity:98.24% - 99.5%
    Color and Shape:Off-White To White Crystalline Powder
    Molecular weight:500.25

    Ref: TM-T1519

  • Desvenlafaxine
    Targetmol
    + Info

    Desvenlafaxine

    CAS:
    Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.
    Formula:C16H25NO2
    Purity:99.46% - 99.81%
    Color and Shape:White Crystalline Powder
    Molecular weight:263.38

    Ref: TM-T1580

  • Dexchlorpheniramine Maleate
    Targetmol
    + Info

    Dexchlorpheniramine Maleate

    CAS:
    Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.
    Formula:C20H23ClN2O4
    Purity:99.58%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:390.86

    Ref: TM-T0785

  • Degarelix acetate(214766-78-6 free base)
    Targetmol
    + Info

    Degarelix acetate(214766-78-6 free base)

    CAS:
    Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
    Formula:C84H107ClN18O18
    Purity:98.66%
    Color and Shape:Solid
    Molecular weight:1692.34

    Ref: TM-T10988L

  • Ogerin
    Targetmol
    + Info

    Ogerin

    CAS:
    Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).
    Formula:C17H17N5O
    Purity:99.5% - 99.75%
    Color and Shape:Solid
    Molecular weight:307.35

    Ref: TM-T16378

  • CymitQuimica logo
    Targetmol
    + Info

    Latozinemab

    Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.
    Purity:> 95%
    Color and Shape:Liquid
    Molecular weight:146.28 kDa

    Ref: TM-T77053

  • MP-A08
    Targetmol
    + Info

    MP-A08

    CAS:
    MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.
    Formula:C27H25N3O4S2
    Purity:97.44%
    Color and Shape:Solid
    Molecular weight:519.64

    Ref: TM-T16128