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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5965 products of "GPCR/G-Protein"

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  • Loratadine

    CAS:
    <p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>
    Formula:C22H23ClN2O2
    Purity:99.71% - 99.98%
    Color and Shape:White Powder
    Molecular weight:382.88
  • AM095 free acid

    CAS:
    AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).
    Formula:C27H24N2O5
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:456.49
  • Heptaminol hydrochloride

    CAS:
    Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.
    Formula:C8H20ClNO
    Purity:98.61%
    Color and Shape:White Crystalline Powder
    Molecular weight:181.71
  • Azacyclonol

    CAS:
    Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.
    Formula:C18H21NO
    Purity:99.46%
    Color and Shape:Solid Powder
    Molecular weight:267.37
  • Lesopitron HCl

    CAS:
    <p>Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.</p>
    Formula:C15H22Cl2N6
    Purity:97.05% - 99.89%
    Color and Shape:Soild
    Molecular weight:357.28
  • Tetrabenazine

    CAS:
    Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.
    Formula:C19H27NO3
    Purity:98% - 99.91%
    Color and Shape:White To Off-White White To Off-White Solid
    Molecular weight:317.42
  • SBI-477

    CAS:
    SBI-477 deactivates MondoA, inhibits TAG synthesis, and boosts glucose uptake in human muscle cells.
    Formula:C24H25N3O6S
    Purity:99.3%
    Color and Shape:Solid
    Molecular weight:483.54
  • Aripiprazole Lauroxil

    CAS:
    Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.
    Formula:C36H51Cl2N3O4
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:660.71
  • Carbinoxamine Maleate Salt

    CAS:
    Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.
    Formula:C20H23ClN2O5
    Purity:99.97%
    Color and Shape:Off-White Solid
    Molecular weight:406.86
  • DSP-4 hydrochloride

    CAS:
    <p>DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.</p>
    Formula:C11H16BrCl2N
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:313.06
  • 6-Iodopravadoline

    CAS:
    6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.
    Formula:C23H25IN2O3
    Purity:99.29%
    Color and Shape:Off-White Solid
    Molecular weight:504.36
  • AB928

    CAS:
    AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
    Formula:C23H22N8O
    Purity:98.09% - >99.99%
    Color and Shape:Solid
    Molecular weight:426.47
  • Risperidone

    CAS:
    Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
    Formula:C23H27FN4O2
    Purity:99.73%
    Color and Shape:Crystalline Solid
    Molecular weight:410.48
  • Sarizotan 2HCl

    CAS:
    Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.
    Formula:C22H23Cl2FN2O
    Purity:98.83%
    Color and Shape:Soild
    Molecular weight:421.34
  • Iloperidone

    CAS:
    Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.
    Formula:C24H27FN2O4
    Purity:99.42%
    Color and Shape:Solid
    Molecular weight:426.48
  • BP 897 hydrochloride

    CAS:
    BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low affinity for D1/D4.
    Formula:C26H32ClN3O2
    Purity:99.42%
    Color and Shape:Solid
    Molecular weight:454
  • Lofepramine

    CAS:
    <p>Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.</p>
    Formula:C26H27ClN2O
    Purity:98.38%
    Color and Shape:Crystals From Methanol Or Acetone Solid
    Molecular weight:418.96
  • Quercetin-3'-o-phosphate TEA


    Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.
    Formula:C21H26NO10P
    Purity:97.04%
    Color and Shape:Soild
    Molecular weight:483.41
  • Evatanepag

    CAS:
    <p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>
    Formula:C25H28N2O5S
    Purity:97.09%
    Color and Shape:Solid
    Molecular weight:468.57
  • UCM-1306

    CAS:
    <p>UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.</p>
    Formula:C14H14FNO2S
    Purity:99.98%
    Color and Shape:Soild
    Molecular weight:279.33