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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • Blonanserin
    Targetmol
    + Info

    Blonanserin

    CAS:
    Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.
    Formula:C23H30FN3
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:367.5

    Ref: TM-T1180

  • KGA-2727
    Targetmol
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    KGA-2727

    CAS:
    <p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>
    Formula:C26H40N4O8
    Purity:98.46%
    Color and Shape:Solid
    Molecular weight:536.62

    Ref: TM-T15656

  • (3aR,9aR)-Fluparoxan
    Targetmol
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    (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H10FNO2
    Purity:97.82%
    Color and Shape:Soild
    Molecular weight:195.19

    Ref: TM-T77566

  • Azatadine dimaleate
    Targetmol
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    Azatadine dimaleate

    CAS:
    <p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.</p>
    Formula:C28H30N2O8
    Purity:99.7% - >99.99%
    Color and Shape:Powder
    Molecular weight:522.55

    Ref: TM-T0236

  • Zolmitriptan
    Targetmol
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    Zolmitriptan

    CAS:
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Formula:C16H21N3O2
    Purity:99.69% - 99.91%
    Color and Shape:White Or Kind Of White Powder
    Molecular weight:287.36

    Ref: TM-T1092

  • Flopropione
    Targetmol
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    Flopropione

    CAS:
    <p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>
    Formula:C9H10O4
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:182.17

    Ref: TM-T0525

  • AH 6809
    Targetmol
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    AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Formula:C17H14O5
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:298.29

    Ref: TM-T14148

  • Dopexamine hydrochloride
    Targetmol
    + Info

    Dopexamine hydrochloride

    CAS:
    <p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>
    Formula:C22H34Cl2N2O2
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:429.42

    Ref: TM-T11318

  • Noradrenaline bitartrate
    Targetmol
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    Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Formula:C12H19NO10
    Purity:99.53% - >99.99%
    Color and Shape:Solid
    Molecular weight:337.28

    Ref: TM-T0871

  • Antazoline hydrochloride
    Targetmol
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    Antazoline hydrochloride

    CAS:
    <p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>
    Formula:C17H19N3·HCl
    Purity:98% - 99.53%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:301.82

    Ref: TM-T0092

  • Mifentidine
    Targetmol
    + Info

    Mifentidine

    CAS:
    <p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>
    Formula:C13H16N4
    Purity:98.34% - 99.73%
    Color and Shape:Solid
    Molecular weight:228.29

    Ref: TM-T68100

  • Bambuterol hydrochloride
    Targetmol
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    Bambuterol hydrochloride

    CAS:
    <p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>
    Formula:C18H30ClN3O5
    Purity:99.53% - 99.61%
    Color and Shape:White Solid
    Molecular weight:403.91

    Ref: TM-T1446

  • Ticlopidine hydrochloride
    Targetmol
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    Ticlopidine hydrochloride

    CAS:
    <p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>
    Formula:C14H15Cl2NS
    Purity:99.85% - >99.99%
    Color and Shape:White Powder
    Molecular weight:300.25

    Ref: TM-T0362

  • Senktide acetate
    Targetmol
    + Info

    Senktide acetate

    <p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>
    Formula:C42H59N7O13S
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:902.02

    Ref: TM-T7633L

  • (R)-Elagolix
    Targetmol
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    (R)-Elagolix

    CAS:
    <p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>
    Formula:C32H30F5N3O5
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:631.59

    Ref: TM-T11174

  • LCKLSL hydrochloride
    Targetmol
    + Info

    LCKLSL hydrochloride

    <p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>
    Formula:C30H58ClN7O8S
    Purity:98.02% - 99.31%
    Color and Shape:Solid
    Molecular weight:712.34

    Ref: TM-T78015

  • SEP-363856 hydrochloride
    Targetmol
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    SEP-363856 hydrochloride

    CAS:
    <p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>
    Formula:C9H14ClNOS
    Purity:99.86% - 99.99%
    Color and Shape:Solid
    Molecular weight:219.73

    Ref: TM-T12899L

  • YNT-185
    Targetmol
    + Info

    YNT-185

    CAS:
    <p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>
    Formula:C33H37N5O5S
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:615.74

    Ref: TM-T39229

  • Ziprasidone hydrochloride
    Targetmol
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    Ziprasidone hydrochloride

    CAS:
    <p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>
    Formula:C21H22CL2N4OS
    Purity:97.97% - 99.82%
    Color and Shape:Solid
    Molecular weight:449.4

    Ref: TM-T0031L

  • CCR2-RA-[R]
    Targetmol
    + Info

    CCR2-RA-[R]

    CAS:
    <p>CCR2-RA-[R] is a C-C chemokine receptor type 2 (CCR2) allosteric antagonist (IC50: 103 nM).</p>
    Formula:C18H19ClFNO3
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:351.8

    Ref: TM-T14900