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Quinazoline and Quinoline Derivatives

Quinazoline and Quinoline Derivatives

Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules. At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.

Found 65624 products of "Quinazoline and Quinoline Derivatives"

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  • Sunitinib

    CAS:
    <p>Sunitinib (SU 11248) is a multi-targeted receptor tyrosine kinase (RTK) inhibitor that inhibits VEGFR2 and PDGFRβ (IC50=80/2 nM).</p>
    Formula:C22H27FN4O2
    Purity:98% - 99.67%
    Color and Shape:Yellow Solid
    Molecular weight:398.47
  • Paliperidone

    CAS:
    <p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>
    Formula:C23H27FN4O3
    Purity:95% - 99.08%
    Color and Shape:Off White To Light Orange Coloured Solid
    Molecular weight:426.48
  • Silodosin

    CAS:
    <p>Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.</p>
    Formula:C25H32F3N3O4
    Purity:99.282% - 99.76%
    Color and Shape:Colorless To Pink Solid
    Molecular weight:495.53
  • Altretamine

    CAS:
    <p>Altretamine (ENT-50852) is an alkylating agent with antineoplastic activity.</p>
    Formula:C9H18N6
    Purity:99.54%
    Color and Shape:Less Crystalline Solid Insoluble In Water (Ntp 1992) Physical Description Colorless Crystalline Solid Insoluble In Water (Ntp 1992)
    Molecular weight:210.28
  • Terazosin hydrochloride

    CAS:
    <p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>
    Formula:C19H26ClN5O4
    Purity:99.69% - 99.91%
    Color and Shape:Solid
    Molecular weight:423.89
  • Ticagrelor

    CAS:
    <p>Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.</p>
    Formula:C23H28F2N6O4S
    Purity:98.08% - 99.77%
    Color and Shape:Solid
    Molecular weight:522.57
  • Lenalidomide

    CAS:
    <p>Lenalidomide (CC-5013) is an orally immunomodulator. Lenalidomide is a ligand for the ubiquitin E3 ligase cereblon (CRBN). Cost-effective and quality-assured.</p>
    Formula:C13H13N3O3
    Purity:98% - 99.97%
    Color and Shape:Yellow Solid
    Molecular weight:259.26
  • Carteolol hydrochloride

    CAS:
    <p>Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.</p>
    Formula:C16H24N2O3·HCl
    Purity:99.84% - 99.91%
    Color and Shape:Solid
    Molecular weight:328.83
  • Dequalinium chloride

    CAS:
    <p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>
    Formula:C30H40Cl2N4
    Purity:99.79% - 99.9%
    Color and Shape:Solid
    Molecular weight:527.59
  • Lomustine

    CAS:
    <p>Lomustine (NSC-79037) is an alkylating agent of value against both hematologic malignancies and solid tumors.</p>
    Formula:C9H16ClN3O2
    Purity:98.36% - 99.44%
    Color and Shape:Solid Solid
    Molecular weight:233.7
  • Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Formula:C22H29N3O4S
    Purity:98.55%
    Color and Shape:Yellowish White Crystalline Powder
    Molecular weight:431.55
  • Buflomedil hydrochloride

    CAS:
    <p>Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.</p>
    Formula:C17H26ClNO4
    Purity:99.7% - 99.91%
    Color and Shape:White Or Off-White Crystalline Powder
    Molecular weight:343.85
  • Dyclonine hydrochloride

    CAS:
    <p>Dyclonine hydrochloride (Dyclonine HCl) , an over the counter throat lozenge, is found in Sucretswith local anesthetic effect .</p>
    Formula:C18H27NO2·HCl
    Purity:99.35%
    Color and Shape:White Crystalline Solid
    Molecular weight:325.87
  • Dasatinib

    CAS:
    <p>Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive.</p>
    Formula:C22H26ClN7O2S
    Purity:99.59% - 99.86%
    Color and Shape:Pale-Yellow Solid
    Molecular weight:488.01
  • Ramelteon

    CAS:
    <p>Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.</p>
    Formula:C16H21NO2
    Purity:97.21% - 99.92%
    Color and Shape:Crystalline Solid
    Molecular weight:259.34
  • Doxylamine succinate

    CAS:
    <p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>
    Formula:C21H28N2O5
    Purity:99.61%
    Color and Shape:5 1 (Ntp 1992)
    Molecular weight:388.46
  • Clofazimine

    CAS:
    <p>Clofazimine, a phenazine dye, has anti-mycobacterial/inflammatory effects, targeting Mycobacterium leprae and others.</p>
    Formula:C27H22Cl2N4
    Purity:98.23% - 99.79%
    Color and Shape:Solid
    Molecular weight:473.4
  • Chlormezanone

    CAS:
    <p>Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.</p>
    Formula:C11H12ClNO3S
    Purity:99.89% - >99.99%
    Color and Shape:Crystals Solid
    Molecular weight:273.74
  • Phenylephrine hydrochloride

    CAS:
    <p>Phenylephrine hydrochloride (NCI-c55641) is a selective agonist of the α1-adrenergic receptor.</p>
    Formula:C9H14ClNO2
    Purity:99.51% - 99.97%
    Color and Shape:Physical Description Odorless White Microcrystalline Powder Bitter Taste Ph (1%
    Molecular weight:203.67
  • Pemirolast potassium

    CAS:
    <p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>
    Formula:C10H7KN6O
    Purity:98.91% - 99.63%
    Color and Shape:Crystals From Dimethylformamide Crystalline Solid
    Molecular weight:266.31
  • Triflusal

    CAS:
    <p>Triflusal (UR1501) is a 2-acetoxy-4-trifluoromethylbenzoic acid and it is an aspirin chemically-related molecule but not a derivative.</p>
    Formula:C10H7F3O4
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:248.16
  • Elsulfavirine

    CAS:
    <p>Elsulfavirine (VM-1500) is an HIV-1 infection reverse transcriptase inhibitor. It is a new anti-HIV drug.</p>
    Formula:C24H17BrCl2FN3O5S
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:629.28
  • Olopatadine hydrochloride

    CAS:
    <p>Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.</p>
    Formula:C21H23NO3·HCl
    Purity:99.62% - 99.64%
    Color and Shape:White Solid
    Molecular weight:373.87
  • Nithiamide

    CAS:
    <p>Nithiamide (CL-5279) is an orally available antiprotozoan agent used in the treatment of vaginal trichomoniasis.</p>
    Formula:C5H5N3O3S
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:187.18
  • Isoprenaline hydrochloride

    CAS:
    <p>Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.</p>
    Formula:C11H18ClNO3
    Purity:98% - 99.65%
    Color and Shape:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)
    Molecular weight:247.719
  • Bendamustine hydrochloride

    CAS:
    <p>Bendamustine hydrochloride (EP-3101) (IC50 of 50 μM) is an alkylating agent associated with DNA damage.</p>
    Formula:C16H21Cl2N3O2·HCl
    Purity:97.71%
    Color and Shape:Solid
    Molecular weight:394.72
  • Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Formula:C15H23N3O4S
    Purity:98.20% - 99.88%
    Color and Shape:White Crystalline Powder
    Molecular weight:341.43
  • Azelastine hydrochloride

    CAS:
    <p>Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.</p>
    Formula:C22H24ClN3O·HCl
    Purity:98% - >99.99%
    Color and Shape:White Crystalline Powder
    Molecular weight:418.36
  • Ozagrel

    CAS:
    <p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>
    Formula:C13H12N2O2
    Purity:97.90% - 99.38%
    Color and Shape:White Powder
    Molecular weight:228.25
  • Duloxetine hydrochloride

    CAS:
    <p>Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.</p>
    Formula:C18H20ClNOS
    Purity:99.93% - >99.99%
    Color and Shape:White Or White Crystalline Powder
    Molecular weight:333.88
  • Lornoxicam

    CAS:
    <p>Lornoxicam (Chlortenoxicam) (chlortenoxicam) is a new nonsteroidal anti-inflammatory drug (NSAID) of the oxicam class with analgesic, anti-inflammatory, and</p>
    Formula:C13H10ClN3O4S2
    Purity:98.74% - 99.28%
    Color and Shape:Crystalline Solid
    Molecular weight:371.82
  • Phenoxybenzamine hydrochloride

    CAS:
    <p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>
    Formula:C18H23Cl2NO
    Purity:98.04% - >99.99%
    Color and Shape:Antihypertensive Drug
    Molecular weight:340.3
  • Dapoxetine hydrochloride

    CAS:
    <p>Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature ejaculation.</p>
    Formula:C21H23NO·HCl
    Purity:99.70% - 99.91%
    Color and Shape:White To Off-White Crystalline Solid
    Molecular weight:341.87
  • Lisinopril dihydrate

    CAS:
    <p>Lisinopril dihydrate (MK-521) is an orally bioavailable, long-acting angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.</p>
    Formula:C21H35N3O7
    Purity:98.83% - 99.22%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:441.52
  • CL-82198

    CAS:
    <p>CL-82198, a selective MMP-13 inhibitor, serves as a pharmacological intervention to halt the progression of osteoarthritis (OA).</p>
    Formula:C17H22N2O3
    Purity:95.91%
    Color and Shape:Solid
    Molecular weight:302.37
  • Nepafenac

    CAS:
    <p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>
    Formula:C15H14N2O2
    Purity:98.94% - 99.43%
    Color and Shape:Solid
    Molecular weight:254.28
  • Phenformin

    CAS:
    <p>Phenformin: a biguanide with anti-cancer, anti-glycemic effects, inhibits skin tumors, enhances keratinocyte differentiation/apoptosis.</p>
    Formula:C10H15N5
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:205.26
  • Bifonazole

    CAS:
    <p>Bifonazole (Bay H-4502) inhibits fungal enzyme cytochrome p450 51, halting ergosterol synthesis, causing cell membrane damage and fungal cell lysis.</p>
    Formula:C22H18N2
    Purity:99.29% - 99.87%
    Color and Shape:Solid
    Molecular weight:310.39
  • Erlotinib

    CAS:
    <p>Erlotinib (NSC-718781) is an EGFR inhibitor (IC50: 2 nM). It is used for the treatment of non-small cell lung cancer.</p>
    Formula:C22H23N3O4
    Purity:98.19% - 99.98%
    Color and Shape:White To Off-White Powder
    Molecular weight:393.44
  • Nebivolol hydrochloride

    CAS:
    <p>Nebivolol hydrochloride is a beta-1 blocker and vasodilator treating hypertension and heart failure in the elderly.</p>
    Formula:C22H25F2NO4·HCl
    Purity:99.77% - >99.99%
    Color and Shape:White To Off-White Powder
    Molecular weight:441.90
  • Vildagliptin

    CAS:
    <p>Vildagliptin (LAF237), an oral DPP-4 inhibitor with hypoglycemic effects, is metabolized and excreted in urine.</p>
    Formula:C17H25N3O2
    Purity:97.81% - >99.99%
    Color and Shape:White Crystalline Powder
    Molecular weight:303.40
  • Diminazene Aceturate

    CAS:
    <p>Diminazene is a trypanocidal agent.</p>
    Formula:C22H29N9O6
    Purity:96.86% - 99.58%
    Color and Shape:Solid
    Molecular weight:515.52
  • Thalidomide

    CAS:
    <p>Thalidomide, a glutamic acid derivative, has teratogenic and immunomodulatory effects.</p>
    Formula:C13H10N2O4
    Purity:98.88% - 99.88%
    Color and Shape:White Solid
    Molecular weight:258.23
  • Epalrestat

    CAS:
    <p>Epalrestat (ONO2235), an aldose reductase inhibitor, helps manage diabetic neuropathy symptoms and slows disease progression.</p>
    Formula:C15H13NO3S2
    Purity:99.2% - 99.54%
    Color and Shape:Deep Red Acicular Crystal
    Molecular weight:319.4
  • Alosetron hydrochloride

    CAS:
    <p>Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.</p>
    Formula:C17H19ClN4O
    Purity:99.90%
    Color and Shape:Off-White Powder
    Molecular weight:330.81
  • Dimenhydrinate

    CAS:
    <p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>
    Formula:C24H28ClN5O3
    Purity:99.57% - 99.77%
    Color and Shape:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Molecular weight:469.96
  • Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Formula:C22H21Cl3N4O
    Purity:98% - 99.91%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:463.79
  • Atazanavir

    CAS:
    <p>Atazanavir (BMS-232632)(BMS-232632) is an highly effective HIV-1 protease inhibitor.</p>
    Formula:C38H52N6O7
    Purity:98% - 99.95%
    Color and Shape:Crystalline Solid
    Molecular weight:704.86
  • Pericyazine

    CAS:
    <p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>
    Formula:C21H23N3OS
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:365.49
  • Zomepirac sodium salt

    CAS:
    <p>Zomepirac sodium salt (McN-2783-21-98) is a prostaglandin synthetase inhibitor.</p>
    Formula:C15H13ClNNaO3
    Purity:98.65% - ≥95%
    Color and Shape:Solid
    Molecular weight:313.71