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Glucocorticoid Receptor

Glucocorticoid Receptor

The glucocorticoid receptor (GR) is a nuclear hormone receptor that mediates the effects of glucocorticoids, a class of steroid hormones involved in the regulation of metabolism, immune response, and stress. Glucocorticoid receptor agonists and antagonists are widely used in the treatment of inflammatory and autoimmune diseases, as well as in cancer therapy. GR modulators are also important tools for studying the physiological and pathological roles of glucocorticoids. At CymitQuimica, we provide a wide range of high-quality glucocorticoid receptor modulators to support your research in endocrinology, immunology, and hormone regulation.

Found 153 products of "Glucocorticoid Receptor"

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  • Amcinonide

    CAS:
    <p>Amcinonide (CL-34699) is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid Hormone Receptor Agonist.</p>
    Formula:C28H35FO7
    Purity:98.33% - 99.62%
    Color and Shape:Solid
    Molecular weight:502.57
  • Mometasone furoate

    CAS:
    <p>Mometasone furoate (Sch32088) is a pregnadienediol derivative ANTI-ALLERGIC AGENT and ANTI-INFLAMMATORY AGENT that is used in the management of ASTHMA and</p>
    Formula:C27H30Cl2O6
    Purity:99.43% - 99.48%
    Color and Shape:Distributed As 0 1% Ointment With A Petrolatum Base
    Molecular weight:521.43
  • Betamethasone dipropionate

    CAS:
    <p>Betamethasone Dipropionate, a synthetic glucocorticoid, modulates gene expression to manage inflammation and autoimmune activity.</p>
    Formula:C28H37FO7
    Purity:98.13% - 99.59%
    Color and Shape:Powder
    Molecular weight:504.59
  • AZD5423

    CAS:
    <p>AZD5423: Inhaled, potent GR modulator, non-steroidal, curbs allergy asthma symptoms.</p>
    Formula:C25H21F4N3O3
    Purity:98.76%
    Color and Shape:Solid
    Molecular weight:487.45
  • Triamcinolone acetonide

    CAS:
    <p>Triamcinolone acetonide (Azmacort) is a Corticosteroid.</p>
    Formula:C24H31FO6
    Purity:99.61% - 99.91%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:434.50
  • Hydrocortisone Valerate

    CAS:
    <p>Hydrocortisone Valerate (Westcort) has anti-inflammatory, antipruritic and vasoconstrictive properties.</p>
    Formula:C26H38O6
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:446.58
  • Triamcinolone

    CAS:
    <p>Triamcinolone (Aristocort) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.</p>
    Formula:C21H27FO6
    Purity:98.59% - 99.60%
    Color and Shape:Solid
    Molecular weight:394.43
  • Esaxerenone

    CAS:
    <p>Esaxerenone (XL-550) is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor.</p>
    Formula:C22H21F3N2O4S
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:466.47
  • Clobetasol propionate

    CAS:
    <p>Clobetasol propionate (CGP9555) exerts its effect by binding to cytoplasmic glucocorticoid receptors and subsequently activates glucocorticoid receptor-mediated</p>
    Formula:C25H32ClFO5
    Purity:99.41%
    Color and Shape:White Crystalline Powder
    Molecular weight:466.97
  • Mirodenafil

    CAS:
    <p>Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.</p>
    Formula:C26H37N5O5S
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:531.67
  • Miricorilant

    CAS:
    <p>Miricorilant (CORT 118335) is a glucocorticoid receptor modulator for the study of digestive and metabolic disorders.</p>
    Formula:C24H23F3N2O2
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:428.45
  • Loteprednol etabonate

    CAS:
    <p>Loteprednol etabonate (Lotemax) is an ophthalmic analog of the corticosteroid prednisolone with anti-inflammatory activity.</p>
    Formula:C24H31ClO7
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:466.95
  • Hydrocortisone

    CAS:
    <p>Hydrocortisone is a synthetic glucocorticoid that aids in metabolism, immunity, and inflammation control.</p>
    Formula:C21H30O5
    Purity:98.4% - 99.95%
    Color and Shape:Plates From Alc Or Iso-Propyl Alc Solid
    Molecular weight:362.46
  • Halcinonide

    CAS:
    <p>Halcinonide (Halciderm), a high-efficiency corticosteroid, is served as an anti-inflammatory agent used in topical preparations.</p>
    Formula:C24H32ClFO5
    Purity:99.32% - 99.93%
    Color and Shape:Solid
    Molecular weight:454.96
  • Fluticasone (propionate)

    CAS:
    <p>Fluticasone propionate (CCI-187881), derived from fluticasone used to remedy asthma and allergic rhinitis, is a high affinity, selective GR agonist.</p>
    Formula:C25H31F3O5S
    Purity:98.98% - >99.99%
    Color and Shape:Crystalline Solid
    Molecular weight:500.57
  • Hydrocortisone acetate

    CAS:
    <p>Hydrocortisone acetate (Cortisol 21-acetate) is the synthetic acetate salt form of hydrocortisone, a corticosteroid with anti-inflammatory and immunosuppressive</p>
    Formula:C23H32O6
    Purity:98.89% - 99.22%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:404.5
  • Prednisolone

    CAS:
    <p>Prednisolone (Hydroretrocortine) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.</p>
    Formula:C21H28O5
    Purity:99.59% - 99.85%
    Color and Shape:Crystals Solid
    Molecular weight:360.44
  • Medroxyprogesterone Acetate

    CAS:
    <p>Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. Farlutin is a long-acting contraceptive.</p>
    Formula:C24H34O4
    Purity:99.05% - 99.44%
    Color and Shape:White Powder
    Molecular weight:386.52
  • Prednisolone disodium phosphate

    CAS:
    <p>Prednisolone disodium phosphate, a synthetic glucocorticoid, has immunomodulating and anti-inflammatory properties.</p>
    Formula:C21H27Na2O8P
    Purity:97.1% - 99.16%
    Color and Shape:Solid
    Molecular weight:484.39
  • Betamethasone valerate

    CAS:
    <p>Betamethasone valerate (Luxiq) is a synthetic glucocorticoid with metabolic, immunosuppressive and anti-inflammatory actions.</p>
    Formula:C27H37FO6
    Purity:99.32% - >99.99%
    Color and Shape:Mixed With A Solvent
    Molecular weight:476.58
  • Prednisolone acetate


    <p>Prednisolone acetate (Omnipred) is the acetate salt form of prednisolone, a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.</p>
    Formula:C23H30O6
    Purity:98.26% - 98.85%
    Color and Shape:White Crystalline Powder
    Molecular weight:402.48
  • Fluocinolone (Acetonide)

    CAS:
    <p>Fluocinolone Acetonide (Flucort-N) is a glucocorticoid derivative used topically in the treatment of various skin disorders.</p>
    Formula:C24H30F2O6
    Purity:99.29% - 99.82%
    Color and Shape:Crystals From Acetone & Hexane Solid
    Molecular weight:452.49
  • Dexamethasone

    CAS:
    <p>Dexamethasone: a glucocorticoid agonist; modulates IL receptors; reduces inflammatory miRNA-155 exosomes in macrophage responses.</p>
    Formula:C22H29FO5
    Purity:98% - 99.91%
    Color and Shape:Crystals From Ether (Ntp 1992)
    Molecular weight:392.46
  • Desonide

    CAS:
    <p>Desonide is a synthetic topical steroid that reduces inflammation by inhibiting key inflammatory mediators.</p>
    Formula:C24H32O6
    Purity:99.5% - 99.74%
    Color and Shape:Solid
    Molecular weight:416.51
  • Cortisone acetate

    CAS:
    <p>Cortisone Acetate is a synthetic or semisynthetic analog of the naturally occurring cortisone hormone produced by the adrenal glands with anti-inflammatory and</p>
    Formula:C23H30O6
    Purity:98.63% - 99.73%
    Color and Shape:Solid
    Molecular weight:402.48
  • Mifepristone

    CAS:
    <p>Mifepristone (C-1073) is a progesterone-receptor (IC50=0.2 nM) and glucocorticoid-receptor antagonist (IC50=2.6 nM). High-Quality, Low-Cost!</p>
    Formula:C29H35NO2
    Purity:98.9% - ≥95%
    Color and Shape:Pale Yellow Solid
    Molecular weight:429.59
  • Cortisone

    CAS:
    <p>Cortisone (17-Hydroxy-11-dehydrocorticosterone) is a corticosteroid with potent glucocorticoid activity.</p>
    Formula:C21H28O5
    Purity:95.48% - 99.5%
    Color and Shape:Solid
    Molecular weight:360.44
  • Medrysone

    CAS:
    <p>Medrysone is a synthetic glucocorticoid for topical use with anti-inflammatory and anti-allergic effects, altering gene expression to reduce inflammation.</p>
    Formula:C22H32O3
    Purity:97.72% - 99.91%
    Color and Shape:Solid
    Molecular weight:344.49
  • Clobetasone butyrate

    CAS:
    <p>Clobetasone butyrate, a synthetic glucocorticoid with topical anti-inflammatory activity, is effective in treating corticosteroid-responsive dermatoses, such as</p>
    Formula:C26H32ClFO5
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:478.98
  • Nimodipine

    CAS:
    <p>Nimodipine (BAY-e 9736), a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.</p>
    Formula:C21H26N2O7
    Purity:99.64% - 99.79%
    Color and Shape:Solid
    Molecular weight:418.44
  • Dexamethasone acetate

    CAS:
    <p>Dexamethasone acetate (NSC 39471) is a potent anti-inflammatory steroid, blocks NF-kB, and lacks salt-retention.</p>
    Formula:C24H31FO6
    Purity:99.22% - 99.65%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:434.50
  • GW-870086

    CAS:
    <p>GW-870086 is an effective anti-inflammatory agent.</p>
    Formula:C31H39F2NO6
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:559.64
  • Dexamethasone Phosphate disodium

    CAS:
    <p>Dexamethasone Phosphate disodium (EGP437. Dex-Phos) is a water-soluble form of the synthetic glucocorticoid dexamethasone.</p>
    Formula:C22H28FNa2O8P
    Purity:99.76% - 99.848%
    Color and Shape:White To Off White Powder
    Molecular weight:516.4
  • Beclometasone dipropionate

    CAS:
    <p>Beclometasone dipropionate (Vancenase) is the dipropionate ester of a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.</p>
    Formula:C28H37ClO7
    Purity:98% - 98.49%
    Color and Shape:Solid
    Molecular weight:521.04
  • Dexamethasone phosphate

    CAS:
    <p>Dexamethasone phosphate is a synthetic adrenal corticosteroid. It also has potent anti-inflammatory properties.</p>
    Formula:C22H30FO8P
    Color and Shape:Solid
    Molecular weight:472.44
  • Nuclear Receptor Compound Library


    <p>A unique collection of 531 nuclear receptor signaling targeted compounds for high throughput and high content screening;</p>
    Color and Shape:Odour Solid
  • Prednicarbate

    CAS:
    <p>Prednicarbate (Hoe 777), a corticosteroid, has antipruritic, anti-inflammatory effects, reduces lymphocytes, and inhibits vasodilators.</p>
    Formula:C27H36O8
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:488.57
  • Zavacorilant

    CAS:
    <p>Zavacorilant is capable of modulating glucocorticoid receptor (GR).</p>
    Formula:C25H26FN7O3S2
    Color and Shape:Solid
    Molecular weight:555.65
  • BI 653048 phosphate

    CAS:
    <p>BI 653048 phosphate is a selective and orally active agonist of nonsteroidal glucocorticoid (GC)(IC50 : 55 nM).</p>
    Formula:C23H28F4N3O8PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:613.52
  • BI 653048

    CAS:
    <p>BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). BI 653048 is also an HCV NS3 protease inhibitor.</p>
    Formula:C23H25F4N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.52
  • Betamethasone acibutate

    CAS:
    <p>Betamethasone acibutate, a glucocorticoid, is derived from Betamethasone.</p>
    Formula:C28H37FO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:504.59
  • (Rac)-Finerenone

    CAS:
    <p>Rac-Finerenone, or (Rac)-BAY 94-8862, is an oral nonsteroidal MR antagonist with high selectivity and an IC50 of 18 nM.</p>
    Formula:C21H22N4O3
    Color and Shape:Solid
    Molecular weight:378.432
  • Methylprednisolone Acetate


    <p>Methylprednisolone Acetate(Depo-Medrate) has the ability to inhibit oxygen free radicals and can be used to treat acute spinal cord injuries.</p>
    Formula:C24H32O6
    Purity:99.74%
    Color and Shape:Off-White Solid
    Molecular weight:416.51
  • Glucocorticoids receptor agonist 1

    CAS:
    <p>GRA-1, an arylpyrazole, is a potent glucocorticoid receptor agonist with robust anti-inflammatory effects and preserves insulin secretion.</p>
    Formula:C20H23FN2O
    Color and Shape:Solid
    Molecular weight:326.41
  • RS 21314

    CAS:
    <p>RS 21314 is a thiol ester corticosteroid that is topical.</p>
    Formula:C24H30F2O5S
    Color and Shape:Solid
    Molecular weight:468.55
  • Deacylcortivazol

    CAS:
    <p>Deacylcortivazol is a potent glucocorticoid that inhibits growth in glucocorticoid-resistant leukemia cells without receptor mediation.</p>
    Formula:C30H36N2O4
    Color and Shape:Solid
    Molecular weight:488.62
  • Hydrocortisone sodium succinate

    CAS:
    <p>Hydrocortisone sodium succinate is a glucocorticoid which is used to alleviate allergic reactions, particularly those of the skin and gums.</p>
    Formula:C25H34NaO8
    Color and Shape:Solid
    Molecular weight:485.529
  • Alclometasone

    CAS:
    <p>Alclometasone is a glucocorticoid that reduces inflammation and treats various skin conditions like eczema and psoriasis.</p>
    Formula:C22H29ClO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.92
  • Ocedurenone

    CAS:
    <p>Ocedurenone, a corticosteroid receptor antagonist, is a compound utilized in the investigation of kidney disease (WO2018054357, compound I).</p>
    Formula:C28H30ClN5O2
    Color and Shape:Solid
    Molecular weight:504.03
  • Dagrocorat hydrochloride

    CAS:
    <p>PF-0251802 HCl is a bio-active chemical.</p>
    Formula:C29H30ClF3N2O2
    Color and Shape:Solid
    Molecular weight:531.01
  • AL-438

    CAS:
    <p>AL-438 is a non-steroidal selective glucocorticoid receptor modulator.</p>
    Formula:C23H25NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:347.45
  • BAY 1003803

    CAS:
    <p>BAY 1003803 is a glucocorticoid receptor agonist for the topical treatment of psoriasis or severe atopic dermatitis.</p>
    Formula:C21H18ClF5N2O4
    Color and Shape:Solid
    Molecular weight:492.83
  • OP-3633

    CAS:
    <p>OP-3633: potent GR antagonist (IC50: 29 nM), low PR agonism, AR antagonism, inhibits GR transcription.</p>
    Formula:C30H39NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.64
  • CP-472555

    CAS:
    <p>CP-472555 is a selective nonsteroidal glucocorticoid receptor antagonist with anti-GR and anti-obesity activity in animal models.</p>
    Formula:C31H32N2O2
    Color and Shape:Solid
    Molecular weight:464.60
  • PPARγ/GR modulator 1


    <p>PPARγ/GR Modulator 1, an orally active dual agonist for the Peroxisome Proliferator-Activated Receptor Gamma (PPARγ) and Glucocorticoid Receptor (GR), exhibits</p>
    Formula:C14H10FNO4
    Color and Shape:Solid
    Molecular weight:275.23
  • EX-A5386

    CAS:
    <p>EX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50/EC50&lt;100nM.</p>
    Formula:C29H27FN4O2
    Purity:99.89%
    Color and Shape:Soild
    Molecular weight:482.55
  • Triamcinolone Benetonide

    CAS:
    <p>Triamcinolone benetonide is a synthetic glucocorticoid corticosteroid exhibiting potent anti-inflammatory properties.</p>
    Formula:C35H42FNO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:623.71
  • Glucocorticoids receptor agonist 2

    CAS:
    <p>Arylpyrazole-based glucocorticoid agonist with potent anti-inflammatory effects; doesn't affect insulin secretion.</p>
    Formula:C25H25FN2O
    Color and Shape:Solid
    Molecular weight:388.48
  • Prednisolone farnesylate

    CAS:
    <p>Prednisolone farnesylate is a novel transdermal corticosteroid with anti-inflammatory activity.</p>
    Formula:C36H50O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:578.78
  • Betamethasone 17-benzoate

    CAS:
    <p>Betamethasone 17-benzoate is a representative steroid. It also can be used in the treatment of recurrent aphothous ulcers (RAU).</p>
    Formula:C29H33FO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:496.57
  • Dexamethasone cipecilate

    CAS:
    <p>Dexamethasone cipecilate is a long-acting intranasal corticosteroid and a highly lipophilic anti-inflammatory corticosteroid.</p>
    Formula:C33H43FO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:570.69
  • Rofleponide

    CAS:
    <p>Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.</p>
    Formula:C25H34F2O6
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:468.53
  • Flucloronide

    CAS:
    <p>Flucloronide is a corticosteroid for topical use on the skin. It has anti-inflammatory properties.</p>
    Formula:C24H29Cl2FO5
    Color and Shape:Solid
    Molecular weight:487.39
  • NR3C1 Protein, Human, Recombinant (His)


    <p>NR3C1 (Nuclear Receptor Subfamily 3 Group C Member 1) is a Protein Coding gene.</p>
    Color and Shape:Lyophilized Powder
    Molecular weight:10.95 kDa (predicted)
  • Prednisolone valerate acetate

    CAS:
    <p>Prednisolone valerate acetate is a prodrug anti-inflammatory and immunosuppressive,converted to the active form of Prednisolone and glucocorticoid receptor.</p>
    Formula:C28H38O7
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:486.6
  • Diflorasone Diacetate

    CAS:
    <p>Diflorasone Diacetate, a topical glucocorticoid, has immunosuppressive and anti-inflammatory properties.</p>
    Formula:C26H32F2O7
    Color and Shape:Crystals
    Molecular weight:494.53
  • Hydrocortisone buteprate

    CAS:
    <p>Hydrocortisone buteprate is a medium-potent, non-halogenated double-ester of hydrocortisone with a highly favorable benefit-to-risk ratio for inflammatory skin disorders.</p>
    Formula:C28H40O7
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:488.61
  • Hydrocortisone cypionate

    CAS:
    <p>Hydrocortisone cypionate is a corticosteroid ester and synthetic glucocorticoid corticosteroid.</p>
    Formula:C29H42O6
    Color and Shape:Solid
    Molecular weight:486.64
  • Desoxycorticosterone pivalate

    CAS:
    <p>DOCP, a mineralocorticoid, treats dogs with adrenal insufficiency.</p>
    Formula:C26H38O4
    Color and Shape:Solid
    Molecular weight:414.58
  • Anti-NR3C1 Antibody (9X89)


    <p>Anti-NR3C1 Antibody (9X89) is an antibody targeting NR3C1. Anti-NR3C1 Antibody (9X89) can be used in ELISA, WB, FCM.</p>
    Color and Shape:Odour Liquid
  • Isoflupredone Acetate

    CAS:
    <p>Isoflupredone Acetate is a corticosteroid with the activity of topical anti-inflammatory.</p>
    Formula:C23H29FO6
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:420.47
  • (20S)-Protopanaxatriol

    CAS:
    <p>(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid</p>
    Formula:C30H52O4
    Purity:95% - 99%
    Color and Shape:Solid
    Molecular weight:476.73
  • Fluorometholone Acetate

    CAS:
    <p>Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.</p>
    Formula:C24H31FO5
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:418.50
  • Mirodenafil dihydrochloride

    CAS:
    <p>Mirodenafil dihydrochloride is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.</p>
    Formula:C26H39Cl2N5O5S
    Purity:99.64% - 99.78%
    Color and Shape:Solid
    Molecular weight:604.59
  • Canrenoate potassium

    CAS:
    <p>Canrenoate potassium (Soldactone) is a synthetic pregnadiene derivative with anti-aldosterone activity.</p>
    Formula:C22H29KO4
    Purity:99.04% - 99.18%
    Color and Shape:Light Yellow To Tan Powder
    Molecular weight:396.56
  • Apararenone

    CAS:
    <p>Apararenone (MT-3995) is a receptor antagonist of mineralocorticoid receptor which can be used to treat non-alcoholic steatohepatitis and diabetic nephropathy.</p>
    Formula:C17H17FN2O4S
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:364.39
  • Beclometasone

    CAS:
    <p>Beclometasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma.</p>
    Formula:C22H29ClO5
    Purity:99.41% - 99.68%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:408.92
  • Desoximetasone

    CAS:
    <p>Desoximetasone (Topicort) is a topical corticosteroid for treating skin conditions like rashes.</p>
    Formula:C22H29FO4
    Purity:99.06% - 99.89%
    Color and Shape:Solid
    Molecular weight:376.46
  • Osilodrostat

    CAS:
    <p>Osilodrostat (LCI699) is a potent inhibitor of human 11β-hydroxylase (CYP11B1) and aldosterone synthase (CYP11B2).Cost-effective and quality-assured.</p>
    Formula:C13H10FN3
    Purity:99.10% - 99.36%
    Color and Shape:Solid
    Molecular weight:227.24
  • Fludrocortisone acetate

    CAS:
    <p>Fludrocortisone acetate (9α-Fludrocortisone acetate) , a glucocorticoid-receptor agonist, binds to cytoplasmic receptors, translocates to the nucleus, and</p>
    Formula:C23H31FO6
    Purity:96.92% - 98.03%
    Color and Shape:Crystalline Solid
    Molecular weight:422.49
  • Fluorometholone

    CAS:
    <p>Fluorometholone (Fluoromethalone) is a corticosteroid, most often used after laser-based refractive surgery.</p>
    Formula:C22H29FO4
    Purity:99% - 99.15%
    Color and Shape:Solid
    Molecular weight:376.46
  • Hydrocortisone hemisuccinate

    CAS:
    <p>Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.</p>
    Formula:C25H34O8
    Purity:98.01% - 98.7%
    Color and Shape:Solid
    Molecular weight:462.53
  • AZD9977

    CAS:
    <p>AZD9977 is a novel, selective modulator of mineralocorticoid receptor .</p>
    Formula:C20H18FN3O5
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:399.37
  • Halobetasol propionate

    CAS:
    <p>Halobetasol propionate (BMY-30056) is the salt of halobetasol, a synthetic corticosteroid with anti-inflammatory, antipruritic, and vasoconstrictor activities.</p>
    Formula:C25H31ClF2O5
    Purity:99.89%
    Color and Shape:Distributed As 0 05% Ointment
    Molecular weight:484.96
  • Fluocinonide

    CAS:
    <p>Fluocinonide (Topsyn) (Vanos) is an effective glucocorticoid steroid, utilized in the treatment as the skin disorders anti-inflammatory agent.</p>
    Formula:C26H32F2O7
    Purity:98.33% - 99.70%
    Color and Shape:Solid
    Molecular weight:494.52
  • Corticosterone

    CAS:
    <p>Corticosterone (Kendall's compound B) is an adrenocortical steroid with salocorticoid and glucocorticoid activity that is orally active.</p>
    Formula:C21H30O4
    Purity:98.44% - ≥95%
    Color and Shape:Solid
    Molecular weight:346.46
  • Velsecorat

    CAS:
    <p>Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).</p>
    Formula:C32H32F2N4O6
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:606.62
  • AL 082D06

    CAS:
    <p>AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR.</p>
    Formula:C23H24ClN3O2
    Purity:99.05% - 99.06%
    Color and Shape:Solid
    Molecular weight:409.91
  • Methylprednisolone succinate

    CAS:
    <p>Methylprednisolone succinate (Methylprednisolone hemisuccinate) is a synthetic glucocorticoid and is widely used as an anti-inflammatory agent.</p>
    Formula:C26H34O8
    Purity:98.41% - 99.82%
    Color and Shape:White Or Almost-White Solid Powder
    Molecular weight:474.54
  • Ciclesonide

    CAS:
    <p>Ciclesonide (Alvesco)(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.</p>
    Formula:C32H44O7
    Purity:99.89% - >99.99%
    Color and Shape:Solid
    Molecular weight:540.69
  • Vamorolone

    CAS:
    <p>Vamorolone (VBP15) is a steroid-like drug that treats muscular dystrophy with fewer side effects and inhibits NF-κB.</p>
    Formula:C22H28O4
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:356.46
  • Diflorasone

    CAS:
    <p>Diflorasone is a synthetic glucocorticoid. It has anti-inflammatory and immunosuppressive effects by acting on gene expression.</p>
    Formula:C22H28F2O5
    Purity:99.02% - 99.92%
    Color and Shape:Solid
    Molecular weight:410.45
  • Beclometasone dipropionate monohydrate

    CAS:
    <p>Beclometasone dipropionate monohydrate, precursor to oral glucocorticoid for inflammation and asthma research.</p>
    Formula:C28H39ClO8
    Color and Shape:Solid
    Molecular weight:539.06
  • Cortodoxone

    CAS:
    <p>Cortodoxone (11-Desoxycortisol) is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.</p>
    Formula:C21H30O4
    Purity:99.26% - 99.87%
    Color and Shape:Solid
    Molecular weight:346.46
  • Osilodrostat phosphate

    CAS:
    <p>Osilodrostat phosphate is a potent oral 11β-hydroxylase inhibitor.</p>
    Formula:C13H13FN3O4P
    Color and Shape:Solid
    Molecular weight:325.23
  • LY404039

    CAS:
    <p>LY404039 (pomaglumetad) is an effective agonist of recombinant human mGlu2(Ki =149 nM)/mGlu3(Ki =92 nM).</p>
    Formula:C7H9NO6S
    Purity:99% - 99.92%
    Color and Shape:Solid
    Molecular weight:235.22
  • Finerenone

    CAS:
    <p>Finerenone (BAY-948862) is a selective and orally nonsteroidal antagonist of the mineralocorticoid receptor (MR). Cost effective and quality assured.</p>
    Formula:C21H22N4O3
    Purity:99.45% - 99.91%
    Color and Shape:Solid
    Molecular weight:378.42
  • Betamethasone disodium phosphate

    CAS:
    <p>Betamethasone disodium phosphate (Betamethasone 21-phosphate disodium salt) has anti-inflammatory activity and may be used in the study of rheumatoid arthritis.</p>
    Formula:C22H28FNa2O8P
    Purity:99.37%
    Color and Shape:White Powder
    Molecular weight:516.41
  • Triamcinolone hexacetonide

    CAS:
    <p>Triamcinolone hexacetonide, an exogenous synthetic corticosteroid, is a GR agonist used in the study of auto-reactive pericarditis and diabetic macular edema.</p>
    Formula:C30H41FO7
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:532.64
  • Hydrocortisone aceponate

    CAS:
    <p>Hydrocortisone aceponate (Hydrocortisone 17-propionate 21-acetate) is an effective topical glucocorticoid used in the form of a cream to treat various skin</p>
    Formula:C26H36O7
    Purity:98.12%
    Color and Shape:Solid
    Molecular weight:460.56
  • Timobesone

    CAS:
    <p>Timobesone is a topical corticosteroid.</p>
    Formula:C22H29FO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.53
  • Flumethasone pivalate

    CAS:
    <p>Flumethasone pivalate: antipruritic, anti-inflammatory, and vasoconstrictor; for adrenocortical suppression, skin atrophy, and telangiectasia studies.</p>
    Formula:C27H36F2O6
    Purity:99.57% - 99.95%
    Color and Shape:Solid
    Molecular weight:494.57
  • Fluticasone furoate

    CAS:
    <p>Fluticasone furoate (Avamys), a potent, trifluorinated steroid with anti-inflammatory effects, treats allergic rhinitis.</p>
    Formula:C27H29F3O6S
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:538.58
  • GSK9027

    CAS:
    <p>GSK9027, a nonsteroidal GR agonist, is a partial 2×GRE reporter gene activator, less potent than dexamethasone.</p>
    Formula:C27H19F4N3O2S
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:525.52
  • Demegestone

    CAS:
    <p>Demegestone: synthetic progestogen, progesterone receptor agonist, treats luteal insufficiency, no androgenic activity.</p>
    Formula:C21H28O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.45
  • Prednisolone hemisuccinate

    CAS:
    <p>Prednisolone hemisuccinate is a soluble glucocorticoid and cortisol exerts anti-inflammatory, immunosuppressive, and antiallergic by binding to GR receptor.</p>
    Formula:C25H32O8
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:460.52
  • Isoflupredone

    CAS:
    <p>Isoflupredone, a synthetic corticosteroid, inhibits inflammation and immune response in animals.</p>
    Formula:C21H27FO5
    Purity:97.62% - 99.85%
    Color and Shape:Solid
    Molecular weight:378.43
  • Paramethasone Acetate

    CAS:
    <p>Paramethasone Acetate is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive effects that can be used in the treatment of systemic lupus</p>
    Formula:C24H31FO6
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:434.50
  • Desisobutyryl-ciclesonide

    CAS:
    <p>Desisobutyryl-ciclesonide is the active metabolite of Ciclesonide with affinity for the glucocorticoid receptor. a glucocorticoid with anti-inflammatory.</p>
    Formula:C28H38O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:470.6
  • RU 752

    CAS:
    <p>RU 752 is an antagonist of mineralocorticoid receptor that inhibits aldosterone synthesis.</p>
    Formula:C22H30O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:358.47
  • J9

    CAS:
    <p>J9 is an inhibitor of Glucocorticoid resistance. J9 reverses Dexamethasone Resistance in T-cell Acute Lymphoblastic Leukemia.</p>
    Formula:C12H12N4
    Color and Shape:Solid
    Molecular weight:212.25
  • Glucocorticoid receptor-IN-2

    CAS:
    <p>Glucocorticoid receptor-IN-2 selectively targets GR with anti-inflammatory effects (IC50: 0.171 nM) and activates MMTV (EC50: 0.94 nM).</p>
    Formula:C25H20F4N6O2
    Color and Shape:Solid
    Molecular weight:512.46
  • INCB13739

    CAS:
    <p>INCB13739 is an 11β-HSD1 inhibitor that can be used in the study of hyperlipidemia and hypertriglyceridemia.</p>
    Formula:C28H25N3O4
    Purity:99.32%
    Color and Shape:Soild
    Molecular weight:467.52
  • RU 28318, potassium salt

    CAS:
    <p>mineralocorticoid receptor (MR) antagonist</p>
    Formula:C25H38KO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.67
  • Fludrocortisone

    CAS:
    <p>Fludrocortisone (Florinef) is a synthetic corticosteroid with moderate glucocorticoid potency and greater mineralocorticoid potency.Cost-effective and quality-assured.</p>
    Formula:C21H29FO5
    Purity:98.56% - 98.66%
    Color and Shape:White Solid
    Molecular weight:380.45
  • (S)-Baxdrostat

    CAS:
    <p>(S)-Baxdrostat is an S-enantiomer of Baxdrostat, which functions as an inhibitor of aldosterone synthase [1].</p>
    Formula:C22H25N3O2
    Color and Shape:Solid
    Molecular weight:363.45
  • Methylprednisolone Aceponate

    CAS:
    <p>Methylprednisolone Aceponate (SH 440), a non-halogenated corticosteroid, is a potent anti-inflammatory agent.</p>
    Formula:C27H36O7
    Purity:99.00% - 99.61%
    Color and Shape:Solid
    Molecular weight:472.57
  • RU 25055

    CAS:
    <p>RU 25055 is a synthetic antiglucocorticoid.</p>
    Formula:C24H26O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:378.53
  • PF-3882845

    CAS:
    <p>PF-3882845, a high affinity MR antagonist (IC50=2.7 nM) for hypertension, also targets progesterone receptor (IC50: 310 nM).</p>
    Formula:C24H22ClN3O2
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:419.9
  • RU 43044

    CAS:
    <p>RU 43044 is a selective glucocorticoid receptor antagonist that has exhibited an antidepressant-like effect.</p>
    Formula:C29H34O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.58
  • Org-34517

    CAS:
    <p>Org-34517, a glucocorticoid receptor (GR) antagonist, is used potentially for the treatment of depression.</p>
    Formula:C28H30O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.54
  • AZD2906

    CAS:
    <p>AZD2906: selective GR agonist with human/rat IC50s - 2.2/0.3 nM (PBMC), 41.6/7.5 nM (blood); induces rat bone marrow micronuclei.</p>
    Formula:C26H25FN4O3
    Color and Shape:Solid
    Molecular weight:460.5
  • Prednisolone Tebutate

    CAS:
    <p>Prednisolone Tebutate is a synthetic glucocorticoid, and is an antiinflammatory and immunosuppressant.</p>
    Formula:C27H38O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:458.59
  • AZD9567

    CAS:
    <p>AZD9567: potent, selective SGRM, oral, IC50=3.8nM, effective in SCW joint inflammation.</p>
    Formula:C27H28F2N4O3
    Purity:98.4%
    Color and Shape:Solid
    Molecular weight:494.53
  • Lorundrostat

    CAS:
    <p>Lorundrostat is an aldosterone synthase inhibitor.</p>
    Formula:C24H33N7O2
    Purity:95.47%
    Color and Shape:Solid
    Molecular weight:451.56
  • Glucocorticoid receptor agonist-1

    CAS:
    <p>Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].</p>
    Formula:C35H39NO6
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:569.69
  • Dagrocorat

    CAS:
    <p>Dagrocorat is a novel and dissociated agonist of glucocorticoid receptor.</p>
    Formula:C29H29F3N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:494.55
  • HP210

    CAS:
    <p>HP210, a selective glucocorticoid receptor modulator (SGRM), can suppress IL-1β and IL-6 mRNA expression, suggesting its utility in investigating inflammation-</p>
    Formula:C22H19N3O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:421.54
  • Spirorenone

    CAS:
    <p>Spirorenone (INN) is a novel aldosterone antagonist with anti-salt corticosteroid activity, used in metabolic disease research.</p>
    Formula:C24H28O3
    Purity:98.28% - 99.84%
    Color and Shape:Solid
    Molecular weight:364.48
  • Halobetasol

    CAS:
    <p>Halobetasol (Ulobetasol), a corticosteroid, is utilized in the research of severe localized psoriasis [1].</p>
    Formula:C22H27ClF2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:428.9
  • Dexamethasone palmitate

    CAS:
    <p>DXP, a lipophilic prodrug of Dexamethasone, has 47x less glucocorticoid receptor affinity; it's an agonist &amp; anti-inflammatory.</p>
    Formula:C38H59FO6
    Purity:99.28%
    Color and Shape:Solid
    Molecular weight:630.87
  • Amebucort

    CAS:
    <p>Amebucort is a synthetic glucocorticoid corticosteroid. It may used for the research of inflammatory disorders.</p>
    Formula:C28H40O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:488.61
  • RU28362

    CAS:
    <p>RU28362 is an agonist of glucocorticoid receptor.</p>
    Formula:C23H28O3
    Color and Shape:Solid
    Molecular weight:352.47
  • Glucocorticoid receptor agonist

    CAS:
    <p>Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.</p>
    Formula:C20H20F4N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.38
  • Glucocorticoid receptor-IN-1

    CAS:
    <p>Glucocorticoid receptor-IN-1 selectively modulates GR with anti-inflammatory effects, represses hMMP1 (IC50: 2.11 nM), and activates MMTV (EC50: 5.59 nM).</p>
    Formula:C24H19F4N7O2
    Color and Shape:Solid
    Molecular weight:513.45
  • Fosdagrocorat

    CAS:
    <p>Fosdagrocorat is an agonist of the dissociated glucocorticoid receptor.</p>
    Formula:C29H30F3N2O5P
    Color and Shape:Solid
    Molecular weight:574.53
  • Baxdrostat

    CAS:
    <p>Baxdrostat is an aldosterone synthase inhibitor.</p>
    Formula:C22H25N3O2
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:363.45
  • Dazucorilant

    CAS:
    <p>Dazucorilant (CORT113176), a selective non-steroidal GR modulator, has high affinity with a K i &lt;1 nM, useful for neurological research.</p>
    Formula:C29H22F4N4O3S
    Color and Shape:Solid
    Molecular weight:582.57
  • ORIC-101

    CAS:
    <p>ORIC-101 is a highly effective and selective glucocorticoid receptor antagonist (EC50: 5.6 nM). It also has anti-cancer activity.</p>
    Formula:C34H47NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:501.74
  • C108297

    CAS:
    <p>C108297: glucocorticoid modulator, combats diet obesity/inflammation, reduces appetite/lipid storage, boosts fat burn.</p>
    Formula:C30H36FN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.69
  • LEO 134310

    CAS:
    <p>LEO 134310: Selective, non-steroidal GR agonist with 14 nM EC50, for topical skin disease treatment.</p>
    Formula:C34H40N2O8
    Color and Shape:Solid
    Molecular weight:604.69
  • Glucocorticoid receptor activator 1

    CAS:
    <p>Glucocorticoid Receptor Activator 1, a phenyl nitrogen-heterocyclic precursor, acts as an activator of the glucocorticoid receptor (GR). By activating GR, it downregulates the expression of pro-inflammatory genes stimulated by TNF, making it useful for inflammation research.</p>
    Formula:C11H15Cl2NO2
    Color and Shape:Solid
    Molecular weight:264.15
  • Glucocorticoid receptor agonist-5

    CAS:
    <p>Glucocorticoid Receptoragonist-5 (compound 4) is an effective glucocorticoid molecule acting as a potent agonist for glucocorticoid receptors. It exhibits anti-inflammatory and immunosuppressive activities and serves as an ADC cytotoxin.</p>
    Formula:C36H40O7
    Color and Shape:Solid
    Molecular weight:584.7
  • 22-Hydroxy mifepristone

    CAS:
    <p>22-Hydroxy Mifepristone (RU 42698) is an orally active hydroxylated alcohol metabolite that exhibits both anti-progestational and anti-glucocorticoid activities. This compound contains an alkyne group and is capable of undergoing copper-catalyzed azide-alkyne cycloaddition (CuAAC) with azide-containing molecules. Furthermore, 22-Hydroxy Mifepristone demonstrates a relative binding affinity of 48% to the human glucocorticoid receptor.</p>
    Formula:C29H35NO3
    Color and Shape:Solid
    Molecular weight:445.59
  • S-HP210


    <p>S-HP210: selective GR modulator, blocks NF-κB (IC50: 1.92 μM), non-toxic to mouse fibroblasts.</p>
    Formula:C22H19N3O2S2
    Color and Shape:Solid
    Molecular weight:421.54
  • JTP-117968

    CAS:
    <p>JTP-117968: Non-steroidal SGRM, glucocorticoid receptor modulator, IC50 = 6.8 nM, offers better inhibitory/activatory balance.</p>
    Formula:C31H31F3N2O2
    Color and Shape:Solid
    Molecular weight:520.59
  • Cort108297

    CAS:
    <p>Cort108297: selective GR modulator/antagonist, high GR affinity (Ki: 0.45nM), no other steroid receptor affinity.</p>
    Formula:C26H25F4N3O3S
    Purity:98.36% - 99.94%
    Color and Shape:Solid
    Molecular weight:535.55
  • ZK 216348

    CAS:
    <p>ZK 216348 also binds to Progesterone and mineralocorticoid receptors (IC50s: 20.4 nM and 79.9 nM, respectively). ZK 216348 is a nonsteroidal selective glucocorticoid receptor agonist (IC50: 20.3 nM). ZK 216348 has an anti-inflammatory activity similar to</p>
    Formula:C24H23F3N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:476.45

    Ref: TM-T17291

    1mg
    Discontinued
    Discontinued product
  • Mapracorat

    CAS:
    <p>Mapracorat (ZK-245186, BOL-303242X) is a selective glucocorticoid receptor agonist,anti-inflammatory agent for atopic dermatitis and allergic conjunctivitis.</p>
    Formula:C25H26F4N2O2
    Color and Shape:Solid
    Molecular weight:462.48

    Ref: TM-T13451L

    1mg
    Discontinued
    Discontinued product
  • (S)-Mapracorat

    CAS:
    <p>(S)-Mapracorat is a selective and less active agonist of the glucocorticoid receptor.</p>
    Formula:C25H26F4N2O2
    Color and Shape:Solid
    Molecular weight:462.48

    Ref: TM-T13451

    1mg
    Discontinued
    Discontinued product
  • Budesonide

    CAS:
    <p>Budesonide (Pulmicort), an anti-inflammatory corticosteroid, has shown the effective glucocorticoid activitie and few mineralocorticoid activities. According to reports, Budesonide has extensively inhibitory effects against multiple cells types and mediators referred to allergic and nonallergic-mediated inflammatory. What's more, the anti-inflammatory action of budesonide has been revealed to contribute to the effectiveness of asthma.</p>
    Formula:C25H34O6
    Purity:99.03% - 99.72%
    Color and Shape:Crystals Solid
    Molecular weight:430.53

    Ref: TM-T0094

    50mg
    Discontinued
    100mg
    Discontinued
    200mg
    Discontinued
    500mg
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    1mL*10mM (DMSO)_old
    Discontinued
    Discontinued product
  • Relacorilant

    CAS:
    <p>Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.</p>
    Formula:C27H22F4N6O3S
    Purity:98.53% - 99%
    Color and Shape:Solid
    Molecular weight:586.56

    Ref: TM-T16727

    1mg
    Discontinued
    5mg
    Discontinued
    10mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    500mg
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    1mL*10mM (DMSO)_old
    Discontinued
    Discontinued product
  • 21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione


    <p>21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione is a valuable organic compound for life sciences research [Catalog No.: T67476, CAS No.: 37413-91-5].</p>
    Formula:C23H26O4
    Color and Shape:Solid
    Molecular weight:366.457

    Ref: TM-T67476

    ne
    Discontinued
    Discontinued product