Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(98 products)
- Adiponectin receptor(5 products)
- CFTR(66 products)
- CGRP Receptor(55 products)
- Calcium Channel(574 products)
- Chloride channel(54 products)
- GABA Receptor(372 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(2 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(55 products)
- Potassium Channel(304 products)
- Proton pump(42 products)
- SGLT(31 products)
- Sodium Channel(257 products)
- TRP/TRPV Channel(95 products)
Show 13 more subcategories
Found 2739 products of "Membrane Transporter/Ion Channel"
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Oxybutynin chloride
CAS:Oxybutynin chloride (Oxybutynin HCl) is an anticholinergic medication used to relieve urinary and bladder difficulties.Formula:C22H32ClNO3Purity:99.27% - >99.99%Color and Shape:White PowderMolecular weight:393.96ML418
CAS:ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.Formula:C19H24ClN3O3Purity:99.3%Color and Shape:SolidMolecular weight:377.87Ref: TM-T16110
1mg37.00€5mg79.00€1mL*10mM (DMSO)84.00€10mg111.00€25mg178.00€50mg288.00€100mg414.00€200mg583.00€NMDA-IN-1
CAS:NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).Formula:C20H23ClFN3OPurity:99.57%Color and Shape:SolidMolecular weight:375.87Hydrochlorothiazide
CAS:Hydrochlorothiazide (HCTZ) 是一种口服有效的噻嗪类的利尿药，可抑制转化 TGF-β/Smad 信号通路。它通过打开钙激活钾 (KCA) 通道发挥直接的血管松弛作用。它改善心脏功能，减少纤维化并具有降压作用。Formula:C7H8ClN3O4S2Purity:99.43% - 99.50%Color and Shape:Crystals Physical Description Crystals Or White Powder (Ntp 1992)Molecular weight:297.741-EBIO
CAS:1-EBIO (1-EBIO) is a calium channel agonist.Formula:C9H10N2OPurity:98.75%Color and Shape:SolidMolecular weight:162.19Meticrane
CAS:Meticrane (Arresten) is a sulphonamide-derivative with thiazide-like diuretic activity.Formula:C10H13NO4S2Purity:99.16%Color and Shape:SolidMolecular weight:275.34GABAA receptor agent 1
CAS:GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.Formula:C13H8ClN3O2Purity:99.31%Color and Shape:SolidMolecular weight:273.67Ref: TM-T11349
1mg35.00€5mg79.00€1mL*10mM (DMSO)86.00€10mg111.00€25mg215.00€50mg323.00€100mg469.00€200mg647.00€NS1652
CAS:NS1652 is an anion conductance inhibitor. NS1652 blocks chloride channel has an IC50 of 1.6 μM in human and mouse red blood cells.
Formula:C15H11F3N2O3Purity:99.62%Color and Shape:SolidMolecular weight:324.25Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Formula:C11H15NO5Purity:99.96%Color and Shape:Crystals From Benzene SolidMolecular weight:241.24Isoguvacine hydrochloride
CAS:Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.Formula:C6H10ClNO2Purity:99.59%Color and Shape:SolidMolecular weight:163.6γ-Aminobutyric acid
CAS:γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.Formula:C4H9NO2Purity:99.95%Color and Shape:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderMolecular weight:103.12Broflanilide
CAS:Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.Formula:C25H14BrF11N2O2Purity:99.82%Color and Shape:SolidMolecular weight:663.29Ref: TM-T10618
1mg50.00€2mg71.00€5mg105.00€1mL*10mM (DMSO)124.00€10mg170.00€25mg339.00€50mg557.00€100mg792.00€VU591
CAS:VU591 is a selective extra-renal potassium channel inhibitor with an IC₅₀ of 0.24 μM.Formula:C16H12N6O5Purity:99.29% - 99.53%Color and Shape:SolidMolecular weight:368.3Ref: TM-T13320L
5mg48.00€1mL*10mM (DMSO)49.00€10mg75.00€25mg133.00€50mg230.00€100mg344.00€500mg740.00€Indapamide
CAS:Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.Formula:C16H16ClN3O3SPurity:98.97% - 99.83%Color and Shape:SolidMolecular weight:365.83Fluxametamide
CAS:Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).Formula:C20H16Cl2F3N3O3Purity:99.49%Color and Shape:SolidMolecular weight:474.26MRZ 2-514
CAS:MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with KiFormula:C11H6BrN3O3Purity:98.459%Color and Shape:SolidMolecular weight:308.09Ref: TM-T12110
1mg92.00€5mg192.00€1mL*10mM (DMSO)212.00€10mg313.00€25mg620.00€50mg1,044.00€100mg1,404.00€Nav1.8-IN-4
CAS:Nav1.8-IN-4 is a potent Nav1.8 channel inhibitor with potential analgesic activity.Nav1.8-IN-4 can be used for pain and neurological related disorders.Formula:C20H14F4N2O3Purity:99.83%Color and Shape:SoildMolecular weight:406.33Ref: TM-T77693
1mg56.00€2mg80.00€5mg118.00€10mg178.00€25mg356.00€50mg580.00€100mg888.00€500mg1,783.00€Omeprazole metabolite Omeprazole sulfone
CAS:Omeprazole metabolite Omeprazole sulfone can inhibit proton pump.Formula:C17H19N3O4SPurity:99.87%Color and Shape:SolidMolecular weight:361.42Ref: TM-T12309
1mg47.00€2mg62.00€5mg92.00€1mL*10mM (DMSO)101.00€10mg145.00€25mg281.00€50mg423.00€100mg608.00€500mg1,251.00€Pentetrazol
CAS:Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.Formula:C6H10N4Purity:99.67% - 99.90%Color and Shape:Bitter Taste Aqueous Solutions Neutral To Litmus (Ntp 1992)Molecular weight:138.173,4,5-Trimethoxycinnamic acid
CAS:3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at theFormula:C12H14O5Purity:98.91%Color and Shape:SolidMolecular weight:238.24E 0747 FA
E 0747 FA is an antiarrhythmic compound that inhibits the voltage of action potential Vmax in Purkinje fibers of porcine heart.E 0747 FA inhibits Na channels in cardiac cells.Formula:C22H30ClN3O6Purity:98.54%Color and Shape:SolidMolecular weight:467.94Dooku1
CAS:Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.Formula:C13H9Cl2N3OSPurity:98.87% - 99.74%Color and Shape:SolidMolecular weight:326.2Ref: TM-T11076
1mg43.00€2mg56.00€1mL*10mM (DMSO)90.00€5mg93.00€10mg133.00€25mg259.00€50mg482.00€100mg695.00€Caloxin 2A1 TFA
Caloxin 2A1 TFA is a PM Ca2+ pump inhibitor that inhibits human red blood cell Ca2+-Mg2+-ATPase leakage.Formula:C66H92F3N19O24Purity:99.89%Color and Shape:SolidMolecular weight:1592.55Oxiracetam
CAS:Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.
Formula:C6H10N2O3Purity:99.67%Color and Shape:White Crystalline PowderMolecular weight:158.16TPC2-A1-P
CAS:TPC2-A1-P is a TPC2 agonist that can differentially activate two-pore channel 2 (TPC2) and mimic the activation of TPC2 with NAADP and PIP (2).Formula:C20H21BrF3NO3Purity:98.49%Color and Shape:SolidMolecular weight:460.29Ref: TM-T36806
1mg92.00€5mg225.00€1mL*10mM (DMSO)226.00€10mg374.00€25mg710.00€50mg1,153.00€100mg1,755.00€Ethaverine hydrochloride
CAS:Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.Formula:C24H30ClNO4Purity:99.66% - 99.90%Color and Shape:SolidMolecular weight:431.96Ref: TM-T0369
2mg42.00€5mg59.00€1mL*10mM (DMSO)81.00€10mg96.00€25mg165.00€50mg236.00€100mg339.00€200mg530.00€Bupivacaine hydrochloride
CAS:Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.Formula:C18H28N2O·HClPurity:99.89% - 99.9%Color and Shape:SolidMolecular weight:324.89Vocacapsaicin hydrochloride
CAS:Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.Formula:C26H42ClN3O4Purity:99.66% - 99.80%Color and Shape:SolidMolecular weight:496.08Prilocaine hydrochloride
CAS:Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.Formula:C13H21ClN2OPurity:99.97%Color and Shape:Needles White Or Off White Crystalline PowderMolecular weight:256.77Lotilaner
CAS:Lotilaner is a parasiticide.Formula:C20H14Cl3F6N3O3SPurity:99.56%Color and Shape:SolidMolecular weight:596.76Ref: TM-T15775
1mg44.00€2mg58.00€5mg94.00€1mL*10mM (DMSO)111.00€10mg144.00€25mg335.00€50mg550.00€100mg882.00€200mg1,188.00€FFN 511
CAS:Fluorescent false neurotransmitter (FFN)Formula:C17H20N2O2Purity:98%Color and Shape:SolidMolecular weight:284.35Tocainide hydrochloride
CAS:Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.Formula:C11H17ClN2OPurity:97%Color and Shape:SolidMolecular weight:228.72Bemegride
CAS:Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.Formula:C8H13NO2Purity:99.89%Color and Shape:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Molecular weight:155.19IK1 inhibitor PA-6
CAS:IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouseFormula:C31H32N4O2Purity:98.9%Color and Shape:SolidMolecular weight:492.61Phenibut
CAS:Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).Formula:C10H13NO2Purity:99.55%Color and Shape:SolidMolecular weight:179.22AZD 7009
CAS:AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.Formula:C23H34N4O5Purity:98.42% - 98.51%Color and Shape:SoildMolecular weight:446.54TRPV4 agonist-1 free base
CAS:TRPV4 agonist-1 free base (OUN67600) is an agonist of transient receptor potential vanilloid 4 (TRPV4;EC50 of 60 nM, in the hTRPV4 Ca2+ assay).Formula:C25H22F2N4O2Purity:99.79%Color and Shape:SolidMolecular weight:448.46Trichlormethiazide
CAS:Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.Formula:C8H8Cl3N3O4S2Purity:98.8% - 99.54%Color and Shape:SolidMolecular weight:380.66NEO 376
CAS:NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.Formula:C20H24ClN3OPurity:99.56%Color and Shape:SolidMolecular weight:357.88Ref: TM-T12207
1mg71.00€5mg133.00€1mL*10mM (DMSO)147.00€10mg205.00€25mg353.00€50mg495.00€100mg665.00€200mg893.00€T16Ainh-A01
CAS:T16Ainh-A01 is a potent TMEM16A chloride channel inhibitor with a 1 μM IC50, targeting CaCC.Formula:C19H20N4O3S2Purity:97.18% - 98.15%Color and Shape:SolidMolecular weight:416.52ATP synthase inhibitor 1
CAS:ATP synthase inhibitor 1 is an inhibitor of the c subunit of the F1/FO-ATP synthase complex.Formula:C17H18ClN3O3S2Purity:99.83%Color and Shape:SolidMolecular weight:411.93Z433927330
CAS:Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).Formula:C20H20N4O3Purity:99.78%Color and Shape:SolidMolecular weight:364.4Ref: TM-T13381
1mg43.00€1mL*10mM (DMSO)92.00€5mg96.00€10mg138.00€25mg264.00€50mg388.00€100mg532.00€200mg705.00€GFB-8438
CAS:GFB-8438 is a potent and subtype selective inhibitor of TRPC5(IC50s of 0.18 and 0.29 μM of hTRPC5 and hTRPC4, respectively).Formula:C16H14ClF3N4O2Purity:99.58%Color and Shape:SolidMolecular weight:386.76Ref: TM-T11394
2mg34.00€5mg50.00€1mL*10mM (DMSO)55.00€10mg77.00€25mg111.00€50mg166.00€100mg236.00€200mg349.00€Mebeverine hydrochloride
CAS:Mebeverine hydrochloride (Colofac Hydrochloride), a β-phenylethylamine derivative, is a potent α1 repector inhibitor, relaxing the muscles in and around the gutFormula:C25H35NO5Purity:99.81% - 99.81%Color and Shape:SolidMolecular weight:429.55Pivagabine
CAS:Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.Formula:C9H17NO3Purity:99.87%Color and Shape:SolidMolecular weight:187.24MK-7622
CAS:MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.Formula:C25H25N3O2Purity:99.77% - 99.8%Color and Shape:SolidMolecular weight:399.48Sulfacarbamide
CAS:Sulfacarbamide (Sulfanilylurea) is a blood sugar-lowering agent.Formula:C7H9N3O3SPurity:95.6% - 99.72%Color and Shape:SolidMolecular weight:215.23Moxidectin
CAS:Moxidectin (CL301423) is an anthelmintic for heartworm/intestinal worms in dogs, cats, horses, cattle, and sheep; oral/topical/injectable.Formula:C37H53NO8Purity:97.38%Color and Shape:Appearance White Or Pale Yellow Amorphous PowderMolecular weight:639.82RUVBL1/2 ATPase-IN-1
CAS:RUVBL1/2 ATPase-IN-1 inhibits RUVBL1/2 ATPase (IC50: 6.0/7.7 μM); useful in cancer research.Formula:C28H28F3N5OPurity:99.92%Color and Shape:SolidMolecular weight:507.55γ-DGG acetate(6729-55-1 free base)
CAS:gamma-DGG acetate(6729-55-1 free base) (γ-D-Glutamylglycine) is a competitive blocker of AMPA receptor.Formula:C9H16N2O7Purity:99.81%Color and Shape:SolidMolecular weight:264.23Ornidazole (Levo-)
CAS:Ornidazole (Levo-) (Levornidazole) is the levo-isomer of Ornidazole.Formula:C7H10ClN3O3Purity:99.8%Color and Shape:SolidMolecular weight:219.63Ropivacaine hydrochloride
CAS:Ropivacaine hydrochloride (Ropivacaine monohydrochloride) is the hydrochloride salt of ropivacaine, a local anesthetic of the amide type with analgesic activityFormula:C17H26N2O·HClPurity:99.85% - 99.95%Color and Shape:SolidMolecular weight:310.86Tertiapin-Q
CAS:Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).Formula:C106H175N35O24S4Purity:98.06% - 98.09%Color and Shape:SolidMolecular weight:2452Doxapram hydrochloride hydrate
CAS:Doxapram hydrochloride hydrate (Doxapram HCl) inhibits TASK-1, TASK-3, TASK-1/TASK-3 heterodimeric channel function with EC50 of 0.41, 37, 9 μM, respectively.Formula:C24H33ClN2O3C24H30N2O2·ClH·H2OPurity:99.64% - >99.99%Color and Shape:SolidMolecular weight:432.99Manidipine dihydrochloride
CAS:Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).Formula:C35H40Cl2N4O6Purity:99.76% - 99.86%Color and Shape:SolidMolecular weight:683.62Oxybutynin
CAS:Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.Formula:C22H31NO3Purity:97.81% - 99.57%Color and Shape:White To Off-White Crystalline PowderMolecular weight:357.49VU0134992 hydrochloride
CAS:VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).Formula:C20H32BrClN2O2Purity:>99.99%Color and Shape:SolidMolecular weight:447.84Norverapamil hydrochloride
CAS:Norverapamil HCl, a Verapamil metabolite, blocks L-type calcium channels and inhibits P-gp function.Formula:C26H37ClN2O4Purity:99.47%Color and Shape:SolidMolecular weight:477.04Ref: TM-T16339
1mg34.00€5mg105.00€1mL*10mM (DMSO)110.00€10mg177.00€25mg299.00€50mg447.00€100mg602.00€200mg842.00€Disopyramide
CAS:Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.Formula:C21H29N3OPurity:99.62%Color and Shape:SolidMolecular weight:339.47DCPIB
CAS:DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μMFormula:C22H28Cl2O4Purity:99.79% - 99.87%Color and Shape:SolidMolecular weight:427.36Ref: TM-T10979
2mg39.00€5mg57.00€1mL*10mM (DMSO)63.00€10mg87.00€25mg177.00€50mg301.00€100mg485.00€200mg690.00€Etifoxine hydrochloride
CAS:Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.Formula:C17H18Cl2N2OPurity:99.36%Color and Shape:SolidMolecular weight:337.24Gabapentin
CAS:Gabapentin (Neurontin) is an Anti-epileptic Agent.Formula:C9H17NO2Purity:99.55% - 99.91%Color and Shape:White To Off-White Crystalline Solid; Crystals From Ethanol/Ether SolidMolecular weight:171.24Pramocaine hydrochloride
CAS:Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.Formula:C17H27NO3·HClPurity:99.15% - 99.61%Color and Shape:Crystals White Or Off White Crystalline PowderMolecular weight:329.865,5-Dimethyloxazolidine-2,4-dione
CAS:5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.Formula:C5H7NO3Purity:99.12%Color and Shape:Drypowder PelletslargecrystalsMolecular weight:129.11Riparin III
CAS:Riparin III is an alcamide isolated from Aniba riparia that has exhibited effects of antidepressant and anxiolytic activities in acute stress behavioral models.Formula:C16H17NO4Purity:95.13%Color and Shape:SolidMolecular weight:287.31PF-04885614
CAS:PF-04885614 is a potent inhibitor of NaV1.8, has potential for neurological and neurodevelopmental diseases treatment.Formula:C13H14F3N3OPurity:98.02%Color and Shape:SolidMolecular weight:285.27Ref: TM-T12421
2mg42.00€5mg64.00€1mL*10mM (DMSO)64.00€10mg92.00€25mg170.00€50mg316.00€100mg447.00€200mg628.00€Mephenesin
CAS:Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.Formula:C10H14O3Purity:99.49%Color and Shape:SolidMolecular weight:182.22Emamectin Benzoate
CAS:Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropodsFormula:C56H81NO15Purity:98.68%Color and Shape:SolidMolecular weight:1008.256Suloctidil
CAS:Suloctidil is a peripheral vasodilator that was formerly used in the management of peripheral and cerebral vascular disorders.Formula:C20H35NOSPurity:99.75% - >99.99%Color and Shape:SolidMolecular weight:337.56GV-58
CAS:GV-58 agonizes N/P-Q-type Ca2+ channels (EC50: 7.21/8.81 μM) with 20x less inhibition on CDK kinases.Formula:C18H26N6OSPurity:97.36%Color and Shape:SolidMolecular weight:374.5Ref: TM-T11517
1mg49.00€5mg137.00€1mL*10mM (DMSO)150.00€10mg205.00€25mg409.00€50mg592.00€100mg827.00€500mg1,648.00€NS13001
CAS:NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).Formula:C17H16ClN7Purity:99.55%Color and Shape:SolidMolecular weight:353.81Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Formula:C10H12ClNO2Purity:98% - >99.99%Color and Shape:1992)Molecular weight:213.66Boc-LRR-AMC TFA
Boc-LRR-AMC TFA is a fluorogenic protease substrate for detecting trypsin-like activity in the 26S proteasome or 20S proteasome core.Formula:C35H53F3N10O9Purity:97.70%Color and Shape:SolidMolecular weight:814.85UK-124114
CAS:Selamectin, a derivative of ivermectin, is a macrocyclic lactone that enhances chloride channels in nematodes, inhibiting H. contortus larval growth.Formula:C43H63NO11Purity:99.31%Color and Shape:SolidMolecular weight:769.96Omeprazole sulfide
CAS:Omeprazole sulfide (Ufiprazole), a metabolite of Omeprazole, functions as a proton pump inhibitor.Formula:C17H19N3O2SPurity:98.83%Color and Shape:White To Slightly Collored Solid Solid CrystallineMolecular weight:329.42Nefiracetam
CAS:Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Formula:C14H18N2O2Purity:97.37%Color and Shape:White To Off-White Crystalline PowderMolecular weight:246.3DSP-2230
CAS:DSP-2230 is a selective blocker of Nav1.7/Nav1.8.Formula:C20H20F3N5O2Purity:97.14%Color and Shape:SolidMolecular weight:419.4Ref: TM-T15174
1mg34.00€5mg66.00€1mL*10mM (DMSO)73.00€10mg99.00€25mg205.00€50mg334.00€100mg537.00€200mg762.00€VU6036720
VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuit
Formula:C20H22ClFN4O2SPurity:98.1%Color and Shape:SoildMolecular weight:436.93Otilonium bromide
CAS:Otilonium bromide (SP63) , an antimuscarinic, is utilized as a spasmolytic agent.Formula:C29H43BrN2O4Purity:98.88% - 99.78%Color and Shape:White PowerMolecular weight:563.57Levamlodipine
CAS:Levamlodipine (S-amlodipine) belongs to the dihydropyridine group of calcium channel blockers.Formula:C20H25ClN2O5Purity:97.21%Color and Shape:White Crystal PowderMolecular weight:408.88Diltiazem hydrochloride
CAS:Diltiazem hydrochloride (RG 83606 HCl) is a benzothiazepine calcium channel blocking agent with vasodilating action.Formula:C22H27ClN2O4SPurity:98% - 99.65%Color and Shape:Odorless White PowderMolecular weight:450.98Synta66
CAS:Synta66 is a store-operated calcium entry channel Orai inhibitor, and used for the research of neurological disease.Formula:C20H17FN2O3Purity:99.57% - 99.84%Color and Shape:SolidMolecular weight:352.36Ref: TM-T13047
2mg34.00€5mg50.00€1mL*10mM (DMSO)55.00€10mg80.00€25mg147.00€50mg227.00€100mg339.00€200mg482.00€4-Aminopyridine
CAS:4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.Formula:C5H6N2Purity:91.61%Color and Shape:SolidMolecular weight:94.11GSK-7975A
CAS:GSK-7975A is a potent and orally available inhibitor of CRAC channel.Formula:C18H12F5N3O2Purity:98.92%Color and Shape:SolidMolecular weight:397.3Ref: TM-T15423
1mg42.00€2mg55.00€1mL*10mM (DMSO)87.00€5mg88.00€10mg130.00€25mg250.00€50mg378.00€100mg570.00€500mg1,189.00€Tetracaine hydrochloride
CAS:Tetracaine HCl (Pontocaine), a potent local anesthetic and antipruritic, is used in eye care and for surface/spinal anesthesia.Formula:C15H25ClN2O2Purity:99.72% - 99.94%Color and Shape:White Or Off White Crystalline PowderMolecular weight:300.82L-Cycloserine
CAS:L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.Formula:C3H6N2O2Purity:99.75% - 99.99%Color and Shape:Crystals White PowderMolecular weight:102.09Flindokalner
CAS:Flindokalner (BMS-204352) modulates potassium channels, enhances Kv7 subtypes and BKca, inhibits Kv7.1 (Ki=3.7μM), GABAA; has anxiolytic effects in vivo.Formula:C16H10ClF4NO2Purity:99.96%Color and Shape:SolidMolecular weight:359.7Eleclazine hydrochloride
CAS:Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).Formula:C21H17ClF3N3O3Purity:99.86%Color and Shape:SolidMolecular weight:451.83Ref: TM-T15207
1mg58.00€5mg110.00€1mL*10mM (DMSO)122.00€10mg166.00€25mg268.00€50mg403.00€100mg532.00€200mg705.00€Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFormula:C15H14FN3O3Purity:99.72% - 99.98%Color and Shape:Less Crystals Colourless CrystalsMolecular weight:303.29AChE/Aβ-IN-1
AChE/Aβ-IN-1 (compound 32) is a potent, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 86 nM and an NMDA receptor antagonist targeting theFormula:C20H25BrN4Color and Shape:SolidMolecular weight:401.34Volixibat
CAS:Volixibat, a selective inhibitor of the bile acid transporter, may treat non-alcoholic steatohepatitis.Formula:C38H51N3O12S2Purity:98%Color and Shape:SolidMolecular weight:805.95Elgodipine
CAS:Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.Formula:C29H33FN2O6Purity:99.84% - 99.98%Color and Shape:SolidMolecular weight:524.58AQP4 (205-215)
CAS:AQP4 (205-215) is a fragment of the water channel protein Aquaporin-4 (AQP4). This protein is an autoimmune antigen in optic neuromyelitis and, upon binding with CD40, is upregulated and presented in B cells. AQP4 is associated with neuromyelitis optica (NMO), an autoimmune inflammatory disease of the central nervous system (CNS).Formula:C48H75N13O17SColor and Shape:SolidMolecular weight:1138.25GsMTx4
CAS:GsMTx-4, mechanosensitive and stretch-activated ion channel inhibitor (CAS 1209500-46-8).Formula:C185H273N49O45S6Purity:98%Color and Shape:SolidMolecular weight:4095.84TRPA1 Antagonist 3
CAS:TRPA1 Antagonist 3 is a compound with photoswitchable properties that acts as an agonist on the TRPA1 channel, providing the ability for optical control.Formula:C11H8ClN3Color and Shape:SolidMolecular weight:217.66Cavα2δ-IN-1
CAS:Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a KiFormula:C18H27N5OColor and Shape:SolidMolecular weight:329.448GX 201
CAS:GX 201 is a selective NaV1.7 inhibitor, IC50 of < 3.2 nM for hNaV1.7.Formula:C25H27ClF4N2O4SPurity:99.81%Color and Shape:SolidMolecular weight:563EVT-401
EVT-401 (P2X7 receptor antagonist-1), a purinergic P2X7 receptor antagonist, demonstrates efficacy in combating neuroinflammation [1].Formula:C22H20F4N2O3Color and Shape:SolidMolecular weight:436.4Jingzhaotoxin III
CAS:NaV1.5 channels blockerFormula:C174H241N47O46S6Purity:98%Color and Shape:SolidMolecular weight:3919.47Conantokin G
CAS:GluN2B-specific NMDA receptor blocker; IC50=480 nM in neurons, ~300 nM in oocytes; neuroprotective.Formula:C88H138N26O44Purity:98%Color and Shape:White Lyophilised SolidMolecular weight:2264.21
