Metabolism
Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.
Subcategories of "Metabolism"
- AhR(41 products)
- Aminopeptidase(67 products)
- CETP(18 products)
- Carbonic Anhydrase(178 products)
- Casein Kinase(130 products)
- DHFR(33 products)
- Decarboxylase(4 products)
- Dehydrogenase(270 products)
- FAAH(64 products)
- FXR(58 products)
- Factor Xa(80 products)
- Fatty Acid Synthase(33 products)
- Ferroptosis(215 products)
- GR(3 products)
- GSNOR(3 products)
- Glucokinase(54 products)
- HIF/HIF Prolyl-Hydroxylase(142 products)
- HMG-CoA Reductase(33 products)
- Hydroxylase(30 products)
- IDO(82 products)
- LDL(8 products)
- Lipase(97 products)
- Lipid(59 products)
- Lipoxygenase(125 products)
- MAO(87 products)
- MPO(2 products)
- NAMPT(36 products)
- P450(6 products)
- PAI-1(25 products)
- PDE(166 products)
- PED(1 products)
- PKM(15 products)
- PPAR(164 products)
- Phospholipase(82 products)
- ROR(42 products)
- Retinoid Receptor(29 products)
- SGK(11 products)
- Thioredoxin(12 products)
- Transferase(30 products)
- Transporter(42 products)
- UGT(4 products)
- Xanthine Oxidase (XO) Inhibitors(9 products)
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Found 8625 products of "Metabolism"
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CAY10486
CAS:<p>CAY10486 blocks ACAT-1/2, which form cholesterol esters, potentially reducing atherosclerosis; inhibits LDL oxidation. IC50 ~60μM; 28% effect at 3μM.</p>Formula:C19H19NO4Color and Shape:SolidMolecular weight:325.36Epiroprim
CAS:<p>Epiroprim (Ro11-8958) is a selective dihydrofolate reductase (DHFR) inhibitor with antibacterial activity, inhibiting Staphylococcus and Streptococcus.</p>Formula:C19H23N5O2Purity:99.68% - >99.99%Color and Shape:SolidMolecular weight:353.42PDE5-IN-5
CAS:<p>PDE5-IN-5 is a selective inhibitor of phosphodiesterase 5 (PDE5) (IC50: 2.0 nM).</p>Formula:C23H20BrN3O4Color and Shape:SolidMolecular weight:482.33TM-1
CAS:<p>TM-1: PDHK inhibitor, IC50 - PDHK1: 2.97μM, PDHK2: 5.2μM, prevents PDHC phosphorylation, inhibits cancer cell growth.</p>Formula:C26H32N2O6Color and Shape:SolidMolecular weight:468.54MRL-871
CAS:<p>MRL-871 is a selective RORγt allosteric inhibitor, reducing IL-17a mRNA production in EL4 cells, interacting with PPARgamma in partial agonistic binding modes.</p>Formula:C22H12ClF3N2O3Purity:99.66%Color and Shape:SolidMolecular weight:444.79ASP3662
CAS:<p>ASP3662/SPI-62: Potent, selective CNS-penetrable 11β-HSD1 inhibitor; potential neuropathic pain treatment.</p>Formula:C19H16ClF3N4O2Color and Shape:SolidMolecular weight:424.8Trandolaprilate hydrate
CAS:<p>Trandolaprilate hydrate, a powerful ACE inhibitor and Trandolapril's main metabolite, is lipophilic with partial c-fos blocking.</p>Formula:C22H32N2O6Color and Shape:SolidMolecular weight:420.5Izumerogant
CAS:<p>Izumerogant is an inverse agonist of the retinoid-related orphan receptor-gamma (RORγ).</p>Formula:C22H18ClF4N5O2Color and Shape:SolidMolecular weight:495.86YCT529 free acid
CAS:<p>YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .</p>Formula:C29H25NO3Color and Shape:SolidMolecular weight:435.51D-Erythro-dihydrosphingosine
CAS:<p>D-Erythro-dihydrosphingosine (C18-Dihydrosphingosine) inhibits arachidonic acid release and cPLA2α activity.</p>Formula:C18H39NO2Purity:99.50% - 99.88%Color and Shape:SolidMolecular weight:301.51Kurasoin B
CAS:<p>Kurasoin B is an inhibitor of protein farnesyltransferase.</p>Formula:C18H17NO2Color and Shape:SolidMolecular weight:279.33S07-2010
CAS:<p>S07-2010 is a pan-Aldo-Keto Reductase 1C3 (AKR1C3) inhibitor with potential anti-cancer activity, inducing apoptosis in A549/DDP cells.</p>Formula:C19H21N3O3SPurity:98.13%Color and Shape:SolidMolecular weight:371.45CAY10761
CAS:<p>CAY10761 inhibits ENPP1 (IC50: 467 μM human, 429 μM snake), mushroom tyrosinase (Ki: 1.9 μM), and urease from different sources (IC50: 0.093-<0.125 mM).</p>Formula:C7H8N4O2S2Color and Shape:SolidMolecular weight:244.29FR-221647
CAS:<p>FR-221647: non-nucleoside adenosine deaminase blocker, moderate efficacy, better pharmacokinetics than EHNA/Pentostatin.</p>Formula:C14H17N3O2Color and Shape:SolidMolecular weight:259.311β-HSD1-IN-10
CAS:<p>11β-HSD1-IN-10, a potent inhibitor of 11β-HSD1 with an IC50 value of 1.8 µM for humans, is suitable for research into obesity, hyperglycemia, and cognitive</p>Formula:C16H10F3NO2Color and Shape:SolidMolecular weight:305.25IQA
CAS:<p>IQA is a casein kinase 2 (CK2) inhibitor.</p>Formula:C17H12N2O3Color and Shape:SolidMolecular weight:292.29103D5R
CAS:<p>103D5R selectively inhibits hif-1α, reducing its levels in hypoxia or with cobalt ions, dose- and time-dependently.</p>Formula:C20H21N3O2Color and Shape:SolidMolecular weight:335.4hCAI/II-IN-2
CAS:<p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>Formula:C12H12N4O5S2Color and Shape:SolidMolecular weight:356.3814-dehydro Zymostenol
CAS:<p>14-dehydro Zymostenol, a cholesterol precursor, boosts MBP+ oligodendrocytes from precursors at 5.8-17 μM.</p>Formula:C27H44OColor and Shape:SolidMolecular weight:384.64Albaconazole
CAS:<p>Albaconazole, a small fungal CYP51A1 inhibitor, treats fungal infections and some musculoskeletal disorders.</p>Formula:C20H16ClF2N5O2Purity:99.27%Color and Shape:SolidMolecular weight:431.82Autotaxin-IN-1
CAS:<p>Autotaxin-IN-1: strong inhibitor for osteoarthritis pain; IC50=2.2 nM; good PK and PK/PD.</p>Formula:C21H23N7O2Purity:98%Color and Shape:SolidMolecular weight:405.45GlcN-6-P Synthase-IN-1
CAS:<p>'GlcN-6-P Synthase-IN-1, IC50 3.47 μM, inhibits GlcN-6-P synthase & CYP3A4. Has antimicrobial activity and CNS penetration.'</p>Formula:C20H21N7SColor and Shape:SolidMolecular weight:391.49DHODH-IN-17
CAS:<p>DHODH-IN-17 is a human DHODH inhibitor with an IC50 of 0.40 μM.</p>Formula:C12H9ClN2O2Purity:99.41% - 99.52%Color and Shape:SolidMolecular weight:248.67TPN729MA
CAS:<p>TPN729MA, a potent PDE5 inhibitor, IC50: 2.28 nM, targets erectile dysfunction research.</p>Formula:C29H40N6O8SColor and Shape:SolidMolecular weight:632.73Hexazinone
CAS:<p>Hexazinone: a triazine herbicide blocks photosynthesis by binding to D-1 protein in photosystem II.</p>Formula:C12H20N4O2Purity:99.99%Color and Shape:SolidMolecular weight:252.31AZD8329
CAS:<p>AZD8329 is an 11β-HSD1 inhibitor that inhibits 11β-HSD2, 17β-HSD1, 17β-HSD3, and can be used to study allergic reactions in humans.</p>Formula:C25H31N3O3Purity:99.31%Color and Shape:SolidMolecular weight:421.53Quetiapine sulfoxide
CAS:<p>Quetiapine sulfoxide: Main metabolite of Quetiapine, a 5-HT agonist & dopamine antagonist antipsychotic.</p>Formula:C21H25N3O3SPurity:98%Color and Shape:Pale Yellow SolidMolecular weight:399.51Loxoprofenol-SRS
CAS:<p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>Formula:C15H20O3Color and Shape:SolidMolecular weight:248.32BRD6897
CAS:<p>BRD6897 is a mitochondrial content inducer that increases the cellular content of mitochondria.</p>Formula:C25H21N3O2S2Purity:97.74%Color and Shape:SolidMolecular weight:459.58MEDS433
CAS:<p>MEDS433 inhibits dihydroorotate dehydrogenase (IC50 1.2 nM) and blocks replication of hCoV-OC43, hCoV-229E, SARS-CoV-2 at nanomolar levels.</p>Formula:C20H11F4N3O2Color and Shape:SolidMolecular weight:401.31(R)-Bromoenol lactone
CAS:<p>(R)-Bromoenol lactone (BEL) irreversibly inhibits iPLA2γ with 0.6 μM IC50, not affecting iPLA2β unless at 20-30 μM doses.</p>Formula:C16H13BrO2Color and Shape:SolidMolecular weight:317.18IDO1-IN-2
CAS:<p>IDO1-IN-2 is a potent and selective IDO1 inhibitor with IC50s of 81 nM, 59 nM (mouse), and 28 nM (rat), respectively. It has anti-cancer activity.</p>Formula:C15H17FN6O4Purity:98%Color and Shape:SolidMolecular weight:364.33PKM2 activator 3
CAS:<p>PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.</p>Formula:C15H11ClF2N2O3SColor and Shape:SolidMolecular weight:372.77SHP2 inhibitor LY6
CAS:<p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>Formula:C30H27Cl2N3O4Color and Shape:SolidMolecular weight:564.46Semotiadil recemate fumarate
CAS:<p>Semotiadil recemate fumarate is the recemate of Semotiadil fumarate. Semotiadil fumarate is a novel antagonist of vasoselective Ca2+ channel.</p>Formula:C33H36N2O10SPurity:98%Color and Shape:SolidMolecular weight:652.71Risarestat
CAS:<p>Risarestat (CT-112) is a potent aldose reductase inhibitor and thyroid hormone receptor (TR) antagonist for the treatment of hypoglycemia.</p>Formula:C16H21NO4SPurity:98.39%Color and Shape:SolidMolecular weight:323.41Rentiapril racemate
CAS:<p>Rentiapril racemate (SA-446 racemate) is the racemate of Rentiapril.Rentiapril racemate has anti-inflammatory activity and may be used in glaucoma research.</p>Formula:C13H15NO4S2Purity:98.96% - >99.99%Color and Shape:SolidMolecular weight:313.39LY367385
CAS:<p>LY367385 is a highly effective and selective mGluR1a antagonist.</p>Formula:C10H11NO4Purity:98%Color and Shape:SolidMolecular weight:209.2ACAT-IN-1 cis isomer
CAS:<p>ACAT-IN-1 cis isomer is a potent ACAT inhibitor (IC50: 100 nM) for the study of immune system-related diseases.</p>Formula:C29H25NO2Purity:>99.99%Color and Shape:SolidMolecular weight:419.51RORγt Inverse agonist 8
CAS:<p>RORγt Inverse agonist 8 is a potent, selective, orally bioavailable RORγt inverse agonist(human RORγt-LBD with an IC50 of 19 nM).</p>Formula:C26H33N7O2Purity:98%Color and Shape:SolidMolecular weight:475.59UK-500001
CAS:<p>UK-500001 is a potent PDE4 inhibitor with robust anti-inflammatory activity.</p>Formula:C26H24F3N3O4Purity:98%Color and Shape:SolidMolecular weight:499.48IDH-C227
CAS:<p>IDH-C227 is a selective and potent inhibitor of IDH1R132H that exhibits anticancer activity.</p>Formula:C30H31FN4O2Color and Shape:SolidMolecular weight:498.59hCAI/II-IN-1
CAS:<p>hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).</p>Formula:C18H29N5O3S3Color and Shape:SolidMolecular weight:459.65TFB-TBOA
CAS:<p>glial glutamate transporter EAAT1 and EAAT2 inhibitor</p>Formula:C19H17F3N2O6Purity:98%Color and Shape:SolidMolecular weight:426.34Enpp-1-IN-6
CAS:<p>Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).</p>Formula:C22H28N4O5SColor and Shape:SolidMolecular weight:460.55UCK2 Inhibitor-2
CAS:<p>UCK2 Inhibitor-2 is a non-competitive inhibitor of uridine-cytidine kinase 2 (UCK2) with IC50=3.8 µM that inhibits UCK2-mediated nucleoside recycling in cells.</p>Formula:C28H23N3O4SPurity:98.76% - 99.25%Color and Shape:SolidMolecular weight:497.57Imazodan hydrochloride
CAS:<p>Imazodan hydrochloride (CI-914 HCl) is a potent and selective type III phosphodiesterase inhibitor used in the treatment of chronic congestive heart failure.</p>Formula:C13H13ClN4OPurity:98.97%Color and Shape:SolidMolecular weight:276.72Teludipine hydrochloride
CAS:Teludipine hydrochloride is a blocker of lipophilic calcium channel.Formula:C28H39ClN2O6Purity:98%Color and Shape:SolidMolecular weight:535.07Fodipir
CAS:<p>Fodipir, the active metabolite of mangafodipir, plays a crucial role in the mechanism of mangafodipir-mediated cytoprotection, specifically mitigating cell</p>Formula:C22H32N4O14P2Purity:98%Color and Shape:SolidMolecular weight:638.46Tralkoxydim
CAS:<p>Tralkoxydim (Tralkoxydime) is an alkyl ketone herbicide. Tralkoxydim works as an ACCase inhibitor.</p>Formula:C20H27NO3Purity:97.44%Color and Shape:SolidMolecular weight:329.43ONO-1603
CAS:<p>ONO-1603, a prolyl endopeptidase inhibitor, is used potentially for the treatment of Alzheimer's disease.</p>Formula:C16H19ClN2O3Purity:98%Color and Shape:SolidMolecular weight:322.79hCAIX-IN-11
CAS:<p>hCAIX-IN-11 inhibits carbonic anhydrases IX & XII with Ki of 32.7 nM & 623.5 nM, respectively.</p>Formula:C21H15ClN4O3Color and Shape:SolidMolecular weight:406.82Sterculic acid
CAS:<p>Sterculic acid inhibits SCD1 with IC50 of 0.9μM, affecting Δ9D desaturase activity.</p>Formula:C19H34O2Color and Shape:SolidMolecular weight:294.47Darexaban glucuronide
CAS:<p>Darexaban glucuronide is the major component in plasma after oral administration of darexaban to humans. Darexaban (YM150) is a direct inhibitor of factor Xa.</p>Formula:C33H38N4O10Color and Shape:SolidMolecular weight:650.68Diaplasinin
CAS:<p>Diaplasinin (PAI-749) is a potent inhibitor of plasminogen activator inhibitor-1 (PAI-1) with antithrombotic activity, used in cardiovascular disease research.</p>Formula:C32H31N5OPurity:99.02%Color and Shape:SolidMolecular weight:501.62(Rac)-Etavopivat
CAS:<p>(Rac)-Etavopivat, an oral PKR activator, targets sickle cell disease and haemoglobinopathies.</p>Formula:C22H23N3O6SColor and Shape:SolidMolecular weight:457.5ARL-67156 trisodium salt hydrate
CAS:<p>ARL-67156 trisodium salt hydrate is an ecto-ATPase inhibitor that prevents metabolism of P2 purinoceptor agonists.</p>Formula:C15H24Br2N5O12P3Color and Shape:SolidMolecular weight:719.11Seviteronel R enantiomer
CAS:<p>Seviteronel R enantiomer (VT-464 R enantiomer) is a Seviteronel isomer produced during the manufacturing process.</p>Formula:C18H17F4N3O3Purity:97.97% - >99.99%Color and Shape:SolidMolecular weight:399.34ZSET-845
CAS:<p>ZSET-845 is an enhancer of cognitive which enhances choline acetyltransferase activity in the hippocampus in the rat.</p>Formula:C21H18N2OPurity:98%Color and Shape:SolidMolecular weight:314.38γ-Methylleucine
CAS:<p>Gamma-Methylleucine (2-Amino-3-tert-butylpropionic acid) is an auxiliary for copper-catalyzed asymmetric Michael reactions.</p>Formula:C7H15NO2Purity:≥98%Color and Shape:SolidMolecular weight:145.2Mevalonic acid
CAS:<p>Mevalonic acid is essential for cell growth and proliferation,Mevalonic acid is a precursor in the mevalonate pathway.</p>Formula:C6H12O4Purity:98%Color and Shape:SolidMolecular weight:148.16ML218
CAS:<p>ML218 is an inhibitor of T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3).ML218 inhibits the synaptic activity of subthalamic nucleus (STN) neurons.</p>Formula:C19H26Cl2N2OPurity:99.2% - 99.45%Color and Shape:SolidMolecular weight:369.33HCAIX-IN-2
CAS:<p>HCAIX-IN-2 (compound 9d) is a selective inhibitor of carbonic anhydrase and acts on hCA IX (Ki: 24.6 nM) and hCA XII (Ki: 45.3 nM).</p>Formula:C19H16N8O4SColor and Shape:SolidMolecular weight:452.45Glucosylceramide synthase-IN-2
CAS:<p>T-690: Potent, BBB-permeable, oral GCS inhibitor; human IC50: 15 nM, mouse IC50: 190 nM; non-competitive with C8 ceramide/UDP glucose.</p>Formula:C22H20F3N3O4Color and Shape:SolidMolecular weight:447.41Choline theophyllinate
CAS:<p>Choline theophyllinate (Oxtriphylline) is the choline salt of theophylline, a small molecule PDE inhibitor that can be used to treat immune system disorders and</p>Formula:C12H21N5O3Purity:98%Color and Shape:SolidMolecular weight:283.33Dimethyl-bisphenol A
CAS:<p>DMBPA inhibits HIF-1α, promotes its degradation by detaching Hsp90, and reduces Vegfa mRNA expression.</p>Formula:C17H20O2Color and Shape:SolidMolecular weight:256.34Fenleuton
CAS:<p>Fenleuton is a 5-lipoxygenase inhibitor.</p>Formula:C17H15FN2O3Purity:98%Color and Shape:SolidMolecular weight:314.31L 656224
CAS:<p>L 656224 is a 5-LO inhibitor.</p>Formula:C20H21ClO3Purity:98%Color and Shape:SolidMolecular weight:344.83LGE-899
CAS:<p>LGE-899 (Sonidegib metabolite M48) is a main metabolite of Sonidegib which is an inhibitor of the hedgehog pathway.</p>Formula:C15H11F3O3Purity:99.93%Color and Shape:SolidMolecular weight:296.24Piritrexim
CAS:<p>Piritrexim (BW 301U) is an orally available fat-soluble dihydrofolate reductase inhibitor with pulmonary toxicity used in the study of uroepithelial carcinoma</p>Formula:C17H19N5O2Purity:98.50% - >99.99%Color and Shape:SolidMolecular weight:325.37Dacisteine
CAS:<p>Dacisteine (N,S-Diacetyl-L-cysteine) is an inhibitor of New Delhi metallo-beta-lactamase-1 (NDM-1, IC50 = 1000 μM).</p>Formula:C7H11NO4SPurity:99.57%Color and Shape:SolidMolecular weight:205.23PGAM1-IN-1
CAS:<p>PGAM1-IN-1 is an inhibitor of phosphoglycerate mutase 1 ( PGAM1 ) with an IC 50 of 6.4 μM [1].</p>Formula:C19H11ClFNO6SPurity:98%Color and Shape:SolidMolecular weight:435.81LAZABEMIDE
CAS:<p>Lazabemide (Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively).</p>Formula:C8H10ClN3OPurity:98%Color and Shape:SolidMolecular weight:199.64Abiraterone decanoate
CAS:<p>Abiraterone decanoate is a prodrug of Abiraterone that provides controlled release and prolonged inhibition of the enzyme CYP17 through intramuscular.</p>Formula:C34H49NO2Purity:99.69%Color and Shape:SolidMolecular weight:503.76AK-106
CAS:<p>AK-106, or AK106-001616, selectively inhibits cPLA2 and has NSAID-like analgesic effects.</p>Formula:C26H25N3O3Color and Shape:SolidMolecular weight:427.4911β-HSD1-IN-1
CAS:<p>11β-HSD1-IN-1 is an inhibitor of 11β-hydroxydehydrogenase 1 (11β-HSD1, IC50: 52 nM), and used for the treatment of pain.</p>Formula:C18H14ClF4N3OPurity:99.84%Color and Shape:SolidMolecular weight:399.77Aldophosphamide
CAS:<p>Aldophosphamide possesses apoptotic antitumor activity.</p>Formula:C7H15Cl2N2O3PPurity:98%Color and Shape:SolidMolecular weight:277.09ML299
CAS:<p>ML299 (VU0463568) is a dual PLD1/2 inhibitor (PLD1 and PLD2, IC50 of 6 nM, 20 nM, respectively).</p>Formula:C23H26BrFN4O2Purity:98%Color and Shape:SolidMolecular weight:489.38Acetyl-CoA Carboxylase-IN-1
CAS:<p>Acetyl-CoA Carboxylase-IN-1 (ACC-IN-1) is a potent acetyl-CoA carboxylase (ACC) inhibitor with antibacterial activity, used in metabolic disease research.</p>Formula:C13H9Br2N5Purity:98.73%Color and Shape:SolidMolecular weight:395.05KT109
CAS:<p>KT109 is a DAGLβ inhibitor (IC50=42nM), lessens LPS allodynia in mice without tolerance, and has no major side effects.</p>Formula:C27H26N4OPurity:98%Color and Shape:SolidMolecular weight:422.52Tanogitran
CAS:<p>Tanogitran, a coagulation factor Xa inhibitor, is used potentially for the treatment of septic shock.</p>Formula:C25H31N7O3Purity:98%Color and Shape:SolidMolecular weight:477.56Crilvastatin
CAS:<p>Crilvastatin (PMD 387) is an HMGCR inhibitor with cholesterol-lowering activity that inhibits cholesterol uptake in rats with hereditary hypercholesterolemia.</p>Formula:C14H23NO3Purity:98.69% - 99.54%Color and Shape:SolidMolecular weight:253.34T-1095A
CAS:<p>T-1095A, a T-1095 metabolite, inhibits SGLTs, lowers blood glucose, improves glucose intolerance in mice, and prevents neuropathy in diabetic rats.</p>Formula:C24H26O9Purity:98%Color and Shape:SolidMolecular weight:458.46α-Glucosidase-IN-3
CAS:<p>α-Glucosidase-IN-3 is an oleanolic acid oxime ester derivative targeting α-glucosidase and α-amylase with an IC50 value of 0.35 μM for α-glucosidase.</p>Formula:C39H53NO4Color and Shape:SolidMolecular weight:599.84IDO1/TDO-IN-3
CAS:<p>IDO1/TDO-IN-3 inhibits IDO1 (IC50: 0.005 μM) and TDO (IC50: 0.004 μM) with strong anti-tumor activity and low toxicity.</p>Formula:C16H6ClF2N3O2Color and Shape:SolidMolecular weight:345.69AGI-14100
CAS:<p>AGI-14100 is a novel and orally available mIDH1 inhibitor.AGI-14100 is used for the treatment of primary human myeloid leukemia.</p>Formula:C29H22ClF4N5O3Purity:99.91%Color and Shape:SolidMolecular weight:599.96POP-IN-2
CAS:<p>Compound 7k (POP-IN-2) is a potent POP inhibitor with Ki of 6 nM, useful in neurodegenerative and cancer studies.</p>Formula:C24H33BN2O5Color and Shape:SolidMolecular weight:440.34OL-135
CAS:<p>OL-135: CNS-accessible, potent, selective FAAH inhibitor with analgesic effects in animals, no motor impairment.</p>Formula:C21H22N2O2Color and Shape:SolidMolecular weight:334.41Oleyl Anilide
CAS:<p>"Oleyl analide (OA) inhibits ACAT (IC50 26 μM), linked to toxic oil syndrome (TOS) with eosinophilia, T-cell activation, and high IL-4, IL-2R, IL-5."</p>Formula:C24H39NOColor and Shape:SolidMolecular weight:357.57ARN19874
CAS:<p>ARN19874 is a selective, reversible uncompetitive N-acylphosphatidylethanolamine phospholipase D (NAPE-PLD) activity inhibitor. With an IC50 of ~34 μM[1].</p>Formula:C19H14N4O4SPurity:98%Color and Shape:SolidMolecular weight:394.4FTase-IN-1
CAS:<p>FTase-IN-1, a potent FTase inhibitor, has an IC50 of 0.35 μM with strong antitumor activity and cytotoxicity.</p>Formula:C23H16N2O2SColor and Shape:SolidMolecular weight:384.45α-Glucosidase-IN-2
CAS:<p>α-Glucosidase-IN-2 (compound 5d) is a potent inhibitor of α-Glucosidase, exhibiting an inhibitory concentration (IC50) of 9.48 μM, and functions as an</p>Formula:C17H11N3O2S2Color and Shape:SolidMolecular weight:353.42OSMI-3
CAS:<p>OSMI-3 is a potent and cell-permeable inhibitor of O-GlcNAc transferase (OGT) for the study of cancer and cardiovascular disease.</p>Formula:C32H35N3O9S2Purity:99.03% - 99.08%Color and Shape:SolidMolecular weight:669.7793-O17O
CAS:<p>93-O17O is a cationic lipidoid used in lipid nanoparticles for spleen-targeted delivery and genome editing in mice.</p>Formula:C44H83N3O6Color and Shape:SolidMolecular weight:750.152'-O-Methyladenosine
CAS:<p>2'-O-Methyladenosine, a methylated adenine residue is found in the urine of normals and adenosine deaminase deficient patients.</p>Formula:C11H15N5O4Purity:99.89%Color and Shape:White SolidMolecular weight:281.27AGN 191701
CAS:<p>AGN 191701 is an agonist of the Retinoid X receptor.</p>Formula:C23H28O2SPurity:98%Color and Shape:SolidMolecular weight:368.53sPLA2-X Inhibitor 31
CAS:<p>sPLA2-X Inhibitor 31 targets sPLA2-X with IC50: 26 nM; less effective on sPLA2-IIa (310 nM), sPLA2-V (2230 nM).</p>Formula:C19H15F3N2O4Purity:98%Color and Shape:SolidMolecular weight:392.33Spiraprilat
CAS:<p>Spiraprilat is an ACE inhibitor. It also is an active metabolite of spirapril.</p>Formula:C20H26N2O5S2Purity:98%Color and Shape:SolidMolecular weight:438.56OMDM-2
CAS:<p>OMDM-2 is a metabolically stable and selective inhibitor of anandamide cellular uptake (ACU), exhibiting a Ki value of 3.0 μM in RBL-2H3 cells.</p>Formula:C27H45NO3Purity:98%Color and Shape:SolidMolecular weight:431.6512(S)-HpETE
CAS:<p>12(S)-HpETE activates human blood leukocyte 5-LOE and mediates induction of c-fos and c-jun, activation of AP-1, and endothelium-dependent vasoconstriction.</p>Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47
