Metabolism
Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.
Subcategories of "Metabolism"
- AhR(41 products)
- Aminopeptidase(67 products)
- CETP(18 products)
- Carbonic Anhydrase(177 products)
- Casein Kinase(130 products)
- DHFR(32 products)
- Decarboxylase(4 products)
- Dehydrogenase(267 products)
- FAAH(63 products)
- FXR(58 products)
- Factor Xa(80 products)
- Fatty Acid Synthase(32 products)
- Ferroptosis(215 products)
- GR(3 products)
- GSNOR(3 products)
- Glucokinase(53 products)
- HIF/HIF Prolyl-Hydroxylase(142 products)
- HMG-CoA Reductase(32 products)
- Hydroxylase(30 products)
- IDO(82 products)
- LDL(8 products)
- Lipase(96 products)
- Lipid(59 products)
- Lipoxygenase(124 products)
- MAO(87 products)
- MPO(2 products)
- NAMPT(36 products)
- P450(6 products)
- PAI-1(25 products)
- PDE(166 products)
- PED(1 products)
- PKM(15 products)
- PPAR(164 products)
- Phospholipase(82 products)
- ROR(42 products)
- Retinoid Receptor(29 products)
- SGK(11 products)
- Thioredoxin(12 products)
- Transferase(30 products)
- Transporter(42 products)
- UGT(4 products)
- Xanthine Oxidase (XO) Inhibitors(9 products)
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Found 8595 products of "Metabolism"
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TMCB
CAS:<p>CK2 and ERK8 inhibitor</p>Formula:C11H9Br4N3O2Purity:98%Color and Shape:SolidMolecular weight:534.82α-Glucosidase-IN-20
CAS:<p>α-Glucosidase-IN-20 (Compound 3B) is a highly effective and orally active inhibitor of α-glucosidase.</p>Formula:C23H21NOSColor and Shape:SolidMolecular weight:359.48Brofaromine
CAS:Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A).Formula:C14H16BrNO2Color and Shape:SolidMolecular weight:310.19Lp-PLA2-IN-11
CAS:<p>Lp-PLA2-IN-11, a potent Lp-PLA2 inhibitor, may be explored for atherosclerosis and Alzheimer's (WO2014114249A1, E145).</p>Formula:C22H20F4N4O3Color and Shape:SolidMolecular weight:464.41DHODH-IN-21
CAS:<p>DHODH-IN-21, orally active DHODH blocker with 1.1 nM IC50, shows anticancer activity, potential for AML research.</p>Formula:C20H19ClF4N6O4Color and Shape:SolidMolecular weight:518.85LEO-29102
CAS:<p>LEO-29102: Potent, selective PDE4 inhibitor, promising for treating skin diseases, phase 2 efficacy in atopic dermatitis.</p>Formula:C20H22Cl2N2O5Color and Shape:SolidMolecular weight:441.31HIF-PHD-IN-2
CAS:<p>HIF-PHD-IN-2 (compound 25) is a highly effective PHD inhibitor, displaying IC50 values below 100 nM for PHD1, PHD2, and PHD3 [1].</p>Formula:C17H15N5O3SColor and Shape:SolidMolecular weight:369.4MB-07729
CAS:<p>MB-07729 inhibits fructose-1,6-bisphosphate with IC50: 189 nM (rat), 121 nM (monkey), 31 nM (human) for diabetes research.</p>Formula:C12H15N2O5PSPurity:99.54% - 99.64%Color and Shape:SolidMolecular weight:330.3α-Amylase-IN-2
CAS:<p>α-Glucosidase-IN-3, an oxime ester derivative of oleanolic acid (OA), exhibits inhibitory activity against α-glucosidase (IC50 = 1.28 µM) and α-amylase (IC50 =</p>Formula:C39H52BrNO4Color and Shape:SolidMolecular weight:678.74Glucosylceramide synthase-IN-1
CAS:<p>Potent oral GCS inhibitor T-036, crosses BBB, targets human (IC50: 31 nM) and mouse GCS (IC50: 51 nM), for Gaucher disease research.</p>Formula:C24H20F4N2O3Color and Shape:SolidMolecular weight:460.42α-Glycosidase-IN-1
CAS:<p>α-Glycosidase-IN-1 (compound MZ7) is a potent inhibitor of α-GLY (α-glycosidase) (IC50: 44.72 nM, Ki: 44.74 nM).</p>Formula:C21H19N9O6S2Color and Shape:SolidMolecular weight:557.56Agn 190727
CAS:<p>Agn 190727 is a retonoic acid receptor that can induce retinoid-induced hypertriglyceridemia.</p>Formula:C20H22O2Color and Shape:SolidMolecular weight:294.3911β-HSD1-IN-12
CAS:<p>11β-HSD1-IN-12 is an 11β-HSD1 inhibitor.11β-HSD1-IN-12 is implicated in the conversion of glucocorticoids in vivo and can be used to study metabolic syndrome</p>Formula:C19H27ClN2O3SPurity:99.68%Color and Shape:SolidMolecular weight:398.95HIF-1α-IN-3
CAS:<p>HIF-1α-IN-3, also known as Compound (S)-3f, is a hypoxia-selective inhibitor of HIF-1α. It exhibits potent antiestrogenic activity [1].</p>Formula:C19H17N5O2Color and Shape:SolidMolecular weight:347.37α-Glucosidase-IN-9
CAS:<p>α-Glucosidase-IN-9 (compound 7) is a highly potent α-glucosidase inhibitor with an IC50 of 55.6 μM, making it suitable for type II diabetes research [1].</p>Formula:C19H12N4OSColor and Shape:SolidMolecular weight:344.39Metyltetraprole
CAS:<p>Metyltetraprole: potent fungicide, effective against Zymoseptoria, low EC50 (0.002 ppm), inhibits respiratory chain.</p>Formula:C19H17ClN6O2Color and Shape:SolidMolecular weight:396.83Delapril
CAS:<p>Delapril is an ACE inhibitor. It blocks the conversion of angiotensin I to angiotensin II.</p>Formula:C26H32N2O5Purity:98%Color and Shape:SolidMolecular weight:452.54Liarozole HCl
CAS:<p>Liarozole HCl: antineoplastic, boosts ATRA levels, impedes cell growth, promotes differentiation, aromatase inhibitor.</p>Formula:C17H14Cl2N4Purity:98%Color and Shape:SolidMolecular weight:345.23Umbralisib sulfate
CAS:<p>Umbralisib sulfate, an oral dual PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), targets CLL T cells for blood cancer research.</p>Formula:C31H26F3N5O7SColor and Shape:SolidMolecular weight:669.63MDK-4823
CAS:<p>MDK-4823 (LMPTP inhibitor1) blocks LMPTP, fighting insulin resistance and diabetes in obesity.</p>Formula:C28H36N4OColor and Shape:SolidMolecular weight:444.61Enpp-1-IN-8
CAS:<p>Enpp-1-IN-8: potent inhibitor of enpp-1, an enzyme breaking down various nucleotide bonds; potential in cancer/infectious disease research.</p>Formula:C19H26N6O4SColor and Shape:SolidMolecular weight:434.51FAAH-IN-7
<p>FAAH-IN-7: Reversible FAAH inhibitor, IC50=8.29 nM, reduces oxidative stress, neuroprotective in neuroinflammation.</p>Formula:C26H29N3O4Color and Shape:SolidMolecular weight:447.53AGI-14100
CAS:<p>AGI-14100 is a novel and orally available mIDH1 inhibitor.AGI-14100 is used for the treatment of primary human myeloid leukemia.</p>Formula:C29H22ClF4N5O3Purity:99.91%Color and Shape:SolidMolecular weight:599.96SYN20028567
CAS:<p>SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].</p>Formula:C20H29N3O3SColor and Shape:SolidMolecular weight:391.53mEH-IN-1
CAS:<p>mEH-IN-1 (Compound 62) is a potent mEH enzyme inhibitor with an IC50 of 2.2 nM, relevant in preeclampsia, hypercholanemia, and cancer research.</p>Formula:C16H17F6NOSColor and Shape:SolidMolecular weight:385.37PDE11-IN-1
CAS:<p>PDE11-IN-1 is a PDE11 inhibitor and can be used for adrenal insufficiency research [1].</p>Formula:C16H10ClN3O3SColor and Shape:SolidMolecular weight:359.79CP 80633
CAS:<p>CP 80633 is a PDE4 inhibitor.</p>Formula:C18H24N2O3Purity:98%Color and Shape:SolidMolecular weight:316.39ATX inhibitor 8
CAS:<p>ATX inhibitor 8 is an inhibitor of the autocrine motor factor Autotaxin (ATX).</p>Formula:C28H26N10OColor and Shape:SolidMolecular weight:518.57hCAIX-IN-14
CAS:<p>hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .</p>Formula:C11H17ClN6O2SColor and Shape:SolidMolecular weight:332.81PKM2 activator 4
CAS:<p>PKM2 Activator 4, a chemical compound, functions as an activator of PKM2 with an activation concentration (AC 50) ranging from 1 to 10 μM.</p>Formula:C16H16N2O4SColor and Shape:SolidMolecular weight:332.37PF-04822163
CAS:<p>PF-04822163 is a potent inhibitor of PDE1 with IC50 value of 0.0024 μM.</p>Formula:C19H17ClN2O2Purity:99.55%Color and Shape:SolidMolecular weight:340.8SLC26A3-IN-3
CAS:<p>SLC26A3-IN-3 (compound 4az), a potent SLC26A3 inhibitor with an IC50 of 40 nM, is utilized for constipation and cystic fibrosis research [1].</p>Formula:C20H17IO5Color and Shape:SolidMolecular weight:464.25Antitumor agent-88
CAS:<p>Antitumor agent-88, a potent antimitotic, arrests G2/M phase, disrupts microtubules in breast cancer, and inhibits CYP1A1 (Ki: 1.4 μM).</p>Formula:C23H30N2O7SColor and Shape:SolidMolecular weight:478.56SPK-601
CAS:<p>SPK-601 is an inhibitor of phosphatidylcholine-specific phospholipase C.</p>Formula:C11H16KOS2Purity:98%Color and Shape:SolidMolecular weight:267.47CX08005
CAS:<p>CX08005 inhibits PTP1B, cuts liver fat, and improves microcirculation in NAFLD.</p>Formula:C28H39NO4Purity:≥98%Color and Shape:SolidMolecular weight:453.61Spirapril
CAS:<p>Spiropril is an ACE inhibitor antihypertensive drug, which belongs to the bicarboxyl group of ACE inhibitors and is used in the treatment of hypertension.</p>Formula:C22H30N2O5S2Color and Shape:SolidMolecular weight:466.61hCA IX-IN-2
<p>hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferative</p>Formula:C23H24N2O4STeColor and Shape:SolidMolecular weight:552.11Disulfamide
CAS:<p>Disulfamide: Oral carbonic anhydrase inhibitor, IC50 0.07 μM, diuretic by blocking Na+/HCO3- reabsorption.</p>Formula:C7H9ClN2O4S2Purity:98.1%Color and Shape:SolidMolecular weight:284.74VU0155056
CAS:<p>VU0155056 is a dual PLD1/2 inhibitor with IC50 < 1 µM in cellular assays, inhibits breast cancer cell invasion.</p>Formula:C25H26N4O2Purity:98.6% - 99.15%Color and Shape:SolidMolecular weight:414.5Arasertaconazole
CAS:<p>Arasertaconazole, a sterol-14-alpha demethylation inhibitor, is used potentially for the treatment of vulvovaginal candcanidiasis.</p>Formula:C20H15Cl3N2OSColor and Shape:SolidMolecular weight:437.77A-908292
CAS:<p>A-908292: potent ACC2 inhibitor with 38 nM IC50, useful for studying fatty acid metabolism.</p>Formula:C18H20N2O4SColor and Shape:SolidMolecular weight:360.43FABP-IN-2
CAS:<p>FABP-IN-2, a novel ligand for FABP3, demonstrates inhibition of both FABP3 and FABP4 with IC50 values of 1.16 μM and 4.27 μM, respectively.</p>Formula:C25H21ClN2O3Color and Shape:SolidMolecular weight:432.9hCAXII-IN-1
CAS:<p>hCAXII-IN-1 selectively inhibits HCA IX/XII, promising for new cancer drug development.</p>Formula:C20H17NO5Color and Shape:SolidMolecular weight:351.35McN3716
CAS:<p>McN3716 is a carnitine palmitoyltransferase I (CPT-1) inhibitor for the study of metabolic diseases.</p>Formula:C18H34O3Purity:>99.99%Color and Shape:SolidMolecular weight:298.46ENPP1 inhibitor 43
CAS:<p>ENPP1 inhibitor 43 is a novel small molecule for cancer immunotherapy.</p>Formula:C16H18N6O3SColor and Shape:SolidMolecular weight:374.42BN82002
CAS:<p>BN82002 (CDC25 Phosphatase Inhibitor I) is a synthetic inhibitor of CDC25 phophatases</p>Formula:C19H25N3O4Purity:98.24%Color and Shape:SolidMolecular weight:359.42PDE4-IN-11
CAS:<p>PDE4-IN-11: Potent PDE4 inhibitor with strong bronchodilatory and anti-inflammatory effects for airway disease research.</p>Formula:C21H19FN2O2Color and Shape:SolidMolecular weight:350.39Xanthine oxidase-IN-4
CAS:<p>Xanthine oxidase-IN-4: an oral XO inhibitor with 0.039 μM IC50, useful for hyperuricemia/gout research.</p>Formula:C15H13N5O2Color and Shape:SolidMolecular weight:295.3PRRSV/CD163-IN-1
CAS:<p>PRRSV/CD163-IN-1 blocks PRRSV GP2a/GP4 and CD163-SRCR5, aiding PRRS research.</p>Formula:C25H24FN5O5S2Color and Shape:SolidMolecular weight:557.62(+)-Cembrene A
CAS:<p>(+)-Cembrene A, a nontoxic α-glucosidase inhibitor to human normal hepatocyte (LO2) cells, exhibits an IC50 value of 30.31 μM.</p>Formula:C20H32Color and Shape:SolidMolecular weight:272.47AVE-8134
CAS:<p>AVE-8134 is an agonist of PPARα. For human and rodent PPARα receptor, the EC50 values are 100 and 3000 nM, respectively.</p>Formula:C22H23NO5Purity:98%Color and Shape:SolidMolecular weight:381.42hCAIX-IN-8
CAS:<p>hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.</p>Formula:C19H16N4O6Color and Shape:SolidMolecular weight:396.35ICI 153110
CAS:<p>ICI 153110: Oral phosphodiesterase inhibitor for treating congestive heart failure, has inotropic, vasodilator effects.</p>Formula:C11H11N3OPurity:98%Color and Shape:SolidMolecular weight:201.22Xanthine oxidase-IN-5
CAS:<p>Xanthine oxidase-IN-5: oral XO inhibitor, IC50 = 0.70 μM, LE = 0.33, LLE = 3.41, reduces uric acid in rats.</p>Formula:C18H16FN3O3Color and Shape:SolidMolecular weight:341.34Endothelial lipase inhibitor-1
CAS:<p>Endothelial lipase inhibitor-1 is a potent endothelial lipase inhibitor with an IC50 of 49 nM.</p>Formula:C22H22N4O4Purity:99.59%Color and Shape:SolidMolecular weight:406.43Lp-PLA2-IN-3
CAS:<p>Lp-PLA2-IN-3: Potent oral inhibitor of human Lp-PLA2 with a 14 nM IC50.</p>Formula:C20H13ClF3N3O3SPurity:99.65%Color and Shape:SolidMolecular weight:467.85Hydroxychlorodenafil
CAS:<p>Hydroxychlorodenafil is a derivative of the phosphodiesterase 5 (PDE5) inhibitor sildenafil.</p>Formula:C19H23ClN4O3Color and Shape:SolidMolecular weight:390.86HS79
CAS:<p>HS-79, a Fasnall enantiomer, selectively inhibits FASN with an IC50 of 1.57 μM, blocking tritiated acetate lipid incorporation.</p>Formula:C19H22N4SPurity:98%Color and Shape:SolidMolecular weight:338.47Deltasonamide 2
CAS:<p>Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.</p>Formula:C30H39ClN6O4S2Purity:98%Color and Shape:SolidMolecular weight:647.25AMG-221
CAS:<p>AMG-221: potent 11β-HSD1 inhibitor, lowers glucose & insulin, reduces obesity in mice.</p>Formula:C14H22N2OSPurity:98%Color and Shape:SolidMolecular weight:266.4Enazadrem
CAS:<p>Enazadrem is a 5-lipoxygenase inhibitor with antiinflammatory activities.</p>Formula:C18H25N3OPurity:98%Color and Shape:SolidMolecular weight:299.41JTP-4819
CAS:<p>JTP-4819: potent PEP inhibitor, may treat Alzheimer's, boosts brain peptides and acetylcholine, aiding memory.</p>Formula:C19H25N3O4Color and Shape:SolidMolecular weight:359.42Enpp-1-IN-10
CAS:<p>Enpp-1-IN-10 inhibits ENPP1 with 3.866 μM Ki, useful in cancer research.</p>Formula:C13H12N6OSColor and Shape:SolidMolecular weight:300.34Andolast
CAS:<p>Andolast (CR-2039) is an anti-allergic for asthma and COPD, inhibiting IgE synthesis and improving airflow.</p>Formula:C15H11N9OColor and Shape:SolidMolecular weight:333.31sEH inhibitor-14
CAS:<p>sEH inhibitor-14, a benzoxazolone-5-urea analogue, acts as an efficient soluble Epoxide Hydrolase (sEH) inhibitor, demonstrating significant activity with an</p>Formula:C16H12F3N3O4Color and Shape:SoildMolecular weight:367.282'-Ethyl Simvastatin
CAS:<p>2'-Ethyl Simvastatin is a Mevinolin analog with HMG-CoA reductase inhibition.</p>Formula:C23H34O5Purity:98%Color and Shape:SolidMolecular weight:390.51MitoTEMPO hydrate
CAS:<p>MitoTEMPO, a mitochondria-targeted antioxidant, scavenges superoxide and alkyl radicals supporting potential therapy for mitochondrial dysfunction.</p>Formula:C29H35N2O2P·Cl·H2OColor and Shape:SolidMolecular weight:528.04PGMI-004A
CAS:<p>PGMI-004A is an effective inhibitor of phosphoglycerate mutase 1 (IC50: 13.1 μM).</p>Formula:C21H12F3NO6SPurity:98%Color and Shape:SolidMolecular weight:463.38Manitimus
CAS:<p>Manitimus is a potent immunosuppressive drug, and is an inhibitor of dehydroorotate dehydrogenase,.</p>Formula:C15H11F3N2O2Purity:99.75% - 99.75%Color and Shape:SolidMolecular weight:308.26ATX inhibitor 11
CAS:<p>ATX inhibitor 11 blocks autotaxin (IC50: 2.7 nM), reduces fibrosis and α-SMA in mice. Useful for lung fibrosis studies.</p>Formula:C32H35N5O6Color and Shape:SolidMolecular weight:585.65UK-371804 HCl
CAS:<p>UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (2700-</p>Formula:C14H17Cl2N5O4SPurity:98%Color and Shape:SolidMolecular weight:422.29(3S,5R)-Fluvastatin sodium
CAS:<p>(3S,5R)-Fluvastatin sodium: synthetic HMG-CoA reductase inhibitor, IC50 8 nM, boosts vascular cell antioxidant defense.</p>Formula:C24H26FNNaO4Purity:98%Color and Shape:SolidMolecular weight:434.463SRPKIN-1
CAS:<p>SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).</p>Formula:C27H21FN2O3SPurity:98%Color and Shape:SolidMolecular weight:472.53AMPD2 inhibitor 1
CAS:<p>AMPD2 inhibitor 1 is an adenosine monophosphate deaminase 2 (AMPD2) inhibitor, useful for studying anorexia in the nervous system.</p>Formula:C25H22N2O2Color and Shape:SolidMolecular weight:382.45Xanthine oxidoreductase-IN-2
CAS:<p>Xanthine oxidoreductase-IN-2 inhibits XOR with 7.2 nM IC50 and shows hypouricemic effects in mice.</p>Formula:C21H19N3O2Color and Shape:SolidMolecular weight:345.39AX 048
CAS:<p>Group IVA cPLA2 inhibitor AX 048 halts arachidonic acid release, preventing prostaglandin production, with XI(50) of 0.022 and ED50 of 1.2 mg/kg.</p>Formula:C22H41NO4Color and Shape:SolidMolecular weight:383.57TUPS
CAS:<p>TUPS is a selective soluble epoxide hydrolase inhibitor which protects against isoprenaline-induced cardiac hypertrophy.</p>Formula:C14H18F3N3O4SColor and Shape:SolidMolecular weight:381.37α-Glucosidase-IN-10
CAS:<p>α-Glucosidase-IN-10 (compound 13) is a potent inhibitor of α-glucosidase (IC50: 92.7 μM). α-Glucosidase-IN-10 can be used to study type II diabetes.</p>Formula:C21H15BrN4O2SColor and Shape:SolidMolecular weight:467.34α-Glucosidase-IN-8
CAS:<p>α-Glucosidase-IN-8 (Compound 4k) is a potent, competitive inhibitor of α-glucosidase. It displays an impressive IC50 value of 0.18 μg/mL [1].</p>Formula:C19H20FN3O2Color and Shape:SolidMolecular weight:341.38Thialysine HCl
CAS:<p>Thialysine HCl is a cytotoxic cysteine derivative that inhibits Escherichia coli, acting as a protein synthesis inhibitor and metabolite.</p>Formula:C5H13ClN2O2SColor and Shape:SolidMolecular weight:200.69hCAIX-IN-6
CAS:<p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>Formula:C18H12N2O4SColor and Shape:SolidMolecular weight:352.36Carbonic anhydrase inhibitor 13
CAS:<p>Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).</p>Formula:C17H15N5O3S2Color and Shape:SolidMolecular weight:401.46IDO1-IN-17
CAS:<p>IDO1-IN-17 (I-4) is an IDO1 inhibitor, with an IC 50 of 0.44 μM in hela cells .</p>Formula:C28H32BrClFN5O2Color and Shape:SolidMolecular weight:604.94FAAH-IN-5
CAS:<p>FAAH-IN-5 (Compound 7) selectively, irreversibly inhibits FAAH (IC50: 10.5 nM) with low PAMPA permeability.</p>Formula:C21H19N3O6SColor and Shape:SolidMolecular weight:441.46IDH2R140Q-IN-1
CAS:<p>IDH2R140Q-IN-1 is a potent inhibitor of IDH2R140Q (IC50: 6.1 nM) and can be used in studies of acute myeloid leukemia.</p>Formula:C22H20F6N6Color and Shape:SolidMolecular weight:482.427-Ketolithocholic acid
CAS:<p>7-Ketolithocholic acid absorbs and reduces endogenous bile acid and cholesterol secretion.</p>Formula:C24H38O4Purity:98.68% - 99.9%Color and Shape:White - Almost White Solid PowderMolecular weight:390.56Rovazolac
CAS:<p>Rovazolac (ALX-101) is a liver x receptor (LXR) modulator used in the study of immune system disorders and atopic dermatitis.</p>Formula:C21H19F3N2O4SPurity:99.35%Color and Shape:SolidMolecular weight:452.45ALDH1A1-IN-2
CAS:<p>ALDH1A1-IN-2 is an aldehyde dehydrogenase 1a1 inhibitor with anticancer activity.ALDH1A1-IN-2 may be used in the study of breast cancer, inflammation or obesity</p>Formula:C25H23ClN4O3SPurity:99.48%Color and Shape:SolidMolecular weight:494.99PKR activator 2
CAS:<p>PKR activator 2 is a potent activator of pyruvate kinase-R (PKR).</p>Formula:C18H16N8OSPurity:98%Color and Shape:SolidMolecular weight:392.44LYS006
CAS:<p>LYS006 is a highly efficient and selective LTA4H (leukotriene A4 hydrolase) inhibitor,for neutrophil-driven inflammatory diseases ulcerative colitis.</p>Formula:C16H14ClFN6O3Purity:99.33%Color and Shape:SoildMolecular weight:392.77CYP3A4-IN-1
CAS:<p>CYP3A4-IN-1 is a potent inhibitor of cytochrome P450 3A4 (CYP3A4) (IC50: 0.085 μM).</p>Formula:C31H37N5O3SColor and Shape:SolidMolecular weight:559.72FXR agonist 4
<p>FXR agonist 4: EC50 of 1.05μM, treats hyperlipidemia, steatosis, insulin resistance, inflammation in DIO mice, for NAFLD research.</p>Formula:C21H28ClN3OColor and Shape:SolidMolecular weight:373.92BAY 73-6691
CAS:<p>BAY 73-6691 is an inhibitor of brain penetrant PDE9A.</p>Formula:C15H12ClF3N4OColor and Shape:SolidMolecular weight:356.73IDO/TDO-IN-1
CAS:<p>IDO/TDO-IN-1 is an orally active dual indoleamine-2,3-dioxygenase (IDO) and tryptophan 2,3-dioxygenase (TDO) inhibitor (IC50s: 9.7 and 47 nM).</p>Formula:C25H24FN5Purity:98%Color and Shape:SolidMolecular weight:413.49KCN1
CAS:<p>KCN1: a synthetic sulfonamide, nanomolar HIF inhibitor with preclinical anti-glioma and anti-pancreatic cancer effects.</p>Formula:C26H27NO5SColor and Shape:SolidMolecular weight:465.56F-1394
CAS:<p>F-1394 is an ACAT inhibitor that reduces atherosclerosis and neointimal thickening without changing serum cholesterol.</p>Formula:C33H61N3O6Color and Shape:SolidMolecular weight:595.85CYP1B1-IN-3
CAS:<p>CYP1B1-IN-3: strong CYP1B1 inhibitor (IC50: 6.6 nM); weak on CYP1A1/CYP1A2; hinders cell migration, invasion; blocks P-gp, AKT/ERK, FAK/SRC, EMT.</p>Formula:C20H16FN3O2S2Color and Shape:SolidMolecular weight:413.49PF-07208254
CAS:<p>PF-07208254, a potent BDK inhibitor, enhances cardiometabolic endpoints in mice [1].</p>Formula:C7H2ClFO2S2Purity:98%Color and Shape:SolidMolecular weight:236.67CM39
CAS:<p>CM39 inhibits ALDH, linked to cancer stem-like cells & chemoresistance.</p>Formula:C19H15FN4OSColor and Shape:SolidMolecular weight:366.41Oxythiamine diphosphate
CAS:<p>Oxythiamine diphosphate is a competitivethiamine pyrophosphate inhibitor(Ki of 30 nM).</p>Formula:C12H17N3O8P2SPurity:98%Color and Shape:SolidMolecular weight:425.29DTP348
CAS:<p>DTP348: Oral carbonic anhydrase IX inhibitor & hypoxic cell radiosensitizer with sulfamide & 5-nitroimidazole components.</p>Formula:C6H11N5O4SColor and Shape:SolidMolecular weight:249.25Nitrefazole
CAS:<p>Nitrefazole: a 4-nitroimidazole, inhibits ALDH enzyme crucial for alcohol metabolism, has potent, durable effects.</p>Formula:C10H8N4O4Color and Shape:SolidMolecular weight:248.19URB-694
CAS:<p>URB-694 is a fatty acid amide hydrolase (FAAH) inhibitor.</p>Formula:C19H21NO3Color and Shape:SolidMolecular weight:311.37Angiogenesis agent 1
CAS:<p>Compound C-31, a salidroside-based glycoside, activates HIF-1α and may aid in diabetic limb ischemia studies.</p>Formula:C20H24O7Purity:98%Color and Shape:SolidMolecular weight:376.411β-HSD1-IN-6
CAS:<p>11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs).</p>Formula:C21H19ClN4OColor and Shape:SolidMolecular weight:378.86WES-1
CAS:<p>WES-1 (Compound 8g), a carbonic anhydrase IX inhibitor (Ki: 55.9 μM), exhibits broad-spectrum antiproliferative activity against various cancer cell lines,</p>Formula:C20H20N4O3SPurity:98%Color and Shape:SolidMolecular weight:396.46(±)-γ-Tocopherol
CAS:<p>(±)-γ-Tocopherol is a form of vitamin E with antioxidant and anti-inflammatory properties.</p>Formula:C28H48O2Color and Shape:SolidMolecular weight:416.68Icomucret
CAS:<p>Icomucret can be used for the Treatment of Dry Eye.</p>Formula:C20H32O3Color and Shape:SolidMolecular weight:320.47CL 242817
CAS:<p>CL 242817 is an inhibitor of angiotensin converting enzyme (ACE).</p>Formula:C18H21NO5SColor and Shape:SolidMolecular weight:363.4311β-HSD1-IN-9
CAS:<p>11β-HSD1-IN-9 is a potent inhibitor of 11β-HSD1, displaying IC50 values of 0.48 µM for human and 1.3 µM for murine variants, respectively.</p>Formula:C13H9F3N2OColor and Shape:SolidMolecular weight:266.22Erythronic acid
CAS:<p>Erythronic acid, an endogenous carbohydrate metabolite, is instrumental for research into metabolism-associated disorders.</p>Formula:C4H8O5Purity:98%Color and Shape:SolidMolecular weight:136.1Methyl-3β-hydroxycholenate
CAS:<p>Methyl-3β-hydroxycholenate (Methyl 3beta-hydroxychol-5-enoate) is a modulator of RORγ.</p>Formula:C25H40O3Purity:98.78%Color and Shape:SolidMolecular weight:388.58FASN-IN-4
CAS:<p>FAS-IN-1 is a potent inhibitor of Fatty acid synthase (FAS) wtih IC50 of 10 nM.</p>Formula:C26H27N3O4SPurity:98%Color and Shape:SolidMolecular weight:477.58BMS-351
CAS:<p>BMS-351: potent, selective CYP17A1 inhibitor, promising for prostate cancer, minimal side effects.</p>Formula:C15H12F3N3Color and Shape:SolidMolecular weight:291.2717β-HSD10-IN-2
CAS:<p>17β-HSD10-IN-2 (compound 11), a benzothiazolylurea-based inhibitor, specifically targets 17β-hydroxysteroid dehydrogenase type 10 (17β-HSD10), avoiding</p>Formula:C15H10ClN3O4SPurity:98%Color and Shape:SolidMolecular weight:363.78Glucocerebrosidase-IN-1
CAS:<p>Glucocerebrosidase-IN-1 inhibits GCase with IC50 of 29.3 μM, Ki 18.5 μM, useful for Gaucher's and Parkinson's research.</p>Formula:C13H27NO3Color and Shape:SolidMolecular weight:245.36AMPD2 inhibitor 2
<p>AMPD2 inhibitor 2: strong h/mAMPD2 blocker, IC50s: 0.1/0.28μM. Potentially assesses AMPD2's role in high-fat diet mice.</p>Formula:C26H27F2N3O3Color and Shape:SolidMolecular weight:467.51ME-143
CAS:<p>ME-143, a 2nd-gen NADH oxidase inhibitor, blocks WNT/β-catenin pathway, active against various cancers in vitro/vivo.</p>Formula:C21H18O4Color and Shape:SolidMolecular weight:334.37SCD1 inhibitor-1
CAS:SCD1 inhibitor-1 is a potent and liver-selective inhibitor of stearoyl-CoA desaturase-1 (SCD1).Formula:C21H23N3NaO3S2Purity:98%Color and Shape:SolidMolecular weight:452.54MDPD
CAS:<p>MDPD boosts AtFAAH, the enzyme degrading NAEs in Arabidopsis, reducing NAE 12:0's growth inhibition.</p>Formula:C21H19N3O3Color and Shape:SolidMolecular weight:361.39hCAXII-IN-4
CAS:<p>hCAXII-IN-4 is a selective and potent CA XII inhibitor with a Ki value of 6.4 nM for human CA XII.</p>Formula:C22H27N5O6SColor and Shape:SolidMolecular weight:489.54Antiproliferative agent-10
<p>Antiproliferative agent-10: Ruthenium(II) complex that blocks cancer cell growth by halting mitochondrial calcium uptake.</p>Formula:C35H36Cl2N7PRuColor and Shape:SolidMolecular weight:757.66Niraparib metabolite M1
CAS:<p>Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1) is the carboxylic acid metabolite of niraparib.</p>Formula:C19H19N3O2Purity:99.65%Color and Shape:SolidMolecular weight:321.37MK-4409
CAS:<p>MK-4409, a potent and selective fatty acid amide hydrolase (FAAH) inhibitor, is being investigated for the treatment of inflammatory and neuropathic pain.</p>Formula:C22H17ClFN3O2SPurity:99.80% - 99.87%Color and Shape:SolidMolecular weight:441.91PDE9-IN-1
CAS:<p>PDE9-IN-1 is a selective and orally bioavailable Inhibitor of PDE9A(IC50 of 8.7 nM).</p>Formula:C17H23FN6O2Purity:99.86%Color and Shape:SolidMolecular weight:362.4IACS-8968
CAS:<p>IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).</p>Formula:C17H18F3N5O2Purity:98%Color and Shape:SolidMolecular weight:381.35Piritrexim
CAS:<p>Piritrexim (BW 301U) is an orally available fat-soluble dihydrofolate reductase inhibitor with pulmonary toxicity used in the study of uroepithelial carcinoma</p>Formula:C17H19N5O2Purity:98.50% - >99.99%Color and Shape:SolidMolecular weight:325.37K134
CAS:<p>K134 is an inhibitor of phosphodiesterase 3. The IC50s of K134 for PDE3A, PDE3B, PDE5, PDE2 and PDE4 are 0.1, 0.28, 12.1, >300 and >300 μM, respectively.</p>Formula:C22H29N3O4Purity:98%Color and Shape:SolidMolecular weight:399.48MitoPBN
CAS:<p>MitoPBN: mitochondria-targeted antioxidant, inhibits UCP1-3 at 250 nM, traps hydroxyl & carbon radicals, prevents lipid peroxidation.</p>Formula:C33H37BrNO2PColor and Shape:SolidMolecular weight:590.542AVE5688
CAS:<p>AVE5688 is an inhibitor of glycogen phosphorylase (GP, IC50s: 430 nM and 915 nM; Kds: 170 nM and 530 nM for rmGPb and rmGPa).</p>Formula:C16H8ClF5N2O5Purity:99.65%Color and Shape:SolidMolecular weight:438.69LY 113174
CAS:<p>LY 113174, a novel nonsteroidal aromatase inhibitor, may prove useful in the treatment of estrogen-dependent diseases.</p>Formula:C17H10Cl2N2Color and Shape:SolidMolecular weight:313.18FC11409B
CAS:<p>FC11409B is a CAIX inhibitor, inhibiting breast cancer invasion and metastasis.</p>Formula:C29H23BF4N2O3SColor and Shape:SolidMolecular weight:566.38SK-216
CAS:<p>SK-216,PAI-1 inhibitor. Reduces tumor angiogenesis. Inhibits VEGF-induced endothelial cell migration. Alleviates pulmonary fibrosis.</p>Formula:C29H29NNa2O6Purity:98.29%Color and Shape:SolidMolecular weight:533.52BI-L 357
CAS:<p>BI-L 357, a prodrug of BL-L 226, is a selective, orally active inhibitor of 5-lipoxygenase.</p>Formula:C18H18O4SColor and Shape:SolidMolecular weight:330.4CS-722 Free base
CAS:<p>CS-722 Free base: synthetic muscle relaxant; inhibits spinal reflex and sodium/calcium currents affecting synaptic activity.</p>Formula:C16H19ClN2O4Purity:99.52%Color and Shape:SolidMolecular weight:338.79PF-04279405
CAS:<p>PF-04279405 is a potent and selective glucokinase activator.</p>Formula:C25H25FN4O4Color and Shape:SolidMolecular weight:464.49Anti-hyperglycemic agent-1
CAS:<p>Anti-hyperglycemic agent 1 is a potent inhibitor of alpha-glucosidase (IC50: 0.53 μM). anti-Hyperglycemic agent 1 can be used to study diabetes.</p>Formula:C20H15BrN2O3Color and Shape:SolidMolecular weight:411.25Enpp-1-IN-17
CAS:<p>Enpp-1-IN-17 (example 274) is a potent inhibitor of ENPP1, exhibiting inhibition constants (Ki values) of 100 nM-1 μM for cGAMP hydrolysis and >1 μM for ATP</p>Formula:C18H24N4O2Color and Shape:SolidMolecular weight:328.41hCAI/II-IN-4
CAS:<p>hCAI/II-IN-4 inhibits hCA I & II (Ki: 16.95 & 15.22 nM), hCA IX (Ki: 27.04 nM), has anti-hypoxia benefits and is low-toxic for AMS research.</p>Formula:C15H15N3O5S2Color and Shape:SolidMolecular weight:381.43THPP-4
CAS:<p>THPP-4 inhibits phosphodiesterase 10A (PDE10A).</p>Formula:C20H21ClN6O2Color and Shape:SolidMolecular weight:412.87α-Glucosidase-IN-6
CAS:<p>α-Glucosidase-IN-6 is a competitive inhibitor of α-glucosidase (IC50: 5.69 μM) and exhibits potential for anti-diabetic studies.</p>Formula:C24H17ClF3NO3SColor and Shape:SolidMolecular weight:491.91SHP2-IN-5
CAS:<p>SHP2-IN-5 (compound 1) is a non-receptor protein tyrosine phosphatase inhibitor targeting SHP2 with an IC50 value of 97 nM, associated with regulating cell</p>Formula:C12H8O6Color and Shape:SolidMolecular weight:248.19Gallopamil hydrochloride
CAS:<p>Gallopamil hydrochloride (Methoxyverapamil hydrochloride) is an antagonist of phenylalkylamine calcium.</p>Formula:C28H41ClN2O5Purity:99.86%Color and Shape:SolidMolecular weight:521.09BMS270394
CAS:<p>BMS270394 is a RARγ agonist used in the study of breast cancer and skin diseases.</p>Formula:C23H26FNO4Color and Shape:SolidMolecular weight:399.46HFI-437
CAS:<p>HFI-437 is a potent, non-peptidic, insulin-regulated aminopeptidase (IRAP) inhibitor with a K i of 20 nM and functions as a cognitive enhancer [1].</p>Formula:C23H20N2O5Color and Shape:SolidMolecular weight:404.42BMS 961
CAS:<p>BMS961 is a potent and selective retinoic acid receptor gamma (RARγ) agonist (IC50: 30 nM).</p>Formula:C23H26FNO4Purity:98%Color and Shape:SolidMolecular weight:399.46Liarozole dihydrochloride
CAS:<p>Liarozole dihydrochloride, an oral CYP450 inhibitor, blocks estrogen and androgens, targeting prostate cancer and skin disorders.</p>Formula:C17H15Cl3N4Purity:98%Color and Shape:SolidMolecular weight:381.69Cycloguanil
CAS:<p>Cycloguanil is an antimalarial.</p>Formula:C11H14ClN5Purity:98%Color and Shape:SolidMolecular weight:251.72AHR-5333
CAS:<p>AHR-5333 an antiallergy agent.</p>Formula:C30H33F2NO4Purity:98%Color and Shape:SolidMolecular weight:509.58FABP4/5-IN-5
CAS:<p>FABP4/5-IN-5 (compound D9) serves as a potent inhibitor of both FABP 4 and FABP 5, demonstrating IC50 values of 4.68 μM and 10.72 μM, respectively. It is notably effective in addressing metabolic disorders such as diabetes mellitus [1].</p>Formula:C23H14ClF2NO4SColor and Shape:SolidMolecular weight:473.88L-693612 HCl
CAS:<p>L-693612 HCl is an inhibitor of carbonic anhydrase.</p>Formula:C14H25ClN2O5S3Purity:98%Color and Shape:SolidMolecular weight:433.01RO6806051
CAS:<p>RO6806051 (compound 12) is a potent dual inhibitor of fatty acid binding proteins 4 and 5 (FABP4 and FABP5), exhibiting excellent selectivity and absorption, distribution, metabolism, and excretion (eADME) properties.</p>Formula:C21H19ClN6Color and Shape:SolidMolecular weight:390.87Methazolamide-d6
CAS:<p>Methazolamide-d6 is a GC/LC-MS standard for measuring methazolamide, a glaucoma drug that lowers eye pressure and fluid, reduces seizures, and combats ROS.</p>Formula:C5H2D6N4O3S2Color and Shape:SolidMolecular weight:242.31BMS-593214
CAS:<p>BMS-593214 is an inhibitor of active site-directed factor VIIa and a non-competitive inhibitor of the VIIa-activated substrate FX.</p>Formula:C31H27N3O4Purity:96.63% - 98.04%Color and Shape:SolidMolecular weight:505.56Quinapril-d5
CAS:<p>Quinapril-d5: An internal standard for quinapril quantification via GC/LC-MS; a prodrug ACE inhibitor for hypertension and heart failure.</p>Formula:C25H25D5N2O5Color and Shape:SolidMolecular weight:443.55Riboflavine phosphate
CAS:<p>Riboflavine phosphate (Flavin mononucleotide) is a derivative of Riboflavin.</p>Formula:C17H21N4O9PPurity:98%Color and Shape:SolidMolecular weight:456.34GNF362
CAS:<p>GNF362 is an ITPKB inhibitor that inhibits Itpka and Itpkc and reverses the migratory stimulatory effect of ITPKA overexpression.</p>Formula:C22H21F3N6Purity:99.63%Color and Shape:SolidMolecular weight:426.44Cefetrizole
CAS:<p>Ceftezole is an α-Glucosidase inhibitor (IC50: 2.1 μM; Ki: 0.578 μM).</p>Formula:C16H15N5O4S3Purity:98%Color and Shape:SolidMolecular weight:437.52Dopropidil
CAS:<p>Dopropidil: anti-angina calcium regulator with anti-ischemic properties in animal models.</p>Formula:C20H35NO2Purity:98%Color and Shape:SolidMolecular weight:321.5SA57
CAS:<p>SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).</p>Formula:C17H23ClN2O3Purity:98%Color and Shape:SolidMolecular weight:338.83FSG67
CAS:<p>FSG67 is an inhibitor of glycerol 3-phosphate acyltransferase (IC 50 =24 μM) [1].</p>Formula:C16H25NO4SPurity:99.76%Color and Shape:SolidMolecular weight:327.44Factor VII-IN-1
CAS:<p>Factor VII-IN-1 (example 43) is an effective Factor VII (FVII) inhibitor (IC50=1.1 μM) with anticoagulant properties.</p>Formula:C15H10BrNO3Purity:99.19%Color and Shape:SolidMolecular weight:332.15α-2,3-sialyltransferase-IN-1
CAS:<p>α-2,3-sialyltransferase-IN-1 is a noncompetitive inhibitor of α-2,3-sialyltransferase(IC50 of 6 μM).</p>Formula:C28H45NO6Purity:98% - 98%Color and Shape:SolidMolecular weight:491.66Gemlapodect
CAS:<p>Gemlapodect (RO554965), a phosphodiesterase 10A (PDE10A) inhibitor, is utilized in schizophrenia research.</p>Formula:C22H21N7O3Color and Shape:SolidMolecular weight:431.45CD 1530
CAS:<p>CD 1530 is an ARγ agonist (Kd:150 nM) with potential anticancer activity for the study of oral carcinogenesis.</p>Formula:C27H26O3Purity:98.13%Color and Shape:SolidMolecular weight:398.49JMS-053
CAS:<p>JMS-053 is a phosphatase DUSP3 inhibitor that inhibits CDC25B and prevents VEGF from disrupting the microvascular endothelial barrier.</p>Formula:C13H8N2O2SPurity:≥98.0%Color and Shape:SolidMolecular weight:256.28Aminopeptidase-IN-1
CAS:<p>Aminopeptidase-IN-1: potent IRAP blocker, Ki 7.7 μM, useful for cognitive/memory disorder research.</p>Formula:C18H16N2O6Purity:98.37%Color and Shape:SolidMolecular weight:356.33Albaconazole
CAS:<p>Albaconazole, a small fungal CYP51A1 inhibitor, treats fungal infections and some musculoskeletal disorders.</p>Formula:C20H16ClF2N5O2Purity:99.27%Color and Shape:SolidMolecular weight:431.82DHODH-IN-17
CAS:<p>DHODH-IN-17 is a human DHODH inhibitor with an IC50 of 0.40 μM.</p>Formula:C12H9ClN2O2Purity:99.41% - 99.52%Color and Shape:SolidMolecular weight:248.67GSK376501A
CAS:<p>GSK376501A is a selective and effective modulator of peroxisome proliferator-activated receptor γ (PPARγ) for the study of type 2 diabetes.</p>Formula:C32H37NO6Purity:>99.99%Color and Shape:SolidMolecular weight:531.64Hexazinone
CAS:<p>Hexazinone: a triazine herbicide blocks photosynthesis by binding to D-1 protein in photosystem II.</p>Formula:C12H20N4O2Purity:99.99%Color and Shape:SolidMolecular weight:252.31TK-642
CAS:<p>TK-642 is a potent and selective SHP2 inhibitor with oral activity, based on pyrazole and pyrazine structures (IC50 = 2.7 nmol/L). It effectively inhibits the proliferation of esophageal carcinoma cells and induces apoptosis, making it useful for studying esophageal cancer.</p>Formula:C17H20ClN7SColor and Shape:SolidMolecular weight:389.91BKIDC-1553
CAS:<p>BKIDC-1553, an orally active antiglycolytic agent and bumped kinase inhibitor-derived compound, has a predicted half-life of approximately 17 hours in humans. It inhibits CYP2C8 and Angiotensin Converting Enzyme, making it suitable for cancer research [1].</p>Formula:C22H23N5O2Color and Shape:SolidMolecular weight:389.45Senazodan
CAS:<p>Senazodan is a sensitiser of Ca2+, and shows inhibition effect on PDE III.</p>Formula:C15H14N4OPurity:98%Color and Shape:SolidMolecular weight:266.3Phosphodiesterase-IN-1
CAS:<p>Phosphodiesterase-IN-1 (Compound 7), a phosphodiesterase (PDE) inhibitor, exhibits anti-Plasmodium and antiproliferative activities. It effectively inhibits P. falciparum (strain 3D7) with an IC 50 value of 0.64 μM [1].</p>Formula:C15H15FN4OColor and Shape:SolidMolecular weight:286.3KD-027
CAS:<p>KD-027 is a novel and long-acting PDE5A(phosphodiesterase 5A) inhibitor with potential antihypertensive activity.</p>Formula:C25H35N7O6SPurity:99.55%Color and Shape:SolidMolecular weight:561.65RO-28-1675
CAS:<p>RO-28-1675 is a direct and selective glucokinase activator, the GK/GKRP complex,insulin secretion and type 2 diabetes.</p>Formula:C18H22N2O3S2Purity:98.13%Color and Shape:SolidMolecular weight:378.51AGI-026
CAS:<p>AGI-026 (AGI-12026) is a novel and potent dual inhibitor of the mutant isocitrate dehydrogenase mIDH1/2 blood-brain barrier, reduce d-2-hydroxyglutarate (2-HG).</p>Formula:C18H15F6N7Purity:99.79% - 99.86%Color and Shape:SolidMolecular weight:443.352-TEDC
CAS:<p>2-TEDC: Potent LOX inhibitor, blocks 5-LOX, 12-LOX, 15-LOX (IC50: 0.09, 0.013, 0.5 μM); aids atherosclerosis research.</p>Formula:C16H13NO4SPurity:99.75%Color and Shape:SolidMolecular weight:315.34DA 3003-2
CAS:<p>DA 3003-2: Potent Cdc25 inhibitor, halts cell division, may aid prostate cancer research.</p>Formula:C15H16ClN3O3Color and Shape:SolidMolecular weight:321.76Asterriquinol D dimethyl ether
CAS:<p>Asterriquinol D dimethyl ether inhibits mouse myeloma (IC50: 28 μg/mL) and Tritrichomonas foetus.</p>Formula:C26H24N2O4Color and Shape:SolidMolecular weight:428.48OMDM-4
CAS:<p>OMDM-4 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 17.7 μM).</p>Formula:C29H43NO3Purity:98%Color and Shape:SolidMolecular weight:453.66Lovastatin hydroxy acid sodium
CAS:<p>Lovastatin Sodium is an HMG-CoA reductase inhibitor.</p>Formula:C24H38NaO6Color and Shape:SolidMolecular weight:445.5412(S)-HpETE
CAS:<p>12(S)-HpETE activates human blood leukocyte 5-LOE and mediates induction of c-fos and c-jun, activation of AP-1, and endothelium-dependent vasoconstriction.</p>Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47LTV-1
CAS:<p>LTV-1 has the potential for autoimmunity treatment. LTV-1 is a potent lymphoid tyrosine phosphatase (LYP) inhibitor in T cells with an IC50 of 508 nM.</p>Formula:C26H20N2O5SColor and Shape:SolidMolecular weight:472.51Entacapone sodium salt
CAS:<p>Entacapone sodium salt, a potent peripheral COMT inhibitor (IC50=151 nM), hinders α-syn/β-amyloid aggregation and protects PC12 cells.</p>Formula:C14H15N3NaO5Purity:98%Color and Shape:SolidMolecular weight:328.28GGsTop
CAS:<p>GGsTop (Nahlsgen) is a GGT inhibitor with anti-aging activity.</p>Formula:C13H18NO7PPurity:98.96%Color and Shape:SolidMolecular weight:331.26IDO-IN-11
CAS:<p>IDO-IN-11 is an indoleamine-2,3-dioxygenase (IDO) inhibitor with IC50s of 0.18 μM (Kinase) and 0.014 μM (Hela Cell).</p>Formula:C19H23BrFN7O4SPurity:98%Color and Shape:SolidMolecular weight:544.4Fadrozole HCl hydrate
CAS:<p>Fadrozole is a selective inhibitor of aromatase. It also effective in the treatment of estrogen-dependent diseases including breast cancer.</p>Formula:C14H13N3ClHH2OPurity:98%Color and Shape:SolidMolecular weight:268.74PSB069
CAS:<p>NTPDase inhibitor</p>Formula:C20H13ClN2NaO5SPurity:98%Color and Shape:SolidMolecular weight:451.84FCE 28654
CAS:<p>FCE 28654 is a water-soluble acyl-CoA inhibitor.</p>Formula:C25H35N2O7PColor and Shape:SolidMolecular weight:506.53Glycogen phosphorylase-IN-1
CAS:<p>Glycogen phosphorylase-IN-1 is an hlGPa inhibitor that can be used in the study of type 2 diabetes and canine lupus.</p>Formula:C17H15ClF2N4O4Purity:97.98% - 98.15%Color and Shape:SolidMolecular weight:412.78IDO1-IN-18
CAS:<p>IDO1-IN-18 (Compound 14) is a potent inhibitor of IDO1. IDO1-IN-18 has potential for cancer disease research.</p>Formula:C23H18F4N2O3Color and Shape:SolidMolecular weight:446.39TM6008
CAS:<p>TM6008 is an inhibitor of prolyl hydroxylase that protects against cell death after hypoxia.</p>Formula:C21H17N5O3Purity:98%Color and Shape:SolidMolecular weight:387.39SCH 42495
CAS:<p>SCH 42495 is an orally active neutral metalloendopeptidase inhibitor. SCH 42495 is the orally active ethyl ester prodrug of SCH 42354.</p>Formula:C20H29NO4S2Purity:98%Color and Shape:SolidMolecular weight:411.58hCAXII-IN-3
CAS:<p>hCAXII-IN-3 (Compound 6o) is a selective inhibitor of human carbonic anhydrase XII (hCAXII) (Ki: 10.0 nM).</p>Formula:C26H20BrN5O3SColor and Shape:SolidMolecular weight:562.44Pimobendan hydrochloride
CAS:<p>Pimobendan hydrochloride is a selective inhibitor of PDE3 (IC50: 0.32 μM).</p>Formula:C19H19ClN4O2Purity:98%Color and Shape:SolidMolecular weight:370.83hDHODH-IN-9
CAS:<p>hDHODH-IN-9 is a potent hDHODH inhibitor, IC50=0.34 μM, toxic to MCF-7/A375 cells, promising for cancer research.</p>Formula:C21H21NO4Color and Shape:SolidMolecular weight:351.4Nampt-IN-9
CAS:<p>Nampt-IN-9 (Compound 8) is a potent inhibitor of NAMPT with anticancer properties.Nampt-IN-9 can be used to study ductal adenocarcinoma of the pancreas.</p>Formula:C26H33N3O4Color and Shape:SolidMolecular weight:451.56SQ 27786
CAS:<p>SQ 27786 is an inhibitor of ACE.</p>Formula:C23H25ClN4O7S2Purity:98%Color and Shape:SolidMolecular weight:569.05
