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PDGFR
Regorafenib
CAS:755037-03-7
Formula:
C21H15ClF4N4O3
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
482.82
Estimated delivery in United States, on Tuesday 25 Jan 2022
Imatinib
Formula:
C29H31N7O
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
493.62
Estimated delivery in United States, on Tuesday 25 Jan 2022
TCS 359
CAS:301305-73-7
Formula:
C18H20N2O4S
Purity:
>98.0%(HPLC)
Color and Shape:
Light yellow to Brown powder to crystal
Molecular weight:
360.43
Estimated delivery in United States, on Tuesday 25 Jan 2022
GW 2580
CAS:870483-87-7
Formula:
C20H22N4O3
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
366.42
Estimated delivery in United States, on Tuesday 25 Jan 2022
GNF5837
CAS:1033769-28-6
GNF-5837 is a specific, and orally bioavailable pan-TRK inhibitor for TrkA/TrkB (IC50: 8/12 nM).
Formula:
C28H21F4N5O2
Purity:
99.29%
Color and Shape:
solid
Molecular weight:
535.49
Estimated delivery in United States, on Thursday 3 Feb 2022
Pazopanib
CAS:444731-52-6
Pazopanib, a small molecule inhibitor, inhibits multiple protein tyrosine kinases with potential antineoplastic activity. Pazopanib …
Formula:
C21H23N7O2S
Purity:
99.84%
Color and Shape:
solid
Molecular weight:
437.52
Estimated delivery in United States, on Thursday 3 Feb 2022
Vatalanib 2HCl
CAS:212141-51-0
Vatalanib (PTK787) (IC50=37 nM) is an inhibitor of VEGFR2/KDR. It exhibits less effective against VEGFR1/Flt-1 …
Formula:
C20H15ClN4·2HCl
Purity:
99.78%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
419.73
Estimated delivery in United States, on Thursday 3 Feb 2022
Tivozanib
CAS:475108-18-0
Tivozanib is an orally bioavailable inhibitor of vascular endothelial growth factor receptors (VEGFRs) 1, 2 …
Formula:
C22H19ClN4O5
Purity:
97.41%
Color and Shape:
solid
Molecular weight:
454.86
Estimated delivery in United States, on Thursday 3 Feb 2022
Bisindolylmaleimide I
CAS:133052-90-1
GF109203X is a potent and highly selective protein kinase C (PKC) inhibitor with a Ki …
Formula:
C25H24N4O2
Purity:
99.08%
Color and Shape:
Orange Solid
Molecular weight:
412.48
Estimated delivery in United States, on Thursday 3 Feb 2022
Cediranib
CAS:288383-20-0
Cediranib (AZD2171) is a highly potent (IC50 < 1 nmol/L) ATP-competitive inhibitor of recombinant KDR tyrosine …
Formula:
C25H27FN4O3
Purity:
97.21%
Color and Shape:
solid
Molecular weight:
450.51
Estimated delivery in United States, on Thursday 3 Feb 2022
JI101
CAS:900573-88-8
JI-101 is an oral multi-kinase inhibitor that targets vascular endothelial growth factor receptor type 2 …
Formula:
C22H20BrN5O2
Purity:
99.41%
Color and Shape:
solid
Molecular weight:
466.34
Estimated delivery in United States, on Thursday 3 Feb 2022
PP58
CAS:212391-58-7
PP58 is an inhibit of PDGFR, FGFR and Src family.
Formula:
C22H19Cl2N5O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
456.32
Estimated delivery in United States, on Thursday 3 Feb 2022
AG 1295
CAS:71897-07-9
AG 1295 is a selective platelet-derived growth factor receptor (PDGFR) tyrosine-kinase inhibitor. AG1295 abolishes autophosphorylation …
Formula:
C16H14N2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
234.3
Estimated delivery in United States, on Thursday 3 Feb 2022
Seralutinib
CAS:1619931-27-9
Seralutinib is an inhibitor of inhaled PDGFR and PDGFR. It is used in the study …
Formula:
C27H27N5O3
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
469.55
Estimated delivery in United States, on Thursday 3 Feb 2022
Crenolanib
CAS:670220-88-9
Crenolanib is an orally bioavailable type III tyrosine kinases inhibitor of PDGFR/ and FLT3 (IC50s: …
Formula:
C26H29N5O2
Purity:
99.28%
Color and Shape:
solid
Molecular weight:
443.54
Estimated delivery in United States, on Thursday 3 Feb 2022
N-(p-Coumaroyl) serotonin
CAS:68573-24-0
N-(p-Coumaroyl) Serotonin is a polyphenol isolated from the seeds of safflower. N-(p-Coumaroyl) serotonin has antioxidant, …
Formula:
C19H18N2O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
322.4
Estimated delivery in United States, on Thursday 3 Feb 2022
Flumatinib mesylate
CAS:895519-91-2
Flumatinib mesylate is a selective inhibitor of c-Abl, PDGFR and c-Kit, effectively overcomes drug resistance …
Formula:
C30H33F3N8O4S
Purity:
99.82%
Color and Shape:
solid
Molecular weight:
658.69
Estimated delivery in United States, on Thursday 3 Feb 2022
Axitinib
CAS:319460-85-0
Axitinib is an orally bioavailable tyrosine kinase inhibitor with IC50s of 0.1, 0.2, 0.1-0.3, 1.7, …
Formula:
C22H18N4OS
Purity:
99.65%
Color and Shape:
Off-White Solid
Molecular weight:
386.47
Estimated delivery in United States, on Thursday 3 Feb 2022
Imatinib
CAS:152459-95-5
matinib is an inhibitor of the receptor tyrosine kinases c-Abl, Bcr-Abl, PDGFR, and c-Kit (IC50: …
Formula:
C29H31N7O
Purity:
99.94%
Color and Shape:
Off White Powder
Molecular weight:
493.6
Estimated delivery in United States, on Thursday 3 Feb 2022
AC710 Mesylate
CAS:1351522-05-8
AC710 Mesylate is a potent PDGFR inhibitor (Kds: 0.6, 1.57, 1, 1.3, 1.0 nM for …
Formula:
C32H46N6O7S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
658.81
Estimated delivery in United States, on Thursday 3 Feb 2022
PDGFR kinase inhibitor 1
CAS:2209053-93-8
PDGFR kinase inhibitor 1 is a highly selective inhibitor of type II PDGFR kinase (PDGFR …
Formula:
C34H34N8O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
586.69
Estimated delivery in United States, on Thursday 3 Feb 2022
Sennoside B
CAS:128-57-4
Sennoside B is an anthranoid. Anthranoid derivatives are used all over the world as a …
Formula:
C42H38O20
Color and Shape:
Light Yellow Crystal
Molecular weight:
862.74
Estimated delivery in United States, on Thursday 3 Feb 2022
Toceranib
CAS:356068-94-5
Toceranib phosphate is an orally active inhibitor of tyrosine kinase (RTK) receptor, and it potently …
Formula:
C22H25FN4O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
396.46
Estimated delivery in United States, on Thursday 3 Feb 2022
Sunitinib Malate
CAS:341031-54-7
Sunitinib is an indolinone-based tyrosine kinase inhibitor. It blocks the tyrosine kinase activities of VEGFR2, …
Formula:
C26H33FN4O7
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
532.56
Estimated delivery in United States, on Thursday 3 Feb 2022
JNJ-10198409
CAS:627518-40-5
JNJ-10198409 is a relatively selective and ATP competitive PDGF-RTK inhibitor (IC50=2 nM). JNJ-10198409 has good …
Formula:
C18H16FN3O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
325.34
Estimated delivery in United States, on Thursday 3 Feb 2022
NSC 86429
CAS:5812-07-7
SU-4312, also known as DMBI, is a potent and selective inhibitor of VEGFR and PDGFR …
Formula:
C17H16N2O
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
264.33
Estimated delivery in United States, on Thursday 3 Feb 2022
Imatinib Mesylate
CAS:220127-57-1
Imatinib mesylate is a tyrosine kinase receptor inhibitor with antineoplastic activity (IC50s: 0.6 μM, 0.1 …
Formula:
C29H31N7O·CH4SO3
Purity:
100.00%
Color and Shape:
White Crystalline Powder
Molecular weight:
589.71
Estimated delivery in United States, on Thursday 3 Feb 2022
Ripretinib
CAS:1442472-39-0
Ripretinib is an orally bioavailable inhibitor of KIT and PDGFRA.
Formula:
C24H21BrFN5O2
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
510.36
Estimated delivery in United States, on Thursday 3 Feb 2022
GZD856
CAS:1257628-64-0
GZD856 is an orally bioavailable PDGFR/ inhibitor (IC50s: 68.6 and 136.6 nM) with anti-lung cancer …
Formula:
C29H27F3N6O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
532.56
Estimated delivery in United States, on Thursday 3 Feb 2022
SU16f
CAS:251356-45-3
SU16f is a potent and selective PDGFR inhibitor (IC50s: 10 nM, 140 nM, 2.29 μM …
Formula:
C24H22N2O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
386.44
Estimated delivery in United States, on Thursday 3 Feb 2022
Avapritinib
CAS:1703793-34-3
Avapritinib is a dual inhibitor of the mutant KIT receptor (KIT D816V, IC50: 0.27 nM) …
Formula:
C26H27FN10
Purity:
96.59%
Color and Shape:
Solid
Molecular weight:
498.56
Estimated delivery in United States, on Thursday 3 Feb 2022
CP673451
CAS:343787-29-1
CP-673451 is a specific inhibitor of PDGFR/ (IC50: 10/1 nM) with antiangiogenic and antitumor activity …
Formula:
C24H27N5O2
Purity:
99.88%
Color and Shape:
solid
Molecular weight:
417.5
Estimated delivery in United States, on Thursday 3 Feb 2022
Telatinib
CAS:332012-40-5
Telatinib is an effective inhibitor of VEGFR2/3, c-Kit, and PDGFR. The IC50s of Telatinib forVEGFR2/3, …
Formula:
C20H16ClN5O3
Purity:
99.81%
Color and Shape:
solid
Molecular weight:
409.83
Estimated delivery in United States, on Thursday 3 Feb 2022
Tyrphostin 9
CAS:10537-47-0
Tyrphostin 9 is an Agricultural acaricide, now superseded. Tyrphostin 9 is firstly designed as an …
Formula:
C18H22N2O
Purity:
98.21%
Color and Shape:
Solid Yellow
Molecular weight:
282.38
Estimated delivery in United States, on Thursday 3 Feb 2022
CEP32496
CAS:1188910-76-0
CEP-32496 is a highly potent inhibitor of BRAF.
Formula:
C24H22F3N5O5
Purity:
95.78%
Color and Shape:
solid
Molecular weight:
517.46
Estimated delivery in United States, on Thursday 3 Feb 2022
Tyrphostin AG1433
CAS:168835-90-3
Tyrphostin AG1433 (SU1433) is an inhibitor of tyrosine kinases, and also a selective PDGFR and …
Formula:
C16H14N2O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
266.29
Estimated delivery in United States, on Thursday 3 Feb 2022
Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))
Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 …
Formula:
C18H18ClN5O3S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
419.88
Estimated delivery in United States, on Thursday 3 Feb 2022
AC710
CAS:1351522-04-7
AC710 is a potent PDGFR inhibitor (Kds: 0.6, 1, 1.57, 1.3, 1 nM for FLT3, …
Formula:
C31H42N6O4
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
562.7
Estimated delivery in United States, on Thursday 3 Feb 2022
Imatinib Mesylate
Formula:
C29H31N7O·CH4O3S
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
589.72
Estimated delivery in United States, on Monday 7 Feb 2022
AG-1296
CAS:146535-11-7
Formula:
C16H14N2O2
Purity:
>98.0%(GC)
Color and Shape:
White to Orange to Green powder to crystal
Molecular weight:
266.30
Estimated delivery in United States, on Monday 7 Feb 2022
Tyrphostin RG 13022
CAS:136831-48-6
Formula:
C16H14N2O2
Purity:
>98.0%(GC)
Color and Shape:
White to Yellow to Green powder to crystal
Molecular weight:
266.30
Estimated delivery in United States, on Monday 7 Feb 2022
Tyrphostin A9
CAS:10537-47-0
Formula:
C18H22N2O
Purity:
>98.0%(GC)
Color and Shape:
Light orange to Yellow to Green powder to crystal
Molecular weight:
282.39
Estimated delivery in United States, on Monday 7 Feb 2022
