GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,058 products)
- Adenosine Receptor(216 products)
- Adrenergic Receptor(3,265 products)
- Bombesin Receptor(37 products)
- Bradykinin Receptor(63 products)
- CXCR(179 products)
- CaSR(31 products)
- Cannabinoid Receptor(226 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(449 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(89 products)
- GPCR19(40 products)
- GRK(43 products)
- GTPase(26 products)
- Glucagon Receptor(210 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(389 products)
- LPA Receptor(22 products)
- Melatonin Receptor(26 products)
- OX Receptor(57 products)
- Opioid Receptor(337 products)
- PAFR(12 products)
- PKA(57 products)
- S1P Receptor(22 products)
- SGLT(33 products)
- Sigma receptor(49 products)
Show 19 more subcategories
Found 6062 products for "GPCR/G-Protein".
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Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Formula:C19H29ClN2O4Purity:99.49%Color and Shape:SolidMolecular weight:384.9Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Formula:C22H23N3O2Purity:99.29% - 99.97%Color and Shape:White SolidMolecular weight:361.44(3aR,9aR)-Fluparoxan
CAS:(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H10FNO2Purity:97.82%Color and Shape:SolidMolecular weight:195.19AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Formula:C17H14O5Purity:97.07%Color and Shape:SolidMolecular weight:298.29Ref: TM-T14148
1mg34.00€5mg63.00€1mL*10mM (DMSO)67.00€10mg92.00€25mg165.00€50mg250.00€100mg401.00€200mg580.00€Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formula:C23H27Cl2N3O2Purity:99.43% - 99.62%Color and Shape:White SolidMolecular weight:448.39Upidosin
CAS:Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.Formula:C31H33N3O4Purity:99.66%Color and Shape:SolidMolecular weight:511.61Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formula:C22H22FN3O3Purity:99.19% - 99.73%Color and Shape:SolidMolecular weight:395.4268Chlorprothixene hydrochloride
CAS:Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formula:C18H18ClNS·HClPurity:99.76% - 99.97%Color and Shape:White SolidMolecular weight:352.32Amiselimod hydrochloride
CAS:Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.Formula:C19H31ClF3NO3Purity:99.55%Color and Shape:SolidMolecular weight:413.9Ref: TM-T10305
1mg35.00€2mg50.00€5mg75.00€1mL*10mM (DMSO)84.00€10mg114.00€25mg203.00€50mg334.00€100mg485.00€200mg700.00€Alverine citrate
CAS:Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.Formula:C26H35NO7Purity:98.53% - 99.43%Color and Shape:SolidMolecular weight:473.57Venlafaxine hydrochloride
CAS:Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Formula:C17H28ClNO2Purity:97.32% - 99.86%Color and Shape:SolidMolecular weight:313.86Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Formula:C22H29N3O4SPurity:99.96%Color and Shape:Yellowish White Crystalline PowderMolecular weight:431.548Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Formula:C22H21Cl3N4OPurity:98% - 99.91%Color and Shape:White SolidMolecular weight:463.79Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFormula:C19H25F3N2O6Purity:99.92% - 99.94%Color and Shape:White SolidMolecular weight:434.41Ref: TM-T1077
1mL*10mM (DMSO)35.00€10mg49.00€25mg65.00€50mg80.00€100mg109.00€200mg161.00€500mg263.00€Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Formula:C19H21N3OPurity:99.44% - 99.84%Color and Shape:SolidMolecular weight:307.39Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formula:C21H24ClNOPurity:99.77% - 99.99%Color and Shape:White SolidMolecular weight:341.88KGA-2727
CAS:KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.Formula:C26H40N4O8Purity:98.46%Color and Shape:SolidMolecular weight:536.62Ref: TM-T15656
1mg109.00€2mg158.00€5mg260.00€1mL*10mM (DMSO)305.00€10mg430.00€25mg710.00€50mg973.00€100mg1,333.00€Zolmitriptan
CAS:Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Formula:C16H21N3O2Purity:99.69% - 99.91%Color and Shape:White SolidMolecular weight:287.36Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H11ClFNO2Purity:99.98%Color and Shape:SolidMolecular weight:231.65Pizotifen
CAS:Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.Formula:C19H21NSPurity:99.93%Color and Shape:White SolidMolecular weight:295.44
