GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,037 products)
- Adenosine Receptor(214 products)
- Adrenergic Receptor(3,159 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(63 products)
- CXCR(165 products)
- CaSR(31 products)
- Cannabinoid Receptor(223 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(447 products)
- Endothelin Receptor(85 products)
- GNRH Receptor(88 products)
- GPCR19(38 products)
- GRK(40 products)
- GTPase(24 products)
- Glucagon Receptor(204 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(390 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(54 products)
- Opioid Receptor(334 products)
- PAFR(12 products)
- PKA(57 products)
- S1P Receptor(18 products)
- SGLT(32 products)
- Sigma receptor(48 products)
Show 19 more subcategories
Found 5940 products for "GPCR/G-Protein".
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Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Formula:C22H23N3O2Purity:99.29% - 99.97%Color and Shape:White SolidMolecular weight:361.44Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formula:C23H27Cl2N3O2Purity:99.43% - 99.62%Color and Shape:White SolidMolecular weight:448.39Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Formula:C19H29ClN2O4Purity:99.49%Color and Shape:SolidMolecular weight:384.9Olinciguat
CAS:Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.Formula:C21H16F5N7O3Purity:99.33% - 99.71%Color and Shape:SolidMolecular weight:509.39Ref: TM-T16383
1mg170.00€5mg430.00€1mL*10mM (DMSO)475.00€10mg620.00€25mg973.00€50mg1,333.00€100mg1,765.00€YNT-185
CAS:YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,Formula:C33H37N5O5SPurity:99.67%Color and Shape:SolidMolecular weight:615.74Urocortin (rat) acetate
Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.Purity:97.76%Color and Shape:White Solid2-Bromo-6-methoxynaphthalene
CAS:2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.Formula:C11H9BrOPurity:98.51%Color and Shape:SolidMolecular weight:237.09Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formula:C22H22FN3O3Purity:99.19% - 99.73%Color and Shape:SolidMolecular weight:395.43CP-809101 hydrochloride
CAS:CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formula:C15H18Cl2N4OPurity:99.5%Color and Shape:Yellow SolidMolecular weight:341.24Amiselimod hydrochloride
CAS:Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.Formula:C19H31ClF3NO3Purity:99.55%Color and Shape:SolidMolecular weight:413.9Ref: TM-T10305
1mg35.00€2mg50.00€5mg75.00€1mL*10mM (DMSO)84.00€10mg114.00€25mg203.00€50mg334.00€100mg485.00€200mg700.00€Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Formula:C19H26ClNO2Purity:99.35%Color and Shape:White SolidMolecular weight:335.87Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Formula:C22H29N3O4SPurity:99.96%Color and Shape:Yellowish White Crystalline PowderMolecular weight:431.55Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Formula:C19H21N3OPurity:99.44% - 99.84%Color and Shape:SolidMolecular weight:307.39Upidosin
CAS:Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.Formula:C31H33N3O4Purity:99.66%Color and Shape:SolidMolecular weight:511.61Venlafaxine hydrochloride
CAS:Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Formula:C17H28ClNO2Purity:97.32% - 99.86%Color and Shape:SolidMolecular weight:313.86AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Formula:C17H14O5Purity:97.59%Color and Shape:SolidMolecular weight:298.29Ref: TM-T14148
1mg34.00€5mg63.00€1mL*10mM (DMSO)67.00€10mg92.00€25mg165.00€50mg250.00€100mg401.00€200mg580.00€Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H11ClFNO2Purity:99.98%Color and Shape:SolidMolecular weight:231.65Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Formula:C25H32F3N3O4Purity:99.28% - 99.76%Color and Shape:White SolidMolecular weight:495.53Ref: TM-T1504
1500mgTo inquire5mg34.00€1mL*10mM (DMSO)35.00€10mg50.00€25mg73.00€50mg92.00€100mg99.00€200mg126.00€Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Formula:C15H23N3O4SPurity:98.20% - 99.88%Color and Shape:White SolidMolecular weight:341.43CYM 50769
CAS:CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).Formula:C24H17ClN2O3Purity:98% - 99.08%Color and Shape:SolidMolecular weight:416.86
