GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,037 products)
- Adenosine Receptor(214 products)
- Adrenergic Receptor(3,159 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(63 products)
- CXCR(165 products)
- CaSR(31 products)
- Cannabinoid Receptor(223 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(447 products)
- Endothelin Receptor(85 products)
- GNRH Receptor(88 products)
- GPCR19(38 products)
- GRK(40 products)
- GTPase(24 products)
- Glucagon Receptor(204 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(390 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(54 products)
- Opioid Receptor(334 products)
- PAFR(12 products)
- PKA(57 products)
- S1P Receptor(18 products)
- SGLT(32 products)
- Sigma receptor(48 products)
Show 19 more subcategories
Found 5940 products for "GPCR/G-Protein".
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Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H11ClFNO2Purity:99.98%Color and Shape:SolidMolecular weight:231.65Alverine citrate
CAS:Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.Formula:C26H35NO7Purity:98.53% - 99.43%Color and Shape:SolidMolecular weight:473.57Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Formula:C22H23N3O2Purity:99.29% - 99.97%Color and Shape:White SolidMolecular weight:361.44CYM 50769
CAS:CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).Formula:C24H17ClN2O3Purity:98% - 99.08%Color and Shape:SolidMolecular weight:416.86Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formula:C23H27Cl2N3O2Purity:99.43% - 99.62%Color and Shape:White SolidMolecular weight:448.39(3aR,9aR)-Fluparoxan
CAS:(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H10FNO2Purity:97.82%Color and Shape:SolidMolecular weight:195.19AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Formula:C17H14O5Purity:97.59%Color and Shape:SolidMolecular weight:298.29Ref: TM-T14148
1mg34.00€5mg63.00€1mL*10mM (DMSO)67.00€10mg92.00€25mg165.00€50mg250.00€100mg401.00€200mg580.00€KGA-2727
CAS:KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.Formula:C26H40N4O8Purity:98.46%Color and Shape:SolidMolecular weight:536.62Ref: TM-T15656
1mg109.00€2mg158.00€5mg260.00€1mL*10mM (DMSO)305.00€10mg430.00€25mg710.00€50mg973.00€100mg1,333.00€Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Formula:C19H26ClNO2Purity:99.35%Color and Shape:White SolidMolecular weight:335.87PF429242 dihydrochloride
CAS:PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).Formula:C25H37Cl2N3O2Purity:99.68%Color and Shape:White ViscousMolecular weight:482.49Prucalopride
CAS:Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.Formula:C18H26ClN3O3Purity:99.99% - >99.99%Color and Shape:White SolidMolecular weight:367.87Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Formula:C22H29N3O4SPurity:99.96%Color and Shape:Yellowish White Crystalline PowderMolecular weight:431.55Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formula:C9H10Cl3N3Purity:99.16% - 99.86%Color and Shape:SolidMolecular weight:266.55Upidosin
CAS:Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.Formula:C31H33N3O4Purity:99.66%Color and Shape:SolidMolecular weight:511.619-Cyclopentyladenine
CAS:9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signalingFormula:C10H13N5Purity:99.98%Color and Shape:White SolidMolecular weight:203.24Naftopidil
CAS:Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-Formula:C24H28N2O3Purity:99.60% - 99.97%Color and Shape:SolidMolecular weight:392.49Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Formula:C25H32F3N3O4Purity:99.28% - 99.76%Color and Shape:White SolidMolecular weight:495.53Ref: TM-T1504
1500mgTo inquire5mg34.00€1mL*10mM (DMSO)35.00€10mg50.00€25mg73.00€50mg92.00€100mg99.00€200mg126.00€Fluvoxamine maleate
CAS:Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFormula:C19H25F3N2O6Purity:99.92% - 99.94%Color and Shape:White SolidMolecular weight:434.41Ref: TM-T1077
1mL*10mM (DMSO)35.00€10mg49.00€25mg65.00€50mg80.00€100mg109.00€200mg161.00€500mg263.00€Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formula:C21H24ClNOPurity:99.77% - 99.99%Color and Shape:White SolidMolecular weight:341.88Olanzapine
CAS:Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Formula:C17H20N4SPurity:99.86% - ≥95%Color and Shape:SolidMolecular weight:312.43
