GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,058 products)
- Adenosine Receptor(216 products)
- Adrenergic Receptor(3,265 products)
- Bombesin Receptor(37 products)
- Bradykinin Receptor(63 products)
- CXCR(179 products)
- CaSR(31 products)
- Cannabinoid Receptor(226 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(447 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(89 products)
- GPCR19(40 products)
- GRK(43 products)
- GTPase(26 products)
- Glucagon Receptor(209 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(389 products)
- LPA Receptor(22 products)
- Melatonin Receptor(26 products)
- OX Receptor(57 products)
- Opioid Receptor(337 products)
- PAFR(12 products)
- PKA(57 products)
- S1P Receptor(22 products)
- SGLT(33 products)
- Sigma receptor(49 products)
Show 19 more subcategories
Found 6055 products for "GPCR/G-Protein".
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Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Formula:C15H23N3O4SPurity:98.20% - 99.88%Color and Shape:White SolidMolecular weight:341.43Lafutidine
CAS:Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.Formula:C22H29N3O4SPurity:99.96%Color and Shape:Yellowish White Crystalline PowderMolecular weight:431.548Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Formula:C22H21Cl3N4OPurity:98% - 99.91%Color and Shape:White SolidMolecular weight:463.79Venlafaxine hydrochloride
CAS:Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Formula:C17H28ClNO2Purity:97.32% - 99.86%Color and Shape:SolidMolecular weight:313.86Serazapine
CAS:Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.Formula:C22H23N3O2Purity:99.29% - 99.97%Color and Shape:White SolidMolecular weight:361.44Fluparoxan hydrochloride
CAS:Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H11ClFNO2Purity:99.98%Color and Shape:SolidMolecular weight:231.65Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Formula:C25H32F3N3O4Purity:99.28% - 99.76%Color and Shape:White SolidMolecular weight:495.53Ref: TM-T1504
1500mgTo inquire5mg34.00€1mL*10mM (DMSO)35.00€10mg50.00€25mg73.00€50mg92.00€100mg99.00€200mg126.00€Metaproterenol hemisulfate
CAS:Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.Formula:C11H17NO3·5H2O4SPurity:98.53% - 99.74%Color and Shape:White SolidMolecular weight:260.3JNJ-18038683
CAS:JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.Formula:C26H28ClN3O7Purity:97.29%Color and Shape:SolidMolecular weight:529.97Ref: TM-T11720
2mg34.00€5mg52.00€1mL*10mM (DMSO)52.00€10mg86.00€25mg161.00€50mg245.00€100mg363.00€200mg515.00€Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formula:C23H27Cl2N3O2Purity:99.43% - 99.62%Color and Shape:White SolidMolecular weight:448.39(3aR,9aR)-Fluparoxan
CAS:(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormula:C10H10FNO2Purity:97.82%Color and Shape:SolidMolecular weight:195.19AH 6809
CAS:AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Formula:C17H14O5Purity:97.07%Color and Shape:SolidMolecular weight:298.29Ref: TM-T14148
1mg34.00€5mg63.00€1mL*10mM (DMSO)67.00€10mg92.00€25mg165.00€50mg250.00€100mg401.00€200mg580.00€KGA-2727
CAS:KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.Formula:C26H40N4O8Purity:98.46%Color and Shape:SolidMolecular weight:536.62Ref: TM-T15656
1mg109.00€2mg158.00€5mg260.00€1mL*10mM (DMSO)305.00€10mg430.00€25mg710.00€50mg973.00€100mg1,333.00€Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formula:C21H24ClNOPurity:99.77% - 99.99%Color and Shape:White SolidMolecular weight:341.88MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.Formula:C24H26F3N3O4Purity:99.98%Color and Shape:SolidMolecular weight:477.48Promazine hydrochloride
CAS:Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Formula:C17H21ClN2SPurity:99.90%Color and Shape:SolidMolecular weight:320.88Naftopidil
CAS:Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-Formula:C24H28N2O3Purity:99.60% - 99.96%Color and Shape:SolidMolecular weight:392.49Zolmitriptan
CAS:Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Formula:C16H21N3O2Purity:99.69% - 99.91%Color and Shape:White SolidMolecular weight:287.36Fluoxetine
CAS:Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.Formula:C17H18F3NOPurity:99.17% - 99.28%Color and Shape:Transparent LiquidMolecular weight:309.33Azatadine dimaleate
CAS:Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.Formula:C28H30N2O8Purity:99.7% - >99.99%Color and Shape:SolidMolecular weight:522.55
