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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5745 products of "GPCR/G-Protein"

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  • Tetrabenazine
    Targetmol
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    Tetrabenazine

    CAS:
    Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.
    Formula:C19H27NO3
    Purity:98% - 99.91%
    Color and Shape:White To Off-White White To Off-White Solid
    Molecular weight:317.42

    Ref: TM-T0719

  • Betaxolol hydrochloride
    Targetmol
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    Betaxolol hydrochloride

    CAS:
    <p>Betaxolol HCl (SL 75212) is a cardioselective beta-blocker for hypertension without reported liver injury.</p>
    Formula:C18H30ClNO3
    Purity:99.48% - 99.56%
    Color and Shape:Solid
    Molecular weight:343.89

    Ref: TM-T0226

  • Nelivaptan
    Targetmol
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    Nelivaptan

    CAS:
    <p>Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.</p>
    Formula:C30H32ClN3O8S
    Purity:98.46% - 99.89%
    Color and Shape:Solid
    Molecular weight:630.11

    Ref: TM-T28153

  • Luzindole
    Targetmol
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    Luzindole

    CAS:
    Luzindole (N-0774) is a selective melatonin receptor antagonist.
    Formula:C19H20N2O
    Purity:98.53%
    Color and Shape:Off-White Amorphous Solid
    Molecular weight:292.37

    Ref: TM-T15795

  • Ebalzotan
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    Ebalzotan

    CAS:
    <p>NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.</p>
    Formula:C19H30N2O2
    Purity:98.09% - 99.41%
    Color and Shape:Solid
    Molecular weight:318.45

    Ref: TM-T68059

  • Rebamipide
    Targetmol
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    Rebamipide

    CAS:
    Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.
    Formula:C19H15ClN2O4
    Purity:99.48% - 99.61%
    Color and Shape:White Powder
    Molecular weight:370.79

    Ref: TM-T1562

  • Vibozilimod
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    Vibozilimod

    CAS:
    Vibozilimod (SCD-044) is S1P receptor-1 (S1PR1) agonist .
    Formula:C29H36ClN3O5
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:542.07

    Ref: TM-T38826

  • Pamabrom
    Targetmol
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    Pamabrom

    CAS:
    Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.
    Formula:C11H18BrN5O3
    Purity:99.84% - >99.99%
    Color and Shape:Coa
    Molecular weight:348.2

    Ref: TM-T1230

  • Azacyclonol
    Targetmol
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    Azacyclonol

    CAS:
    Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.
    Formula:C18H21NO
    Purity:99.46%
    Color and Shape:Solid Powder
    Molecular weight:267.37

    Ref: TM-T0318

  • Roluperidone
    Targetmol
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    Roluperidone

    CAS:
    <p>Roluperidone (CYR-101) is a novel cyclic amide derivative.</p>
    Formula:C22H23FN2O2
    Purity:96.46% - 97.77%
    Color and Shape:Solid
    Molecular weight:366.43

    Ref: TM-T15034

  • Cloperastine hydrochloride
    Targetmol
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    Cloperastine hydrochloride

    CAS:
    <p>Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.</p>
    Formula:C20H25Cl2NO
    Purity:97.74% - 99.42%
    Color and Shape:Solid
    Molecular weight:366.33

    Ref: TM-T0723

  • Mirtazapine
    Targetmol
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    Mirtazapine

    CAS:
    <p>Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.</p>
    Formula:C17H19N3
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:265.35

    Ref: TM-T0137

  • DREADD agonist 21
    Targetmol
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    DREADD agonist 21

    CAS:
    <p>DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).</p>
    Formula:C17H18N4
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:278.35

    Ref: TM-T11095L

  • Seganserin
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    Seganserin

    CAS:
    <p>Seganserin, a 5-HT2 antagonist, negates fluoxetine and quipazine's effects on hyperphagia, depression, and pain.</p>
    Formula:C29H27F2N3O
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:471.54

    Ref: TM-T68141

  • Degarelix acetate(214766-78-6 free base)
    Targetmol
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    Degarelix acetate(214766-78-6 free base)

    CAS:
    Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
    Formula:C84H107ClN18O18
    Purity:98.66%
    Color and Shape:Solid
    Molecular weight:1692.34

    Ref: TM-T10988L

  • Efloxate
    Targetmol
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    Efloxate

    CAS:
    <p>Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.</p>
    Formula:C19H16O5
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:324.33

    Ref: TM-T0151

  • Promethazine
    Targetmol
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    Promethazine

    CAS:
    Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
    Formula:C17H20N2S
    Purity:99.76%
    Color and Shape:Crystals
    Molecular weight:284.42

    Ref: TM-T0445

  • Delequamine
    Targetmol
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    Delequamine

    CAS:
    Delequamine (RS 15385-197) is a TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.
    Formula:C18H26N2O3S
    Purity:99.39%
    Color and Shape:Solid
    Molecular weight:350.48

    Ref: TM-T68051

  • CymitQuimica logo
    Targetmol
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    Leronlimab

    CAS:
    <p>Leronlimab (PRO 140), a humanized IgG4 monoclonal antibody, targets CCR5 to combat HIV and cancer.</p>
    Purity:SDS-PAGE:95.0%;SEC-HPLC:99.6%
    Color and Shape:Liquid
    Molecular weight:146.66 kDa

    Ref: TM-T77059

  • Brefonalol HCl
    Targetmol
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    Brefonalol HCl

    Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.
    Formula:C22H29ClN2O2
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:388.93

    Ref: TM-T30586L