GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,003 products)
- Adenosine Receptor(247 products)
- Adrenergic Receptor(3,010 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(60 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(215 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(435 products)
- Endothelin Receptor(83 products)
- GNRH Receptor(82 products)
- GPCR19(33 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(190 products)
- Hedgehog/Smoothened(48 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(321 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5838 products of "GPCR/G-Protein"
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Takeda103A
CAS:<p>Takeda103A (CMPD103A) is the GRK2-dependent bovine tubulin oxidation effective inhibitor.</p>Formula:C24H23F2N7OPurity:97.17%Color and Shape:SolidMolecular weight:463.48Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formula:C21H26ClNPurity:99.99%Color and Shape:Crystalline SolidMolecular weight:327.90Tripelennamine citrate
CAS:Tripelennamine citrate, an ethylenediamine derivative, blocks H1 receptors to treat allergies and anaphylaxis.Formula:C22H29N3O7Color and Shape:SolidMolecular weight:447.488OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).Formula:C79H125N23O22Purity:98.52%Color and Shape:SolidMolecular weight:1748.98Brimonidine
CAS:<p>Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P.</p>Formula:C11H10BrN5Purity:99.626%Color and Shape:Yellow SolidMolecular weight:292.13SB-334867 free base
CAS:SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.Formula:C17H13N5O2Purity:99.67% - >99.99%Color and Shape:SolidMolecular weight:319.32KB-5492 anhydrous
CAS:KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.Formula:C27H34N2O10Color and Shape:SolidMolecular weight:546.576-fluoro-DL-Tryptophan
CAS:<p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>Formula:C11H11FN2O2Purity:99.25%Color and Shape:Off-White PowderMolecular weight:222.22Melanin Concentrating Hormone, salmon acetate
Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.Formula:C91H143N27O26S4Purity:99.41%Color and Shape:SolidMolecular weight:2157Sarpogrelate hydrochloride
CAS:<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Formula:C24H32ClNO6Purity:99.73%Color and Shape:Colorless LiquidMolecular weight:465.97Eprazinone dihydrochloride
CAS:Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.Formula:C24H32N2O2·2HClPurity:99.25%Color and Shape:A White Or Almost White CrysMolecular weight:453.44Senktide
CAS:<p>Senktide is an agonist of tachykinin NK3 receptor.</p>Formula:C40H55N7O11SPurity:99.84% - >99.99%Color and Shape:White PowderMolecular weight:841.97Azaperone
CAS:Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.Formula:C19H22FN3OPurity:98.73%Color and Shape:White Or Off-White CrystallineMolecular weight:327.4Dexmedetomidine
CAS:Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.Formula:C13H16N2Purity:99% - >99.99%Color and Shape:SolidMolecular weight:200.28JNJ-31020028
CAS:<p>JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).</p>Formula:C34H36FN5O2Purity:95.92% - 99.65%Color and Shape:SolidMolecular weight:565.68Amylin, amide, rat acetate(124447-81-0,free base)
Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 receptors and variably of AMY2 receptors.Formula:C169H276N52O55S2Purity:98.93%Color and Shape:SolidMolecular weight:3980.45Piperoxan hydrochloride
CAS:Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.Formula:C14H20ClNO2Purity:99.61%Color and Shape:SolidMolecular weight:269.77Isocorynoxeine
CAS:Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Formula:C22H26N2O4Purity:98% - 99.9%Color and Shape:SolidMolecular weight:382.45HAEGTFTSDVSSYLE
<p>HAEGTFTSDVSSYLE is a peptide. GLP-I analog contains the sequence.</p>Formula:C71H103N17O28Purity:>99.99%Color and Shape:SolidMolecular weight:1642.71Cilansetron Hydrochloride
CAS:Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Formula:C20H24ClN3O2Color and Shape:SolidMolecular weight:373.88GLP-1(7-37) acetate(106612-94-6 free base)
CAS:<p>Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.</p>Formula:C151H228N40O47Purity:98.89%Color and Shape:SolidMolecular weight:3355.67Rizatriptan sulfate
CAS:Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Formula:C15H21N5O4SColor and Shape:SolidMolecular weight:367.42BRL-15572 hydrochloride
CAS:<p>BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.</p>Formula:C25H28Cl2N2OColor and Shape:SolidMolecular weight:443.41Relenopride hydrochloride
CAS:Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.Formula:C24H31Cl2FN4O4Color and Shape:SolidMolecular weight:529.43RFRP3(human) acetate(311309-27-0 free base)
RFRP-3(human) acetate inhibits gonadotropin, blocks Ca2+ mobilization, acts on NPFF1 receptors, and has an IC50 of 0.7 nM against cAMP production.Formula:C47H76N14O12Purity:97.09%Color and Shape:SolidMolecular weight:1029.19Vericiguat
CAS:<p>Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.</p>Formula:C19H16F2N8O2Purity:98.86% - 99.93%Color and Shape:SolidMolecular weight:426.38WIN 55,212-2 Mesylate
CAS:WIN 55,212-2 Mesylate ((R)-(+)-WIN 55212) is a potent aminoalkylindole cannabinoid (CB) receptor agonist with Kis of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively. Cannabinoid analogue WIN 55,212-2 Mesylate exhibited a novel anticancer effect against human tumors.Formula:C28H30N2O6SPurity:98% - 99.71%Color and Shape:White To Off-White SolidMolecular weight:522.61[Leu31,Pro34]-Neuropeptide Y (porcine)
CAS:[Leu31,Pro34]-Neuropeptide Y (porcine), is a selective and high affinity agonist of neuropeptide Y (NPY) Y1 receptor with anxiolytic effects.Formula:C190H286N54O56Purity:99.39%Color and Shape:SolidMolecular weight:42231-(1-Naphthyl) piperazine hydrochloride
CAS:<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Formula:C14H17ClN2Purity:98.27%Color and Shape:SolidMolecular weight:248.75ML-031
CAS:ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.Formula:C19H20N2O3Purity:99.21%Color and Shape:SolidMolecular weight:324.37Ralinepag
CAS:Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human andFormula:C23H26ClNO5Purity:99.79% - 99.85%Color and Shape:SolidMolecular weight:431.91Tianeptine sodium salt
CAS:<p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。</p>Formula:C21H24ClN2NaO4SPurity:99.82%Color and Shape:SolidMolecular weight:458.93Parmodulin 2
CAS:<p>ML161 (Parmodulin 2) inhibits PAR1, blocking platelet activation and thrombin-induced activity (IC50: 0.26μM).</p>Formula:C17H17BrN2O2Purity:97.35% - 99.95%Color and Shape:SolidMolecular weight:361.23E7046
CAS:E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.Formula:C22H18F5N3O4Purity:99.86%Color and Shape:SolidMolecular weight:483.4Cerlapirdine hydrochloride
CAS:Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Formula:C22H24ClN3O3SColor and Shape:SolidMolecular weight:445.96SKF 38393 hydrochloride
CAS:<p>SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.</p>Formula:C16H17NO2·HClPurity:99.1% - 99.51%Color and Shape:SolidMolecular weight:291.77SB 242084 dihydrochloride
CAS:SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.Formula:C21H21Cl3N4O2Color and Shape:SolidMolecular weight:467.78idalopirdine
CAS:Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Formula:C20H19F5N2OPurity:99.73%Color and Shape:SolidMolecular weight:398.37Dobutamine hydrochloride
CAS:<p>Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.</p>Formula:C18H24ClNO3Purity:97.15% - 99.94%Color and Shape:SolidMolecular weight:337.84Montelukast sodium
CAS:<p>Montelukast sodium (MK0476), an oral leukotriene antagonist for asthma, can cause rare liver injury.</p>Formula:C35H35ClNNaO3SPurity:99.14% - 99.89%Color and Shape:White To Off-White Crystalline PowderMolecular weight:608.17Rimegepant
CAS:View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.Formula:C28H28F2N6O3Purity:99.1% - 99.99%Color and Shape:SolidMolecular weight:534.56Betazole dihydrochloride
CAS:<p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>Formula:C5H11Cl2N3Purity:99.12%Color and Shape:SolidMolecular weight:184.067L-745870 hydrochloride
CAS:<p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>Formula:C18H20Cl2N4Purity:97.36%Color and Shape:SolidMolecular weight:363.28MEN 10207 acetate
MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.Formula:C59H72N14O12Purity:99.18%Color and Shape:SolidMolecular weight:1169.29Alprenolol hydrochloride
CAS:<p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>Formula:C15H24ClNO2Purity:99.79%Color and Shape:SolidMolecular weight:285.817-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Formula:C10H6F3NO2Purity:97.31% - 97.84%Color and Shape:Yellow PowderMolecular weight:229.16(+)-PD 128907 hydrochloride
CAS:<p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>Formula:C14H20ClNO3Purity:97.76%Color and Shape:SolidMolecular weight:285.77MK-571 sodium
CAS:MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.Formula:C26H27ClN2O3S2·NaPurity:97.86% - 99.58%Color and Shape:SolidMolecular weight:537.07Olanzapine HCl
CAS:Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Formula:C17H21ClN4SColor and Shape:SolidMolecular weight:348.89Ibutamoren Mesylate
CAS:<p>Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.</p>Formula:C28H40N4O8S2Purity:97.98% - ≥98%Color and Shape:SolidMolecular weight:624.77Pirenperone
CAS:<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Formula:C23H24FN3O2Purity:99.2%Color and Shape:SolidMolecular weight:393.45Buserelin Acetate (57982-77-1 free base)
CAS:<p>Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).</p>Formula:C62H90N16O15Purity:99.31% - 99.78%Color and Shape:SolidMolecular weight:1299.48Prazosin
CAS:<p>Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.</p>Formula:C19H21N5O4Purity:99.86%Color and Shape:White To Tan Powder SolidMolecular weight:383.4Mecamylamine hydrochloride
CAS:<p>Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.</p>Formula:C11H22ClNPurity:99.76% - >99.99%Color and Shape:White SolidMolecular weight:203.75ICI 89406
CAS:ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.Formula:C19H22N4O3Purity:99.92%Color and Shape:SolidMolecular weight:354.4Terazosin hydrochloride dihydrate
CAS:<p>Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).</p>Formula:C19H25N5O4·HCl·2H2OPurity:99.81%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:459.92Galanin (1-16), mouse, porcine, rat
CAS:Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons.Formula:C78H116N20O21Purity:98.65%Color and Shape:White PowderMolecular weight:1669.88Spiperone hydrochloride
CAS:5-HT2A serotonin and selective D2-like dopamine receptor antagonistFormula:C23H27ClFN3O2Purity:98%Color and Shape:SolidMolecular weight:431.93β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.Formula:C120H178N34O37SPurity:99.64%Color and Shape:SolidMolecular weight:2720.97Azepexole
CAS:Azepexole is a selective α2-adrenoceptor agonist that exhibits greater than 300-fold selectivity for the α2-adrenoceptor over the α1-adrenoceptor.Formula:C9H15N3OColor and Shape:SolidMolecular weight:181.23Tetracosactide acetate
CAS:Cosyntropin (acetate) stimulates the release of corticosteroids such as cortisol from the adrenal gland.Formula:C138H214N40O33SPurity:99.76%Color and Shape:SolidMolecular weight:2993.54BPTU
CAS:<p>BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).</p>Formula:C23H22F3N3O3Purity:99.37% - 99.89%Color and Shape:SolidMolecular weight:445.43Bay 59-3074
CAS:<p>Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).</p>Formula:C18H13F6NO4SPurity:97.68% - 99.69%Color and Shape:SolidMolecular weight:453.36Epinastine
CAS:Epinastine (WAL801) is an antihistamine, mast cell stabilizer, and H1 antagonist with anti-allergic properties.Formula:C16H15N3Purity:99.94%Color and Shape:SolidMolecular weight:249.31Nomifensine maleate
CAS:<p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>Formula:C20H22N2O4Purity:98.46%Color and Shape:SolidMolecular weight:354.4MHP
CAS:MHP (Methyl caprooyl tyrosinate) is an activator of sphingosine kinase (SPHK1), and significantly stimulates CAMP mRNA and protein production in KC.Formula:C16H23NO4Purity:98.58%Color and Shape:SolidMolecular weight:293.36SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formula:C17H19Cl2NOPurity:98% - 99.83%Color and Shape:SolidMolecular weight:324.24Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formula:C21H33Cl3N4OPurity:99.78% - >99.99%Color and Shape:SolidMolecular weight:463.87ABT-702 dihydrochloride
CAS:ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.Formula:C22H21BrCl2N6OPurity:98.42% - 98.98%Color and Shape:SolidMolecular weight:536.25Irdabisant hydrochloride
CAS:<p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>Formula:C18H24ClN3O2Color and Shape:SolidMolecular weight:349.86Blarcamesine
CAS:<p>Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.</p>Formula:C19H23NOPurity:99.87%Color and Shape:SolidMolecular weight:281.39Mosapride Citrate
CAS:Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.Formula:C21H25ClFN3O3·C6H8O7Purity:99.70%Color and Shape:White PowderMolecular weight:614.02Exendin-4
CAS:<p>Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.</p>Formula:C184H282N50O60SPurity:97.71% - 99.78%Color and Shape:SolidMolecular weight:4186.57Desipramine
CAS:<p>Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.</p>Formula:C18H22N2Color and Shape:SolidMolecular weight:266.38Hemokinin 1 (mouse) acetate(208041-90-1 free base)
<p>Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.</p>Formula:C63H104N22O17SPurity:98.33%Color and Shape:SolidMolecular weight:1473.72Tasimelteon
CAS:<p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>Formula:C15H19NO2Purity:98.93% - 99.93%Color and Shape:SolidMolecular weight:245.32GW 405833
CAS:GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFormula:C23H24Cl2N2O3Purity:99.82% - 99.93%Color and Shape:SolidMolecular weight:447.35Hydroxyzine
CAS:<p>Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.</p>Formula:C21H27ClN2O2Purity:99.54% - ≥95%Color and Shape:Oil SolidMolecular weight:374.9Siponimod hemifumarate
CAS:Siponimod (BAF-312) is a potent S1P receptor modulator for multiple sclerosis research.Formula:C62H74F6N4O10Color and Shape:SolidMolecular weight:1149.282Olodaterol hydrochloride
CAS:<p>Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist that exerts its pharmacological effect by binding and activating β2-AR.</p>Formula:C21H27ClN2O5Purity:99.11%Color and Shape:SolidMolecular weight:422.9Pramlintide acetate(151126-32-8 free base)
CAS:<p>Pramlintide acetate is a polypeptide analogue of human amylin. It serves as an antidiabetic agent and exhibits antineoplastic activity in colorectal cancer.</p>Formula:C173H271N51O55S2Purity:>99.99%Color and Shape:SolidMolecular weight:4009ML401
CAS:ML401 is a selectively EBI2(GPR183) receptor antagonist(IC50 of 1.03 nM) .Formula:C20H20BrClN2OPurity:99.13%Color and Shape:SolidMolecular weight:419.74Carcinine ditrifluoroacetate Acetate
<p>Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.</p>Formula:C14H20F6N4O7Purity:98.18%Color and Shape:SolidMolecular weight:470.32GUANABENZ
CAS:GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.Formula:C8H8Cl2N4Purity:98.31%Color and Shape:White Solid From Acetonitrile SolidMolecular weight:231.08ACH-000143
CAS:ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Formula:C13H16ClN3O3Purity:98.15%Color and Shape:SolidMolecular weight:297.74Bexagliflozin
CAS:<p>Bexagliflozin (EGT1442) is a potent, selective sodium glucose co-transporter 2 (SGLT2) inhibitor with IC50 values of 2 nM for human SGLT2.</p>Formula:C24H29ClO7Purity:98.99% - 99.89%Color and Shape:SolidMolecular weight:464.94Puerarin
CAS:<p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>Formula:C21H20O9Purity:98.90% - 99.21%Color and Shape:Yellow Brown Fine PowderMolecular weight:416.38Exo1
CAS:Exo1 is an inhibitor of the exocytic pathwayFormula:C15H12FNO3Purity:98.75%Color and Shape:SolidMolecular weight:273.26Adrenocorticotropic Hormone (ACTH) (4-10) TFA
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .Formula:C46H60F3N13O12SPurity:98.49%Color and Shape:SolidMolecular weight:1076.12A2B receptor antagonist 2
CAS:<p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>Formula:C12H15N5Purity:100%Color and Shape:SolidMolecular weight:229.28Bosentan (hydrate)
CAS:Bosentan hydrate (Ro 47-0203) is a competitive and dual antagonist of endothelin-1 at the endothelin-A (ET-A) and endothelin-B (ET-B) receptors.Formula:C27H29N5O6S·H2OPurity:99.31% - 99.86%Color and Shape:White PowderMolecular weight:569.63Atrasentan sodium
CAS:Atrasentan (ABT-627) is an oral ETA receptor blocker with potential cancer-fighting properties, inhibiting angiogenesis and tumor growth.Formula:C29H37N2NaO6Color and Shape:SolidMolecular weight:532.61Terutroban
CAS:<p>Terutroban, a thromboxane prostaglandin receptor antagonist, affects the progression of atherosclerosis.</p>Formula:C20H22ClNO4SPurity:99.53%Color and Shape:SolidMolecular weight:407.91Tiapride
CAS:<p>Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.</p>Formula:C15H24N2O4SColor and Shape:SolidMolecular weight:328.43Rolapitant hydrochloride hydrate
CAS:Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.Formula:C25H29ClF6N2O3Color and Shape:SolidMolecular weight:554.95Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formula:C10H8N6OColor and Shape:SolidMolecular weight:228.21Phenylephrine
CAS:<p>Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).</p>Formula:C9H13NO2Purity:99.5% - 99.89%Color and Shape:SolidMolecular weight:167.21Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormula:C22H15F3N2O7SPurity:99.33%Color and Shape:SolidMolecular weight:508.42Bradykinin (acetate)
CAS:Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Formula:C52H77N15O13Purity:>99.99%Color and Shape:SolidMolecular weight:1120.26Etilevodopa hydrochloride
CAS:Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.Formula:C11H16ClNO4Purity:95.00%Color and Shape:SolidMolecular weight:261.7Mesdopetam hemitartrate
CAS:Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.Formula:C28H42F2N2O12S2Purity:99.98%Color and Shape:SolidMolecular weight:700.77ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE
CAS:<p>ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE targets the prostaglandin E2 receptor EP2 subtype (human)</p>Formula:C14H15NO2SPurity:99.98%Color and Shape:SolidMolecular weight:261.34ARC-239
CAS:<p>ARC-239 is an agonist of α2-adrenergic receptor.</p>Formula:C24H29N3O3Color and Shape:SolidMolecular weight:407.514F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Formula:C22H26FNO·C2H2O4Purity:97.34%Color and Shape:SolidMolecular weight:429.49Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formula:C19H25NOSPurity:98.08% - 99.59%Color and Shape:SolidMolecular weight:315.47Isoxsuprine Free Base
CAS:Isoxsuprine Free Base relaxes uterine/vascular muscles, dilates arteries, treats peripheral vascular disease, and premature labor.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38Clozapine N-Oxide
CAS:View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Formula:C18H19ClN4OPurity:98.65% - 99.94%Color and Shape:SolidMolecular weight:342.82Doxazosin
CAS:<p>Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.</p>Formula:C23H25N5O5Purity:99.47% - 99.87%Color and Shape:SolidMolecular weight:451.48Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formula:C68H87N17O15Purity:99.98%Color and Shape:SolidMolecular weight:1382.55ZM241385
CAS:<p>ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.</p>Formula:C16H15N7O2Purity:97.02% - 99.69%Color and Shape:SolidMolecular weight:337.34PAR-2-IN-1
CAS:<p>PAR-2-IN-1 (IUN76750) is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.</p>Formula:C12H14ClN3O2Purity:99.75%Color and Shape:SolidMolecular weight:267.71Intepirdine
CAS:<p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>Formula:C19H19N3O2SPurity:98% - 98.63%Color and Shape:SolidMolecular weight:353.44RO1138452
CAS:RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).Formula:C19H23N3OPurity:97.01% - 99.34%Color and Shape:SolidMolecular weight:309.41BAY 41-8543
CAS:<p>BAY 41-8543 is a nitric oxide (NO)-independent stimulator of soluble guanylyl cyclase (sGC).</p>Formula:C21H21FN8OPurity:99.86%Color and Shape:SolidMolecular weight:420.44Enavogliflozin
CAS:<p>Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.</p>Formula:C24H27ClO6Purity:97.37%Color and Shape:SolidMolecular weight:446.92Haloperidol lactate
CAS:Haloperidol lactate: a potent antipsychotic for acute/chronic schizophrenia and polyarousal syndrome research.Formula:C24H29ClFNO5Color and Shape:SolidMolecular weight:465.95Renzapride hydrochloride
CAS:Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors.Formula:C16H23Cl2N3O2Color and Shape:SolidMolecular weight:360.28Thonzylamine
CAS:<p>Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.</p>Formula:C16H22N4OPurity:99.45%Color and Shape:SolidMolecular weight:286.37Alcaftadine
CAS:<p>Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.</p>Formula:C19H21N3OPurity:98% - 98.65%Color and Shape:SolidMolecular weight:307.39Evatanepag sodium
CAS:Evatanepag (CP-533536), an EP2-specific PGE2 agonist, promotes bone growth and heals fractures in rats with a single dose.Formula:C25H27N2NaO5SColor and Shape:SolidMolecular weight:490.55Dasotraline
CAS:Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.Formula:C16H15Cl2NColor and Shape:SolidMolecular weight:292.2Regadenoson hydrate
CAS:Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.Formula:C15H20N8O6Purity:98%Color and Shape:SolidMolecular weight:408.37Temanogrel hydrochloride
CAS:Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.Formula:C24H29ClN4O4Color and Shape:SolidMolecular weight:472.97T-1095
CAS:T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) and facilitative glucose transporter 2 (GLUT2).Formula:C26H28O11Purity:99.78%Color and Shape:SolidMolecular weight:516.49GR 125743
CAS:GR 125743 is a novel antagonist of 5-HT1B/1D receptor.Formula:C25H28N4O2Purity:99.76%Color and Shape:SolidMolecular weight:416.52GW842166X
CAS:<p>GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.</p>Formula:C18H17Cl2F3N4O2Purity:99.47%Color and Shape:SolidMolecular weight:449.25lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formula:C31H36FN3O4SPurity:95.83% - 99.95%Color and Shape:SolidMolecular weight:565.7Bindarit
CAS:<p>Bindarit is a selective inhibitor of monocyte chemoattractant proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.Cost-effective and quality-assured.</p>Formula:C19H20N2O3Purity:98.35% - 98.55%Color and Shape:SolidMolecular weight:324.37Xamoterol
CAS:Xamoterol is a cardiac stimulant.Formula:C16H25N3O5Color and Shape:SolidMolecular weight:339.39PAR-4 Agonist Peptide, amide TFA
CAS:PAR-4 agonist peptide doesn't affect PAR-1/PAR-2; blocked by PAR-4 antagonist.Formula:C36H49F3N8O9Purity:99.72%Color and Shape:SolidMolecular weight:794.82JNJ-10229570
CAS:<p>JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland</p>Formula:C22H19N3O2SPurity:98.41%Color and Shape:SolidMolecular weight:389.47N-ACETYLTRYPTAMINE
CAS:<p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>Formula:C12H14N2OPurity:98.79%Color and Shape:PowderMolecular weight:202.25Tesmilifene fumarate
CAS:Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。Formula:C23H29NO5Purity:99.86%Color and Shape:SolidMolecular weight:399.48Alimemazine hemitartrate
CAS:Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formula:C18H22N2SC4H6O6Purity:98.16% - 99.69%Color and Shape:SolidMolecular weight:448.53Protease-Activated Receptor-1, PAR-1 Agonist acetate
PAR-1 Agonist acetate is a selective PAR-1 agonist that mimics thrombin action.Formula:C37H62N10O11Purity:98.1800%Color and Shape:SolidMolecular weight:822.95PD 168568
CAS:PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.Formula:C22H27N3OColor and Shape:SolidMolecular weight:349.47Bradykinin (2-9)
CAS:Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.Formula:C44H61N11O10Purity:>99.99%Color and Shape:SolidMolecular weight:904.02Clebopride
CAS:Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.Formula:C20H24ClN3O2Color and Shape:SolidMolecular weight:373.88NGB 2904
CAS:NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Formula:C28H29Cl2N3OPurity:98.79%Color and Shape:SolidMolecular weight:494.46S 14506 HCl
CAS:S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).Formula:C24H26FN3O2Color and Shape:SolidMolecular weight:407.48Pimavanserin
CAS:<p>Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.</p>Formula:C25H34FN3O2Purity:97.84% - 99.69%Color and Shape:Pale Yellow To Pale Orange SolidMolecular weight:427.55Substance P 1-9 aceate
Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.Formula:C54H81N15O14Purity:99.01%Color and Shape:SolidMolecular weight:1164.31Cinacalcet hydrochloride
CAS:<p>Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-</p>Formula:C22H23ClF3NPurity:99.96% - >99.99%Color and Shape:Off-White To Tan SolidMolecular weight:393.87CP 376395
CAS:CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist.Formula:C21H30N2OPurity:99.86% - 99.94%Color and Shape:SolidMolecular weight:326.48GSK2018682
CAS:<p>GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).</p>Formula:C22H21ClN4O4Purity:99.04%Color and Shape:SolidMolecular weight:440.88Napitane Mesylate
CAS:Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.Formula:C23H29NO5SPurity:98%Color and Shape:SolidMolecular weight:431.55Apraclonidine
CAS:Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.Formula:C9H10Cl2N4Color and Shape:SolidMolecular weight:245.11[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 andFormula:C76H103N21O18SPurity:99.75%Color and Shape:SolidMolecular weight:1630.82Tafluprost
CAS:Tafluprost, a prostaglandin analog, is the selective agonist of fluoroprostaglandin (FP) receptor PGF2α.Formula:C25H34F2O5Purity:97.7% - 99.67%Color and Shape:LiquidMolecular weight:452.53Etrasimod
CAS:Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).Formula:C26H26F3NO3Purity:98.52% - 99.73%Color and Shape:SolidMolecular weight:457.48Brexpiprazole HCl
CAS:Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.Formula:C25H27N3O2S·xHClPurity:99.05%Color and Shape:SolidMolecular weight:433.6Pardoprunox hydrochloride
CAS:Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)Formula:C12H16ClN3O2Purity:98.95% - 99.13%Color and Shape:SolidMolecular weight:269.73CJC-1295 acetate(863288-34-0 free base)
CJC-1295 acetate is a synthetic GHRH analogue and GHS.Formula:C154H256N44O44Purity:97.29%Color and Shape:SolidMolecular weight:3428.01AM281
CAS:AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.Formula:C21H19Cl2IN4O2Purity:98.6% - >99.99%Color and Shape:White To Off-White SolidMolecular weight:557.21PEN (human) aceate
PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein ProSAAS, is an endogenous ligand of GPR83.Formula:C99H163N27O34Purity:99.25%Color and Shape:SolidMolecular weight:2275.51ACTH 11-24 acetate(4237-93-8 free base)
CAS:ACTH 11-24 acetate is a cortisol-stimulating adrenocorticotrophin fragment and a competitive antagonist of ACTH 1-39 and 1-10.Formula:C79H138N24O18Purity:>99.99%Color and Shape:SolidMolecular weight:1712.12CYM 50358 hydrochloride (1314212-39-9 free base)
CAS:CYM50358 HCl is an S1P4 antagonist.Formula:C20H19Cl3N2O2Purity:99.57%Color and Shape:SolidMolecular weight:425.73Laropiprant sodium
<p>Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.</p>Color and Shape:SolidPNU 22394 hydrochloride
CAS:PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonistFormula:C13H17ClN2Purity:97.83%Color and Shape:SolidMolecular weight:236.74ANP(1-28) Acetate (human, porcine)
CAS:<p>Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.</p>Formula:C129H207N45O41S3Purity:98.24%Color and Shape:SolidMolecular weight:3140.5CYN 154806 TFA
CAS:<p>CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.</p>Formula:C58H69F3N12O16S2Purity:99.7%Color and Shape:SolidMolecular weight:1311.36BAR501
CAS:BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。Formula:C26H46O3Purity:99.29% - 99.68%Color and Shape:SolidMolecular weight:406.64Tecalcet Free Base
CAS:Tecalcet Free Base is an oral calcium receptor agonistFormula:C18H22ClNOColor and Shape:SolidMolecular weight:303.83Alosetron (Hydrochloride(1:X))
CAS:<p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>Formula:C17H18ClN4OColor and Shape:SolidMolecular weight:329.11691TG6-10-1
CAS:TG6-10-1 is an EP2 antagonist.Formula:C23H23F3N2O4Purity:99.66% - ≥95%Color and Shape:SolidMolecular weight:448.43Ganirelix Acetate
CAS:Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFormula:C82H117ClN18O15Purity:96.05%Color and Shape:SolidMolecular weight:1630.4Taminadenant
CAS:<p>Taminadenant is an adenosine receptor antagonist.</p>Formula:C10H8BrN7Purity:99.11%Color and Shape:SolidMolecular weight:306.12CPI-444
CAS:CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.Formula:C20H21N7O3Purity:98.78%Color and Shape:SolidMolecular weight:407.43CID 16020046
CAS:<p>CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.</p>Formula:C25H19N3O4Purity:99.03%Color and Shape:SolidMolecular weight:425.44Riociguat
CAS:Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth muscle and is used to treat severe pulmonary arterialFormula:C20H19FN8O2Purity:99.28% - 99.95%Color and Shape:SolidMolecular weight:422.42Mozavaptan
CAS:Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.Formula:C27H29N3O2Purity:98.98% - 99.12%Color and Shape:SolidMolecular weight:427.54Betaxolol
CAS:Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.Formula:C18H29NO3Purity:99.01%Color and Shape:White Crystalline SolidMolecular weight:307.43PF-06882961 Tris
CAS:PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C35H41FN6O7Purity:98.74% - 99.79%Color and Shape:SolidMolecular weight:676.7Neuropeptide SF(mouse,rat) acetate
Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) & 12.1 nM (NPFF2), enhancing ASIC3 current.Formula:C42H69N13O12Purity:98.37%Color and Shape:SolidMolecular weight:948.08Dimemorfan phosphate
CAS:<p>Dimemorfan phosphate (3,17-dimethylmorphinan) is a sigma 1 receptor agonist. Dimemorfan phosphate is used as a potent antitussive.</p>Formula:C18H25N·H3O4PPurity:99.65%Color and Shape:SolidMolecular weight:353.4Cinanserin
CAS:Cinanserin is a serotonin 5-HT2 antagonist.Formula:C20H24N2OSColor and Shape:SolidMolecular weight:340.48NIBR189
CAS:<p>NIBR189 is a potent and selective antagonist of EBI2 (GPR183) receptor (IC50 of 11 and 15 nM for human and mouse EBI2 receptors, respectively)</p>Formula:C21H21BrN2O3Purity:97%Color and Shape:ColourlessMolecular weight:429.31Talnetant
CAS:Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and modulate dopamine.Formula:C25H22N2O2Purity:97.88%Color and Shape:SolidMolecular weight:382.45Eprazinone
CAS:Erazinone is a mucus dissolver and bronchospasm reliever.Formula:C24H32N2O2Color and Shape:SolidMolecular weight:380.52Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Formula:C20H20ClF5N2OPurity:99.77%Color and Shape:SolidMolecular weight:434.83Neuropeptide EI, rat acetate
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.Formula:C65H102N16O25Purity:95.55%Color and Shape:SolidMolecular weight:1507.6Fexofenadine
CAS:Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Formula:C32H39NO4Purity:99.35%Color and Shape:White To Off-White SolidMolecular weight:501.66Betazole
CAS:Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.Formula:C5H9N3Color and Shape:SolidMolecular weight:111.15Ipragliflozin
CAS:<p>Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.</p>Formula:C21H21FO5SPurity:99.38% - 99.70%Color and Shape:SolidMolecular weight:404.45Mebhydrolin
CAS:<p>Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.</p>Formula:C19H20N2Purity:99.3% - ≥98%Color and Shape:SolidMolecular weight:276.38Risperidone hydrochloride
CAS:Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).Formula:C23H28ClFN4O2Color and Shape:SolidMolecular weight:446.95Tropisetron
CAS:Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.Formula:C17H20N2O2Purity:99.68%Color and Shape:White SolidMolecular weight:284.35Exo-1
CAS:Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism of various nutrients, asFormula:C15H12FNO3Purity:99.45%Color and Shape:SolidMolecular weight:273.26Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Formula:C18H18ClNOSPurity:99.78%Color and Shape:SolidMolecular weight:331.86LGnRH-III, lamprey acetate(147859-97-0 free base)
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretionFormula:C61H78N18O16Purity:99.66%Color and Shape:SolidMolecular weight:1319.385-Iodotubercidin
CAS:<p>5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.</p>Formula:C11H13IN4O4Purity:99.98%Color and Shape:Tan SolidMolecular weight:392.15SB399885
CAS:<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Formula:C18H21Cl2N3O4SPurity:98.94%Color and Shape:SolidMolecular weight:446.35Glucagon (19-29), human acetate
Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.Formula:C63H93N15O20SPurity:98.11%Color and Shape:SolidMolecular weight:1412.57Cinaciguat hydrochloride
CAS:Cinaciguat( BAY582667, BAY58-2667) is a soluble guanosine cyclase activator that can prevent cardiac dysfunction in rat models of type 1 diabetes.Formula:C36H40ClNO5Color and Shape:SolidMolecular weight:602.17Bosentan
CAS:Bosentan is a competitive endothelin receptor antagonist, used for treating pulmonary arterial hypertension.Formula:C27H29N5O6SPurity:99.74% - 99.84%Color and Shape:Pale Yellow To Off-White SolidMolecular weight:551.614Syk Inhibitor II dihydrochloride dihydrate
CAS:Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.Formula:C14H21Cl2F3N6O3Color and Shape:SolidMolecular weight:449.26Naftopidil dihydrochloride
CAS:Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.Formula:C24H28N2O3·2HClPurity:99.76%Color and Shape:White SolidMolecular weight:465.41α-MSH
CAS:α-MSH (MSH, amide) is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.Formula:C77H109N21O19SPurity:99.10% - 99.67%Color and Shape:White PowderMolecular weight:1664.89SLF1081851 TFA
CAS:SLF1081851 (TFA) inhibits Spns2, IC50 at 1.93 μM for S1P release, crucial for development and immunity.Formula:C23H34F3N3O3Color and Shape:SolidMolecular weight:457.538ABT-724
CAS:ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)Formula:C17H19N5Purity:99.73%Color and Shape:SolidMolecular weight:293.37
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